Cisapride
... cisapride", issued 1999-Sep-21 Maclennan S, Augood C, Cash-Gibson L, Logan S, Gilbert RE (April 2010). "Cisapride treatment for ... Cisapride is still available in the United States and Canada for use in animals, and is commonly prescribed by veterinarians to ... Cisapride has been used for the treatment of gastroesophageal reflux disease (GERD). There is no evidence it is effective for ... Cisapride is a gastroprokinetic agent, a drug that increases motility in the upper gastrointestinal tract. It acts directly as ...
Constipation
Cisapride is widely available in third world countries, but has been withdrawn in most of the west. It has not been shown to ... Aboumarzouk, Omar M; Agarwal, Trisha; Antakia, Ramez; Shariff, Umar; Nelson, Richard L (19 January 2011). "Cisapride for ...
Phenylpropanolamine
"Unsafe Drugs- nimesulide, Cisapride, Phenylpropanolamine Banned". 27 January 2011. "Madras High Court Revokes Ban on ...
Metoclopramide
... is a substituted benzamide; cisapride and mosapride are structurally related. Metoclopramide was first described ...
Grapefruit-drug interactions
Gross AS, Goh YD, Addison RS, Shenfield GM (April 1999). "Influence of grapefruit juice on cisapride pharmacokinetics". ... Examples of such known CYP3A4 inhibitors include cisapride (Propulsid), erythromycin, itraconazole (Sporanox), ketoconazole ( ...
Drug of last resort
... such as cisapride. Aminoglycosides - their use is extremely restricted due to risk of hearing loss and kidney damage; ... Cisapride - used for severe gastroesophageal reflux disease (GERD); carries risk of heart arrhythmias; Clomethiazole - a ...
Paracetamol
AUC increases are also observed with nizatidine and cisapride. The effect is explained by these drugs inhibiting ...
Nefazodone
Contraindications include the coadministration of terfenadine, astemizole, cisapride, pimozide, or carbamazepine. Nefazodone is ...
Diazepam
Cisapride may enhance the absorption, and therefore the sedative activity, of diazepam. Small doses of theophylline may inhibit ... Bateman DN (1986). "The action of cisapride on gastric emptying and the pharmacodynamics and pharmacokinetics of oral diazepam ...
Intestinal pseudo-obstruction
Prucalopride, pyridostigmine, metoclopramide, cisapride, erythromycin and octreotide are medications that aim to enhance ...
5-HT4 receptor
Tropisetron - partial agonist BIMU-8 Cisapride CJ-033,466 - partial agonist ML-10302 Mosapride Prucalopride Renzapride RS-67506 ... "Overexpression of serotonin4 receptors in cisapride-responsive adrenocorticotropin-independent bilateral macronodular adrenal ...
Prokinetic agent
As such, the relatively poor selectivity profile of cisapride versus other receptors (especially hERG [human ether-a-go-go K+] ... Some of these prokinetic agents, such as mosapride and cisapride, classic benzamides, have only moderate affinity for 5HT4 ... Benzamide Cisapride Domperidone Itopride Mosapride Metoclopramide Prucalopride Renzapride Tegaserod Mitemcinal Levosulpiride ...
Simeticone
"A randomized placebo-controlled trial of simethicone and cisapride for the treatment of patients with functional dyspepsia". ...
Sir William Arbuthnot Lane, 1st Baronet
Medical treatment with laxatives, enemas and prokinetic agents, such as cisapride, does not relieve the burdensome symptoms. ...
Serotonin receptor agonist
Cisapride and tegaserod are 5-HT4 receptor partial agonists that were used to treat disorders of gastrointestinal motility. ...
Mosapride
... drug information - Drugs Update India Kii Y, Ito T (May 1997). "Effects of 5-HT4-receptor agonists, cisapride, ...
CJ-033466
Toga T, Kohmura Y, Kawatsu R (October 2007). "The 5-HT(4) agonists cisapride, mosapride, and CJ-033466, a Novel potent compound ... In animal tests it stimulated gastrointestinal motility with 30 times the potency of cisapride, and with lower affinity for the ...
Itopride
The affinity of cisapride for 5-HT4 receptors in the heart has been implicated in the undesirable cardiac effects of cisapride ... Itopride belongs to the same benzamide group as cisapride, a drug found to affect QT interval and possibly predispose those ... Moreover, itopride has no affinity for the 5-HT4 receptors, unlike other benzamides such as cisapride and mosapride, which are ... unlike cisapride and mosapride, as it is metabolized by a different enzyme set. New molecular studies on guinea pig ventricular ...
Terence Young (politician)
Johnson prescription drug cisapride (brand name in Canada: Prepulsid). Young became a consumer advocate after this incident, ...
Erythromycin
Other examples include terfenadine (Seldane, Seldane-D), astemizole (Hismanal), cisapride (Propulsid, withdrawn in many ...
Velusetrag
... to earlier generation 5-HT agonists like cisapride and tegaserod. In a large clinical trial in patients with chronic idiopathic ...
5-HT3 antagonist
Certain prokinetic drugs such as cisapride, renzapride and metoclopramide, although not 5-HT3 antagonists proper, possess some ...
Chiral switch
... and cisapride to norcisapride. A summary is presented in the table below. Drug repurposing and chiral switches are part of the ...
Atazanavir
... cisapride, St. John's wort, lovastatin, simvastatin, sildenafil, indinavir, or nevirapine. Atazanavir inhibits the enzyme UDP ...
Sucralfate
... cisapride + sucralfate can significantly improve symptoms and quality of life and was more cost-effective than ranitidine ...
Ketoconazole
... cisapride, nisoldipine, dofetilide, pimozide And is not recommended: carbamazepine, phenytoin gastric acid suppressants: ...
Clarithromycin
... cisapride, pimozide, astemizole, terfenadine, ergotamine, ticagrelor, ranolazine or dihydroergotamine is not recommended. It ...
List of MeSH codes (D03)
... cisapride MeSH D03.383.621.147 - clopamide MeSH D03.383.621.160 - cyproheptadine MeSH D03.383.621.160.500 - loratadine MeSH ...
Brazilian Controlled Drugs and Substances Act
Cyclopentolate Cisapride Citalopram Clomacran Clomethiazole Clomipramine Chloralodol Chlorpromazine Chlorprothixene Clotiapine ...
Prucalopride
... differs from other 5-HT4 agonists such as tegaserod and cisapride, which at therapeutic concentrations also ...