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*  Patent EP3175840A1 - Dermal filler compositions - Google Patents
Non-limiting examples of aminoamide local anesthetics include articaine, bupivacaine, cinchocaine (dibucaine), etidocaine, ... This seems to increase the number of amide bonds formed with respect to the number of ester bonds. It is believed that since ... aminoamide local anesthetics and aminoester local anesthetics. The amount of an anesthetic agent included in a composition ... An anesthetic agent is preferably a local anesthetic agent, i.e., an anesthetic agent that causes a reversible local anesthesia ...
  http://www.google.com.au/patents/EP3175840A1?cl=en&hl=en&output=html_text
*  Bupivacaine - Wikipedia
Bupivacaine is contraindicated in patients with known hypersensitivity reactions to bupivacaine or amino-amide anesthetics. It ... bupivacaine is an amino-amide anesthetic; the aromatic head and the hydrocarbon chain are linked by an amide bond rather than ... the amino-amide anesthetics are more stable and less likely to cause allergic reactions. Unlike lidocaine, the terminal amino ... It is a local anaesthetic of the amide group. Bupivacaine was discovered in 1957. It is on the World Health Organization's List ...
  https://en.wikipedia.org/wiki/Bupivacaine
*  Vasoconstriction Potency Induced by Aminoamide Local Anesthetics Correlates with Lipid Solubility
G. L. Weinberg, R. Ripper, P. Murphy et al., "Lipid infusion accelerates removal of bupivacaine and recovery from bupivacaine ... including amides and esters) of local anesthetics enhances potency and lipid solubility [3]. Lipid solubility is a major ... Aminoamide local anesthetics induce vasoconstriction in vivo and in vitro. The goals of this in vitro study were to investigate ... Vasoconstriction Potency Induced by Aminoamide Local Anesthetics Correlates with Lipid Solubility. Hui-Jin Sung,1 Seong-Ho Ok,2 ...
  https://www.hindawi.com/journals/bmri/2012/170958/
*  Naropin (Ropivacaine Hcl): Side Effects, Interactions, Warning, Dosage & Uses
... bupivacaine (another member of the amino amide class of local anesthetics) was inadvertently rapidly injected intravenously. ... Ropivacaine is a member of the amino amide class of local anesthetics and is supplied as the pure S-(-)-enantiomer. Local ... Naropin® Injection contains ropivacaine HCl, which is a member of the amino amide class of local anesthetics. Naropin ( ... Because amide-type local anesthetics such as ropivacaine are metabolized by the liver, these drugs, especially repeat doses, ...
  https://www.rxlist.com/naropin-drug.htm
*  DERMAL FILLER COMPOSITIONS INCLUDING ANTIOXIDANTS - Patent application
Non-limiting examples of aminoamide local anesthetics include articaine, bupivacaine, cinchocaine (dibucaine), etidocaine, ... PEG amide. In this embodiment, the degree of conjugation may be between about 20 mol % and about 32 mol %. [0092] In another ... aminoamide local anesthetics and aminoester local anesthetics. The amount of an anesthetic agent included in a composition ... An anesthetic agent is preferably a local anesthetic agent, i.e., an anesthetic agent that causes a reversible local anesthesia ...
  http://www.patentsencyclopedia.com/app/20130210760
*  Sciatic Nerve Blockade in Infant, Adolescent, and Adult Rats :, A Comparison of Ropivacaine with Bupivacaine | Anesthesiology ...
Ropivacaine is an amino-amide local anesthetic recently released for clinical use in the United States and many other countries ... Badgwell JM, Heavner JE, Kytta J: Bupivacaine toxicity in young pigs is age-dependent and is affected by volatile anesthetics. ... Akerman B, Hellberg I-B, Trossvik C: Primary evaluation of the local anaesthetic properties of the amino amide agent ... Reiz S, Haggmark S, Johansson G, Nath S: Cardiotoxicity of ropivacaine-A new amide local anesthetic agent. Acta Anesthesiol ...
  http://anesthesiology.pubs.asahq.org/article.aspx?articleid=1946679
*  Pharmaceutical Bupivacaine - chembj.net
All three of these anesthetics contain an amide linkage between the aromatic nucleus and the amino. They differ in this respect ... Product Name:Bupivacaine. Synonyms:MARCAINE;BUPIVACAINE;BUPIVACAINE BASE;(.+/-.)-1-Butyl-2′,6′-pipecoloxylidide;1-Butyl-2-(2,6- ... Bupivacaine Application:. Bupivacaine is indicated for local anaesthesia including infiltration. Bupivacaine often is ... Bupivacaine is an anesthetic (numbing medicine) that blocks the nerve impulses that send pain signals to your brain. ...
  http://www.chembj.net/product/bupivacaine/
*  Patent US5149320 - Composite anesthetic article and method of use - Google Patents
... wherein the anesthetic comprises from about 0.5 to about 2.0% by weight of the composition, the composition further containing ... the composition containing a local parenteral anesthetic which in normal doses gives an acid pH of from about 2.5 to about 6.9 ... An aqueous composition for reducing pain at the site of injection of local parenteral anesthetic material, for improving the ... As background information, the free esters or amides of local anesthetics such as Lidocaine, Mepivacaine and Bupivacaine are ...
  http://www.google.com/patents/US5149320?dq=6,712,702
*  14252-80-3 Pharmaceutical Raw Materials Bupivacaine Hydrochloride HCL Powder - pharmaceuticalsteroids
Buy 14252-80-3 Pharmaceutical Raw Materials Bupivacaine Hydrochloride HCL Powder direct from Pharmaceutical Raw Materials of ... All three of these anesthetics contain an amide linkage between the aromatic nucleus and the amino or piperidine group. They ... 1, Bupivacaine HCL Profile:. Product Name: Bupivacaine hydrochloride. Synonyms: Bupivacaine HCL, Bupivacaine HCI, Sensorcaine. ... Usage: Long-acting local anesthetic (amide type); A local anesthetic used for peripheral nerve block, infiltration, and ...
  http://pharmaceuticalsteroids.sale.pysqlite.org/pz67253e4-14252-80-3-pharmaceutical-raw-materials-bupivacaine-hydrochloride-hcl-powder.html
*  PRIME PubMed | anesthetics topical mucosal journal articles from PubMed
PubMed Journal articles for anesthetics topical mucosal were found in PRIME PubMed. Download Prime PubMed App to iPhone or iPad ... Combining amino amide salts in mucoadhesive films enhances needle-free buccal anesthesia in adults. [Randomized Controlled ... The effects of local anesthetics (LAs), namely, lidocaine (LDC), prilocaine (PLC), mepivacaine (MPV), bupivacaine (BPV), ... The effects of local anesthetics (LAs), namely, lidocaine (LDC), prilocaine (PLC), mepivacaine (MPV), bupivacaine (BPV), ...
  https://www.unboundmedicine.com/medline/research/anesthetics__topical_mucosal_
*  Management of Local Anesthetic Toxicity
Local Anesthetic Pharm Amino esters and Amino amides Metabolism Protein binding Lipophilichydrophilic balance Hydrogen Ion ... B = bupivacaine, N + B = nimodipine 200 [micro sign]g/kg + bupivacaine, V + B = verapamil 150 [micro sign]g/kg + bupivacaine. ... CVS Newer amino amide local anesthetics potential to cause CNS toxicity Indicators of CVS toxicity Mechanism of toxicity ... Alterations in the pharmacokinetic properties of amide local anesthetics following local anesthetic induced convulsions. Acta ...
  http://slidegur.com/doc/157297/management-of-local-anesthetic-toxicity
*  STABILIZATION OF QUINOL COMPOSITION SUCH AS CATECHOLAMINE DRUGS - Patent application
... anesthetic, such as an amino ester local anesthetic (e.g., procaine) or an amino amide local anesthetics (e.g., lidocaine). See ... or an amino ester linkage (e.g., --NH--(C═O)--, as found in lidocaine, prilocalne, bupivacaine) that is situated between (i) ... of local anesthetics, including amino ester local anesthetics (e.g., procaine) and amino amide local anesthetics (e.g., ... amino ester anesthetic and an amino amide anesthetic. 34. A stable pharmaceutical formulation according to claim 1 wherein the ...
  http://www.patentsencyclopedia.com/app/20120029085
*  Levobupivacaine - Wikipedia
... is a local anaesthetic drug belonging to the amino amide group. It is the S-enantiomer of bupivacaine. Levobupivacaine ... Burlacu CL, Buggy DJ (April 2008). "Update on local anesthetics: focus on levobupivacaine". Ther Clin Risk Manag. 4 (2): 381-92 ... Compared to bupivacaine, levobupivacaine is associated with less vasodilation and has a longer duration of action. It is ... ISBN 0-9757919-2-3 Gulec D (Apr 2014). "Intrathecal bupivacaine or levobupivacaine: which should be used for elderly patients ...
  https://en.wikipedia.org/wiki/Levobupivacaine
*  Nerve Block - Pain.dieutridau.com - All for Pain Relief !
Lidocaine and bupivacaine are both amide anesthetics and may have allergic cross-sensitivity. Procaine, an ester anesthetic, ... The 2 main classes of local anesthetics currently in use are amino esters and amino amides. Both inhibit ionic fluxes required ... Lidocaine is the most commonly used anesthetic. If longer anesthesia is required, another amide anesthetic, such as bupivacaine ... separated in the middle by an amino-ester or an amino-amide. This forms the basis of classification of local anesthetics into 2 ...
  https://pain.dieutridau.com/management/nerve-block.html
*  Lidoderm Topical application Advanced Patient Information - Drugs.com
Therapeutic Class: Anesthetic, Local. Chemical Class: Amino Amide. Uses For Lidoderm. Lidocaine topical jelly or ointment is ... Lidocaine belongs to the family of medicines called local anesthetics. This medicine prevents pain by blocking the signals at ... This medicine does not cause unconsciousness as general anesthetics do when used for surgery. ...
  https://www.drugs.com/cons/lidoderm-topical-application.html
*  LMX 4 Topical application Advanced Patient Information - Drugs.com
Therapeutic Class: Anesthetic, Local. Chemical Class: Amino Amide. Uses For LMX 4. Lidocaine topical jelly or ointment is used ... Local Anesthesia lidocaine ophthalmic, cocaine topical, Marcaine, bupivacaine, Novocain, tetracaine topical, ropivacaine, ... Lidocaine belongs to the family of medicines called local anesthetics. This medicine prevents pain by blocking the signals at ... This medicine does not cause unconsciousness as general anesthetics do when used for surgery. ...
  https://www.drugs.com/cons/lmx-4-topical-application.html
*  Solarcaine First Aid Lidocaine Spray Topical application Advanced Patient Information - Drugs.com
Therapeutic Class: Anesthetic, Local. Chemical Class: Amino Amide. Uses For Solarcaine First Aid Lidocaine Spray. Lidocaine ... Lidocaine belongs to the family of medicines called local anesthetics. This medicine prevents pain by blocking the signals at ... This medicine does not cause unconsciousness as general anesthetics do when used for surgery. ...
  https://www.drugs.com/cons/solarcaine-first-aid-lidocaine-spray-topical-application.html
*  Burn-O-Jel Topical application Advanced Patient Information - Drugs.com
Therapeutic Class: Anesthetic, Local. Chemical Class: Amino Amide. Slideshow. Lyrica: 12 Things You Need to Know ... Lidocaine belongs to the family of medicines called local anesthetics. This medicine prevents pain by blocking the signals at ... This medicine does not cause unconsciousness as general anesthetics do when used for surgery. ...
  https://www.drugs.com/cons/burn-o-jel-topical-application.html
*  Buprenorphine Enhances and Prolongs the Postoperative Analgesic Effect of Bupivacaine in Patients Receiving Infragluteal...
... were also excluded if they were receiving long-term opioid analgesic therapy or reported a history of allergy to amino-amide LA ... local anesthetic block + intramuscular placebo; group 2: intramuscular control = local anesthetic block + intramuscular ... Gao F, Waters B, Seager J, Dowling C, Vickers MD: Comparison of bupivacaine plus buprenorphine with bupivacaine alone by caudal ... local anesthetic block + intramuscular placebo; group 2: intramuscular control = local anesthetic block + intramuscular ...
  http://anesthesiology.pubs.asahq.org/article.aspx?articleid=2085796
*  Lidocaine and tetracaine Topical application Advanced Patient Information - Drugs.com
Chemical Class: Amino Amide. Slideshow. FDA-Approved Weight Loss Drugs: Can They Help You? ... Topical anesthetics. Related Drugs. Local Anesthesia lidocaine ophthalmic, cocaine topical, bupivacaine, Marcaine, tetracaine ... Lidocaine and tetracaine combination belongs to a group of medicines known as topical local anesthetics. It deadens the nerve ... Lidocaine and tetracaine does not cause unconsciousness as general anesthetics do when used for surgery. ...
  https://www.drugs.com/cons/lidocaine-and-tetracaine-topical-application.html
*  Levobupivacaine Hydrochloride - Levobupivacaine Hydrochloride Suppliers, Buyers, Wholesalers and Manufacturers - ecplaza.net
... is a local anaesthetic drug belonging to the amino amide group. It is the S-enantiomer of bupivacaine.It is the hydrochloride ... Local Anesthetic Levobupivacaine HCL / Levobupivacaine Hydrochloride Powder. 99% Local Anesthetic Levobupivacaine HCL / ... Levobupivacaine Hydrochloride Local Anesthetic Powder CAS 27262-48-2. Levobupivacaine Hydrochloride Local Anesthetic Powder CAS ... Quality Pharmaceutical Raw Material Local Anesthetic Procaine HCl, Procaine Hydrochloride. Pain Killer Local Anesthetic APIS ...
  https://www.ecplaza.net/Levobupivacaine-Hydrochloride--everything
*  Resuscitation with Lipid Emulsion:Dose-dependent Recovery from Cardiac Pharmacotoxicity Requires a Cardiotonic Effect |...
J-T Lipid emulsion-mediated reversal of toxic-dose aminoamide local anesthetic-induced vasodilation in isolated rat aorta.. ... A Antimetastatic potential of amide-linked local anesthetics: Inhibition of lung adenocarcinoma cell migration and inflammatory ... DL Lipid infusion accelerates removal of bupivacaine and recovery from bupivacaine toxicity in the isolated rat heart.. Reg ... E and F) Same as A and B but for median rate-pressure product normalized to baseline (averaged over 20s before bupivacaine ...
  http://anesthesiology.pubs.asahq.org/article.aspx?articleid=1917827&resultClick=3
*  Book Text
Useful agents for interscalene block are primarily the amino amides. Lidocaine and mepivacaine produce 2 to 3 hours of surgical ... Plain bupivacaine produces surgical anesthesia lasting 4 to 6 hours; the addition of epinephrine may prolong the anesthesia to ... This point may be moot if one is planning to use a combined regional and general anesthetic technique, which allows control of ... Even when a long-acting local anesthetic is chosen for the interscalene technique, usually phrenic nerve, and thus pulmonary, ...
  http://polanest.webd.pl/pliki/varia/books/AtRegAn/micro189.lib3.hawaii.edu_3a2127/das/book/body/0/1353/15.html@tocnode=52418254&fromurl=15.html
*  side effects of dental anaesthetic list - side effects of dental anaesthetic for sale
... is a local anaesthetic drug belonging to the amino amide group. It is the S-enantiomer of bupivacaine. The hydrochlorid ... White Powder Effective Local Anesthetic Bupivacaine CAS 2180-92-9 for Reduce-Pain ... White Powder Effective Local Anesthetic Bupivacaine CAS 2180-92-9 for Reduce-Pain ... Long Acting Local Anesthetic Agents Procaine Without Side Effects 59-46-1 Quick Detail: Product Name: Procaine Synonyms: ...
  http://www.chinacsw.com/side-effects-of-dental-anaesthetic-wholesale
*  Lidocaine - Wikipedia
... the first amino amide-type local anesthetic, was first synthesized under the name 'xylocaine' by Swedish chemist Nils Löfgren ... Bupivacaine is a safe alternative in this case. Impaired liver function - people with lowered hepatic function may have an ... Serious adverse drug reaction to lidocaine or amide local anesthetics Hypersensitivity to corn and corn-related products (corn- ... Longer-acting substances such as bupivacaine are sometimes given preference for spinal and epidural anaesthesias; lidocaine, ...
  https://en.wikipedia.org/wiki/Lidocaine