The pharmacokinetics of dydrogesterone have been reviewed. Dydrogesterone, also known as 6-dehydro-9β,10α-progesterone or as 9β ... Chemical syntheses of dydrogesterone have been published. Dydrogesterone is a progestin which was first synthesized by Duphar ... Dydrogesterone is readily absorbed with oral administration. The absolute bioavailability of dydrogesterone is on average 28%. ... There have been no harmful effects exhibited due to the use of dydrogesterone while pregnant. Dydrogesterone is safe to use ...
Dydrogesterone is associated with a lower risk than other progestins such as medroxyprogesterone acetate and norethisterone, ... with dydrogesterone as Femoston, Femoston Conti; and with nomegestrol acetate as Zoely. Estradiol valerate is available with ...
It shows greater potency than dydrogesterone in bioassays. Harper MJ (1977). Jucker E (ed.). "Contraception--retrospect and ...
Similarly to dydrogesterone and progesterone, trengestone has no androgenic or estrogenic activity. Trengestone appears to be a ... One tablet per day is administered from the 5th [...] Both dydrogesterone and trengestone can inhibit ovulation in the rat and ... ISBN 978-90-219-0144-2. Trengestone, contrary to [dydrogesterone], not only does not inhibit ovarian activity while exerting a ... For instance, unlike other progestogens, trengestone and dydrogesterone do not increase body temperature (i.e., have no ...
... is the parent compound of a group of progestins consisting of the marketed progestins dydrogesterone (6- ... May 2011). "Selectivity and potency of the retroprogesterone dydrogesterone in vitro". Steroids. 76 (6): 607-615. doi:10.1016/j ...
... is a progestin and the major active metabolite of dydrogesterone. It appears that dydrogesterone is a prodrug of 20α-DHD, as it ... Olbrich M, Weigl K, Kahler E, Mihara K (October 2016). "Dydrogesterone metabolism in human liver by aldo-keto reductases and ... 20α-DHD has progestogenic activity similarly to dydrogesterone, but is far less potent in comparison. 20α-Dihydroprogesterone ... May 2011). "Selectivity and potency of the retroprogesterone dydrogesterone in vitro". Steroids. 76 (6): 607-615. doi:10.1016/j ...
It is unclear if these findings may explain the different risks of breast cancer observed with progesterone, dydrogesterone, ... and dydrogesterone weakly stimulate proliferation. As such, progesterone differs from some but not all progestins in the ... "Selectivity and potency of the retroprogesterone dydrogesterone in vitro". Steroids. 76 (6): 607-15. doi:10.1016/j.steroids. ...
Dydrogesterone did not increase the risk of VTE associated with oral estrogen (odds ratio (OR) 0.9, 95% CI 0.4-2.3). Other ... Oral estrogens plus dydrogesterone appears to have lower VTE risk relative to inclusion of other progestins. Norpregnane ... The retroprogesterone derivatives dydrogesterone and trengestone are atypical progestogens and unlike all other clinically used ... Some research has found that oral progesterone and dydrogesterone with short-term use (. 5 years), oral progesterone and ...
In terms of the effects of progestogens on sex drive, one study assessed the use of dydrogesterone to improve sexual desire in ... Schindler AE (February 2011). "Dydrogesterone and other progestins in benign breast disease: an overview". Archives of ... Almost all progestins, with the exception of dydrogesterone, have antigonadotropic effects. Galactogogues such as the ... dydrogesterone, norethisterone acetate, and drospirenone. Progestins in general largely have the same progestogenic effects ...
94-. ISBN 978-93-5090-958-4. The natural preparations of P4 include progesterone, dydrogesterone, and medrogestone. Carter WF, ...
Dydrogesterone did not increase the risk of VTE associated with oral estrogen (odds ratio (OR) 0.9, 95% CI 0.4-2.3). Other ... Stevenson JC, Panay N, Pexman-Fieth C (September 2013). "Oral estradiol and dydrogesterone combination therapy in ... or estrogen-dydrogesterone (RR = 1.16) but was increased for estrogen combined with other progestins (RR = 1.69). These ... or with the atypical progestin dydrogesterone (OR = 1.10). In accordance, another study found similarly that the risk of breast ...
"Dydrogesterone: pharmacological profile and mechanism of action as luteal phase support in assisted reproduction". Reprod. ...
"Oral dydrogesterone for luteal support in frozen-thawed embryo transfer artificial cycles: A pilot randomized controlled trial ... "Oral dydrogesterone vs. vaginal progesterone capsules for luteal-phase support in women undergoing embryo transfer: a ... "Oral dydrogesterone versus intravaginal micronized progesterone gel for luteal phase support in IVF: a randomized clinical ...
The only exception among progestins is dydrogesterone, which has shown similar risk to that of oral progesterone. Breast cancer ... with a respective example from each group including dydrogesterone, medroxyprogesterone acetate, medrogestone, and promegestone ... the French E3N study showed significant associations of both estrogen plus oral progesterone and estrogen plus dydrogesterone ...
Similarly to progesterone, dydrogesterone, and hydroxyprogesterone caproate, quingestrone is a pure progestogen and lacks any ... Along with the retroprogesterone derivative dydrogesterone, quingestrone has been described as a "true" progesterone derivative ...
... transdermal testosterone and oral dydrogesterone (a progestin). After six weeks of treatment, the group treated with ... "Effects of transdermal testosterone or oral dydrogesterone on hypoactive sexual desire disorder in transsexual women: results ...
In 1977, the FDA determined that there was no adequate evidence that progestogens (including progesterone, dydrogesterone, and ... In general, pregnane derivatives (e.g., progesterone, dydrogesterone, hydroxyprogesterone caproate, medroxyprogesterone acetate ... dydrogesterone, and allylestrenol. Doses of 19-nortestosterones required for virilization are 10 to 20 mg/day, far in excess of ... and dydrogesterone (Duphaston) in 1962. The first case reports of fetal masculinization of external genitalia of female infants ...
... may refer to: Prödel, former German municipality Dydrogesterone, by trade name Prodel This disambiguation page lists ...
... is said to have very similar properties to those of dydrogesterone, a pure progestogen and close analogue of progesterone. PGA ... which have almost exactly the same properties as dydrogesterone.] "Gestovis". South African Medical Journal. 40 (5): 99. ...
... and dydrogesterone. The medication has also been studied in the treatment of gynecological disorders such as amenorrhea, ...
Other progestogens including medroxyprogesterone acetate, lynestrenol, allylestrenol, dydrogesterone, and normethandrone have ...
The combination of natural oral progesterone or the atypical progestin dydrogesterone with estrogen has been associated with ...
... dydrogesterone, drospirenone) Selective progesterone receptor modulators (e.g., ulipristal acetate, telapristone acetate, ...
... dydrogesterone (INN) dihydrocodeine (INN) Dymelor Dyna-Hex Dynabac Dynacirc Dynapen Dyrenium (Articles with short description, ...
... and dydrogesterone Androgens - bioidentical testosterone and dehydroepiandrosterone (DHEA), and synthetic anabolic steroids ...
The molecular formula C21H28O2 (molar mass: 312.44 g/mol) may refer to: 11-Dehydroprogesterone Demegestone Dydrogesterone ...
Algestone acetophenide Allylestrenol Chlormadinone acetate Cyproterone acetate Demegestone Dimethisterone Dydrogesterone ...
... dydrogesterone Selective progesterone receptor modulators (PR mixed agonists/antagonists) Examples: mifepristone, ulipristal ...
... dydrogesterone), have been discovered in high-throughput screening that enhance TLX's ability of transcription repression with ...
Dydrogesterone (progestin) Megestrol acetate (progestin, antineoplastic, appetite stimulant) Canrenone (aldosterone antagonist ...