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*  Bradykinin receptor B1
BDKRB1 bradykinin receptor B1". Seabrook GR, Bowery BJ, Hill RG. "Bradykinin receptors in mouse and rat isolated superior ... The B1 receptor is one of two of G protein-coupled receptors that have been found which bind bradykinin and mediate responses ... Bradykinin receptor B1 (B1) is a G-protein coupled receptor encoded by the BDKRB1 gene in humans. Its principal ligand is ... "Bradykinin Receptors: B1". IUPHAR Database of Receptors and Ion Channels. International Union of Basic and Clinical ...
*  Bradykinin receptor B2
... is a G-protein coupled receptor for bradykinin, encoded by the BDKRB2 gene in humans. The B2 receptor is ... "Entrez Gene: BDKRB2 bradykinin receptor B2". "Bradykinin Receptors: B2". IUPHAR Database of Receptors and Ion Channels. ... also potentiates bradykinin action on B2 receptors. Kallidin also signals through the B2 receptor. An antagonist for the ... "Two B1 and B2 bradykinin receptor antagonists fail to inhibit the Ca2+ response elicited by bradykinin in human skin ...
*  Bradykinin receptor
There are two Bradykinin receptors: the B1 receptor and the B2 receptor. Bradykinin receptor B1 (B1) is a G-protein coupled ... The bradykinin receptor family is a group of G-protein coupled receptors whose principal ligand is the protein bradykinin. ... The B1 receptor is one of two G protein-coupled receptors that have been found which bind bradykinin and mediate responses to ... "Bradykinin Receptors". IUPHAR Database of Receptors and Ion Channels. International Union of Basic and Clinical Pharmacology. ...
*  Dynorphin
The group found that it acts on the bradykinin receptor as well as KOR. The N-terminal tyrosine of dynorphin A is necessary to ... type glutamate receptor. Different dynorphins show different receptor selectivities and potencies at receptors. Big dynorphin ... Blocking bradykinin receptors in the lumbar region of the spinal cord reversed persistent pain. A multiple pathway system might ... Lai J, Luo MC, Chen Q, Ma S, Gardell LR, Ossipov MH, Porreca F (December 2006). "Dynorphin A activates bradykinin receptors to ...
*  Hereditary angioedema
Icatibant inhibits the bradykinin B2 receptor, and was approved in Europe and the USA. In hereditary angioedema, specific ... Icatibant (marketed as Firazyr) is a selective bradykinin receptor antagonist, which has been approved in Europe and was ... bradykinin receptor antagonist (Icatibant, Firazyr®, Jerini/Shire) in Europe; kallikrein inhibitor(Ecallantide, Kalbitor®, Dyax ... This results in increased amounts of bradykinin which promotes swelling. The condition may be inherited from a person's parents ...
*  Calreticulin
Abd Alla J, Reeck K, Langer A, Streichert T, Quitterer U (Sep 2009). "Calreticulin enhances B2 bradykinin receptor maturation ... binding of androgen receptor to its hormone-responsive DNA element and can inhibit androgen receptor and retinoic acid receptor ... The amino terminus of calreticulin interacts with the DNA-binding domain of the glucocorticoid receptor and prevents the ... Thus, calreticulin can act as an important modulator of the regulation of gene transcription by nuclear hormone receptors. ...
*  Relaxin/insulin-like family peptide receptor 4
"Identification and characterisation of GPR100 as a novel human G-protein-coupled bradykinin receptor". British Journal of ... RXFP4 relaxin/insulin-like family peptide receptor 4". "Relaxin Family Peptide Receptors: RXFP4". IUPHAR Database of Receptors ... Relaxin/insulin-like family peptide receptor 4, also known as RXFP4, is a human G-protein coupled receptor. GPR100 is a member ... Takeda S, Kadowaki S, Haga T, Takaesu H, Mitaku S (June 2002). "Identification of G protein-coupled receptor genes from the ...
*  THOP1
"EP24.15 interacts with the angiotensin II type I receptor and bradykinin B2 receptor". Cell Biochem. Funct. 23 (3): 195-204. ...
*  G protein-coupled receptor
In kidney cells, the bradykinin receptor B2 has been shown to interact directly with a protein tyrosine phosphatase. The ... transmembrane domain receptors, 7TM receptors, heptahelical receptors, serpentine receptor, and G protein-linked receptors ( ... G protein-coupled receptors database List of MeSH codes (D12.776) Metabotropic receptor Orphan receptor Pepducins, a class of ... is a receptor that can bind with stimulative signal molecules, while inhibitory hormone receptor (Ri) is a receptor that can ...
*  Serafim Guimarães
"Crosstalk between presynaptic angiotensin receptors, bradykinin receptors and α2-autoreceptors in sympathetic neurons: a study ... Veins and their receptors remained favourites. Guimarães has summarized the knowledge on blood vessels, their nerves and their ... Th influence of drugs is determined not only by their pharmacodynamics, especially the existence of receptors, but also their ... ISBN 978-3-437-16888-8 S. Guimarães, M. Q. Paiva, D. Moura (1998). "Different receptors for angiotensin II at pre- and ...
*  Apelin
... and bradykinin B2 receptors". J. Biol. Chem. 279 (9): 7901-8. doi:10.1074/jbc.M306377200. PMID 14645236. O'Dowd BF, Heiber M, ... a seven-transmembrane receptor related to angiotensin-type 1 receptor in blood pressure in vivo". J. Biol. Chem. 279 (25): ... The apelin receptor is expressed early during the embryonic development of the heart, where it regulates the migration of cell ... Apelin receptor is also expressed in the neurons of brain areas involved in regulating water and food intake. Apelin injection ...
*  Rubottom oxidation
Isaka, N.; Tamiya, M.; Hasegawa, A.; Ishiguro, M. (2011). "A Concise Total Synthesis of the Non-Peptide Bradykinin B1 Receptor ... that exhibits anti-inflammatory as well as analgesic properties due to its antagonistic action with the bradykinin receptor. ...
*  Apelin receptor
2004). "Agonist-independent nuclear localization of the Apelin, angiotensin AT1, and bradykinin B2 receptors". J. Biol. Chem. ... The apelin receptor (also known as the APJ receptor) is a G protein-coupled receptor which binds apelin and Apela/ELABELA/ ... "Apelin Receptor: APJ". IUPHAR Database of Receptors and Ion Channels. International Union of Basic and Clinical Pharmacology. ... 2004). "Regulatory roles for APJ, a seven-transmembrane receptor related to angiotensin-type 1 receptor in blood pressure in ...
*  Neurturin
... has been shown to upregulate B1 (bradykinin) receptors in neurons of mice, indicating a possible influence on pain ... Vellani V, Zachrisson O, McNaughton PA (Oct 2004). "Functional bradykinin B1 receptors are expressed in nociceptive neurones ... Neurturin signaling is mediated by the activation of a multi-component receptor system including the Ret tyrosine kinase (RET ... Neurturin preferentially binds to the GFRα2 co-receptor. Upon assembly of the complex, specific tyrosine residues are ...
*  GRK4
2001). "Determination of bradykinin B2 receptor in vivo phosphorylation sites and their role in receptor function". J. Biol. ... 2003). "Desensitization of human renal D1 dopamine receptors by G protein-coupled receptor kinase 4". Kidney Int. 62 (3): 790-8 ... 2006). "The D1 dopamine receptor is constitutively phosphorylated by G protein-coupled receptor kinase 4". Mol. Pharmacol. 69 ( ... G protein-coupled receptor kinase 4 is an enzyme that in humans is encoded by the GRK4 gene. This gene encodes a member of the ...
*  Icatibant
... acts as a bradykinin inhibitor by blocking the binding of native bradykinin to the bradykinin B2 receptor. Icatibant ... which is a selective and specific antagonist of bradykinin B2 receptors. Bradykinin is a peptide-based hormone that is formed ... Bradykinin plays an important role as the mediator of pain. Surplus bradykinin is responsible for the typical symptoms of ... These symptoms are mediated by activation of bradykinin B2 receptors. ...
*  Julian Downward
... "p21ras-induced responsiveness of phosphatidylinositol turnover to bradykinin is a receptor number effect". Proceedings of the ... Downward, David Julian Harry (1986). The structure and function of the receptor for epidermal growth factor (PhD thesis). ... he went on to characterise growth factor receptor complexes mediating Ras nucleotide exchange, and to demonstrate that GTP- ... supervised by Michael Waterfield at the Imperial Cancer Research Fiund where he investigated Epidermal growth factor receptor, ...
*  Menarini
"Antagonism of bradykinin B2 receptor prevents inflammatory responses in human endothelial cells by quenching the NF-kB pathway ...
*  B2
... a subgroup of the Anatomical Therapeutic Chemical Classification System Bradykinin receptor B2, a human gene Proanthocyanidin ...
*  B1
... , B.I, B.1 or B-1 may refer to: Bradykinin receptor B1, a human gene Cinnamtannin B1, a condensed tannin found in cinnamon ...
*  Kallidin
... to bradykinin with an additional lysine residue added at the N-terminal end and signals through the bradykinin receptor. Stefan ... It can be converted to bradykinin by the aminopeptidase enzyme. It can be a substrate for carboxypeptidase M and N. Kallidin is ...
*  Epoxyeicosatrienoic acid
... bradykinin or acetylcholine acting through their respective Bradykinin receptor B2 and muscarinic acetylcholine receptor M1 or ... some studies implicate EET binding to an unidentified Cell surface receptor and/or Gs protein-linked G protein-coupled receptor ... "CYP3A4 mediates growth of estrogen receptor-positive breast cancer cells in part by inducing nuclear translocation of phospho- ... express hyperactive sEH and show reduced vasodilation responses to bradykinin. Other studies find that women with pregnancy- ...
*  Index of biochemistry articles
... bombesin receptor - Bone morphogenetic protein - bradykinin - bradykinin receptor - BRCA1 - buffer solution - C-terminus - C4 ... interleukin receptor - interleukin-1 receptor - interleukin-2 receptor - interleukin-3 - interleukin-3 receptor - intermediate ... G protein-coupled receptor - G3P - GABA - GABA receptor - GABA-A receptor - gag-onc fusion protein - galanin - gamete - gamma- ... IgE receptor - IGF type 1 receptor - IGF type 2 receptor - IgG - IgM - immediate-early protein - immune cell - immune system - ...
*  Rhodopsin-like receptors
IPR003904 Bradykinin receptor InterPro: IPR000496 Bradykinin receptor B1 (BDKRB1, BRB1) Bradykinin receptor B2 (BDKRB2, BRB2) ... chemokine receptor (DARC, DUFF) G Protein-coupled Receptor 30 (GPER, CML2, GPCR estrogen receptor) Angiotensin II receptor ... kappa Opioid receptor (OPRK1, OPRK) mu Opioid receptor (OPRM1, OPRM) Nociceptin receptor (OPRL1, OPRX) Somatostatin receptor ... Motilin receptor (MLNR, GPR38) Anaphylatoxin receptors InterPro: IPR002234 C3a receptor (C3AR1, C3AR) C5a receptor (C5AR1, C5AR ...
*  C1-inhibitor
... a plasma kallikrein inhibitor and the bradykinin receptor antagonist icatibant. The activation of the complement cascade can ... which leads to the production of the vasoactive peptide bradykinin. Also, C4 and C2 cleavage goes unchecked, resulting in auto- ...
*  Oh Uhtaek
2002). "Bradykinin-12-lipoxygenase-VR1 signaling pathway for inflammatory hyperalgesia". Proc. Natl. Acad. Sci. USA. 99 (15): ... 2008). "TMEM16A Confers Receptor Activated Calcium-dependent Chloride Conductance". Nature. 455 (7217): 1210-5. Bibcode: ... J Neurosci (2002) 2000 : Hwang SW et al., Direct activation of capsaicin receptors by products of lipoxygenases: Endogenous ... Nature (2008) 2002 : Shin J et al., Bradykinin-12-lipoxygenase-VR1 signaling pathway for inflammatory hyperalgesia. Proc Natl ...