Prostaglandin receptors or prostanoid receptors represent a sub-class of cell surface membrane receptors that are regarded as ... Prostanoid receptor Eicosanoid receptor Prostaglandin Tsuboi K, Sugimoto Y, Ichikawa A (2002). "Prostanoid receptor subtypes". ... IUPHAR GPCR Database - Prostanoid receptors Prostaglandin+Receptors at the U.S. National Library of Medicine Medical Subject ... receptors belonging to the Subfamily A14 of the rhodopsin-like receptor family except for the Prostaglandin DP2 receptor which ...

Prostaglandin receptors Prostanoid receptors Prostaglandin DP2 receptor Eicosanoid receptor GRCh38: Ensembl release 89: ... is primarily a receptor for prostaglandin D2 (PGD2). The receptor is a member of the Prostaglandin receptors belonging to the ... The Prostaglandin D2 receptor 1 (DP1), a G protein-coupled receptor encoded by the PTGDR1 gene (also termed PTGDR), ... role of the DP-receptor". Prostaglandins & Other Lipid Mediators. 107: 48-55. doi:10.1016/j.prostaglandins.2013.07.001. PMID ...

Prostaglandin DP1 receptor Prostaglandin receptors Prostanoid receptors Eicosanoid receptor GRCh38: Ensembl release 89: ... DP2 along with Prostaglandin DP1 receptor are receptors for prostaglandin D2 (PGD2). Activation of DP2 by PGD2 or other cognate ... with the C5a receptor, Formyl peptide receptor 1, and Formyl peptide receptor 2 receptors. DP2 has little or no such amino acid ... "Entrez Gene: GPR44 G protein-coupled receptor 44". "PTGDR2 prostaglandin D2 receptor 2". Gene Resources NCBI. Marchese A, ...

Eicosanoid receptor Prostaglandin E2 receptor 1 (EP1) Prostaglandin E2 receptor 2 (EP2) Prostaglandin E2 receptor 4 (EP4) ... Prostaglandin EP3 receptor (53kDa), also known as EP3, is a prostaglandin receptor for prostaglandin E2 (PGE2) encoded by the ... "PTGER3 prostaglandin e receptor 3 [Homo sapiens (human)] - Gene - NCBI". "Entrez Gene: PTGER1 prostaglandin E receptor 1 ( ... prostaglandin DP, E2, and E4 receptors (see Prostaglandin receptors). When initially bound to PGE2 or other of its agonists, it ...

PTGER1 Prostaglandin E2 receptor 2 (EP2) - PTGER2 Prostaglandin E2 receptor 3 (EP3) - PTGER3 Prostaglandin E2 receptor 4 (EP4 ... The prostaglandin E2 (PGE2) receptors are G protein-coupled receptors that bind and are activated by prostaglandin E2. They are ... Prostaglandin receptors Prostanoid receptors Prostaglandin Peluffo, M.C.; Stanley, J.; Braeuer, N.; Rotgeri, A.; Fritzemeier, K ... members of the prostaglandin receptors class of receptors and include the following Protein isoforms: Prostaglandin E2 receptor ...

Prostaglandin receptors Prostanoid receptors Prostaglandin E2 receptor 2 (EP2) Prostaglandin E2 receptor 3 (EP3) Prostaglandin ... Prostaglandin E2 receptor 1 (EP1) is a 42kDa prostaglandin receptor encoded by the PTGER1 gene. EP1 is one of four identified ... of available EP1 receptors) is ~20 nM and that of PGE1 ~40 for the mouse receptor and ~25 nM for PGE2 with the human receptor. ... "Airway smooth muscle prostaglandin-EP1 receptors directly modulate beta2-adrenergic receptors within a unique heterodimeric ...

Prostanoid receptors Prostaglandin receptors Prostaglandin E2 receptor 1 (EP1) Prostaglandin E2 receptor 3 (EP3) Prostaglandin ... Prostaglandin E2 receptor 2, also known as EP2, is a prostaglandin receptor for prostaglandin E2 (PGE2) encoded by the human ... "PTGER2 prostaglandin e receptor 2 [Homo sapiens (human)] - Gene - NCBI". Woodward DF, Jones RL, Narumiya S (September 2011). " ... "PTGER2 prostaglandin E receptor 2 (human)". Entrez Gene. National Center for Biotechnology Information, U.S. National Library ...

... (FP) is a receptor belonging to the prostaglandin (PG) group of receptors. FP binds to and mediates ... Prostaglandin F2 alpha Prostaglandin receptors Eicosanoid receptor GRCh38: Ensembl release 89: ENSG00000122420 - Ensembl, May ... "Cloning of the rat and human prostaglandin F2 alpha receptors and the expression of the rat prostaglandin F2 alpha receptor". ... "PTGFR prostaglandin F receptor [Homo sapiens (Human)] - Gene - NCBI". Zhang J, Gong Y, Yu Y (2010). "PG F(2α) Receptor: A ...

Prostaglandin E2 receptor 1 (EP1) Prostaglandin E2 receptor 2 (EP2) Prostaglandin E2 receptor 3 (EP3) Eicosanoid receptor ... Prostaglandin E2 receptor 4 (EP4) is a prostaglandin receptor for prostaglandin E2 (PGE2) encoded by the PTGER4 gene in humans ... "Entrez Gene: PTGER4 prostaglandin E receptor 4 (subtype EP4)". Archived from the original on 2010-12-05. "EP4 receptor - ... Pang L, Cai Y, Tang EH, Irwin MG, Ma H, Xia Z (2016). "Prostaglandin E Receptor Subtype 4 Signaling in the Heart: Role in ...

The prostaglandin D2 (PGD2) receptors are G protein-coupled receptors that bind and are activated by prostaglandin D2. Also ... They include the following proteins: Prostaglandin D2 receptor 1 (DP1) - PTGDR1 Prostaglandin D2 receptor 2 (DP2) - PTGDR2 The ... They also discovered PGD2 receptors on dopaminergic cells but not on microglia. Eicosanoid receptor Prostaglandin E2 receptor ... "The pharmacology of the prostaglandin D2 receptor 2 (DP2) receptor antagonist, fevipiprant". Pulmonary Pharmacology & ...

Hla T (April 2001). "Sphingosine 1-phosphate receptors". Prostaglandins. 64 (1-4): 135-142. doi:10.1016/s0090-6980(01)00109-5. ... Sphingosine-1-phosphate receptor 2, also known as S1PR2 or S1P2, is a human gene which encodes a G protein-coupled receptor ... "Lysophospholipid Receptors: S1P2". IUPHAR Database of Receptors and Ion Channels. International Union of Basic and Clinical ... "The Sphingolipid Receptor S1PR2 Is a Receptor for Nogo-A Repressing Synaptic Plasticity". PLOS Biology. 12 (1): e1001763. doi: ...

Hla T (Apr 2001). "Sphingosine 1-phosphate receptors". Prostaglandins. 64 (1-4): 135-142. doi:10.1016/s0090-6980(01)00109-5. ... Sphingosine-1-phosphate receptor 5 also known as S1PR5 is a human gene which encodes a G protein-coupled receptor which binds ... "Lysophospholipid Receptors: S1P5". IUPHAR Database of Receptors and Ion Channels. International Union of Basic and Clinical ... A-971432 Sphingosine 1-phosphate receptor agonists: a patent review (2010-2012) Lysophospholipid receptor GRCh38: Ensembl ...

PGD2: DP-(PGD2) (PGD2 receptor) DP1 (PTGDR1) - PTGDR1; DP1 is a receptor for Prostaglandin D2; relative potencies in binding to ... PGE2: EP-(PGE2) (PGE2 receptor) EP1-(PGE2) (PTGER1) - PTGER1; EP1 is a receptor for prostaglandin E2; relative potencies in ... The TP receptor is expressed in most human cells types as two alternatively spliced isoforms, TP receptor-α and TP receptor β, ... Prostanoids and Prostaglandin receptors Prostanoids are prostaglandins (PG), thromboxanes (TX), and prostacyclins (PGI). Seven ...

Tager AM, Luster AD (2004). "BLT1 and BLT2: the leukotriene B(4) receptors". Prostaglandins Leukot. Essent. Fatty Acids. 69 (2- ... Leukotriene B4 receptor 1 is a protein that in humans is encoded by the LTB4R gene. Eicosanoid receptor Etalocib, an antagonist ... "Leukotriene Receptors: BLT1". IUPHAR Database of Receptors and Ion Channels. International Union of Basic and Clinical ... G protein-coupled receptors, All stub articles, Transmembrane receptor stubs). ...

Interactions with PAF and benzodiazepine receptors". Prostaglandins. 40 (6): 571-83. doi:10.1016/0090-6980(90)90002-D. PMID ... However israpafant binds far more tightly to the platelet-activating factor receptor, with an IC50 of 0.84nM for inhibiting PAF ... Israpafant (Y-24180) is a drug which acts as a selective antagonist for the platelet-activating factor receptor, and was ... while it binds only weakly to benzodiazepine receptors, with a Ki of 3680nM. Israpafant has been found to inhibit the ...

Prostaglandins ligate a sub-family of cell surface seven-transmembrane receptors, G-protein-coupled receptors. These receptors ... the most abundant prostaglandin - is generated from the action of prostaglandin E synthases on prostaglandin H2 (prostaglandin ... prostaglandin D2 (PGD2), prostaglandin E2 (PGE2), and prostaglandin F2α (PGF2α). Examples of prostaglandin antagonists are: ... DP1-2 receptors bind to PGD2). The diversity of receptors means that prostaglandins act on an array of cells and have a wide ...

... activation of its prostaglandin F receptor and prostaglandin E2-induced activation of its prostaglandin EP1 receptor receptor ... and prostaglandin D2-induced activation of its prostaglandin DP1 receptor cause TP receptor desensitization by activating ... These receptor down regulating events are triggered by the G protein-coupled receptor kinases mobilized during TP receptor ... The thromboxane receptor is one among the five classes of prostanoid receptors and was the first eicosanoid receptor cloned. ...

The Prostacyclin receptor, also termed the prostaglandin I2 receptor or just IP, is a receptor belonging to the prostaglandin ( ... PGI2 Prostaglandin receptors Eicosanoid receptor GRCh38: Ensembl release 89: ENSG00000160013 - Ensembl, May 2017 GRCm38: ... role of the DP-receptor". Prostaglandins & Other Lipid Mediators. 107: 48-55. doi:10.1016/j.prostaglandins.2013.07.001. PMID ... "PTGIR prostaglandin I2 receptor [Homo sapiens (Human)] - Gene - NCBI". Claar D, Hartert TV, Peebles RS (February 2015). "The ...

"The cannabinoid receptors". Prostaglandins & Other Lipid Mediators. 68-69: 619-31. doi:10.1016/S0090-6980(02)00060-6. PMID ... Cannabinoid receptor type 1 (CB1) receptors are thought to be one of the most widely expressed Gαi protein-coupled receptors in ... a class of cell membrane receptors in the G protein-coupled receptor superfamily. As is typical of G protein-coupled receptors ... There are two known subtypes of cannabinoid receptors, termed CB1 and CB2. The CB1 receptor is expressed mainly in the brain ( ...

Prostaglandins & Other Lipid Mediators. 89 (3-4): 105-11. doi:10.1016/j.prostaglandins.2009.07.001. PMC 2751869. PMID 19615459 ... "The nuclear receptor peroxisome proliferator-activated receptor-alpha mediates the anti-inflammatory actions of ... Prostaglandins & Other Lipid Mediators. 89 (3-4): 105-11. doi:10.1016/j.prostaglandins.2009.07.001. PMC 2751869. PMID 19615459 ... A main target of PEA is proposed to be the peroxisome proliferator-activated receptor alpha (PPAR-α). PEA also has affinity to ...

Prostaglandins & Other Lipid Mediators. 89 (3-4): 82-8. doi:10.1016/j.prostaglandins.2009.05.003. PMID 19460454. Al Mahri S, ... Free fatty acid receptor 1 (FFAR1), also known as G-protein coupled receptor 40 (GPR40), is a rhodopsin-like G-protein coupled ... Free fatty acid receptor Free fatty acid receptor 4 GRCh38: Ensembl release 89: ENSG00000126266 - Ensembl, May 2017 GRCm38: ... an orally available G protein-coupled receptor 40/free fatty acid receptor 1 agonist, enhances glucose-dependent insulin ...

Bradshaw HB, Lee SH, McHugh D (September 2009). "Orphan endogenous lipids and orphan GPCRS: A good match". Prostaglandins Other ... N-Arachidonyl glycine receptor (NAGly receptor), also known as G protein-coupled receptor 18 (GPR18), is a protein that in ... Along with the other previously "orphan" receptors GPR55 and GPR119, GPR18 has been found to be a receptor for endogenous lipid ... G protein-coupled receptors, Biology of bipolar disorder, All stub articles, Transmembrane receptor stubs). ...

G protein-coupled receptor 119 also known as GPR119 is a G protein-coupled receptor that in humans is encoded by the GPR119 ... Prostaglandins & Other Lipid Mediators. 89 (3-4): 105-111. doi:10.1016/j.prostaglandins.2009.07.001. PMC 2751869. PMID 19615459 ... "Entrez Gene: GPR119 G protein-coupled receptor 119". Brown AJ (November 2007). "Novel cannabinoid receptors". British Journal ... G protein-coupled receptors, All stub articles, Transmembrane receptor stubs). ...

Rosen H (September 2005). "Chemical approaches to the lysophospholipid receptors". Prostaglandins Other Lipid Mediat. 77 (1-4 ... Sphingosine-1-phosphate receptor 1 (S1P receptor 1 or S1PR1), also known as endothelial differentiation gene 1 (EDG1) is a ... "Lysophospholipid Receptors: S1P1". IUPHAR Database of Receptors and Ion Channels. International Union of Basic and Clinical ... S1PR1 has been shown to interact with 5-HT1A receptor, GNAI1, and GNAI3. Lysophospholipid receptor GRCh38: Ensembl release 89: ...

Ishii S, Nagase T, Shimizu T (2002). "Platelet-activating factor receptor". Prostaglandins Other Lipid Mediat. 68-69: 599-609. ... "Platelet-Activating Factor Receptor". IUPHAR Database of Receptors and Ion Channels. International Union of Basic and Clinical ... The platelet-activating factor receptor (PAF-R) is a G-protein coupled receptor which binds platelet-activating factor. It is ... G protein-coupled receptors, All stub articles, Transmembrane receptor stubs). ...

Matsuoka T, Narumiya S (September 2007). "Prostaglandin receptor signaling in disease". TheScientificWorldJournal. 7: 1329-47. ... formyl peptide receptors (FPR), Chemokines - chemokine receptors (CCR or CXCR), and Leukotrienes - leukotriene receptors (BLT ... Thousands of MCP receptors are known to be encoded across the bacterial kingdom. These receptors may bind attractants or ... The Che proteins alter the tumbling frequency, and alter the receptors. The proteins CheW and CheA bind to the receptor. The ...

doi:10.1016/j.prostaglandins.2011.09.001. PMID 21945326. Matsuoka T, Narumiya S (2007). "Prostaglandin receptor signaling in ... E. J. Corey received it in chemistry in 1990 largely for his synthesis of prostaglandins. Eicosanoid receptors Edwards IJ, ... Hata AN, Breyer RM (2004). "Pharmacology and signaling of prostaglandin receptors: multiple roles in inflammation and immune ... Biosynthesis of prostaglandins); b) PGF synthase which converts PGH2 to PGF2α; c) Prostaglandin D2 synthase which converts PGH2 ...

"Cellular signalling of cysteinyl leukotriene type 1 receptor variants CysLT₁-G300S and CysLT₁-I206S". Prostaglandins, ... Other cysLT receptors include cysteinyl leukotriene receptor 2 (i.e. CysLTR2) and GPR99 (also termed the oxoglutarate receptor ... "Leukotriene Receptors: CysLT1". IUPHAR Database of Receptors and Ion Channels. International Union of Basic and Clinical ... Cysteinyl leukotriene receptor 1, also termed CYSLTR1, is a receptor for cysteinyl leukotrienes (LT) (see leukotrienes# ...

Characterization of receptors". Hypertension. 19 (2): 49-55. doi:10.1161/01.hyp.19.2_suppl.ii49. PMID 1735595. Phillips, PA. " ... Increased levels of bradykinin stimulate in the production of prostaglandin E2 and nitric oxide, which cause vasodilation and ... Jaiswal N, Diz DI, Chappell MC, Khosia MC, Ferrario CM (1992). "Stimulation of endothelial cell prostaglandin production by ... Effects of angiotensin converting enzyme inhibition and angiotensin II type 1 receptor blockade". Basic Research in Cardiology ...

Di Marzo V, De Petrocellis L, Fezza F, Ligresti A, Bisogno T (2002). "Anandamide receptors". Prostaglandins, Leukotrienes, and ... but instead activate other receptors (e.g. peroxisome proliferator-activated receptors (PPAR)-α/γ, G-protein coupled receptors ... Beside the CB1 receptors being triggers of the generation of ceramides that mediate neuronal cell fate, the skin CB1 receptor ... OEA acting mostly at peroxisome proliferator‐activated receptor‐α (PPAR‐α) nuclear receptors and, to some extent, TRPV1 ...