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*  AID 47971 - In vivo beta adrenergic receptor blocking potency was determined by inhibition of tachycardia produced by...
In vivo beta adrenergic receptor blocking potency was determined by inhibition of tachycardia produced by isoproterenol (0.2 mg ...
  https://pubchem.ncbi.nlm.nih.gov/bioassay/47971
*  Characterization of a potentially reversible increase in beta-adrenergic receptors in isolated, neonatal rat cardiac myocytes...
The number of beta-adrenergic receptors was unchanged at 1.2 hours, increased at 1.5-2 hours, and decreased at 3 hours. Thus: ... After 4 hours incubation in potassium cyanide and 2-deoxyglucose, there was a 43% increase in beta-adrenergic receptor number, ... The purpose of this study was to evaluate potential relationships among beta-adrenergic receptor changes, high energy phosphate ... the increased beta-adrenergic receptor density in moderately injured myocytes can be reversed upon removal of the injurious ...
  https://www.semanticscholar.org/paper/Characterization-of-a-potentially-reversible-in-in-Buja-Muntz/30ad456422a57e9acecc669ab325b830fa694ae9
*  ADCY6 Gene - GeneCards | ADCY6 Protein | ADCY6 Antibody
Mediates vasodilatation after activation of beta-adrenergic receptors by isoproterenol (PubMed:17916776). Contributes to bone ... Mediates vasodilatation after activation of beta-adrenergic receptors by isoproterenol (PubMed:17916776). Contributes to bone ... Functions in signaling cascades downstream of beta-adrenergic receptors in the heart and in vascular smooth muscle cells ( ... Functions in signaling cascades downstream of beta-adrenergic receptors in the heart and in vascular smooth muscle cells ( ...
  http://www.genecards.org/cgi-bin/carddisp.pl?gene=ADCY6&origene_gfpshrna_trans=8
*  ADCY6 gene - Genetics Home Reference
Mediates vasodilatation after activation of beta-adrenergic receptors by isoproterenol (PubMed:17916776). Contributes to bone ... Functions in signaling cascades downstream of beta-adrenergic receptors in the heart and in vascular smooth muscle cells ( ... Functions in signaling cascades downstream of the VIP and SCT receptors in pancreas and contributes to the regulation of ... Catalyzes the formation of the signaling molecule cAMP downstream of G protein-coupled receptors (PubMed:17916776, PubMed: ...
  https://ghr.nlm.nih.gov/gene/ADCY6
*  Medihaler-Iso - FDA prescribing information, side effects and uses
Isoproterenol acts directly on beta-adrenergic receptors of tissues supplied by sympathetic nerves. The beta-adrenergic effects ... This may come about by increasing the sensitivity of the beta-adrenergic receptors to isoproterenol. No adverse cardiovascular ... Drug class: adrenergic bronchodilators. Consumer resources. Professional resources. *Isoproterenol Hydrochloride (AHFS ... Beta-adrenergic blocking drugs such as propranolol antagonize the cardiac, bronchodilating, and vasodilating effects of ...
  https://www.drugs.com/pro/medihaler-iso.html
*  DailyMed - ALBUTEROL SULFATE- albuterol syrup
While it is recognized that beta2-adrenergic receptors compared with isoproterenol. While it is recognized that beta2- ... Beta-Blockers. Beta-adrenergic receptor blocking agents not only block the pulmonary effect of beta-agonists, such as albuterol ... adrenergic receptors are the predominant receptors in bronchial smooth muscle, data indicate that there is a population of beta ... studies have demonstrated that albuterol has a preferential effect on beta2-adrenergic receptors compared with isoproterenol. ...
  https://dailymed.nlm.nih.gov/dailymed/drugInfo.cfm?setid=c7713a63-af2a-40d3-8deb-cbb92d5f1cd3
*  CiNii 論文 - スポーツ心臓とは : スポーツに対する循環系
Plasma catecholamine, beta-adrenergic receptors, and isoproterenol sensitivity in endurance trained and non-endurance trained ... Effects of physical training on β-adrenergic receptors in rat myocardial tissue SYLVESTRE-GERVAIS L. ... Autonomic mechanisms of training bradycardia:β-adrenergic receptors in humans WILLIAMS R. S. ...
  http://ci.nii.ac.jp/naid/10008827960
*  anti-ADCY6 antibody | A Cyclase V/VI Polyclonal Antibody-NP 056085.1
Mediates vasodilatation after activation of beta-adrenergic receptors by isoproterenol (PubMed:17916776). Contributes to bone ... Adrenergic Signaling In Cardiomyocytes Pathway Diagram. Adrenergic Signaling In Cardiomyocytes Pathway antibodies. Adrenergic ... Functions in signaling cascades downstream of beta-adrenergic receptors in the heart and in vascular smooth muscle cells ( ... Macrophage Receptor MARCO (MARCO) ELISA Kit. • Thyroglobulin (TG) Antibody • Thymosin Beta 4 (TMSbeta4) ELISA Kit. • Diamine ...
  https://www.mybiosource.com/prods/Antibody/Polyclonal/A-Cyclase-V-VI/ADCY6/datasheet.php?products_id=8521014&cacheID=a0166add1aec9dcaebcdcf7f02b2150e&att=6
*  Cardiovascular Response to Beta-Adrenergic Blockade or Activation in 23 Inbred Mouse Strains
Strain-dependent beta-adrenergic receptor function influences myocardial responses to isoproterenol stimulation in mice. Am J ... Effects of chronic beta-adrenergic receptor stimulation in mice. J Mol Cell Cardiol. 1997;29:2735-2746. [PubMed] ... Atenolol (ate) and isoproterenol (iso) were chosen for their antagonist effects on β-adrenergic receptors. Ate is a β-blocker ... Pharmacogenetics and response to beta-adrenergic receptor antagonists in heart failure. Clin Pharmacol Ther. 2005;77:123-126. [ ...
  http://pubmedcentralcanada.ca/pmcc/articles/PMC2722085/?lang=en-ca
*  Combivent (Ipratropium Bromide and Albuterol Sulfate): Side Effects, Interactions, Warning, Dosage & Uses
... studies have demonstrated that albuterol has a preferential effect on beta2-adrenergic receptors compared with isoproterenol. ... Beta-receptor blocking agents and albuterol inhibit the effect of each other. Beta-receptor blocking agents should be used with ... While it is recognized that beta2-adrenergic receptors are the predominant receptors on bronchial smooth muscle, recent data ... of cardiac beta-adrenergic receptors. The precise function of these receptors, however, is not yet established (see WARNINGS). ...
  https://www.rxlist.com/combivent-drug.htm
*  Proventil HFA (Albuterol Inhalation): Side Effects, Interactions, Warning, Dosage & Uses
... studies have demonstrated that albuterol has a preferential effect on beta2-adrenergic receptors compared with isoproterenol. ... Beta-Blockers. Beta-adrenergic-receptor blocking agents not only block the pulmonary effect of beta-agonists, such as PROVENTIL ... While it is recognized that beta2-adrenergic receptors are the predominant receptors on bronchial smooth muscle, data indicate ... of cardiac beta-adrenergic receptors. The precise function of these receptors has not been established. (See WARNINGS, ...
  https://www.rxlist.com/proventil-drug.htm
*  Effects of Securigera securidaca Extract on Lipolysis and Adipogenesis in Diabetic Rats
... a nonselective beta adrenergic receptor agonist. As expected, 1 μM isoproterenol led to significant elevation in glycerol ... The tissues were treated with vehicle (basal lipolysis) or isoproterenol (stimulated lipolysis) in the absence or presence of S ... μM isoproterenol (ISO) for 90 min. Concentration of SS is shown in parentheses (μg/mL). Data are presented as means ± SEM of 6 ... isoproterenol, penicillin-streptomycin, type-II collagenase, 3-(4,5-dimethyl-2-thiazolyl)-2,5-diphenyl-2H-tetrazolium bromide ( ...
  https://www.hindawi.com/journals/cholesterol/2014/582106/
*  DailyMed - ALBUTEROL- albuterol sulfate tablet
... studies have demonstrated that albuterol has a preferential effect on beta2-adrenergic receptors compared with isoproterenol. ... Beta-Blockers Beta-adrenergic receptor blocking agents not only block the pulmonary effect of beta-agonists, such as albuterol ... While it is recognized that beta2-adrenergic receptors are the predominant receptors in bronchial smooth muscle, data indicate ... are at least in part attributable to stimulation through beta-adrenergic receptors of intracellular adenyl cyclase, the enzyme ...
  https://dailymed.nlm.nih.gov/dailymed/drugInfo.cfm?setid=1c1f3881-2b68-4bdb-a12f-8134fe8ba961
*  Pirbuterol - DrugBank
... studies have demonstrated that pirbuterol has a preferential effect on beta-2 Adrenergic receptors compared with isoproterenol ... While it is recognized that beta-2 adrenergic receptors are the predominant receptors in bronchial smooth muscle, data indicate ... The precise function of these receptors has not been established. The pharmacologic effects of beta adrenergic agonist drugs, ... are at least in proof attributable to stimulation through beta adrenergic receptors of intracellular adenyl cyclase, the enzyme ...
  https://www.drugbank.ca/drugs/DB01291
*  Differences in the Ca2+ response resulting from neurotransmitter stimulations of rat parotid acini and ducts. - PubMed - NCBI
... the beta-adrenergic receptor agonist isoproterenol increased the [Ca2+](i) in only the ductal cells. Additionally, the effects ... Although there was no difference in the alpha1-adrenergic receptor agonist phenylephrine-induced Ca2+ mobilization between ... parotid acini have a greater sensitivity to cholinergic and substance P stimulation and a lesser sensitivity to beta-adrenergic ... In light of these results, substance P and isoproterenol will be useful for identifying parotid acini and ducts, respectively. ...
  https://www.ncbi.nlm.nih.gov/pubmed/20096649?access_num=20096649&link_type=MED&dopt=Abstract
*  Acute and chronic intrarenal alpha- and beta- adrenergic receptor stimulation of renin release in the conscious dog. |...
At the end of the chronic isoproterenol infusion period, beta-adrenergic receptor refractoriness was demonstrated, as PRA did ... Acute and chronic intrarenal alpha- and beta- adrenergic receptor stimulation of renin release in the conscious dog.. C R Ayers ... Acute and chronic intrarenal alpha- and beta- adrenergic receptor stimulation of renin release in the conscious dog. ... Acute and chronic intrarenal alpha- and beta- adrenergic receptor stimulation of renin release in the conscious dog. ...
  http://hyper.ahajournals.org/content/3/5/615
*  Propranolol treatment externalizes beta-adrenergic receptors in guinea pig myocardium and prevents further externalization by...
... as assessed by isoproterenol-stimulated adenylate cyclase activity. After chronic propranolol treatment, ischemia did not ... of beta-adrenergic receptors from a light vesicle fraction to the sarcolemma contributes to up-regulation of beta-receptors ... fractions of beta-adrenergic receptors were used to examine the effects of propranolol on receptor translocation in guinea pig ... Propranolol treatment externalizes beta-adrenergic receptors in guinea pig myocardium and prevents further externalization by ...
  http://circres.ahajournals.org/content/60/1/108
*  Screening for potential beta 2-adrenergic receptor antagonists using CypHer5E and IN Cell Analyzer 1000 ( ...
For live-cell receptor internalization studies a,Screening,for,potential,beta,2-adrenergic,receptor,antagonists,using,CypHer5E, ... used to obtain dose-response and rank-order potency data for both agonist and antagonist treatment of β2-adrenergic receptor ... Introduction CypHer ™ 5 a pH sensitive dye has shown utility in β2-adrenergic receptor agonist screening (1). CypHer5 has been ... Agonist: isoproterenol (Sigma) Antagonist: alprenolol (Sigma) Hoechst™ 33342 (Molecular Probes) Poly-D-lysine, 5 mg (Sigma) 96- ...
  http://www.bio-medicine.org/biology-technology/Screening-for-potential-beta-2-adrenergic-receptor-antagonists-using-CypHer5E-and-IN-Cell-Analyzer-1000-1255-1/
*  Brugada Syndrome - The Clinical Advisor
Isoproterenol, beta-adrenergic receptor agonist, infusion increases inward Ca current and restores the action potential dome, ... alpha-adrenergic agonists, beta-adrenergic blockers, tricyclic or tetracyclic antidepressants, a combination of glucose and ... ST segment elevation and arrhythmias in patients with Brugada syndrome are enhanced by vagotonic agents or beta-adrenergic ... Antiarrhythmic agents such as amiodarone and beta-blockers have been shown to be ineffective. Class Ic antiarrhythmic drugs (eg ...
  https://www.clinicaladvisor.com/cardiology/brugada-syndrome/article/583183/
*  beta.3 adrenergic receptor agonists and uses thereof - Patent # 6706743 - PatentGenius
... beta..sub.3 adrenergic receptor agonists of structural Formula (I), ##STR1##the stereoisomers and prodrugs thereof, and the ... beta..sub.3 adrenergic receptor-mediated diseases, conditions, or disorders in a mammal which methods comprise administering to ... beta..sub.1, .beta..sub.2, or .beta..sub.3 adrenergic receptor. Thenon-selective, full .beta.-adrenergic agonist isoproterenol ... beta..sub.3 Receptor Selectivity Over .beta..sub.1 and .beta..sub.2 Adrenergic Receptors. In vitro .beta..sub.3 receptor ...
  http://www.patentgenius.com/patent/6706743.html
*  Interactions of Hallucinogens with the Glutamatergic System: Permissive Network Effects Mediated Through Cortical Layer V...
... of beta-1 and beta-2 adrenergic receptors in the antidepressant-like effects of centrally administered isoproterenol. J ... Behavioral effects of beta adrenergic agonists and antidepressant drugs after down-regulation of beta-2 adrenergic receptors by ... Nicholas AP, Pieribone VA, Hokfelt T (1993) Cellular localization of messenger RNA for beta-1 and beta-2 adrenergic receptors ... O'Donnell JM (1988) Behavioral consequences of activation of beta adrenergic receptors by clenbuterol: evidence for mediation ...
  https://link.springer.com/chapter/10.1007%2F7854_2017_480
*  Regulation of cardiac beta-adrenergic receptors by captopril. Implications for congestive heart failure. | Circulation
... captopril treatment did not diminish the down-regulation of mononuclear leukocyte beta 2-adrenergic receptors by isoproterenol ... Captopril treatment led to an up-regulation of cardiac beta 1- but not mononuclear leukocyte beta 2-adrenergic receptors and an ... Regulation of cardiac beta-adrenergic receptors by captopril. Implications for congestive heart failure.. A S Maisel, C ... Regulation of cardiac beta-adrenergic receptors by captopril. Implications for congestive heart failure. ...
  http://circ.ahajournals.org/content/80/3/669
*  Beta-2 adrenergic receptor - Wikipedia
... or isoproterenol (USAN) levosalbutamol (INN) or levalbuterol (USAN) orciprenaline (INN) or metaproterenol (USAN) pirbuterol ... Other adrenergic receptors Alpha-1 adrenergic receptor Alpha-2 adrenergic receptor Beta-1 adrenergic receptor Beta-3 adrenergic ... The beta-2 adrenergic receptor (β2 adrenoreceptor), also known as ADRB2, is a cell membrane-spanning beta-adrenergic receptor ... "Insulin stimulates sequestration of beta-adrenergic receptors and enhanced association of beta-adrenergic receptors with Grb2 ...
  https://en.wikipedia.org/wiki/Beta-2_adrenergic_receptor
*  History of catecholamine research - Wikipedia
... he called beta adrenotropic receptor (now β-adrenoceptor or β-adrenergic receptor). ″This concept of two fundamental types of ... "Blocking of inhibitory adrenergic receptors by a dichloro analog of isoproterenol". Journal of Pharmacology and Experimental ... he called alpha adrenotropic receptor (now α-adrenoceptor or α-adrenergic receptor), while the receptor with the second rank ... J. W. Black; A. F. Crowther; R. G. Shanks; A. C. Dornhorst (1964). "A new adrenergic beta-receptor antagonist". The Lancet. 283 ...
  https://en.wikipedia.org/wiki/History_of_catecholamine_research
*  Sympathomimetic drug - Wikipedia
Also, if the amine has bulky substituents, then it will have greater beta adrenergic receptor activity, but if the substituent ... Other examples include phenylephrine, isoproterenol, and dobutamine. Stimulation of the D1 receptor by dopaminergic agonists ... then it will favor the alpha adrenergic receptors. Direct stimulation of the α- and β-adrenergic receptors can produce ... The presence of hydroxy group in the benzene ring at 3rd and 4th position shows maximum alpha- and beta-adrenergic activity.[ ...
  https://en.wikipedia.org/wiki/Sympathomimetic_drug