Impromidine (INN) is a highly potent and specific histamine H2 receptor agonist. It has been used diagnostically as a gastric ... Histamine agonists Durant G, Duncan W, Ganellin C, Parsons M, Blakemore R, Rasmussen A (1978). "Impromidine (SK&F 92676) is a ...
"Impromidine" is a descriptor in the National Library of Medicines controlled vocabulary thesaurus, MeSH (Medical Subject ... This graph shows the total number of publications written about "Impromidine" by people in this website by year, and whether " ... Below are the most recent publications written about "Impromidine" by people in Profiles. ...
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File:Impromidine.png. Impromidine.png File missing. * File:Indigo original synthesis.png ...
Rupatadine is a second generation, non-sedating, long-acting histamine antagonist with selective peripheral H1 receptor antagonist activity. It further blocks the receptors of the platelet-activating factor (PAF) according to in vitro and in vivo studies.[2] Rupatadine possesses anti-allergic properties such as the inhibition of the degranulation of mast cells induced by immunological and non-immunological stimuli, and inhibition of the release of cytokines, particularly of the TNF in human mast cells and monocytes.[3] ...
Impromidine [D03.383.129.308.445] * Levamisole [D03.383.129.308.480] * Losartan [D03.383.129.308.507] ...
Histamine agonists that possessed an imidazole nucleus (2- and 4-methylhistamine) were affected, whereas impromidine, 2 ...
... rat cortical pieces by histamine was antagonized with the blended H2/H3 receptor agonist/antagonists burimamide and impromidine ...
Impromidine [D03.383.129.308.445] * Levamisole [D03.383.129.308.480] * Losartan [D03.383.129.308.507] ...
A strong organic base existing primarily as guanidium ions at physiological pH. It is found in the urine as a normal product of protein metabolism. It is also used in laboratory research as a protein denaturant. (From Martindale, the Extra Pharmacopoeia, 30th ed and Merck Index, 12th ed) It is also used in the treatment of myasthenia and as a fluorescent probe in HPLC ...
Nizamutdinova IT, Dusio GF, Gasheva OY, Skoog H, Tobin R, Peddaboina C, Meininger CJ, Zawieja DC, Newell-Rogers MK, Gashev AA. Mast cells and histamine are triggering the NF-?B-mediated reactions of adult and aged perilymphatic mesenteric tissues to acute inflammation. Aging (Albany NY). 2016 11 21; 8(11):3065-3090 ...
Taking erythromycin or ketoconazole while taking fexofenadine does increase the plasma levels of fexofenadine, but this increase does not influence the QT interval. The reason for this effect is likely due to transport-related effects, specifically involving p-glycoprotein (p-gp).[17] Both erythromycin and ketoconazole are inhibitors of p-gp, a transporter protein involved in preventing the intestinal absorption of fexofenadine. When p-gp is inhibited, fexofenadine may be better absorbed by the body, increasing its plasma concentration by more than what was intended.[medical citation needed] Fexofenadine is not to be taken with apple, orange, or grapefruit juice because they could decrease absorption of the drug. Therefore, it should be taken with water.[17] Grapefruit juice can significantly reduce the plasma concentration of fexofenadine.[20] Antacids containing aluminium or magnesium should not be taken within 15 minutes of fexofenadine as they reduce the absorption of fexofenadine by almost ...
Madani N, Princiotto AM, Mach L, Ding S, Prevost J, Richard J, Hora B, Sutherland L, Zhao CA, Conn BP, Bradley T, Moody MA, Melillo B, Finzi A, Haynes BF, Smith Iii AB, Santra S, Sodroski J. A CD4-mimetic compound enhances vaccine efficacy against stringent immunodeficiency virus challenge. Nat Commun. 2018 06 18; 9(1):2363 ...
This graph shows the total number of publications written about "Fluspirilene" by people in this website by year, and whether "Fluspirilene" was a major or minor topic of these publications ...
Liu J, Xu N, Wang X, Wang Y, Wu Q, Li X, Pan D, Wang L, Xu Y, Yan J, Li X, Yu L, Yang M. Quantitative radio-thin-layer chromatography and positron emission tomography studies for measuring streptavidin transduced chimeric antigen receptor T cells. J Chromatogr B Analyt Technol Biomed Life Sci. 2021 Oct 01; 1182:122944 ...
This graph shows the total number of publications written about "Etomidate" by people in this website by year, and whether "Etomidate" was a major or minor topic of these publications ...
Impromidine [D02.078.370.500] Impromidine * 3-Iodobenzylguanidine [D02.078.370.510] 3-Iodobenzylguanidine * Methylguanidine [ ...
Alcaftadine is an antagonist at three of the histamine receptors (1, 2 and 4). The main indication for Alcaftadine is for prevention of allergic conjunctivitis. By blocking these three receptors, Alcaftadine has been shown to significantly reduce the effects of allergens. This effect on histamine receptors seems to show lower rates of itching, eosinophil recruitment and redness after exposure to an allergen.[6] The effect of alcaftadine seemed to reduce the amount of eosinophil cells significantly as compared to olopatadine 0.1%. When animal models were used to test alcaftadine, alcaftadine 0.25% seemed to show superior results for decreasing E-cadherin expression as compared to placebo. The reduction of E-cadherin means decreased junctions which would lead to progression of allergic conjunctivitis.[7] ...
This graph shows the total number of publications written about "Fluspirilene" by people in this website by year, and whether "Fluspirilene" was a major or minor topic of these publications ...
impromidine Hs. Antagonist. 5.2 pKi 94 ⤻. pKi 5.2 [94] ...
Impromidine [D02.078.370.500] * 3-Iodobenzylguanidine [D02.078.370.510] * Methylguanidine [D02.078.370.570] * Mitoguazone [ ...
Agonists: Amthamine * Betazole * Dimaprit * Histamine * HTMT * Impromidine * UR-AK49. Antagonists: Bisfentidine Burimamide * ...
Given alone, impromidine facilitated the evoked overflow, whereas burimamide, pheniramine and ranitidine had no effect. The ... The inhibitory effect of histamine was antagonized by impromidine and burimamide, but was not affected by pheniramine, ...
6. Gastric secretory studies in humans with impromidine (SK&F 92676)--a specific histamine H2 receptor agonist.. Hunt RH; Mills ...
Impromidine,create,30-MAR-07,(null),(null) C65903,Impromidine_Hydrochloride,create,30-MAR-07,(null),(null) C65904,Imuracetam, ...
Dose-response curve analysis of gastric secretory responses in the dog and man to impromidine: a new histamine-H2-receptor ...
Impromidine Entry term(s):. Hydrochloride, Impromidine. Impromidine Hydrochloride. Impromidine Oxalate (1:2). Impromidine ... Impromidine - Preferred Concept UI. M0026470. Scope note. A highly potent and specific histamine H2 receptor agonist. It has ...
Impromidine (substance). Code System Preferred Concept Name. Impromidine (substance). Concept Status. Published. ...
Impromidine Hydrochloride Impromidine Oxalate (1:2) Impromidine Trihydrochloride SK&F-92676 SKF-92676 Pharm Action. Histamine ... use IMPROMIDINE (NM) to search IMPROMIDINE 1980-92. History Note. 93; was IMPROMIDINE (NM) 1979-92. Date Established. 1993/01/ ... Impromidine Oxalate (1:2) Narrower Concept UI. M0329222. Registry Number. 63169-77-7. Terms. Impromidine Oxalate (1:2) ... Impromidine Hydrochloride Narrower Concept UI. M0329223. Registry Number. E57WP5Y41J. Terms. Impromidine Hydrochloride ...
Impromidine Hydrochloride Impromidine Oxalate (1:2) Impromidine Trihydrochloride SK&F-92676 SKF-92676 Pharm Action. Histamine ... use IMPROMIDINE (NM) to search IMPROMIDINE 1980-92. History Note. 93; was IMPROMIDINE (NM) 1979-92. Date Established. 1993/01/ ... Impromidine Oxalate (1:2) Narrower Concept UI. M0329222. Registry Number. 63169-77-7. Terms. Impromidine Oxalate (1:2) ... Impromidine Hydrochloride Narrower Concept UI. M0329223. Registry Number. E57WP5Y41J. Terms. Impromidine Hydrochloride ...
Impromidine Impromidine is a highly potent and specific histamine H2 receptor agonist. It has been used diagnostically as a ...
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Treatment with oral clotrimazole blocks Ca(2+)-activated K+ transport and reverses erythrocyte dehydration in transgenic SAD mice. A model for therapy of sickle cell disease. J Clin Invest. 1994 Apr; 93(4):1670-6 ...
... hippocampus 5 Impromidine Cimetidine No Postsynaptic Gs Caudate-putamen, cerebral cortex, amygdala. ...
HISTAMINE AGENTS IMPROMIDINE HISTAMINE AGENTS KETOTIFEN HISTAMINE AGENTS LORATADINE HISTAMINE AGENTS MECLIZINE HISTAMINE AGENTS ... HISTAMINE AGONISTS IMPROMIDINE HISTAMINE AGONISTS ANTAZOLINE HISTAMINE ANTAGONISTS ASTEMIZOLE HISTAMINE ANTAGONISTS ... NEUROTRANSMITTERS AND NEUROTRANSMITTER IMPROMIDINE NEUROTRANSMITTERS AND NEUROTRANSMITTER INDORAMIN NEUROTRANSMITTERS AND ... NEUROTRANSMITTER AGENTS IMPROMIDINE NEUROTRANSMITTER AGENTS INDORAMIN NEUROTRANSMITTER AGENTS IODOCYANOPINDOLOL ...
Buzdar AU, Smith R, Vogel C, Bonomi P, Keller AM, Favis G, Mulagha M, Cooper J. Fadrozole HCL (CGS-16949A) versus megestrol acetate treatment of postmenopausal patients with metastatic breast carcinoma: results of two randomized double blind controlled multiinstitutional trials. Cancer. 1996 Jun 15; 77(12):2503-13 ...
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An antihypertensive agent that acts by inhibiting selectively transmission in post-ganglionic adrenergic nerves. It is believed to act mainly by preventing the release of norepinephrine at nerve endings and causes depletion of norepinephrine in peripheral sympathetic nerve terminals as well as in tissues ...
This graph shows the total number of publications written about "Robenidine" by people in this website by year, and whether "Robenidine" was a major or minor topic of these publications ...
Impromidine [D03.383.129.308.445] * Levamisole [D03.383.129.308.480] * Losartan [D03.383.129.308.507] ...
Agonists: Amthamine * Betazole * Dimaprit * Histamine * HTMT * Impromidine * UR-AK49. Antagonists: Bisfentidine Burimamide * ...