*  Frontiers | Variation in the oxytocin receptor gene is associated with behavioral and neural correlates of empathic accuracy |...
We investigated the effect of variation in the oxytocin receptor gene (OXTR) and the serotonin transporter gene (SLC6A4) on the ... We investigated the effect of variation in the oxytocin receptor gene (OXTR) and the serotonin transporter gene (SLC6A4) on the ... Heinrichs, M., von Dawans, B., and Domes, G. (2009). Oxytocin, vasopressin, and human social behavior. Front. Neuroendocrinol. ... We investigated the effect of variation in the oxytocin receptor gene (OXTR) and the serotonin transporter gene (SLC6A4) on the ...
  https://www.frontiersin.org/articles/10.3389/fnbeh.2014.00423/full
*  Plus it
... gonadotropin-releasing hormone receptor, and V2 vasopressin receptor, or truncated V2 and CCR5 receptor mutants with their wild ... B1 Bradykinin Receptor Homo-Oligomers in Receptor Cell Surface Expression and Signaling: Effects of Receptor Fragments. Dong ... B1 Bradykinin Receptor Homo-Oligomers in Receptor Cell Surface Expression and Signaling: Effects of Receptor Fragments. Dong ... B1 Bradykinin Receptor Homo-Oligomers in Receptor Cell Surface Expression and Signaling: Effects of Receptor Fragments. Dong ...
  http://molpharm.aspetjournals.org/content/67/1/309
*  Local Overexpression of V1a-Vasopressin Receptor Enhances Regeneration in Tumor Necrosis Factor-Induced Muscle Atrophy
vasopressin receptor gene," Genomics, vol. 31, no. 3, pp. 327-334, 1996. View at Publisher · View at Google Scholar ... Local Overexpression of V1a-Vasopressin Receptor Enhances Regeneration in Tumor Necrosis Factor-Induced Muscle Atrophy. ... M. Alvisi, V. de Arcangelis, L. Ciccone et al., "V1a vasopressin receptor expression is modulated during myogenic ... α in astrocytes by a V1 vasopressin receptor agonist: a cAMP response element-binding protein-dependent mechanism," The Journal ...
  https://www.hindawi.com/journals/bmri/2014/235426/ref/
*  Biased Agonist Pharmacochaperones: Small Molecules in the Toolbox for Selectively Modulating GPCR Activity | SpringerLink
... biased agonists as well as pharmacological chaperones have demonstrated the potential to harness G protein-coupled receptor ... Lolait SJ, Carroll AM, McBride OW, et al (1992) Cloning and characterization of a vasopressin V2 receptor and possible link to ... In most of the cases, it is associated with inactivating mutations of the renal arginine vasopressin V2 receptor leading to ... Robben JH, Sze M, Knoers NV, et al (2007) Functional rescue of vasopressin V2 receptor mutants in MDCK cells by ...
  https://link.springer.com/chapter/10.1007/7355_2017_14
*  Vasopressin receptor 1A - Wikipedia
V1a vasopressin receptor antidiuretic hormone receptor 1A SCCL vasopressin subtype 1a receptor V1-vascular vasopressin receptor ... Vasopressin receptor 1A (V1AR), or arginine vasopressin receptor 1A (officially called AVPR1A) is one of the three major ... "Vasopressin and Oxytocin Receptors: AVPR1A". IUPHAR Database of Receptors and Ion Channels. International Union of Basic and ... the vasopressin receptor AVPR1A distribution differs both between and within species; vasopressin production occurs in the ...
  https://en.wikipedia.org/wiki/Vasopressin_receptor_1A
*  Long-Term Administration and Outcomes of Tolvaptan for Hepatic Edema | OMICS International
Tolvaptan is an oral vasopressin V2 receptor antagonist that became available as therapy for decompensated hepatic cirrhosis- ... Objective: Tolvaptan is an oral vasopressin V2 receptor antagonist that became available as therapy for decompensated hepatic ... In 2013, tolvaptan an oral vasopressin V2 receptor antagonist became available for treatment of fluid retention associated with ... A highly potent human vasopressin V2-receptor antagonist: pharmacological profile and aquaretic effect by single and multiple ...
  https://www.omicsonline.org/open-access/longterm-administration-and-outcomes-of-tolvaptan-for-hepatic-edema-2167-0889-1000220.php?aid=92501
*  Vasopressin V1a Receptors Mediate Posthemorrhagic Systemic Hypertension Thereby Determining Rebleeding Rate and Outcome After...
Application of the V1 Receptor Antagonist. The selective antagonist [deamino-Pen1, O-Me-Tyr2, Arg8]-vasopressin17 (V-1880; Lot ... Role of vasopressin V(1a) and V2 receptors for the development of secondary brain damage after traumatic brain injury in mice. ... Role of arginine vasopressin V1 and V2 receptors for brain damage after transient focal cerebral ischemia. J Cereb Blood Flow ... Increased expression of vasopressin V1a receptors after traumatic brain injury. J Neurotrauma. 2004;21:1090-1102. ...
  http://stroke.ahajournals.org/content/43/1/227
*  Frontiers | The Non-Peptide Arginine-Vasopressin v1a Selective Receptor Antagonist, SR49059, Blocks the Rewarding, Prosocial,...
However, there is growing evidence that the oxytocin/vasopressin system can modulate some the effects of MDMA. In this study, ... However, there is growing evidence that the oxytocin/vasopressin system can modulate some the effects of MDMA. In this study, ... Taken together, these findings show that the oxytocin/vasopressin system is involved in the rewarding, pro-social and ... alone or in combination with the V1a vasopressin antagonist, SR49059 (0.01-1 ng/kg), before carrying out conditioned place ...
  https://www.frontiersin.org/articles/10.3389/fpsyt.2017.00146/full
*  Application # 2011/0124658. SUBSTITUTED OXINDOLE DERIVATIVES AND THEIR USE AS VASOPRESSIN RECEPTOR LIGANDS - Patents.com
... to medicaments comprising them and to their use for the prophylaxis and/or treatment of diseases vasopressin dep ... 1.) a selectivity for the vasopressin V1b receptor over the vasopressin V1a receptor, i.e. the quotient of the binding affinity ... a selectivity for the vasopressin V1b receptor over the vasopressin V2 receptor, i.e. the quotient of the binding affinity to ... receptor subtypes (for example vasopressin V1a, vasopressin V2 and/or oxytocin). [0083] A further preferred embodiment relates ...
  http://patents.com/us-20110124658.html
*  CUL5 - Wikipedia
It was first titled VACM-1, for vasopressin-activated, calcium-mobilizing receptor. Since then, VACM-1 has been shown to be ... "Expression of all known vasopressin receptor subtypes by small cell tumors implies a multifaceted role for this neuropeptide". ... 1999). "VACM-1 receptor is specifically expressed in rabbit vascular endothelium and renal collecting tubule". Am J Physiol. ... 1999). "VACM-1 receptor is specifically expressed in rabbit vascular endothelium and renal collecting tubule". Am. J. Physiol. ...
  https://en.wikipedia.org/wiki/CUL5
*  Frontiers | Role of the Oxytocin Receptor Expressed in the Rostral Medullary Raphe in Thermoregulation During Cold Conditions |...
Additionally, increased expression of the β3-adrenergic receptor gene, Adrb3 was observed in brown adipose tissue. These ... Additionally, increased expression of the β3-adrenergic receptor gene, Adrb3 was observed in brown adipose tissue. These ... and the oxytocin receptor (Oxtr) may be involved in the regulation of food intake in mammals. We therefore suspected the Oxt/ ... and the oxytocin receptor (Oxtr) may be involved in the regulation of food intake in mammals. We therefore suspected the Oxt/ ...
  https://www.frontiersin.org/articles/10.3389/fendo.2015.00180/full
*  KAKEN - Research Projects | Elucidation of Roles for Free Radicals in the AV3V Mechanism Regulating ADH Secretion (KAKENHI...
1998 - 2000, Research Category:Grant-in-Aid for Scientific Research (C), Section:一般, Research Field:Environmental physiology ( ... Negligible role of catecholaminergic receptors in the anteroventral third ventricular region in mediating vasopressin-releasing ... Negligible role of catecholaminergic receptors in the anteroventral third ventricular region in mediating vasopressin-releasing ... Negligible role of catecholaminergic receptors in the anteroventral third ventricular region in mediating vasopressin-releasing ...
  https://kaken.nii.ac.jp/grant/KAKENHI-PROJECT-10670059/
*  5-HT1A receptor - wikidoc
The receptor does not affect vasopressin or renin secretion, unlike the 5-HT2 receptors.[57][58] It has been suggested that ... The serotonin 1A receptor (or 5-HT1A receptor) is a subtype of serotonin receptor (5-HT receptor) that binds the ... Receptor oligomers. The 5-HT1A receptor forms heterodimers with the following receptors: 5-HT7,[81] 5-HT1B, 5-HT1D, GABAB2, ... The 5-HT1A receptor is the most widespread of all the 5-HT receptors. In the central nervous system, 5-HT1A receptors exist in ...
  http://wikidoc.org/index.php/5-HT1A_receptor
*  Effects of long-term vasopressin receptor stimulation on medullary blood flow and arterial pressure | Regulatory, Integrative...
... and a specific vasopressin V1 receptor agonist (V1AG; [Phe2, Ile3, Orn8]- vasopressin) on the renal medullary blood flow and ... vasopressin; 5) could be prevented if a selective vasopressin V1 receptor antagonist was administered simultaneously into the ... 1995) Control of renal medullary blood flow by vasopressin V1 and V2 receptors. Am. J. Physiol. 269(Regulatory Integrative Comp ... 1997) Localization of the vasopressin V1 and V2 receptors within the renal cortical and medullary circulation. Am. J. Physiol. ...
  http://ajpregu.physiology.org/content/275/5/R1420
*  Index by author - December 01, 1998, 287 (3) | Journal of Pharmacology and Experimental Therapeutics
OPC-41061, a Highly Potent Human Vasopressin V2-Receptor Antagonist: Pharmacological Profile and Aquaretic Effect by Single and ... OPC-41061, a Highly Potent Human Vasopressin V2-Receptor Antagonist: Pharmacological Profile and Aquaretic Effect by Single and ... OPC-41061, a Highly Potent Human Vasopressin V2-Receptor Antagonist: Pharmacological Profile and Aquaretic Effect by Single and ... OPC-41061, a Highly Potent Human Vasopressin V2-Receptor Antagonist: Pharmacological Profile and Aquaretic Effect by Single and ...
  http://jpet.aspetjournals.org/content/287/3.index-by-author
*  Basal Forebrain Cholinergic System and Memory | Springer for Research & Development
Ameliorative effect of vasopressin-(4-9) through vasopressin V(1A) receptor on scopolamine-induced impairments of rat spatial ... Galanin receptor/neuropeptide y receptor interactions in the central nervous system. Curr Protein Pept Sci 15(7):666-672PubMed ... Effects of a single administration of oxytocin or vasopressin and their interactions with two selective receptor antagonists on ... Acetylcholine Learning Modulation Consolidation GABA Glutamate Noradrenaline Hypocretin Orexin Vasopressin Oxytocin Substance P ...
  https://rd.springer.com/chapter/10.1007/7854_2016_467
*  5-HT1A receptor - Wikipedia
The receptor does not affect vasopressin or renin secretion, unlike the 5-HT2 receptors. It has been suggested that oxytocin ... The serotonin 1A receptor (or 5-HT1A receptor) is a subtype of serotonin receptor (5-HT receptor) that binds the ... The serotonin 1A receptor is encoded by the HTR1A gene. The 5-HT1A receptor is the most widespread of all the 5-HT receptors. ... 5-HT1A receptors in the dorsal raphe nucleus are co-localized with neurokinin 1 (NK1) receptors and have been shown to inhibit ...
  https://en.wikipedia.org/wiki/5-HT1A_receptor
*  Effects of oxytocin and arginine vasopressin on the proliferation and differentiation of a serotonergic cell line |...
The neuropeptides oxytocin and arginine vasopressin (AVP) are involved in the regulation of social behavior and cognition. The ... Oxytocin receptor within the breast: biological function and distribution. Anticancer Res 18:2181-2186 PubMed ... Morrison TR, Melloni RH Jr (2014) The role of serotonin, vasopressin, and serotonin/vasopressin interactions in aggressive ... Chen Q, Patel R, Sales A, Oji G, Kim J, Monreal AW, Brinton RD (2000) Vasopressin-induced neurotrophism in cultured neurons of ...
  https://www.springermedizin.de/effects-of-oxytocin-and-arginine-vasopressin-on-the-proliferatio/14224878
*  Estrogen receptor beta - Wikipedia
"Differential colocalization of estrogen receptor β (ER-β) with oxytocin and vasopressin in the paraventricular and supraoptic ... nuclear receptor subfamily 3, group A, member 2), is one of two main types of estrogen receptor, a nuclear receptor which is ... ER-β is a member of the family of estrogen receptors and the superfamily of nuclear receptor transcription factors. The gene ... Leo C, Li H, Chen JD (February 2000). "Differential mechanisms of nuclear receptor regulation by receptor-associated ...
  https://en.wikipedia.org/wiki/Estrogen_receptor_beta
*  Anterograde Trafficking of G Protein-Coupled Receptors: Function of the C-Terminal F(X)6LL Motif in Export from the Endoplasmic...
Robben JH, Sze M, Knoers NV, and Deen PM (2006) Rescue of vasopressin V2 receptor mutants by chemical chaperones: specificity ... adenosine A2b receptor; AA3R, adenosine A3 receptor; HH1R, histamine H1 receptor; ML1A, melatonin type 1A receptor; ML1B, ... receptor; D5DR, dopamine D(5) receptor; 5HT1A, human 5-hydroxytryptamine 1A receptor; 5HT1E, 5-hydroxytryptamine 1E receptor; ... 5, A and B). Among these GPCRs, 21 receptors (49%) have either Ile (16 receptors) or Leu residues (5 receptors) (Fig. 5A), and ...
  http://molpharm.aspetjournals.org/content/75/4/751.full
*  SUBSTITUTED OXINDOLE DERIVATIVES AND THEIR USE AS VASOPRESSIN RECEPTOR LIGANDS - Patent application
1.) a selectivity for the vasopressin V1b receptor over the vasopressin V1a receptor, i.e. the quotient of the binding affinity ... a selectivity for the vasopressin V1b receptor over the vasopressin V2 receptor, i.e. the quotient of the binding affinity to ... receptor subtypes (for example vasopressin V1a, vasopressin V2 and/or oxytocin). [0083] A further preferred embodiment relates ... Vasopressin V1b Receptor Binding Assay: Substances: [0214] The test substances were dissolved in a concentration of 10-2 M in ...
  http://www.patentsencyclopedia.com/app/20120322809
*  Inhibition of the CRF1 receptor influences the activity of antidepressant drugs in the forced swim test in rats
... vasopressin, and somatostatin in depressed patients and healthy controls: response to amitriptyline treatment. Depress Anxiety ... The aim of our study was to assess the influence of SN003, a CRF1 receptor blocker, on the activity of imipramine and ... A high CRF1 receptor density has been detected in the cerebral cortex, cerebellum, olfactory bulb, medial septum, hippocampus, ... Inhibition of the CRF1 receptor influences the activity of antidepressant drugs in the forced swim test in rats. Andrzej Wróbel ...
  http://pubmedcentralcanada.ca/pmcc/articles/PMC5509780/
*  Plus it
North W. G., Fay M. J., Longo K. A., Du J. L. Expression of all known vasopressin receptor subtypes by small cell tumors ... Coulson J. M., Stanley J., Staff D., Woll J. P. Evaluation of vasopressin (AVP) and V1a receptor expression in SCLC cell lines ... 1a ⇓ ) is a morphological variant cell line that we have found to express low levels of vasopressin by nested RT-PCR (data not ... Friedmann A. S., Malott K. A., Memoli V. A., Pai S. I., Yu X. M., North W. G. Products of vasopressin gene expression in small- ...
  http://cancerres.aacrjournals.org/content/60/7/1840
*  Congestive heart failure in rats is associated with increased collecting duct vasopressin sensitivity and vasopressin type 2...
... heart failure in rats is associated with increased collecting duct vasopressin sensitivity and vasopressin type 2 receptor ...
  http://www.forskningsdatabasen.dk/catalog/255852519
*  SMART: Secondary literature for NH domain
... these data suggest that LSCPR2 represents an ancestral receptor to the vasopressin/oxytocin receptor family in the vertebrates ... We have cloned a receptor, named LSCPR, for vasopressin-related Lys-conopressin in Lymnaea stagnalis. Lys-conopressin evokes Ca ... A novel G protein-coupled receptor mediating both vasopressin- and oxytocin-like functions of Lys-conopressin in Lymnaea ... Co-evolution of ligand-receptor pairs in the vasopressin/oxytocin superfamily of bioactive peptides. ...
  http://smart.embl.de/smart/show_secondary.cgi?domain=NH