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*  Beta-adrenergic-receptor kinase
... beta-adrenergic-receptor] kinase, beta-adrenergic receptor-specific kinase, beta-AR kinase, beta-ARK, beta-ARK 1, beta-ARK 2, ... beta-adrenergic receptor] Thus, the two substrates of this enzyme are ATP and beta-adrenergic receptor, whereas its two ... beta-adrenergic receptor] phosphotransferase. Other names in common use include ATP:beta-adrenergic-receptor phosphotransferase ... beta-receptor kinase, GRK2, GRK3, beta-adrenergic-receptor kinase (phosphorylating), beta2ARK, betaARK1, beta-adrenoceptor ...
*  Beta adrenergic receptor kinase
"Overexpression of beta-arrestin and beta-adrenergic receptor kinase augment desensitization of beta 2-adrenergic receptors". J ... "Desensitization of the isolated beta 2-adrenergic receptor by beta-adrenergic receptor kinase, cAMP-dependent protein kinase, ... Beta adrenergic receptor kinase has been shown to interact with: Beta-gamma complex, G protein GIT1, GNAQ, PDE6G, PRKCB1 and ... Beta adrenergic receptor kinase (also referred to as βARK or BARK) is a serine/threonine intracellular kinase. It is activated ...
*  Beta adrenergic receptor kinase-2
Overall, the beta adrenergic receptor kinase 2 has 85% amino acid similarity with beta adrenergic receptor kinase 1, with the ... Beta-adrenergic receptor kinase 2 (beta-ARK-2) also known as G-protein-coupled receptor kinase 3 (GRK3) is an enzyme that in ... The beta-adrenergic receptor kinase specifically phosphorylates the agonist-occupied form of the beta-adrenergic and related G ... 1991). "Cloning, expression, and chromosomal localization of beta-adrenergic receptor kinase 2. A new member of the receptor ...
*  Beta adrenergic receptor kinase carboxyl-terminus
... (also βARKct) is a peptide composed of the last 194 amino acid residues of ... the carboxyl-terminus of beta adrenergic receptor kinase 1 (βARK1). It binds the βγ subunits of G proteins located in the ... White DC, Hata JA, Shah AS, Glower DD, Lefkowitz RJ, Koch WJ (May 2000). "Preservation of myocardial β-adrenergic receptor ... The sympathetic nervous system increases norepinephrine release to stimulate β-adrenergic receptors (βARs) located on heart ...
*  Beta-3 adrenergic receptor
Other adrenergic receptors Alpha-1 adrenergic receptor Alpha-2 adrenergic receptor Beta-1 adrenergic receptor Beta-2 adrenergic ... The beta-3 adrenergic receptor (β3 adrenoreceptor), also known as ADRB3, is a beta-adrenergic receptor, and also denotes the ... "Molecular characterization of the mouse beta 3-adrenergic receptor: relationship with the atypical receptor of adipocytes". ... Beta adrenergic receptors are involved in the epinephrine- and norepinephrine-induced activation of adenylate cyclase through ...
*  Beta-1 adrenergic receptor
Other adrenergic receptors Alpha-1 adrenergic receptor Alpha-2 adrenergic receptor Beta-2 adrenergic receptor Beta-3 adrenergic ... The beta-1 adrenergic receptor (β1 adrenoreceptor), also known as ADRB1, is a beta-adrenergic receptor, and also denotes the ... "The cardiac beta-adrenergic receptor. Structural similarities of beta 1 and beta 2 receptor subtypes demonstrated by ... "beta 1-adrenergic receptor association with PSD-95. Inhibition of receptor internalization and facilitation of beta 1- ...
*  Beta-2 adrenergic receptor
Other adrenergic receptors Alpha-1 adrenergic receptor Alpha-2 adrenergic receptor Beta-1 adrenergic receptor Beta-3 adrenergic ... The beta-2 adrenergic receptor (β2 adrenoreceptor), also known as ADRB2, is a cell membrane-spanning beta-adrenergic receptor ... "Insulin stimulates sequestration of beta-adrenergic receptors and enhanced association of beta-adrenergic receptors with Grb2 ... Frielle T, Caron MG, Lefkowitz RJ (May 1989). "Properties of the beta 1- and beta 2-adrenergic receptor subtypes revealed by ...
*  Ersentilide
... is a beta adrenergic receptor antagonist. Lombardi, F; Terranova, P (2006). "Pharmacological treatment of atrial ...
*  Sulfinalol
... is a beta adrenergic receptor antagonist. The methyl group on a sulfoxide is sufficiently acidic to substitute for ... "Studies on the mechanism of the acute antihypertensive and vasodilator actions of several beta-adrenoceptor antagonists". J. ...
*  GPCR oligomer
Limbird LE, Meyts PD, Lefkowitz RJ (June 1975). "Beta-adrenergic receptors: evidence for negative cooperativity". Biochem. ... and hetero-oligomerization of β2-adrenergic receptor in receptor trafficking, signaling pathways and receptor pharmacology". ... "The size of the mammalian lung beta 2-adrenergic receptor as determined by target size analysis and immunoaffinity ... Receptor homodimers - which consist of two identical GPCRs - are the simplest homomeric GPCR oligomers. Receptor heterodimers ...
*  Toliprolol
... is a beta adrenergic receptor antagonist. Stephenson, KA; Wilson, AA; Meyer, JH; Houle, S; Vasdev, N (2008). "Facile ... radiosynthesis of fluorine-18 labeled beta-blockers. Synthesis, radiolabeling, and ex vivo biodistribution of 18F-(2S and 2R)-1 ...
*  Iodopindolol
A new beta adrenergic receptor probe". Journal of cyclic nucleotide research. 7 (1): 13-26. PMID 6265511. ... Iodopindolol is a beta-adrenergic selective antagonist tagged by radioisotopic iodine. Pindolol Ezrailson, E. G.; Garber, A. J ...
*  Primidolol
... is a beta adrenergic receptor antagonist. J. Augstein, D. A. Cox and A. L. Ham., DE 2238504 (1973). Chem. Abstr. jte ...
*  Adenylyl cyclase
Beta adrenergic receptor kinase pathway G Proteins. PDB-101. Reece J, Campbell N (2002). Biology. San Francisco: Benjamin ... Sodeman W, Sodeman T (2005). "Physiologic- and Adenylate Cyclase-Coupled Beta-Adrenergic Receptors". Sodeman's Pathologic ... Neve, Kim A.; Seamans, Jeremy K.; Trantham-Davidson, Heather (August 2004). "Dopamine receptor signaling". Journal of Receptor ... Isoforms II, IV and IX are stimulated by beta gamma subunits of the G protein. Isoforms I, V and VI are most clearly inhibited ...
*  Midodrine
Desglymidodrine does not stimulate cardiac beta-adrenergic receptors. Desglymidodrine diffuses poorly across the blood-brain ... which is an α1-receptor agonist and exerts its actions via activation of the alpha-adrenergic receptors of the arteriolar and ...
*  History of hypertension
Black JW, Crowther AF, Shanks RG, Smith LH, Dornhorst AC (May 1964). "A new adrenergic beta receptor antagonist". Lancet. 1 ( ... The first member was verapamil, a derivative of papaverine that was initially thought to be a beta blocker and used for angina ... More recently angiotensin receptor blockers and renin inhibitors have also been introduced as antihypertensive agents. Esunge ... The British physician James W. Black developed beta blockers in the early 1960s; these were initially used for angina, but ...
*  Falintolol
... is a beta-adrenergic receptor antagonist. Conti, P; Dallanoce, C; De Amici, M; De Micheli, C; Klotz, KN (1998). " ... "Synthesis of new delta 2-isoxazoline derivatives and their pharmacological characterization as beta-adrenergic receptor ...
*  Pacrinolol
... is a beta adrenergic receptor antagonist. Stache, U; Fritsch, W; Fehlhaber, HW (1987). "Synthesis of the highly ... cardioselective beta-sympatholytic pacrinolol". Arzneimittel-Forschung. 37 (11): 1217-21. PMID 2894210. ...
*  Anxiolytic
Jefferson, James W. (1974). "Beta-Adrenergic Receptor Blocking Drugs in Psychiatry". Archives of General Psychiatry. 31 (5): ... Beta-receptor blockers such as propranolol and oxprenolol, although not anxiolytics, can be used to combat the somatic symptoms ... Noyes, Russell (1982). "Beta-blocking drugs and anxiety". Psychosomatics. 23 (2): 155-70. doi:10.1016/s0033-3182(82)73433-4. ... Its mechanism of action remains poorly defined, with GABAergic, NGF and BDNF release promoting, MT1 receptor agonism, MT3 ...
*  Tolamolol
... is a beta adrenergic receptor antagonist. Curtis-Prior, PB; Gadd, AL (1990). "Beta-adrenoceptor antagonists and human ...
*  Pafenolol
... is a beta adrenergic receptor antagonist. Lennernäs, H; Regårdh, CG (1993). "Dose-dependent intestinal absorption and ... significant intestinal excretion (exsorption) of the beta-blocker pafenolol in the rat". Pharmaceutical Research. 10 (5): 727- ...
*  Tienoxolol
... is a beta adrenergic receptor antagonist. Mahé, N; Do, B; Nicolaï, B; Rietveld, IB; Barrio, M; Tamarit, JL; Céolin, ...
*  Procinolol
... is a beta adrenergic receptor antagonist. Singh, KP (1983). "Influence of beta-adrenoceptor antagonists on ...
*  Tiprenolol
... is a beta adrenergic receptor antagonist. Allen, JD; Shanks, RG (1974). "Effects of tiprenolol, practolol and ...
*  Spirendolol
... is a beta adrenergic receptor antagonist. Mostaghim, R; Maddox, YT; Ramwell, PW (1986). "Endothelial potentiation ... of relaxation response to beta adrenoceptor blocking agents". The Journal of Pharmacology and Experimental Therapeutics. 239 (3 ...
*  Meldonium
... has also been found to induce anticonvulsant and antihypnotic effects involving alpha 2-adrenergic receptors as well ... Studies have shown that meldonium increases cognition and mental performance by reducing amyloid beta deposition in the ... oxide production via stimulation of the M3 muscarinic acetylcholine receptor or specific gamma-butyrobetaine ester receptors. ... known as beta oxidation). Carnitine is mainly absorbed from the diet, but can be formed through biosynthesis. To produce ...