• Oxanamide (Quiactin) is an anxiolytic and muscle relaxant which can produce sedative and hypnotic effects in sufficiently high doses. (wikipedia.org)
  • Xanax belongs to the benzodiazepine class of drugs, prescribed primarily for its sedative and anxiolytic (anti-anxiety) properties. (oxfordbusinessgroup.com)
  • A centrally acting skeletal muscle relaxant whose mechanism of action is not completely understood but may be related to its sedative actions. (rxmedworld.co)
  • Carisoprodol is a central nervous system depressant that acts as a sedative and skeletal muscle relaxant. (rxmedworld.co)
  • Diazepam is a benzodiazepine that exerts anxiolytic, sedative, muscle- relaxant, anticonvulsant and amnestic effects. (virtualpsychcentre.com)
  • Diazepam has similar sedative and hypnotic effects as barbiturates , but unlike the older drugs, diazepam is a more effective anxiolytic, it is much less likely to result in lethal overdose, and it is said to have a lower potential for abuse and dependence. (virtualpsychcentre.com)
  • Belonging to the azaspirodecanedione drug class, 2 buspirone is a serotonin 5-HT 1A receptor agonist that is not chemically or pharmacologically related to benzodiazepines, barbiturates, and other sedative/anxiolytic drugs. (arlen.com.br)
  • Buspirone hydrochloride tablets, USP are an antianxiety agent that is not chemically or pharmacologically related to the benzodiazepines, barbiturates, or other sedative/anxiolytic drugs. (arlen.com.br)
  • A class of psychoactive drugs that are commonly used for their sedative, hypnotic, anxiolytic, anticonvulsant, and muscle relaxant properties. (globalcocaineshop.se)
  • Thе etizolam mоlесulе differs frоm a bеnzоdіаzеріnе in thаt thе bеnzеnе rіng hаѕ bееn rерlасеd bу a thіорhеnе rіng and triazole ring hаѕ bееn fuѕеd, аnxіоlуtіс, аntісоnvulѕаnt, hурnоtіс, sedative аnd (globalcocaineshop.se)
  • Etizolam is known for its sedative, anxiolytic (anti-anxiety), and muscle relaxant effects. (globalcocaineshop.se)
  • Alpha-1-containing rесерtоrѕ mеdіаtе thе sedative еffесtѕ of еtіzоlаm whеrеаѕ alpha-2 аnd аlрhа-3 ѕubunіt-соntаіnіng rесерtоrѕ mediate the anxiolytic еffесt. (globalcocaineshop.se)
  • Rohypnol is known for its strong sedative properties, which can induce drowsiness, muscle relaxation, and a calming effect on the central nervous system. (welevelup.com)
  • Benzodiazepines work by enhancing the effects of the neurotransmitter gamma-aminobutyric acid (GABA) in the brain, leading to sedative, anxiolytic (anti-anxiety), muscle relaxant, and anticonvulsant effects. (welevelup.com)
  • An anxiolytic benzodiazepine derivative with anticonvulsant, sedative, and amnesic properties. (minclinic.ru)
  • The net neuro-inhibitory effects result in the observed sedative, hypnotic, anxiolytic, and muscle relaxant properties. (minclinic.ru)
  • This calming effect gives benzodiazepines their sedative, hypnotic (sleep-inducing), anxiolytic (anti-anxiety), anticonvulsant, and muscle relaxant properties. (tripsitter.com)
  • Other pharmacological agents producing sedation (sedatives and agents used off-label for sedative side-effects) should be used cautiously for the treatment of insomnia due to the increased risk of next day sleepiness as well as for known toxicities and adverse side effects. (springer.com)
  • It has been termed anxioselective because it lacks anticonvulsant, sedative, or muscle-relaxant properties. (cemona.es)
  • It belongs to the class of drugs known as benzodiazepines, but unlike other benzodiazepines, it does not have sedative, muscle relaxant, or memory-impairing effects. (modapharma.org)
  • Using prolonged-release morphine sulfate tablets in combination with other central nervous system inhibitors (e.g. sedatives, anxiolytics, hypnotics, antipsychotics, muscle relaxants, other opioids) may result in hypotension and severe sedation and coma, or respiratory depression. (bestmedico.co)
  • In this brief overview, medications used to treat insomnia such as hypnotics, sedatives, medications inducing sedation as a side effect, medications directed at the sleep-associated circadian neuroendocrine system, and agents utilized in treating insomnia-inducing sleep diagnoses such as restless leg syndrome are discussed. (springer.com)
  • Medications for treating insomnia are classified as hypnotics, sedatives, medications inducing sedation as a side effect, medications directed at the sleep-associated circadian neuroendocrine system, and agents utilized in treating insomnia-inducing sleep diagnoses such as restless leg syndrome (RLS) (Curry et al. (springer.com)
  • Ambien is a member of the drug class sedatives, hypnotics, and anxiolytics. (practicalanxietysolutions.com)
  • It is classed with other anxiolytics (drugs that reduce Anxiety), sedatives, and hypnotics that have different mechanisms of action from other medications in their respective classes. (practicalanxietysolutions.com)
  • The most frequently prescribed medications are in the class of antipsychotics and antihistamines, followed by anxiolytics/sedatives. (bvsalud.org)
  • Due to the risk of respiratory depression with concomitant use of skeletal muscle relaxants and opioids, consider prescribing naloxone for the emergency treatment of opioid overdose [see Dosage and Administration (2.2) , Warnings and Precautions (5.3 , 5.5) ]. (medlibrary.org)
  • If a decision is made to prescribe estazolam concomitantly with opioids, prescribe the lowest effective dosages and minimum durations of concomitant use, and follow patients closely for signs and symptoms of respiratory depression and sedation. (dvago.pk)
  • Advise both patients and caregivers about the risks of respiratory depression and sedation when estazolam is used with opioids. (dvago.pk)
  • CNS Depressant/Alcohol Interaction Additive pharmacodynamic effects may be expected when KADIAN is used in conjunction with alcohol, other opioids, or illicit drugs that cause central nervous system depression. (clustermed.info)
  • Follow patients for signs and symptoms of respiratory depression and sedation. (nih.gov)
  • Monitor patients for respiratory depression and sedation at frequent intervals. (medlibrary.org)
  • If a CYP3A4 inducer is discontinued, consider a acetaminophen and codeine phosphate tablets dosage reduction and monitor for signs of respiratory depression and sedation at frequent intervals. (medlibrary.org)
  • limit dosages and durations to the minimum required and follow patients for signs and symptoms of respiratory depression and sedation ( 5.4 ). (drugs.com)
  • Follow patients closely for signs of respiratory depression and sedation. (medlibrary.org)
  • Monitor closely for signs of respiratory depression and sedation. (medscape.com)
  • Chloridiazepide binds to stereospecific benzodiazepine (BZD) binding sites on GABA (A) receptor complexes at several sites within the central nervous system , including the limbic system and reticular formation. (minclinic.ru)
  • Diazepam , first marketed as Valium , is a medicine of the benzodiazepine family that acts as an anxiolytic. (worldsbest.rehab)
  • Tofisopam is a benzodiazepine that acts on the central nervous system to produce anxiolytic (anxiety-reducing) effects. (modapharma.org)
  • Flumusa is an anxiolytic drug (tranquilizer), a derivative of triazolo-benzodiazepine. (medicatione.com)
  • Carisoprodol is used together with rest and physical therapy to treat skeletal muscle conditions such as pain or injury. (rxmedworld.co)
  • Carisoprodol should only be used for short periods (up to two or three weeks) because there is no evidence of its effectiveness in long term use and most skeletal muscle injuries are generally of short duration. (rxmedworld.co)
  • Carisoprodol is used as a skeletal muscle relaxant. (rxmedworld.co)
  • Rather than acting directly on skeletal muscle, carisoprodol interrupts neuronal communication within the reticular formation and spinal cord, resulting in sedation and alteration in pain perception. (rxmedworld.co)
  • Morphine may enhance the neuromuscular blocking action of skeletal muscle relaxants and produce an increased degree of respiratory depression. (medlibrary.org)
  • This effect affects skeletal muscle functions and decreases muscle tone to promote the relaxation of large and small muscles. (medszee.com)
  • When taken in large doses, a Buspar high is characterized by symptoms like sedation, dizziness, sleepiness, and extreme calm. (cemona.es)
  • The concomitant use of cimetidine can potentiate morphine effects and increase risk of hypotension, respiratory depression, profound sedation, coma, and death. (medlibrary.org)
  • The concomitant use of PGP-inhibitors can increase the exposure to morphine by about two-fold and can increase risk of hypotension, respiratory depression, profound sedation, coma, and death. (medlibrary.org)
  • An uncontrolled trial on patients treated in a clinical gynecology practice published in 1959 found that oxanamide was efficacious in the treatment of anxiety resulting from premenstrual syndrome, menopause, and various other causes, with minimal sedation or other side effects. (wikipedia.org)
  • Xanax is an FDA-approved anxiolytic used to treat conditions such as anxiety, muscle spasms, seizures, and epilepsy. (medszee.com)
  • This leads to a decrease in anxiety, muscle tension, and seizures. (naturalmedicineseries.com)
  • Buspar is a discontinued branded version of buspirone, an anxiolytic medication that treats anxiety disorders. (cemona.es)
  • For decades, the gold standard for treating depression and anxiety has been antidepressants and anxiolytic medications. (goodnesslover.com)
  • Essential oils and the constituents in them exhibit different pharmacological activities, such as antinociceptive, anxiolytic-like, and anticonvulsant effects. (mdpi.com)
  • It is also used to relieve muscle spasms and to provide sedation before medical procedures. (virtualpsychcentre.com)
  • Buspirone anxiolytic can't provide sedation and relaxation so it is not a benzo. (arlen.com.br)
  • Acute higher doses of the methadone drug induce analgesia, sedation, respiratory depression and coma. (rapidtest.com)
  • Effects on the Central Nervous System The principal actions of therapeutic value of morphine are analgesia and sedation. (clustermed.info)
  • α2-agonists are used primarily for sedation, analgesia, and management of delirium. (bvsalud.org)
  • Monitor patients for signs of respiratory depression that may be greater than otherwise expected and decrease the dosage of morphine sulfate extended-release tablets and/or the muscle relaxant as necessary. (medlibrary.org)
  • Effects on the Gastrointestinal Tract and Other Smooth Muscle Gastric, biliary and pancreatic secretions are decreased by morphine. (clustermed.info)
  • Hostile monkeys were made tame by oral drug doses which did not cause sedation. (minclinic.ru)
  • The chart is based an anxiolytic equivalencies, all doses listed are compared against Valium (Diazepam) 10mgs as a control. (seacolors.eu)
  • Activated postsynaptic 5-HT1A receptors promote hyperpolarization to released 5-HT on pyramidal neurons.8, The anxiolytic action of buspirone is mainly thought to arise from the interaction at presynaptic 5-HT1A autoreceptors. (arlen.com.br)
  • Buspirone belongs to a class of drugs called anxiolytics. (arlen.com.br)
  • Most of these effects are thought to result from a facilitation of the action of gamma aminobutyric acid (GABA), an inhibitory neurotransmitter in the central nervous system . (virtualpsychcentre.com)
  • GABA can block specific signals in your central nervous system and thus produce a calming effect. (tripsitter.com)
  • Once absorbed, Xanax enhances the effects of GABA, modifying nerve communication in the central nervous system (CNS). (medszee.com)
  • Estazolam binds to the gamma-aminobutyric acid (GABA) receptor at a site distinct from the inhibitory neurotransmitter GABA binding site in the limbic system of the central nervous system (CNS). (dvago.pk)
  • They work by enhancing the effects of a neurotransmitter called gamma-aminobutyric acid (GABA) in the brain, which helps to calm the central nervous system. (naturalmedicineseries.com)
  • Ambien slows down the brain and central nervous system by stimulating the neurotransmitter GABA (CNS). (practicalanxietysolutions.com)
  • Opiate Opioid analgesics are comprised of a large group of substances that control pain by depressing the central nervous system. (rapidtest.com)
  • These active ingredients contribute to chamomile's anti-inflammatory, antispasmodic, and smooth muscle-relaxing effects, particularly in the gastrointestinal tract. (beauty104.com.tw)
  • Etіzоlаm іѕ a CNS depressant wіth anxiolytic, anticonvulsant, ѕеdаtіvе-hурnоtіс and muscle rеlаxаnt effects. (globalcocaineshop.se)
  • Tofisopam also has some affinity for other receptors such as serotonin receptors and dopamine receptors, which may contribute to its anxiolytic effects. (modapharma.org)
  • Antidepressants, antiseizure drugs, and other central nervous system (CNS)-active drugs may also be used for chronic or neuropathic pain and are first-line therapy for some conditions. (msdmanuals.com)
  • After stopping use of a CYP2D6 inhibitor, consider reducing the dosage of acetaminophen and codeine phosphate tablets and monitor the patient for signs and symptoms of respiratory depression or sedation. (medlibrary.org)
  • Symptoms of respiratory issues and sedation may be seen in newborns whose mothers used Zolpidem during the third trimester of pregnancy. (practicalanxietysolutions.com)
  • The Methadone drug acts on the central nervous and cardiovascular systems to produce respiratory and circulatory depression. (rapidtest.com)
  • 5.13)Risks of Use in Patients with Increased Intracranial Pressure, Brain Tumors, Head Injury, or Impaired Consciousness: Monitor for sedation and respiratory depression. (drugcentral.org)
  • Signs of overdose include respiratory depression, muscle weakness, somnolence (general depressed activity). (minclinic.ru)
  • This effect is a precursor to sedation as it slows down CNS and brain activity by affecting specific receptors. (medszee.com)
  • The term " muscle relaxant" is used to refer to two major 1 They work by depressing the central nervous system to relax and calm the entire body, not just the muscles. (seacolors.eu)
  • The drug dosage which effectively blocked the vicious reaction was well below the dose which caused sedation in these animals. (minclinic.ru)
  • The Methadone drug also produces miosis and increases the tone of smooth muscle in the lower gastrointestinal tract while decreasing the amplitude of contractions. (rapidtest.com)
  • It is used as an adjunct in the symptomatic treatment of musculoskeletal conditions associated with painful muscle spasm. (rxmedworld.co)
  • It is also used as a premedication for inducing sedation, anxiolysis, or amnesia before certain medical procedures (e.g., endoscopy). (worldsbest.rehab)
  • It can be taken orally (by mouth), as a suppository inserted into the rectum, intramuscularly (injected into muscle), intravenously (injection into a vein) or used as a nasal spray. (worldsbest.rehab)