*  Steroid‐induced androgen receptor-oestradiol receptor β-Src complex triggers prostate cancer cell proliferation | The EMBO...
An oestradiol antagonist (ICI 182,780) prevents complex assembly and pathway activation not only by oestradiol but also by ... Antagonist cross‐inhibition in MCF‐7 and T47D cells of androgen or oestradiol action. To answer the question of whether the ... Antagonist cross‐inhibition of signalling pathway activation by androgen or oestradiol in LNCaP cells. Based on the effects of ... Antagonist cross‐inhibition of LNCaP growth stimulated by androgen or oestradiol. LNCaP cells were maintained for 4 days under ...
  http://emboj.embopress.org/content/19/20/5406?ijkey=cb9909929b3c3ec1ee605549dc94c8ed1734ed9c&keytype2=tf_ipsecsha
*  Anabolic steroid-induced hypogonadism - towards a unified hypothesis of anabolic steroid action
Enclomiphene is an estradiol antagonist, while zuclomipheneis an estradiol agonist. The addition of tamoxifen to clomiphene ... Estradiol has a much larger, inhibitory effect than . AAS treatment for these conditions is towards disease-asso- testosterone ... These need to be followed up with well- mers, which have opposite effects upon the estradiol receptor controlled clinical ... Estradiol modulates the pulsatile secretion of athletes: effects upon hostility and aggression. Hum Psychopharmacol ...
  http://marysfamilymedicine.org/a/asih.net1.html
*  Markaverich BM[au] - PubMed - NCBI
Type II [3H]estradiol binding site antagonists: inhibition of normal and malignant prostate cell growth and proliferation. ... Effects of estradiol-17 alpha on nuclear occupancy of the estrogen receptor, stimulation of nuclear type II sites and uterine ... Nuclear type II [3H]estradiol binding site ligands: inhibition of ER-positive and ER-negative cell proliferation and c-Myc and ... The effect of low dose continuous exposure to estradiol on the estrogen receptor (type I) and nuclear type II sites. ...
  https://www.ncbi.nlm.nih.gov/pubmed?cmd=search&term=Markaverich+BM%5Bau%5D&dispmax=50
*  Estrogen Dominance, Natural Progesterone and Men | DrDekel.com
The male hormone, testosterone, is an antagonist to estradiol (E2). It is made from progesterone. Men normally continue to ... When the level of testosterone decreases, the relative level of estradiol in men increases. Estradiol, turns on BCL2 oncogene ( ... Men produce estrogen (Estradiol) but in much lower amount than women. Men also produce progesterone, but about half the amount ...
  http://www.drdekel.com/content/estrogen-dominance-natural-progesterone-and-men
*  List of MeSH codes (D06) - Wikipedia
File "2006 MeSH Trees".) MeSH D06.347.360.315 --- estrogen antagonists MeSH D06.347.360.315.300 --- estradiol antagonists MeSH ... ethinyl estradiol MeSH D06.472.334.851.437.968.500.250 --- ethinyl estradiol-norgestrel combination MeSH D06.472.334.851. ... estradiol congeners MeSH D06.472.334.851.437.249 --- equilenin MeSH D06.472.334.851.437.374 --- equilin MeSH D06.472.334.851. ... 437.500 --- estradiol MeSH D06.472.334.851.437.750 --- estriol MeSH D06.472.334.851.437.750.320 --- estetrol MeSH D06.472. ...
  https://en.wikipedia.org/wiki/List_of_MeSH_codes_(D06)
*  MEDLINE Data Changes - 2015. NLM Technical Bulletin. 2014 Nov-Dec
Dopa Decarboxylase /antagonists & inhibitors. Aromatic Amino Acid Decarboxylase Inhibitors. Estradiol /antagonists & inhibitors ... Receptor, Bradykinin B1 /antagonists & inhibitors. Bradykinin B1 Receptor Antagonists. Receptor, Bradykinin B2 /antagonists & ... Receptor, Endothelin A /antagonists & inhibitors. Endothelin A Receptor Antagonists. Receptor, Endothelin B /antagonists & ... Receptors, CCR5 /antagonists & inhibitors. CCR5 Receptor Antagonists. Receptors, Dopamine D2 /antagonists & inhibitors. ...
  https://www.nlm.nih.gov/pubs/techbull/nd14/nd14_medline_data_changes_2015.html
*  Levothyroxine - Wikipedia
Antagonists: 3,17β-Estradiol. *3α-Androstanol. *3α-Androstenol. *3β-Androstanol ...
  https://en.wikipedia.org/wiki/Levothyroxine
*  5α-Dihydroprogesterone - Wikipedia
Antagonists: 3,17β-Estradiol. *3α-Androstanol. *3α-Androstenol. *3β-Androstanol ...
  https://en.wikipedia.org/wiki/5-alpha-dihydroprogesterone
*  The Link between "The Pill" and Prostate Cancer
Fortunately, testosterone is also antagonist to estrogens like estradiol, which may explain why men with low testosterone are ... Like women, men also make estrogens such as estradiol, although (usually) in much lower amounts than women. ... Even the characteristically "male" hormone testosterone can be converted into estradiol via the hormone aromatase - which is ...
  https://articles.mercola.com/sites/articles/archive/2012/01/02/use-of-pill-raise-prostate-cancer-risk.aspx
*  Effects of Transdermal 17β-Estradiol on Left Ventricular Anatomy and Performance in Hypertensive Women | Hypertension
It is known that 17β-estradiol has a powerful calcium antagonist effect on both vascular smooth muscle cells and cardiac fibers ... 17β-Estradiol attenuates voltage-dependent Ca2+ currents in A7r5 vascular smooth muscle cell line. Am J Physiol. 1994;266:C975- ... 17β-estradiol was administered in the form of self-adhesive cutaneous patches, which provided a cutaneous absorption rate of 50 ... Effects of Transdermal 17β-Estradiol on Left Ventricular Anatomy and Performance in Hypertensive Women. Maria Grazia Modena, ...
  http://hyper.ahajournals.org/content/34/5/1041
*  Patente US6906086 - Methods for inhibiting bone loss - Google Patentes
... and actually serve as potent antagonists of natural estrogens such as estradiol. In contrast to the report of Feldmann, S. et ... Estradiol, as expected, caused a large increase in eosinophil infiltration.. Little or no difference was detectable between ... Richards J, Imagawa W, Balakrishnan A, Edery M, Nandi S. The lack of effect of phenol red or estradiol on the growth response ... Synergistic actions of estradiol and the insulin-like growth factor Somatomedin-C on swine ovarian (granulosa) cells. ...
  http://www.google.es/patents/US6906086?hl=es&dq=flatulence
*  Plus it
We also defined the E217βG antagonist, tamoxifen, as a novel substrate and stimulator of ABCC10. In addition, a number of ... LTC4, the estrogen estradiol-glucuronide (E217βG) and glutathione are physiologic substrates for ABCC1, and induce ABCC1 ATPase ... 3C inset). The compound tamoxifen is frequently used in breast cancer treatments as an estrogen receptor antagonist, based on ... Using crude membranes in an ABCC10 overexpression system, we found that the ABCC10 transport substrates estrogen estradiol- ...
  http://cancerres.aacrjournals.org/content/72/24/6457
*  Drug Information Portal - U.S. National Library of Medicine - Quick Access to Quality Drug Information
Blocks aromatization of testosterone to estradiol; aromatase antagonist. Category:. * Info Enzyme Inhibitors ...
  https://druginfo.nlm.nih.gov/drugportal/rn/633-35-2
*  Frontiers | Estradiol Binds to Insulin and Insulin Receptor Decreasing Insulin Binding in vitro | Endocrinology
200 nM estradiol shifted the binding curve of insulin to its receptor 0.8 log units to the right. Conclusions: Estradiol ... 200 nM estradiol shifted the binding curve of insulin to its receptor 0.8 log units to the right. Conclusions: Estradiol ... Main Results: Estradiol bound to insulin with a Kd of 12 x 10-9 M and to the insulin receptor with a Kd of 24 x 10-9 M, while ... Main Results: Estradiol bound to insulin with a Kd of 12 x 10-9 M and to the insulin receptor with a Kd of 24 x 10-9 M, while ...
  https://www.frontiersin.org/articles/10.3389/fendo.2014.00118/full
*  Science--Whitacre et. al
... the estrogen antagonist tamoxifen or by antibody to estradiol (63). Collectively, these observations indicate that estrogens ... both IL-10 and IFN-γ production were increased in the presence of estradiol (31). Sex steroid regulation of cytokine production ... progesterone or estradiol alone suppressed disease, whereas medroxyprogesterone potentiated EAE (53). Similarly, estrogen ...
  http://www.sciencemag.org/site/feature/data/983519.xhtml
*  Protocols and Video Articles Authored by Peng Jin (Translated to Danish)
In cultured COLO205 cells, the effect of estradiol (E2) and antagonist ICI182.780 on the expression of hMLH1 and hMSH2 was ... Alterations in selective serum hormone levels, including FSH, LH and 17β-estradiol, are seen in this mouse model, which mimics ...
  https://www.jove.com/author/Peng_Jin?language=Danish
*  Chromatin Remodeling and Pregnancy-Induced Differentiation | SpringerLink
... content and chromatin texture of human breast epithelial cells transformed with 17-beta-estradiol and the estrogen antagonist ... Mello ML, Russo P, Russo J, Vidal BC (2009) Entropy of Feulgen-stained 17-beta-estradiol-transformed human breast epithelial ... prevents the transformed phenotypes induced by 17 beta-estradiol in human breast epithelial cells. Cell Biol Int 33:1135-1143 ...
  https://link.springer.com/chapter/10.1007/978-1-4614-4884-6_7
*  Recycle (100 Capsules) Reviews - AnabolicMinds.com
One possibility is that the kelp may be acting as an estrogen antagonist by preventing estradiol from binding with its estrogen ...
  http://anabolicminds.com/forum/product-review/211085-recycle-100-capsules.html
*  PPT - Physiology of Penile Erection and Pathophysiology of Erectile Dysfunction PowerPoint Presentation - ID:1091514
Treatment with flutamide, estradiol, or a gonadotropin-releasing hormone antagonist in addition to castration further depresses ... α-Adrenoceptor Blockers- positive effect on erection for α antagonists, particularly those acting on the α1 receptor - drugs ... β antagonists also exert an inhibitory effect within the CNS, perhaps leading to lowered sex hormone levels - nonselective ... Angiotensin II receptor antagonists, have a beneficial effect on existing sexual dysfunction at baseline ...
  https://www.slideserve.com/halle/physiology-of-penile-erection-and-pathophysiology-of-erectile-dysfunction
*  Fulvestrant (F)/Goserelin (G) vs Anastrozole (A)/G vs G for Premenopausal Women - Full Text View - ClinicalTrials.gov
Estradiol. Estrogen Antagonists. Hormone Antagonists. Hormones, Hormone Substitutes, and Hormone Antagonists. Physiological ... a plasma estradiol in the premenopausal range (≥20 pg/mL), ④ if in case of chemotherapy induced amenorrhea, a plasma estradiol ... Fulvestrant is an ER antagonist with no agonist effects, which binds, blocks and degrades the ER. Fulvestrant is comparable to ... Estrogen Receptor Antagonists. Estrogens. Hormones. Aromatase Inhibitors. Steroid Synthesis Inhibitors. Enzyme Inhibitors. ...
  https://clinicaltrials.gov/ct2/show/NCT01266213
*  Patent US20070269522 - Transdermal Drug Delivery Device with Translucent Protective Film - Google Patents
... anti-ulceratives such as H2 antagonists; steroidal hormones (e.g., progesterone, testosterone, estradiol); antivirals and/or ... The average concentration of estradiol in samples not exposed to UV radiation was 20.45 mg per gram of adhesive. The average ... Some examples include, clonidine, estradiol, nicotine, nitroglycerine, scopolamine, and fentanyl, which are commercially ... estradiol, an acrylate copolymer adhesive, and Kollidon VA 64. The resulting adhesive formulation was knife coated onto a ...
  http://www.google.ca/patents/US20070269522
*  Nina S Stachenfeld, PhD | Yale School of Medicine
... a saline load in gonadotropin-releasing hormone antagonist-pretreated premenopausal women receiving progesterone or estradiol- ... Mechanisms contributing to low orthostatic tolerance in women: the influence of oestradiol Wenner, M.M., Haddadin, A.S., Taylor ... While the women are suppressed, we add-back controlled levels of estradiol and progesterone to test the hypothesis of interest ... Over my first seven years at Yale we demonstrated that estradiol, with and without progesterone, alters the osmotic regulation ...
  http://medicine.yale.edu/intranet/facultybydept/nina_stachenfeld-2.profile
*  Optimizing Ovulation Induction in the Poor Responder - Full Text View - ClinicalTrials.gov
6 Luteal estradiol and GnRH antagonist administration prior to controlled ovarian hyperstimulation for in vitro fertilization ( ... Drug Information available for: Estradiol Estradiol cypionate Estradiol valerate Estradiol acetate Estradiol hemihydrate ... Estradiol. Polyestradiol phosphate. Estradiol 3-benzoate. Estradiol 17 beta-cypionate. Estradiol valerate. Contraceptive Agents ... Group 1: Luteal estradiol • Starting cycle day 20, two 0.1 mg/d transdermal estradiol patch will be applied every other day ...
  https://clinicaltrials.gov/ct2/show/study/NCT01200537?show_desc=Y
*  Process for the production of microcapsules - Patent # 5648096 - PatentGenius
C. Sex hormones (female/male)/anabolic steroids/hormone antagonists, e.g. estradiol, estradiolvalerate, estradiolbenzoate, ... The production of microcapsules, containing a hormone: 25 g 17-beta-estradiol were dissolved in a mixture of 125 ml anhydrous ... The production of microcapsules containing a hormone: 10 g 17-beta-estradiol were dissolved in a mixture of 100 ml anhydrous ... opioid antagonists, e.g.naloxone, nalorphin, levallorphan, and opioid analgesics, e.g. morphine, hydromorphone, oxycodone, ...
  http://www.patentgenius.com/patent/5648096.html