Theophylline, which is used mostly in asthma, is also contraindicated.[citation needed] Erythromycin and doxycycline can have a ...
... information about the value of theophylline and other methylxanthines as prophylaxis against exercise-induced asthma. The use ... The name 'theophylline' derives from "Thea"-the former genus name for tea + Legacy Greek φύλλον (phúllon, "leaf") + -ine. The ... Theophylline, also known as 1,3-dimethylxanthine, is a drug that inhibits phosphodiesterase and blocks adenosine receptors. It ... Theophylline and other methylxanthines are often used for their performance-enhancing effects in sports, as these drugs ...
Like theophylline, it is a xanthine derivative. Doxophylline is used to treat chronic respiratory diseases such as asthma and ... In animal and human studies, it has shown similar efficacy to theophylline but with significantly fewer side effects. In ... From a pharmacokinetic point of view, doxofylline importantly differs from theophylline also because it lacks the ability to ... theophylline" (PDF). Expert Review of Pharmacoeconomics & Outcomes Research. 17 (5): 503-510. doi:10.1080/14737167.2017.1301815 ...
"Concomitant bitolterol mesylate aerosol and theophylline for asthma therapy, with 24 hr electrocardiographic monitoring". The ... Nathan RA, Bodman SF, Storms WW, Mingo TS (June 1986). "Bitolterol mesylate aerosol in adults with steroid-dependent asthma: a ... The drug, alone or in co-administration with theophylline, doesn't show cardiotoxic effect. The U.S. Food and Drug ... Chemistry, pharmacokinetics, pharmacodynamics, adverse effects and clinical efficacy in asthma". Pharmacotherapy. 5 (3): 127- ...
... and is used to treat asthma. The therapeutic dose of theophylline, however, is many times greater than the levels attained from ... Some people use caffeine-containing beverages such as coffee or tea to try to treat their asthma. Evidence to support this ... The weak stimulant effect of chocolate may be due to a combination of theobromine and theophylline, as well as caffeine. A ... Welsh EJ, Bara A, Barley E, Cates CJ (January 2010). Welsh EJ (ed.). "Caffeine for asthma". The Cochrane Database of Systematic ...
Its most common use is in the treatment of airway obstruction from asthma or COPD. Aminophylline is a nonselective adenosine ... It is more soluble in water than theophylline. White or slightly yellowish granules or powder, having a slight ammoniacal odor ... Intravenous aminophylline can be used for acute exacerbation of symptoms and reversible airway obstruction in asthma and other ... Aminophylline can lead to theophylline toxicity. Aminophylline has been found to decrease the sedative effects of propofol and ...
The combination of theophylline and ephedrine was first used in the 1940s as a treatment for asthma, and the addition of a ... "Global Strategy for Asthma Management and Prevention". Global Initiative for Asthma. "FDA Announces Final Rule on Ephedrine ... Theophylline relaxes the bronchial smooth muscle and pulmonary artery smooth muscle. In addition, it also reduces the airway ... Tedral was first marketed by the pharmaceutical company Eli Lilly and Company in the 1950s as a treatment for asthma and other ...
Treatments with corticosteroids and theophylline for inflammatory lung diseases interfere with HAT/HDAC activity to turn off ... gene expression data demonstrated increased activity of HAT and decreased level of HDAC activity in patients with Asthma. ...
It should be used in patients 12 years of age and older with or without concurrent theophylline and/or inhaled corticosteroid. ... Pirbuterol is used in asthma for reversal of acute bronchospasm, and also as a maintenance medication to prevent future attacks ... is a short-acting β2 adrenoreceptor agonist with bronchodilating action used in the treatment of asthma, available (as ...
... and the drug theophylline used in asthma patients are known to cause lower intestinal sphincter relaxation. Gastro-esophageal ... Asthma is a respiratory disease that can begin or worsen due to exposure at work and is characterized by episodic narrowing of ... Occupational asthma has a variety of causes, including sensitization to a specific substance, causing an allergic response; or ... Exposure to various substances can also worsen pre-existing asthma. People who work in isocyanate manufacturing, who use latex ...
... derivative that was introduced in hope of being a long-acting replacement for theophylline in the treatment of asthma. It is an ...
Available in oral and injectable form, theophylline is a long-acting bronchodilator that prevents asthma episodes. It belongs ... However, it will not stop an asthma attack already in progress. Because it has no effect on asthma symptoms when used alone, it ... and theophylline (long-acting). These are quick-relief or "rescue" medications that provide quick, temporary relief from asthma ... For this reason, it plays a secondary role in acute asthma treatment. Dry throat is the most common side effect. If the ...
It has fewer side effects as compared to theophylline. Caffeine improves airway function in asthma, increasing forced ... Welsh EJ, Bara A, Barley E, Cates CJ (January 2010). "Caffeine for asthma". The Cochrane Database of Systematic Reviews. 2010 ( ...
... is a short-acting β2 adrenoreceptor agonist used in the treatment of asthma. It was patented in 1965 and came into ... Virchow JC (1999). "Reproterol: beta-2-agonist, theophylline, or both?". Respiration; International Review of Thoracic Diseases ... what's best for exercise-induced asthma?". Sleep & Breathing = Schlaf & Atmung. 16 (4): 1229-35. doi:10.1007/s11325-011-0638-2 ...
Ibudilast, a neuroprotective and bronchodilator drug used mainly in the treatment of asthma and stroke. It inhibits PDE4 to the ... A metabolite of caffeine, theophylline, is a more potent PDE inhibitor. Diazepam, a benzodiazepine anxiolytic, amnesic, ... asthma and rheumatoid arthritis. PDE4D inhibition, along with PDE4A inhibition also appears to be responsible for the ...
Under his leadership, the company developed sustained-release Theo-Dur (theophylline), which became the nation's best-selling ... asthma remedy at the time, and cardiovascular drug Nitro-Dur. Key Pharmaceuticals was sold to Schering-Plough Corporation in ...
... s such as epinephrine, theophylline and salbutamol orally have been used to treat asthma, but inhaled adrenergic drugs ... Chu, Eric K.; Drazen, Jeffrey M. (1 June 2005). "Asthma". American Journal of Respiratory and Critical Care Medicine. 171 (11 ... Doig RL (February 1905). "Epinephrin; especially in asthma". California State Journal of Medicine. 3 (2): 54-5. PMC 1650334. ... asthma, nasal congestion and, in case of cocaine, as local anesthetics. Drugs used to treat obesity are called anorectics and ...
It is also preferred due to the former term giving the false impression that asthma is caused by exercise. In a patient with ... Other: Other prescription and over-the-counter medications, such as theophylline, cromolyn, and montelukast are indicated for ... National Asthma Education and Prevention Program (2007). "Expert Panel 3 (EPR-3): guidelines for the diagnosis and management ... The condition has a number of causes, the most common being emphysema as well as asthma. Exer an otherwise asymptomatic ...
Phosphodiesterase (PDE) inhibitors, such as theophylline, have been used to treat COPD for centuries; however, the clinical ... 1999). "Ariflo (SB 207499), a second generation phosphodiesterase 4 inhibitor for the treatment of asthma and COPD: from ... is a drug which was developed for the treatment of respiratory disorders such as asthma and chronic obstructive pulmonary ... potent and selective inhibitors of phosophodiesterase 4 for the treatment of asthma". Journal of Medicinal Chemistry. 41 (6): ...
Acute exacerbations of chronic respiratory diseases, mainly asthma and chronic obstructive pulmonary disease (COPD), are ... assessed as emergencies and treated with oxygen therapy, bronchodilators, steroids or theophylline, have an urgent chest X-ray ...
PIPPA Position Inspection Palpation Percussion Auscultation ASTHMA Adrenergic agonists Steroids Theophylline Hydration Masked ... rheumatoid arthritis Epilepsy Asthma Diabetes Strokes VAMP THIS: Vices (tobacco, alcohol, other drugs, sexual risks) Allergies ... ". "ASTHMA". Archived from the original on 2015-07-13. Retrieved 2015-04-24. "COPD Assessment Test" (PDF). "PULMONARY EDEMA" ( ...
His group investigated the role of neuropeptides in asthma and he proposed the axon reflex mechanism of asthma Their ... He also showed that theophylline was able to restore HDAC2 and reverse steroid resistance in COPD by selectively inhibiting ... His research explored mechanisms of severe asthma and in particular steroid-resistance in asthma, identifying several molecular ... Asthma as an axon reflex. Lancet 1986;i:242-245.PMID 2418322 Barnes PJ, Karin M. Nuclear factor-κB: a pivotal transcription ...
Theophylline is a non-selective agent. In contrast, meribendan is a highly selective inhibitor. Also, meribendan has a higher ... inhaled RPL-554 delivered via a nebulizer was in development for COPD and had been studied in asthma. Mutschler, Ernst; Schäfer ... theophylline) and papaverine. The active site of PDE3 can be considered as a summary of ideas about receptor topography ...
It is not available in the U.S. As other LABAs, bambuterol is used in the long-term management of persistent asthma. It should ... Concomitant administration of bambuterol with corticosteroids, diuretics, and xanthine derivatives (such as theophylline) ... Bambuterol (INN) is a long-acting β adrenoceptor agonist (LABA) used in the treatment of asthma; it also is a prodrug of ... 2009). "Bronchodilators and Anti-asthma Drugs". Martindale: The complete drug reference (36th ed.). London: Pharmaceutical ...
Theophylline and caffeine are nonselective adenosine antagonists that are used to stimulate respiration in premature infants. ... and makes them medically useful for the treatment of conditions such as asthma, but less suitable for use in scientific ... Xanthine derivatives such as caffeine and theophylline act as non-selective antagonists at A1 and A2A receptors in both heart ... The adenosine receptors are commonly known for their antagonists caffeine, theobromine, and theophylline, whose action on the ...
Daly JW, Padgett WL, Shamim MT (July 1986). "Analogues of caffeine and theophylline: effect of structural alterations on ... notably in the treatment of asthma or influenza symptoms. In contrast to other, more potent stimulants like sympathomimetic ... Several stimulants are derived from xanthine, including caffeine, theophylline, and theobromine. Xanthine is a product on the ... theophylline, and 7-methylxanthine (heteroxanthine), among others, affect the airways, increase heart rate and force of ...
Methylxanthines (e.g. caffeine found in coffee, theophylline found in tea, or theobromine found in chocolate) have a purine ... ISBN 978-1-4641-8652-3. Brown RA, Spina D, Page CP (March 2008). "Adenosine receptors and asthma". British Journal of ... The recommended dose may be increased in patients on theophylline since methylxanthines prevent binding of adenosine at ... Common contraindications for adenosine include Asthma, traditionally considered an absolute contraindication. This is being ...
... is a selective β2 adrenergic receptor agonist used in the treatment of asthma. Hexoprenaline is also used in some ... theophylline) increase its action General anaesthetics (e.g., halothane) and adrenergic receptor agonists may increase the risk ... a review of its pharmacological properties and therapeutic efficacy with particular reference to asthma". Drugs. 14 (1): 1-28. ...
As of December 2013[update], olodaterol is not approved for the treatment of asthma. It is administered in an inhaler called ... and theophylline), tricyclic antidepressants, and monoamine oxidase inhibitors could increase the likelihood of adverse effects ... for example in an asthma attack. On 29 January 2013 the U.S. Food and Drug Administration (FDA) Pulmonary-Allergy Drugs ...
... they play a central role in asthma, eczema, itch (from various causes), allergic rhinitis and allergic conjunctivitis. ... step in sodium fluoride-induced histamine secretion is inhibited by theophylline. Vasodilation and increased permeability of ...