... and etonogestrel are eliminated exclusively as metabolites 50% in urine and 35% in feces. Desogestrel, also known ... Neither desogestrel nor etonogestrel are bound by corticosteroid-binding globulin. Desogestrel is a prodrug of etonogestrel (3- ... Desogestrel was synthesized in 1972 at Organon [...] Holtsclaw JA (2007). Progress Towards the Total Synthesis of Desogestrel ... Contraindications of desogestrel include: Allergy to desogestrel or any other ingredients Active thrombosis (deep vein ...

Examples: desogestrel, nomegestrol acetate, norgestimate. Third generation: Approved for marketing between 1990 and 2000. ... Studies have found that combined birth control pills containing newer-generation progestins such as desogestrel, gestodene, ... Combined birth control with less androgenic or antiandrogenic progestins like desogestrel, gestodene, and drospirenone may have ... desogestrel, and etonogestrel. The androgens that have been used in combination with these progestins include testosterone, ...

Taken together, like desogestrel, gestodene appears to have a low potential for androgenic effects. Gestodene has relatively ... Kaplan B (1995). "Desogestrel, norgestimate, and gestodene: the newer progestins". Ann Pharmacother. 29 (7-8): 736-42. doi: ... 966-. ISBN 978-0-7817-7968-5. Chez RA (May 1989). "Clinical aspects of three new progestogens: desogestrel, gestodene, and ... London RS (November 1992). "The new era in oral contraception: pills containing gestodene, norgestimate, and desogestrel". ...

150 μg desogestrel (AU, EU, RU, UK: Marvelon, BR: Microdiol, US: Desogen, MSD; US: Ortho-Cept, Ortho-McNeil; RU: Regulon, ... ethinylestradiol/desogestrel combination with 7 tablets 25 μg/100 μg, 7 tablets 25 μg/125 μg, 7 tablets 25 μg/150 μg, followed ... triphasic ethinylestradiol/desogestrel combination with 7 tablets 35 μg/50 μg, 7 tablets 30 μg/100 μg, 7 tablets 30 μg/150 μg ( ... 150 μg desogestrel (UK: Mercilon, Organon; HU: Novynette, Richter Gedeon) 75 μg gestodene (UK: Femodette, Bayer; RU: Logest, ...

"Kimidess (Desogestrel and Ethinyl Estradiol Tablets, USP and Ethinyl Estradiol Tablets, USP), 0.15 mg/0.02 mg and 0.01 mg". ... "Cyred EQ- desogestrel and ethinyl estradiol kit". DailyMed. Archived from the original on 11 July 2021. Retrieved 10 July 2021 ... "Bekyree- desogestrel and ethinyl estradiol and ethinyl estradiol kit". DailyMed. Archived from the original on 11 July 2021. ... "Cesia- desogestrel and ethinyl estradiol kit". DailyMed. Archived from the original on 11 July 2021. Retrieved 10 July 2021. " ...

Third-generation progestins (desogestrel, norgestimate and elsewhere, gestodene) were introduced to maintain the potent ... Third generation COCPs are sometimes defined as those containing the progestins desogestrel or gestodene; and sometimes defined ... with desogestrel (DSG) 1.82, with gestodene 1.86, with drospirenone (DRSP) 1.64, and with cyproterone acetate 1.88. In ... desogestrel, gestodene) or antiandrogen activity (cyproterone acetate, chlormadinone acetate, drospirenone, dienogest, ...

It was investigated in combination with desogestrel as a birth control pill, but resulted in unacceptable menstrual bleeding ... Schubert W, Cullberg G (1987). "Ovulation inhibition with 17 beta-estradiol cyclo-octyl acetate and desogestrel". Acta Obstet ...

Examples include gestodene, desogestrel, and etonogestrel, which are CYP3A4 and CYP2C19 inhibitors. In addition, these ... while the combination of 30 µg/day EE and 150 µg/day desogestrel increased them by 100%. EE shows strong and disproportionate ... to 4-fold with desogestrel and gestodene, 3.5- to 4-fold with drospirenone and dienogest, and 4- to 5-fold with cyproterone ... The combination of 30 µg/day EE and 150 µg/day desogestrel, a progestin with relatively weak androgenicity than levonorgestrel ...

Besides levonorgestrel itself, this group includes desogestrel, dienogest, etonogestrel, gestodene, norelgestromin, ...

In 1981, desogestrel was marketed as a new low dose oral contraceptive under the trade names Marvelon and Desogen.32 Glasier A ... Desogestrel (3-deketoetonogestrel), a prodrug of etonogestrel, was introduced for medical use in 1981. Norplant was used ... A closely related and more widely known and used progestin, desogestrel, is a prodrug of etonogestrel in the body. Etonogestrel ... Etonogestrel is the C3 ketone derivative of desogestrel and the C11 methylene derivative of levonorgestrel and is also known as ...

However, the 3-keto group is initially missing in the case of desogestrel and norgestimate. They are prodrugs which undergo ...

However, the 3-keto group is initially missing in the case of desogestrel and norgestimate. They are prodrugs which undergo ...

Third-generation gonanes (desogestrel, gestodene, and norgestimate) have been developed to reduce unwanted side effects of ... desogestrel, etonogestrel, gestodene, norgestimate, dienogest (actually a 17α-cyanomethyl-19-nortestosterone derivative), and ...

Desogestrel 75 µg (brand name Cerzette) was marketed in Europe in 2002 and was the most recent POP to be introduced. It differs ... 2424-. ISBN 978-1-4557-1126-0. In 2002, a POP containing desogestrel 75 ug/day, a dose sufficient to inhibit ovulation in ... Commercially available progestogen-only pills include the following common or widely used formulations: Desogestrel 75 µg (e.g ... by those containing desogestrel. Greenberg (19 February 2016). Exploring the Dimensions of Human Sexuality. Jones & Bartlett ...

Along with desogestrel, it is one of the only progestins that is widely available as a progestogen-only "mini pill" for birth ...

The progestins drospirenone and desogestrel minimize the androgenic side effects but increase the risks of blood clots and are ...

Conversely, this would be the case less or not at all with progestins that are less androgenic, like desogestrel and gestodene ... Birth control pills containing progestins such as desogestrel, gestodene, drospirenone, and cyproterone acetate have been found ... desogestrel, drospirenone, or gestodene overall were associated with a risk of VTE of about 1.3- to 2.0-fold compared to that ... whereas this may occur less or not at all with weakly androgenic progestins like desogestrel and antiandrogenic progestins like ...

... additive effects between desogestrel and testosterone enanthate in suppression of spermatogenesis, pituitary-testicular axis, ...

Progestin treatment with desogestrel and norgestimate appears to have fewer androgenic side effects and may be safer to use in ...

It shares this property with lynestrenol (17α-ethynylestr-4-en-17β-ol), desogestrel (11-methylene-17α-ethynyl-18-methylestr-4- ...

... to 4-fold with desogestrel and gestodene, 3.5- to 4-fold with drospirenone and dienogest, and 4- to 5-fold with cyproterone ...

... examples include: 19-norpregnane (from pregnane), desogestrel, ethylestrenol, etynodiol diacetate, ethinylestradiol ...

... desogestrel, levonorgestrel, and drospirenone strongly stimulate proliferation and medroxyprogesterone acetate, dienogest, and ...

... with desogestrel (DSG) 1.82, with gestodene 1.86, with drospirenone (DRSP) 1.64, and with cyproterone acetate 1.88. Venous ...

... by codename A brand name of desogestrel Azala (disambiguation) Azalea (disambiguation) This disambiguation page lists articles ...

Ethinylestradiol and desogestrel (Bekyree, Cyclessa, Desogen, Emoquette, Enskyce, Isibloom, Kariva, Kimidess, Mircette, Ortho- ...

Estradiol/estriol/norethisterone acetate Estradiol/desogestrel Estradiol cyclooctyl acetate/desogestrel Estradiol/ ...

... a brand name of desogestrel Hannah (disambiguation) This disambiguation page lists articles associated with the title Hana. If ...

... ethinyloestradiol with desogestrel, and ethinyloestradiol with levonorgestrel), and two formulations of the progestogen-only ...

Desogestrel Unclassified progestin: Drospirenone, Cyproterone acetate Extended or continuous use of COCPs has been used for ...