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*  Flutamide Cheap Price - Buy Flutamide Online Europe
Bicalutamide". Horm Cancer. Duffy, P. and Phillips, Y. Y. Caffeine consumption decreases the response to bronchoprovocation ... Therefore, blocking these androgens can provide powerful treatment for prostate cancer, especially metastatic disease. Taylor, ... "Marked symptom reduction in two women with bulimia nervosa treated with the testosterone receptor antagonist flutamide. What ... Overview of phase II trials on combined androgen treatment in patients with metastatic prostate cancer. Cancer. 1993; 72: 3888- ...
  http://flutamide.inam.info
*  Cyproterone acetate - Wikipedia
CPA is a potent androgen receptor (AR) competitive antagonist. It directly blocks endogenous androgens such as testosterone and ... Other important antiandrogens besides CPA include spironolactone and bicalutamide. The drug is available widely throughout the ... CPA is known to possess the following pharmacological activity: Androgen receptor (AR) antagonist/very weak partial agonist ( ... ISBN 978-1-84076-013-2. Singh, Shankar; Gauthier, Sylvain; Labrie, Fernand (2000). "Androgen Receptor Antagonists ( ...
  https://en.wikipedia.org/wiki/Cyproterone_acetate
*  WO 2009/124396 A1 - Polymorphisms Predictive Of Platinum-coordinating Compound-induced Ototoxicity - The Lens - Free & Open...
... androgen antagonists such as flutamide and bicalutamide; and gonadotropin- releasing hormone analogs such as leuprolide. ... estrogen antagonists such as tamoxifen and anastrozole; androgens such as testosterone propionate and fluoxymesterone and ... hormones and antagonists, and miscellaneous agents. Examples of alternate names are indicated in brackets. Examples of ... DNA synthesis antagonists such as estramustine phosphate; and triazines such as dacarbazine (DTIC, dimethyl- ...
  https://www.lens.org/lens/patent/111-217-672-730-519/fulltext
*  A Study of Enzalutamide Versus Bicalutamide in Castrate Men With Metastatic Prostate Cancer - Full Text View - ClinicalTrials...
Bicalutamide. Androgen Antagonists. Hormone Antagonists. Hormones, Hormone Substitutes, and Hormone Antagonists. Physiological ... Ongoing androgen deprivation therapy with a Luteinizing Hormone Receptor Hormone (LHRH) agonist or antagonist at a stable dose ... Active Comparator: Bicalutamide Participants received bicalutamide 50 mg orally once daily until confirmed radiographic disease ... A Study of Enzalutamide Versus Bicalutamide in Castrate Men With Metastatic Prostate Cancer. The safety and scientific validity ...
  https://clinicaltrials.gov/ct2/show/NCT01288911
*  Bioequivalence of Bicalutamide New Formulation in Japan - Full Text View - ClinicalTrials.gov
Bicalutamide. Androgen Antagonists. Hormone Antagonists. Hormones, Hormone Substitutes, and Hormone Antagonists. Physiological ... Bioequivalence of Bicalutamide New Formulation in Japan. The safety and scientific validity of this study is the responsibility ... To investigate the bioequivalence of ICI176,334-1 by assessment of t1/2 (half time) of bicalutamide [ Time Frame: Blood samples ... The purpose of this study is to investigate the bioequivalence of Bicalutamide new formation with Casodex commercial tablet ( ...
  https://clinicaltrials.gov/ct2/show/NCT01416870
*  Bicalutamide With or Without Enzastaurin in Treating Patients With Prostate Cancer - Full Text View - ClinicalTrials.gov
Bicalutamide. Androgen Antagonists. Hormone Antagonists. Hormones, Hormone Substitutes, and Hormone Antagonists. Physiological ... RATIONALE: Androgens can cause the growth of prostate cancer cells. Antihormone therapy, such as bicalutamide, may lessen the ... PURPOSE: This randomized phase II trial is studying bicalutamide to see how well it works compared with giving bicalutamide ... It is not yet known whether giving bicalutamide together with enzastaurin is more effective than bicalutamide alone in treating ...
  https://clinicaltrials.gov/ct2/show/NCT00685633
*  Antineoplaston Therapy in Treating Patients With Stage III or Stage IV Prostate Cancer - Full Text View - ClinicalTrials.gov
Bicalutamide. Androgen Antagonists. Hormones, Hormone Substitutes, and Hormone Antagonists. Physiological Effects of Drugs. ... Phase II Study of Antineoplastons A10 and AS2-1 Capsules With Total Androgen Blockade in Patients With Stage III or IV ... Drug: antineoplaston A10 Drug: antineoplaston AS2-1 Drug: bicalutamide Drug: flutamide Drug: leuprolide acetate Procedure: ... Determine the antitumor activity of antineoplastons A10 and AS2-1 capsules in combination with total androgen blockade in ...
  https://clinicaltrials.gov/ct2/show/NCT00003517
*  Safety and Efficacy Study of Enzalutamide Versus Bicalutamide in Men With Prostate Cancer - Full Text View - ClinicalTrials.gov
Bicalutamide. Androgen Antagonists. Hormone Antagonists. Hormones, Hormone Substitutes, and Hormone Antagonists. Physiological ... Willing to maintain androgen deprivation therapy with a gonadotropin releasing hormone (GnRH) agonist/antagonist or has had a ... Bicalutamide In Men With Prostate Cancer Who Have Failed Primary Androgen Deprivation Therapy. ... Randomized to bicalutamide and receiving bicalutamide at the time of study unblinding; ...
  https://clinicaltrials.gov/ct2/show/NCT01664923?term=Medivation&rank=6
*  SECRETED PROTEIN ACIDIC AND RICH IN CYSTEINE (SPARC) AS CHEMOTHERAPEUTIC SENSITIZERS - Patent application
... androgen antagonists such as flutamide and bicalutamide; and gonadotropin-releasing hormone analogs such as leuprolide. ... estrogen antagonists, tamoxifen, anastrozole; androgens, testosterone propionate, fluoxymesterone, androgen antagonists, ... estrogen antagonists such as tamoxifen and anastrozole; androgens such as testosterone propionate and fluoxymesterone and ... Examples of chemotherapeutic agents include alkylating agents, antimetabolites, natural products, hormones and antagonists, and ...
  http://www.patentsencyclopedia.com/app/20130196929
*  Bicalutamide) Casodex vs Placebo in Non-metastatic Early Prostate Cancer
androgen antagonists. *prostate neoplasms. *Prostatic Neoplasms. .map{width:100%;height:300px;margin-bottom:15px}. Name. ... A Randomized, Double-Blind, Parallel-Group Trial Comparing Bicalutamide (Casodex) 150mg Once Daily With Placebo in Patients ... A Randomized, Double-Blind, Parallel-Group Trial Comparing Bicalutamide (Casodex) 150mg Once Daily With Placebo in Patients ...
  http://www.knowcancer.com/cancer-trials/NCT00673205/
*  S1216, Phase III ADT+TAK-700 vs. ADT+Bicalutamide for Metastatic Prostate Cancer - Full Text View - ClinicalTrials.gov
Androgens. Bicalutamide. Hormones. Hormones, Hormone Substitutes, and Hormone Antagonists. Physiological Effects of Drugs. ... A Phase III Randomized Trial Comparing Androgen Deprivation Therapy + TAK-700 With Androgen Deprivation Therapy + Bicalutamide ... Active Comparator: ADT + Bicalutamide LHRH agonist - given as approved for androgen deprivation at a dose necessary to maintain ... ADT+Bicalutamide for Metastatic Prostate Cancer (S1216). This study is ongoing, but not recruiting participants. ...
  https://clinicaltrials.gov/show/NCT01809691
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The main active ingredient is a nonsteroidal androgen antagonist Bicalutamide.. Andarine selectively connected to the androgen ... LGD-4033 has an excellent ability to bind to androgen receptors on muscle cells with very high affinity (Ki ~ 1 nM) and ... These processes are controlled by the size and frequency of the GnRH pulses and feedback from androgens and estrogens. Low ... Andarine (GTX-007S-4) is a very popular non-steroidal selective androgen receptor modulator (SARM), developed by GTX, Inc. to ...
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*  Bicalutamide and Goserelin or Leuprolide Acetate With or Without Cixutumumab in Treating Patients With Newly Diagnosed...
Androgens. Leuprolide. Goserelin. Bicalutamide. Hormones. Hormones, Hormone Substitutes, and Hormone Antagonists. Physiological ... Active Comparator: Arm II (androgen deprivation therapy) Patients receive androgen deprivation therapy comprising bicalutamide ... Patients receive androgen deprivation therapy comprising bicalutamide PO QD on days 1-28 and either goserelin acetate SC or ... Androgens can cause the growth of prostate cancer cells. Antihormone therapy, such as bicalutamide, goserelin, or leuprolide ...
  https://clinicaltrials.gov/ct2/show/NCT01120236?term=SWOG+0925&rank=1
*  Suberoylanilide hydroxamic acid (vorinostat) represses androgen receptor expression and acts synergistically with an androgen...
... and blocking the effects of androgens with an AR antagonist, bicalutamide, result in markedly enhanced sensitivity to SAHA, ... Evaluation of Interaction between SAHA and the Anti-Androgen Bicalutamide. Dose-response curves were generated for bicalutamide ... represses androgen receptor expression and acts synergistically with an androgen receptor antagonist to inhibit prostate cancer ... represses androgen receptor expression and acts synergistically with an androgen receptor antagonist to inhibit prostate cancer ...
  http://mct.aacrjournals.org/content/6/1/51
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*  China Prostate Cancer Treatment Drugs Industry Forecasts Analysis: MarketReportsOnline
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*  Ligand-Specific Dynamics of the Androgen Receptor at Its Response Element in Living Cells
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  http://pubmedcentralcanada.ca/pmcc/articles/PMC1820481/?lang=en-ca
*  Bicalutamide Supplier | CAS 90357-06-5 | ICI 176,334 | Casodex | Tocris Bioscience
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*  Abstract 2460: Discovery of potent androgen receptor antagonists for treating CRPC and AR+ breast cancer. | Cancer Research
Androgen Receptor (AR) antagonists have been used in clinic to treat prostate cancer. One example is bicalutamide (Casodex®), ... Abstract 2460: Discovery of potent androgen receptor antagonists for treating CRPC and AR+ breast cancer.. Youzhi Tong, Chunyun ... Discovery of potent androgen receptor antagonists for treating CRPC and AR+ breast cancer. [abstract]. In: Proceedings of the ... MDV3100, a more potent AR antagonist (∼5x vs bicalutamide) without residual agonism, has demonstrated excellent efficacy in ...
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*  Comparison of bicalutamide with other antiandrogens - Wikipedia
Rathkopf D, Scher HI (2013). "Androgen receptor antagonists in castration-resistant prostate cancer". Cancer Journal. 19 (1): ... As such, although bicalutamide has not been compared head-to-head to CPA or spironolactone in the treatment of androgen- ... ISBN 978-1-60327-829-4. Singh SM, Gauthier S, Labrie F (February 2000). "Androgen receptor antagonists (antiandrogens): ... This article is a comparison of bicalutamide, a nonsteroidal antiandrogen (NSAA), with other antiandrogens. Bicalutamide and ...
  https://en.wikipedia.org/wiki/Comparison_of_bicalutamide_with_other_antiandrogens
*  EPI-001 - Wikipedia
Masiello D, Cheng S, Bubley GJ, Lu ML, Balk SP (Jul 2002). "Bicalutamide functions as an androgen receptor antagonist by ... EPI-001 is an antagonist of the androgen receptor (AR) that acts by binding covalently to the N-terminal domain (NTD) of the AR ... Unlike antiandrogens such as bicalutamide, EPI-001 does not cause the AR to bind to androgen response elements on the DNA of ... 2009). "A novel androgen receptor splice variant is up-regulated during prostate cancer progression and promotes androgen ...
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*  Flutamide - Wikipedia
"Bicalutamide Functions as an Androgen Receptor Antagonist by Assembly of a Transcriptionally Inactive Receptor". Journal of ... Flutamide acts as a selective antagonist of the androgen receptor (AR), competing with androgens like testosterone and ... Helsen C, Van den Broeck T, Voet A, Prekovic S, Van Poppel H, Joniau S, Claessens F (Aug 2014). "Androgen receptor antagonists ... Sundblad C, Landén M, Eriksson T, Bergman L, Eriksson E (2005). "Effects of the androgen antagonist flutamide and the serotonin ...
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*  SWOG-9346, Hormone Therapy in Treating Men With Stage IV Prostate Cancer - Full Text View - ClinicalTrials.gov
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*  Familial male-limited precocious puberty - Wikipedia
Alternatively, the combination of the androgen receptor antagonist bicalutamide and the aromatase inhibitor anastrozole may be ... "Treatment of familial male-limited precocious puberty with bicalutamide and anastrozole". The Journal of Pediatrics. 149 (3): ...
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