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*  Insulin Downregulates Alpha-2 Adrenergic Receptors in Cultured Glial Cells | SpringerLink
Neuronal and glial cells in culture contain a2-adrenergic receptors, in preparation.Google Scholar ... Glial Cell Insulin Receptor Synaptic Cleft Scatchard Analysis Saturation Experiment This is a preview of subscription content, ... D. W. Clarke, F. T. Boyd, Jr., M. S. Kappy, and M. K. Raizada, Insulin binds to specific receptors and stimulates 2-deoxy-D- ... F. T. Boyd, Jr., and M. K. Raizada, Effects of insulin and tunicamycin on neuronal insulin receptors in culture, Am. J. Phvsiol ...
  https://link.springer.com/chapter/10.1007/978-1-4684-5380-5_17
*  Selective modification of renal alpha 2-adrenergic receptors in Milan hypertensive rat strain. | Hypertension
Cerebral and renal alpha-adrenergic receptors play an important role in the control of blood pressure. We studied alpha- ... Binding of the selective alpha 1-adrenergic antagonist [3H]prazosin and the alpha 2-adrenergic antagonist [3H]rauwolscine was ... In the cerebral cortex, no between-strain differences in alpha 1-adrenergic and alpha 2-adrenergic receptor density and ... adrenergic receptors in the cerebral and renal cortex of Milan hypertensive strain (MHS) and normotensive strain (MNS) rats, a ...
  http://hyper.ahajournals.org/content/10/5/505
*  Alpha-2 adrenergic receptor - Wikipedia
"Identification of duplicated fourth alpha2-adrenergic receptor subtype by cloning and mapping of five receptor genes in ... signal through the α2-adrenergic receptor in the central and peripheral nervous systems. The α2A adrenergic receptor is ... where it sits alongside the more plentiful α1-adrenergic receptor. The α2-adrenergic receptor binds both norepinephrine ... Saunders, C; Limbird, LE (November 1999). "Localization and trafficking of alpha2-adrenergic receptor subtypes in cells and ...
  https://en.wikipedia.org/wiki/Alpha-2_adrenergic_receptor
*  Routine Glucose Monitoring in Postoperative Pheochromocytoma Patients: Yes or No? | SpringerLink
Desensitization of beta-adrenergic receptors by pheochromocytoma. Endocrinology. 1984;114:1272-8.CrossRefPubMedGoogle Scholar ... Tsujimoto G, Honda K, Hoffman BB, Hashimoto K. Desensitization of postjunctional alpha 1- and alpha 2-adrenergic receptor- ... An ultra short-acting Beta-adrenergic blocker. Chest. 1988;93:398-403.CrossRefPubMedGoogle Scholar ... Alpha and beta-blockade further blunt the body's natural response to hypoglycemia which is usually tachycardia, palpitations, ...
  https://link.springer.com/chapter/10.1007%2F978-3-319-92860-9_28
*  Alpha-2A adrenergic receptor - Wikipedia
The alpha-2A adrenergic receptor (α2A adrenoceptor), also known as ADRA2A, is an α2 adrenergic receptor, and also denotes the ... the sites for beta-adrenergic receptor kinase-mediated phosphorylation and desensitization of the alpha 2A-adrenergic receptor ... ADRA2A adrenergic, alpha-2A-, receptor". "α2A-adrenoceptor". IUPHAR Database of Receptors and Ion Channels. International Union ... Handy DE, Gavras H (Nov 1992). "Promoter region of the human alpha 2A adrenergic receptor gene". The Journal of Biological ...
  https://en.wikipedia.org/wiki/Alpha-2A_adrenergic_receptor
*  Table of neurotransmitter actions in the ANS - Wikipedia
Elliott, J. (1997). "Alpha-adrenoceptors in equine digital veins: Evidence for the presence of both alpha1 and alpha2-receptors ... "Effects of 3-Adrenergic Receptor Activation on Rat Urinary Bladder Hyperactivity Induced by Ovariectomy". Journal of ... ISBN 0-7817-7311-3. Schmitz, JM; Graham, RM; Sagalowsky, A; Pettinger, WA (1981). "Renal alpha-1 and alpha-2 adrenergic ... "Involvement of alpha-1 and alpha-2 adrenoceptors in the postlaparotomy intestinal motor disturbances in the rat". Gut. 28 (8): ...
  https://en.wikipedia.org/wiki/Table_of_neurotransmitter_actions_in_the_ANS
*  Role of autonomic nervous system in the pathomechanism of hypertension | Zamojski | Arterial Hypertension
The effect of thyroid hormone on adrenergic receptors. In: Oppenheimer JH. ed. Molecular Basis of Thyroid Hormone Action. ... Alpha 2- and beta-adrenergic receptor binding and action in gluteal adipocytes from patients with hypothyroidism and ... Role of endothelin and endothelin A-type receptor in adaptation of the carotid body to chronic hypoxia. Am J Physiol Lung Cell ... Grassi G. Adrenergic overdrive as the link among hypertension, obesity, and impaired thermogenesis: lights and shadows. ...
  https://journals.viamedica.pl/arterial_hypertension/article/view/44202
*  Apraclonidine Hydrochloride Monograph for Professionals - Drugs.com
Adrenergic alpha1 and alpha2 binding sites are present in bovine retinal blood vessels. Invest Ophthalmol Vis Sci. 1987; 28: ... 3H]Para-Amino-clonidine: a novel ligand which binds with high affinity to α-adrenergic receptors. Life Sci. 1979; 25:769-74. ... Interaction of clonidine and clonidine analogues with α-adrenergic receptors of neuroblastoma × glioma hybrid cells and rat ... Aqueous flow is reduced by the alpha-adrenergic agonist, apraclonidine hydrochloride (ALO 2145). Ophthalmology. 1988; 95:1217- ...
  https://www.drugs.com/monograph/apraclonidine-hydrochloride.html
*  US5583144A - Methods for treating erectile impotence - Google Patents
... the receptors being classified as either alpha or beta subtypes. Alpha-adrenergic receptor antagonism causes relaxation of the ... Nitrosated and nitrosylated alpha-adrenergic receptor antagonist compounds US6514934B1 (en) 1996-02-02. 2003-02-04. Nitromed, ... Nitrosated and nitrosylated alpha-adrenergic receptor antagonists, compositions and methods of use ... Nitrosated and nitrosylated alpha-adrenergic receptor antagonist compounds, compositions and their uses ...
  https://patents.google.com/patent/US5583144?oq=7751826
*  Effect of Circulating Epinephrine on Platelet Function and Hematocrit | Hypertension
Fréden K, Lundborg P, Vilén L, Kutti J. The peripheral platelet count in response to adrenergic alpha- and beta-1-receptor ... Agonistic and antagonistic effects of various alpha-adrenergic agonists in human platelets. Naunyn Schmiedebergs Arch Pharmacol ... Cloning and expression of a human kidney cDNA for an alpha2-adrenergic receptor subtype. Proc Natl Acad Sci U S A. 1988;85:6301 ... Subtypes of alpha2-adrenoceptors: pharmacological and molecular biological evidence converge. Trends Pharmacol Sci. 1988;9:356- ...
  http://hyper.ahajournals.org/content/25/5/1096.full
*  US20090081277A1 - Pharmaceutical formulations and methods for treating ocular conditions - Google Patents
... adrenergic blocker or beta.-adrenergic agonist, e.g. ephidrine, epinephrine, etc.; aldose reductase inhibitor, e.g. epalrestat ... Ocular therapy using alpha-2 adrenergic receptor compounds having enhanced anterior clearance rates ... Additionally, the drug delivery system can comprise a glucocorticoid receptor blocker (such as RU-486) to help reduce ... Ocular therapy using alpha-2 adrenergic receptor compounds having enhanced anterior clearance rates ...
  https://patents.google.com/patent/US20090081277A1/en
*  Systemic Dysregulation in the Development of Hepatocellular Carcinoma | SpringerLink
Hein L, Altman J D, Kobilka B K. Two functionally distinct alpha2-adrenergic receptors regulate sympathetic neurotransmission. ... NMR structural analysis of alpha-bungarotoxin and its complex with the principal alpha-neurotoxinbinding sequence on the alpha ... Alpha 1-adrenergic effects and liver regeneration. Hepatology, 1987, 7: 1189-11894.PubMedCrossRefGoogle Scholar ... Cloning of the gene and cDNA for mammalian beta-adrenergic receptor and homology with rhodopsin. Nature, 1986, 321: 75-79. ...
  https://link.springer.com/chapter/10.1007/978-3-642-28702-2_2
*  Prochlorperazine (Professional Patient Advice) - Drugs.com
... exhibits a strong alpha-adrenergic and anticholinergic blocking effect and depresses the release of hypothalamic and ... IM (as edisylate): 5 to 10 mg 1 to 2 hours before anesthesia induction or to control symptoms during or after surgery; may ... IM (as mesylate): 5 to 10 mg 1 to 2 hours before anesthesia induction; may repeat once if needed during surgery; ... 18 to 39 kg: 2.5 mg 3 times/day or 5 mg 2 times/day as needed (maximum: 15 mg/day) ...
  https://www.drugs.com/ppa/prochlorperazine.html
*  Synephrine - Wikipedia
The potency of synephrine at adrenergic receptors of the β-class (regardless of sub-type) is much lower than at α-receptors. ... differences in activity at alpha-1 and alpha-2 adrenergic receptors." J. Pharmacol. Exp. Ther. 224 559-566. T. Hibino, M. ... An adrenergic antagonist selective for α1 receptors. Reversal of reserpine-induced hypothermia by a drug is a classical test ... The binding of racemic synephrine to cloned human adrenergic receptors has been examined: Ma and co-workers found that ...
  https://en.wikipedia.org/wiki/Synephrine
*  1 - Bollinger bands and macd forex strategy
Midodrine stimulates alpha-one adrenergic receptors. Then, for guest operating systems, right after the project build. 1987), ... ing of CaM to the receptor (118,119,121). Therefore, the SLNs identified may not be histopathologically infiltrated Chapter 6 ... 2 248. Earlymineralization[11] .. reacts with and strategy forex bollinger macd bands. Currently, there are QC ranges for Amx, ... 2-2-(azanediyl)bis[N-(2,6-dimethylphenyl)acetamide], the weakness is in the proximal muscle groups. If the two teams have ...
  http://signali-forex.com/bollinger-bands-and-macd-forex-strategy.html
*  YOHIMBE: Uses, Side Effects, Interactions and Warnings - WebMD
Brodde, O. E., Anlauf, M., Arroyo, J., Wagner, R., Weber, F., and Buck, K. D. Hypersensitivity of adrenergic receptors and ... Evidence for activation of both adrenergic and cholinergic nervous pathways by yohimbine, an alpha 2-adrenoceptor antagonist. ... Implications for the beta-adrenergic receptor hypothesis of antidepressant action. Arch.Gen.Psychiatry 1986;43(12):1155-1161. ... Hui, K. K., Yu, J. L., Chan, W. F., and Tse, E. Interaction of berberine with human platelet alpha 2 adrenoceptors. Life Sci. ...
  https://www.webmd.com/vitamins-supplements/ingredientmono-759-yohimbe.aspx
*  Angiotensin II Decreases a Resting K+ Conductance in Rat Bulbospinal Neurons of the C1 Area | Circulation Research
Alpha(2A)-adrenergic receptors are present in lower brainstem catecholaminergic and serotonergic neurons innervating spinal ... In a previous study, we found that the predominant catecholaminergic receptors of bulbospinal C1 adrenergic cells are α2- ... adrenergic receptors that couple to inwardly rectifying K+ channels.17 In the present experiment, we examined the responses of ... 32 This conductance is the target of several G protein-coupled receptors found commonly on neurons, such as receptors to ...
  http://circres.ahajournals.org/content/78/2/274
*  Dopamine Uptake Inhibitor-Induced Rotation in 6-Hydroxydopamine-Lesioned Rats Involves Both D1 and D2 Receptors but Is...
Henry B, Fox SH, Peggs D, Crossman AR, and Brotchie JM (1999) The alpha2-adrenergic receptor antagonist idazoxan reduces ... Fox SH and Brotchie JM (2000) 5-HT(2C) receptor antagonists enhance the behavioural response to dopamine D(1) receptor agonists ... Actions of alpha2 adrenoceptor ligands at alpha2A and 5-HT1A receptors: the antagonist, atipamezole and the agonist, ... amphetamine-induced rotation in unilateral substantia nigra-lesioned rats by alpha 1 as compared to alpha 2 agonists and ...
  http://jpet.aspetjournals.org/content/312/3/1124
*  Textbook of Psychiatry/Psychopharmacology - Wikibooks, open books for an open world
Prazosin is an alpha-1-adrenergic receptor antagonist. Like clonidine, it is an antihypertensive which can decrease anxiety ... Hydroxyzine is an antihistamine with less affinity for muscarinic and alpha-1-adrenergic receptors than other antihistamines. ... but may have similar receptor occupancy to the more potent SGAs.(Seeman, 2002) It has alpha-adrenergic antagonism and ... Buprenorphine is an opioid mu-receptor partial agonist (with very high affinity for this receptor) that is used as an ...
  https://en.wikibooks.org/wiki/Textbook_of_Psychiatry/Psychopharmacology
*  The autonomic nervous system at high altitude | SpringerLink
Gavras I, Manolis AJ, Gavras H (2001) The alpha2 -adrenergic receptors in hypertension and heart failure: experimental and ... reduction in β-adrenergic receptor density in both left and right ventricles. They also reported an increase in α1-adrenergic ... adrenergic receptors. Studies in rats following prolonged exposure to hypobaric hypoxia have shown a decreased β-adrenergic ... found no change in α1-adrenergic receptor density in either left or right ventricle. Density of adenosine receptors has also ...
  https://link.springer.com/article/10.1007%2Fs10286-006-0395-7
*  Alpha blocker - Wikipedia
However, the most common type of alpha blocker is usually an α1 blocker. Non-selective α-adrenergic receptor antagonists ... are a class of pharmacological agents that act as antagonists on α-adrenergic receptors (α-adrenoceptors). Historically, alpha- ... Alpha-Blockers)" (PDF). British Hypertension Society. "CV Pharmacology , Alpha-Adrenoceptor Antagonists (Alpha-Blockers)". ... This is done by binding to the alpha receptors in smooth muscle or blood vessels. α-blockers can bind both reversibly and ...
  https://en.wikipedia.org/wiki/Alpha_blocker
*  The Latent Inhibition Model of Schizophrenia | SpringerLink
... adrenergic receptors: I. Receptorial, neurochemical, and electrophysiological profile. J Pharmacol Exp Ther. 292: 38-53.Google ... potential antipsychotic displaying marked antagonist properties at alpha(1)- and alpha(2)-adrenergic receptors: II. Functional ... Meltzer, H.Y. and Nash, J.F. (1991) Effects of antipsychotic drugs on serotonin receptors. Pharmacol Rev. 43: 587-604.PubMed ... potential antipsychotic displaying marked antagonist properties at alpha(1)- and alpha(2)- ...
  https://link.springer.com/chapter/10.1007/978-1-4757-4860-4_12
*  The Analgesic Action of Nitrous Oxide Is Dependent on the Release of Norepinephrine in the Dorsal Horn of the Spinal Cord |...
... inhibits nociceptive inputs to sacral dorsal horn nociceptive neurons through alpha2-adrenergic receptors. J Neurophysiol 1998 ... Clearly, if an adrenergic receptor mediates the action in the spinal cord, then an endogenous pathway that releases ... Camarata PJ, Yaksh TL: Characterization of the spinal adrenergic receptors mediating the spinal effects produced by the ... 3. Block of opiate receptors with naltrexone suppressed N2O-evoked norepinephrine release. ( A ) In the absence of naltrexone ( ...
  http://anesthesiology.pubs.asahq.org/article.aspx?articleid=1946596
*  WO1995005464A1 - B7-2: ctla4/cd28 counter receptor - Google Patents
... beta-adrenergic receptor, folate receptor, cholesterol side chain cleavage enzyme, and a host of other cDNAs. It should be ... The pCMV vectors have been used to express the LDL receptor, nuclear factor 1 , Gs alpha polypeptide, polypeptide phosphatase, ... Ctl4a receptor, fusion proteins containing it and uses thereof EP0613944A2 (en) * 1993-01-22. 1994-09-07. Bristol-Myers Squibb ... Ctl4a receptor, fusion proteins containing it and uses thereof EP0613944A2 (en) * 1993-01-22. 1994-09-07. Bristol-Myers Squibb ...
  https://patents.google.com/patent/WO1995005464A1/en
*  Phencyclidine-Induced Deficits in Prepulse Inhibition of Startle are Blocked by Prazosin, an Alpha-1 Noradrenergic Antagonist |...
PPI-disruptive effect of PCP may be mediated in part by alpha-1 adrenergic receptors and that antagonism ofalpha-1 receptors ... In addition to its actions on DA and 5-HT receptors, clozapine also has a high affinity foralpha-1, alpha-2 and muscarinic M1 ... These latter antipsychotics have antagonistic actions at several receptors, including alpha-1 and alpha-2 adrenergic, M1 ... A shared feature of these compounds is a high affinity foralpha-1 adrenergic receptors (Moore et al., 1993;Coward et al., 1989 ...
  http://jpet.aspetjournals.org/content/283/2/666