*  Insulin Downregulates Alpha-2 Adrenergic Receptors in Cultured Glial Cells | SpringerLink
Neuronal and glial cells in culture contain a2-adrenergic receptors, in preparation.Google Scholar ... Glial Cell Insulin Receptor Synaptic Cleft Scatchard Analysis Saturation Experiment This is a preview of subscription content, ... D. W. Clarke, F. T. Boyd, Jr., M. S. Kappy, and M. K. Raizada, Insulin binds to specific receptors and stimulates 2-deoxy-D- ... F. T. Boyd, Jr., and M. K. Raizada, Effects of insulin and tunicamycin on neuronal insulin receptors in culture, Am. J. Phvsiol ...
  https://link.springer.com/chapter/10.1007/978-1-4684-5380-5_17
*  Selective modification of renal alpha 2-adrenergic receptors in Milan hypertensive rat strain. | Hypertension
Cerebral and renal alpha-adrenergic receptors play an important role in the control of blood pressure. We studied alpha- ... Binding of the selective alpha 1-adrenergic antagonist [3H]prazosin and the alpha 2-adrenergic antagonist [3H]rauwolscine was ... In the cerebral cortex, no between-strain differences in alpha 1-adrenergic and alpha 2-adrenergic receptor density and ... adrenergic receptors in the cerebral and renal cortex of Milan hypertensive strain (MHS) and normotensive strain (MNS) rats, a ...
  http://hyper.ahajournals.org/content/10/5/505
*  Alpha-2 adrenergic receptor - Wikipedia
"Identification of duplicated fourth alpha2-adrenergic receptor subtype by cloning and mapping of five receptor genes in ... signal through the α2-adrenergic receptor in the central and peripheral nervous systems. The α2A adrenergic receptor is ... where it sits alongside the more plentiful α1-adrenergic receptor. The α2-adrenergic receptor binds both norepinephrine ... Saunders, C; Limbird, LE (November 1999). "Localization and trafficking of alpha2-adrenergic receptor subtypes in cells and ...
  https://en.wikipedia.org/wiki/Alpha-2_adrenergic_receptor
*  Alpha-2A adrenergic receptor - Wikipedia
The alpha-2A adrenergic receptor (α2A adrenoceptor), also known as ADRA2A, is an α2 adrenergic receptor, and also denotes the ... the sites for beta-adrenergic receptor kinase-mediated phosphorylation and desensitization of the alpha 2A-adrenergic receptor ... ADRA2A adrenergic, alpha-2A-, receptor". "α2A-adrenoceptor". IUPHAR Database of Receptors and Ion Channels. International Union ... Handy DE, Gavras H (Nov 1992). "Promoter region of the human alpha 2A adrenergic receptor gene". The Journal of Biological ...
  https://en.wikipedia.org/wiki/Alpha-2A_adrenergic_receptor
*  Table of neurotransmitter actions in the ANS - Wikipedia
Elliott, J. (1997). "Alpha-adrenoceptors in equine digital veins: Evidence for the presence of both alpha1 and alpha2-receptors ... "Effects of 3-Adrenergic Receptor Activation on Rat Urinary Bladder Hyperactivity Induced by Ovariectomy". Journal of ... ISBN 0-7817-7311-3. Schmitz, JM; Graham, RM; Sagalowsky, A; Pettinger, WA (1981). "Renal alpha-1 and alpha-2 adrenergic ... "Involvement of alpha-1 and alpha-2 adrenoceptors in the postlaparotomy intestinal motor disturbances in the rat". Gut. 28 (8): ...
  https://en.wikipedia.org/wiki/Table_of_neurotransmitter_actions_in_the_ANS
*  US5583144A - Methods for treating erectile impotence - Google Patents
... the receptors being classified as either alpha or beta subtypes. Alpha-adrenergic receptor antagonism causes relaxation of the ... Nitrosated and nitrosylated alpha-adrenergic receptor antagonist compounds US6514934B1 (en) 1996-02-02. 2003-02-04. Nitromed, ... Nitrosated and nitrosylated alpha-adrenergic receptor antagonists, compositions and methods of use ... Nitrosated and nitrosylated alpha-adrenergic receptor antagonist compounds, compositions and their uses ...
  https://patents.google.com/patent/US5583144?oq=7751826
*  Effect of Circulating Epinephrine on Platelet Function and Hematocrit | Hypertension
Fréden K, Lundborg P, Vilén L, Kutti J. The peripheral platelet count in response to adrenergic alpha- and beta-1-receptor ... Agonistic and antagonistic effects of various alpha-adrenergic agonists in human platelets. Naunyn Schmiedebergs Arch Pharmacol ... Cloning and expression of a human kidney cDNA for an alpha2-adrenergic receptor subtype. Proc Natl Acad Sci U S A. 1988;85:6301 ... Subtypes of alpha2-adrenoceptors: pharmacological and molecular biological evidence converge. Trends Pharmacol Sci. 1988;9:356- ...
  http://hyper.ahajournals.org/content/25/5/1096.full
*  US20090081277A1 - Pharmaceutical formulations and methods for treating ocular conditions - Google Patents
... adrenergic blocker or beta.-adrenergic agonist, e.g. ephidrine, epinephrine, etc.; aldose reductase inhibitor, e.g. epalrestat ... Ocular therapy using alpha-2 adrenergic receptor compounds having enhanced anterior clearance rates ... Additionally, the drug delivery system can comprise a glucocorticoid receptor blocker (such as RU-486) to help reduce ... Ocular therapy using alpha-2 adrenergic receptor compounds having enhanced anterior clearance rates ...
  https://patents.google.com/patent/US20090081277A1/en
*  Systemic Dysregulation in the Development of Hepatocellular Carcinoma | SpringerLink
Hein L, Altman J D, Kobilka B K. Two functionally distinct alpha2-adrenergic receptors regulate sympathetic neurotransmission. ... NMR structural analysis of alpha-bungarotoxin and its complex with the principal alpha-neurotoxinbinding sequence on the alpha ... Alpha 1-adrenergic effects and liver regeneration. Hepatology, 1987, 7: 1189-11894.PubMedCrossRefGoogle Scholar ... Cloning of the gene and cDNA for mammalian beta-adrenergic receptor and homology with rhodopsin. Nature, 1986, 321: 75-79. ...
  https://link.springer.com/chapter/10.1007/978-3-642-28702-2_2
*  Prochlorperazine (Professional Patient Advice) - Drugs.com
... exhibits a strong alpha-adrenergic and anticholinergic blocking effect and depresses the release of hypothalamic and ... IM (as edisylate): 5 to 10 mg 1 to 2 hours before anesthesia induction or to control symptoms during or after surgery; may ... IM (as mesylate): 5 to 10 mg 1 to 2 hours before anesthesia induction; may repeat once if needed during surgery; ... 18 to 39 kg: 2.5 mg 3 times/day or 5 mg 2 times/day as needed (maximum: 15 mg/day) ...
  https://www.drugs.com/ppa/prochlorperazine.html
*  1 - Bollinger bands and macd forex strategy
Midodrine stimulates alpha-one adrenergic receptors. Then, for guest operating systems, right after the project build. 1987), ... ing of CaM to the receptor (118,119,121). Therefore, the SLNs identified may not be histopathologically infiltrated Chapter 6 ... 2 248. Earlymineralization[11] .. reacts with and strategy forex bollinger macd bands. Currently, there are QC ranges for Amx, ... 2-2-(azanediyl)bis[N-(2,6-dimethylphenyl)acetamide], the weakness is in the proximal muscle groups. If the two teams have ...
  http://signali-forex.com/bollinger-bands-and-macd-forex-strategy.html
*  YOHIMBE: Uses, Side Effects, Interactions and Warnings - WebMD
Brodde, O. E., Anlauf, M., Arroyo, J., Wagner, R., Weber, F., and Buck, K. D. Hypersensitivity of adrenergic receptors and ... Evidence for activation of both adrenergic and cholinergic nervous pathways by yohimbine, an alpha 2-adrenoceptor antagonist. ... Implications for the beta-adrenergic receptor hypothesis of antidepressant action. Arch.Gen.Psychiatry 1986;43(12):1155-1161. ... Hui, K. K., Yu, J. L., Chan, W. F., and Tse, E. Interaction of berberine with human platelet alpha 2 adrenoceptors. Life Sci. ...
  https://www.webmd.com/vitamins-supplements/ingredientmono-759-yohimbe.aspx
*  Synephrine - Wikipedia
The potency of synephrine at adrenergic receptors of the β-class (regardless of sub-type) is much lower than at α-receptors. ... differences in activity at alpha-1 and alpha-2 adrenergic receptors." J. Pharmacol. Exp. Ther. 224 559-566. T. Hibino, M. ... An adrenergic antagonist selective for α1 receptors. Reversal of reserpine-induced hypothermia by a drug is a classical test ... The binding of racemic synephrine to cloned human adrenergic receptors has been examined: Ma and co-workers found that ...
  https://en.wikipedia.org/wiki/Synephrine
*  Angiotensin II Decreases a Resting K+ Conductance in Rat Bulbospinal Neurons of the C1 Area | Circulation Research
Alpha(2A)-adrenergic receptors are present in lower brainstem catecholaminergic and serotonergic neurons innervating spinal ... In a previous study, we found that the predominant catecholaminergic receptors of bulbospinal C1 adrenergic cells are α2- ... adrenergic receptors that couple to inwardly rectifying K+ channels.17 In the present experiment, we examined the responses of ... 32 This conductance is the target of several G protein-coupled receptors found commonly on neurons, such as receptors to ...
  http://circres.ahajournals.org/content/78/2/274
*  Textbook of Psychiatry/Psychopharmacology - Wikibooks, open books for an open world
Prazosin is an alpha-1-adrenergic receptor antagonist. Like clonidine, it is an antihypertensive which can decrease anxiety ... Hydroxyzine is an antihistamine with less affinity for muscarinic and alpha-1-adrenergic receptors than other antihistamines. ... but may have similar receptor occupancy to the more potent SGAs.(Seeman, 2002) It has alpha-adrenergic antagonism and ... Buprenorphine is an opioid mu-receptor partial agonist (with very high affinity for this receptor) that is used as an ...
  https://en.wikibooks.org/wiki/Textbook_of_Psychiatry/Psychopharmacology
*  Dopamine Uptake Inhibitor-Induced Rotation in 6-Hydroxydopamine-Lesioned Rats Involves Both D1 and D2 Receptors but Is...
Henry B, Fox SH, Peggs D, Crossman AR, and Brotchie JM (1999) The alpha2-adrenergic receptor antagonist idazoxan reduces ... Fox SH and Brotchie JM (2000) 5-HT(2C) receptor antagonists enhance the behavioural response to dopamine D(1) receptor agonists ... Actions of alpha2 adrenoceptor ligands at alpha2A and 5-HT1A receptors: the antagonist, atipamezole and the agonist, ... amphetamine-induced rotation in unilateral substantia nigra-lesioned rats by alpha 1 as compared to alpha 2 agonists and ...
  http://jpet.aspetjournals.org/content/312/3/1124
*  Alpha blocker - Wikipedia
However, the most common type of alpha blocker is usually an α1 blocker. Non-selective α-adrenergic receptor antagonists ... are a class of pharmacological agents that act as antagonists on α-adrenergic receptors (α-adrenoceptors). Historically, alpha- ... Alpha-Blockers)" (PDF). British Hypertension Society. "CV Pharmacology , Alpha-Adrenoceptor Antagonists (Alpha-Blockers)". ... This is done by binding to the alpha receptors in smooth muscle or blood vessels. α-blockers can bind both reversibly and ...
  https://en.wikipedia.org/wiki/Alpha_blocker
*  The Latent Inhibition Model of Schizophrenia | SpringerLink
... adrenergic receptors: I. Receptorial, neurochemical, and electrophysiological profile. J Pharmacol Exp Ther. 292: 38-53.Google ... potential antipsychotic displaying marked antagonist properties at alpha(1)- and alpha(2)-adrenergic receptors: II. Functional ... Meltzer, H.Y. and Nash, J.F. (1991) Effects of antipsychotic drugs on serotonin receptors. Pharmacol Rev. 43: 587-604.PubMed ... potential antipsychotic displaying marked antagonist properties at alpha(1)- and alpha(2)- ...
  https://link.springer.com/chapter/10.1007/978-1-4757-4860-4_12
*  WO1995005464A1 - B7-2: ctla4/cd28 counter receptor - Google Patents
... beta-adrenergic receptor, folate receptor, cholesterol side chain cleavage enzyme, and a host of other cDNAs. It should be ... The pCMV vectors have been used to express the LDL receptor, nuclear factor 1 , Gs alpha polypeptide, polypeptide phosphatase, ... Ctl4a receptor, fusion proteins containing it and uses thereof EP0613944A2 (en) * 1993-01-22. 1994-09-07. Bristol-Myers Squibb ... Ctl4a receptor, fusion proteins containing it and uses thereof EP0613944A2 (en) * 1993-01-22. 1994-09-07. Bristol-Myers Squibb ...
  https://patents.google.com/patent/WO1995005464A1/en
*  Phencyclidine-Induced Deficits in Prepulse Inhibition of Startle are Blocked by Prazosin, an Alpha-1 Noradrenergic Antagonist |...
PPI-disruptive effect of PCP may be mediated in part by alpha-1 adrenergic receptors and that antagonism ofalpha-1 receptors ... In addition to its actions on DA and 5-HT receptors, clozapine also has a high affinity foralpha-1, alpha-2 and muscarinic M1 ... These latter antipsychotics have antagonistic actions at several receptors, including alpha-1 and alpha-2 adrenergic, M1 ... A shared feature of these compounds is a high affinity foralpha-1 adrenergic receptors (Moore et al., 1993;Coward et al., 1989 ...
  http://jpet.aspetjournals.org/content/283/2/666
*  GNAI2 - Wikipedia
McClue SJ, Milligan G (Sep 1990). "The alpha 2B adrenergic receptor of undifferentiated neuroblastoma x glioma hybrid NG108-15 ... Osawa S, Dhanasekaran N, Woon CW, Johnson GL (Nov 1990). "G alpha i-G alpha s chimeras define the function of alpha chain ... GNAI2 has been shown to interact with: EYA2, GPSM2, Interleukin 8 receptor, alpha, MDFI, RGS5, and RIC8A. GRCh38: Ensembl ... Inhibition of adenylyl cyclase activity by muscarinic receptor-activated and constitutively activated G(o) alpha". The Journal ...
  https://en.wikipedia.org/wiki/GNAI2
*  Serafim Guimarães - Wikipedia
... alpha inhibitory and beta inhibitory adrenergic receptors in the guinea-pig stomach". Archives internationales de ... S. Guimarães, W. Osswald (1969). "Adrenergic receptors in the veins of the dog". European Journal of Pharmacology. 5 (2): 188- ... "Crosstalk between presynaptic angiotensin receptors, bradykinin receptors and α2-autoreceptors in sympathetic neurons: a study ... Veins and their receptors remained favourites. Guimarães has summarized the knowledge on blood vessels, their nerves and their ...
  https://en.wikipedia.org/wiki/Serafim_Guimar%C3%A3es
*  Clonidine Evokes Vasodepressor Responses via α2-Adrenergic Receptors in Gigantocellular Reticular Formation | Journal of...
1988) Alpha-2A and alpha-2B adrenergic receptor subtypes: Antagonist binding in tissues and cell lines containing only one ... 1994) Alpha2A-adrenergic receptors are present in lower brainstem catecholaminergic and serotonergic neurons innervating spinal ... Milner TA, Rosin DL, Lee A and Aicher SA (1998) Alpha2A-adrenergic receptors are primarily presynaptic heteroreceptors in the ... adrenergic receptor. GiDA. gigantocellular depressor area. MAP. mean arterial pressure. HR. heart rate. aCSF. artificial ...
  http://jpet.aspetjournals.org/content/289/2/688
*  Smaller cardiac cell size and reduced extra-cellular collagen might be beneficial for hearts of Ames dwarf mice
Rapamycin inhibits alpha 1-adrenergic receptor-stimulated cardiac myocyte hypertrophy but not activation of hypertrophy- ... Prolactin receptor signal transduction pathways and actions determined in prolactin receptor knockout mice. Biochem Soc Trans. ... Growth hormone receptor deficiency in mice results in reduced systolic blood pressure and plasma renin, increased aortic eNOS ... Flyvbjergs, insulin, and insulin A, Kopchick JJ Deletion, but not antagonism, of the mouse growth hormone receptor results in ...
  http://www.ijbs.com/v06p0475.htm
*  Evidence for the Role of Membrane Receptor Lateral Movement in GTP-Binding Protein-Mediated Signal Transduction | SpringerLink
... direct measurements indicate that plasma membrane polypeptide hormone receptors are mobile within the plane of the lipid ... Role of fry subunits of G proteins in targeting the (3-adrenergic receptor kinase to membrane-bound receptors. Science 1992; ... Lateral mobility of tetramethylrhodamine (TMR) labelled G protein alpha and beta gamma subunits in NG 108-15 cells. Cell Signal ... multiple sites of regulation by 3-adrenergic receptor and Mg-' studied in reconstituted receptor-G, vesicles. J Biol Chem 1986 ...
  https://link.springer.com/chapter/10.1007/978-1-4757-0680-2_5