Saralasin - Wikipedia
Saralasin is a competitive angiotensin II receptor antagonist with partial agonist activity. The aminopeptide sequence for ... Saralasin was used to distinguish renovascular hypertension from essential hypertension prior to its discontinuation in January ... Tsang S, Ip S, Wong T, Che C, Leung P (2003). "Differential effects of saralasin and ramiprilat, the inhibitors of renin- ... Ip S, Tsang S, Wong T, Che C, Leung P (2003). "Saralasin, a nonspecific angiotensin II receptor antagonist, attenuates ...
Saralasin
Literature References: A specific antagonist of angiotensin II. Prepn: Sipos et al., DE 2127393 corresp to US 3751404 (1972, 1973 to Norwich Pharmacal). Activity studies: Pals et al., Circ. Res. 29, 673 (1971); Pals, Fulton, Arch. Int. Pharmacodyn. Ther. 204, 20 (1973); Solomon, Buckley, J. Pharm. Sci. 63, 1109 (1974); Streeten et al., N. Engl. J. Med. 292, 657 (1975). Comprehensive review of the acetate: C. T. Huang et al., in Pharmacological and Biochemical Properties of Drug Substances vol. 3, M. E. Goldberg, Ed. (Am. Pharm. Assoc., Washington, DC, 1981) pp 176-225. ...
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Saralasin-induced inhibition of ovulation in the in vitro perfused ratovary is not replicated by the angiotensin II type-2 ...
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... saralasin def: "A partial angiotensin II receptor agonist which is used as an antihypertensive agent." [] synonym: "CHEBI: ...
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... but Hales et al and Previtt and LefHer were not able to confirm positive effects of saralasin or captopril in preventing ...
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... saralasin def: "A partial angiotensin II receptor agonist which is used as an antihypertensive agent." [] synonym: "CHEBI: ...
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DeCS 2009 - February 20, 2009 version
1-Sar-8-Ala Angiotensin II use Saralasin 1-Sar-8-Ile Angiotensin II use 1-Sarcosine-8-Isoleucine Angiotensin II ...
DeCS 2008 - May 16, 2008 version
1-Sar-8-Ala Angiotensin II use Saralasin. 1-Sar-8-Ile Angiotensin II use 1-Sarcosine-8-Isoleucine Angiotensin II ...
DeCS 2009 - February 20, 2009 version
1-Sar-8-Ala Angiotensin II use Saralasin 1-Sar-8-Ile Angiotensin II use 1-Sarcosine-8-Isoleucine Angiotensin II ...
DeCS 2010 - February 12, 2010 version
1-Sar-8-Ala Angiotensin II use Saralasin 1-Sar-8-Ile Angiotensin II use 1-Sarcosine-8-Isoleucine Angiotensin II ...
DeCS 2010 - February 12, 2010 version
1-Sar-8-Ala Angiotensin II use Saralasin 1-Sar-8-Ile Angiotensin II use 1-Sarcosine-8-Isoleucine Angiotensin II ...
DeCS 2013 - July 15, 2013 version
1-Sar-8-Ala Angiotensin II use Saralasin 1-Sar-8-Ile Angiotensin II use 1-Sarcosine-8-Isoleucine Angiotensin II ...
DeCS 2008 - May 16, 2008 version
1-Sar-8-Ala Angiotensin II use Saralasin. 1-Sar-8-Ile Angiotensin II use 1-Sarcosine-8-Isoleucine Angiotensin II ...