... (furethylnorlevorphanol) is an opioid analgesic drug from the morphinan series that was discovered by the ... Synthetic analgesics - Aralkyl substitution on nitrogen of morphinan. UNODC Bulletin on Narcotics 1958 p 23-42. Hellerbach J, ... morphinans", published 1961-01-31 Nathan B. Eddy, Hedwig Besendorf and Béla Pellmont. ... Schnider O, Besendorf H, Pellmont B (1966). "Morphinans". Synthetic Analgesics. Part IIA. Pergamon Press. Bulletin on Narcotics ...
Morphinans. International series of monographs on organic chemistry. Pergamon Press. v t e. ... "Process for making morphinan derivatives and products available thereby", published 1956-03-22, issued 1959-05-05 US patent ... 2970147, Andre Grussner, Joseph Hellerbach, Otto Schnider, "3-hydroxy-N-(heterocyclic-ethyl)-morphinans", published 1958-11-26 ...
... morphinan series. 5. Synthesis and biological properties of (+)-naloxone". Journal of Medicinal Chemistry. 21 (4): 398-400. doi ...
Benzazocine Azocine Morphinan Kar, Ashutosh (2005). Medicinal Chemistry - Google Books. ISBN 9788122415650. Cittern PA, Kapoor ...
Benzomorphan Azocine Morphinan Ginsburg, David (1950). "The synthesis of morphan (2-azabicyclo[3.3.1]nonane)". Journal of ...
... is a plant-isolate morphinan. A plant-derived morphinan as a novel lead compound active against malaria liver stages ...
Morphinans Butorphanol. Comes in tartrate salt form; sparingly soluble in water, insoluble in most organic solvents; degrades ...
Synthesis of morphine-like alkaloids in chemistry describes the total synthesis of the natural morphinan class of alkaloids ... Hong CY, Kado N, Overman LE (November 1993). "Asymmetric synthesis of either enantiomer of opium alkaloids and morphinans. ...
Elements of the morphine structure have been used to create completely synthetic drugs such as the morphinan family ( ... Hong CY, Kado N, Overman LE (November 1993). "Asymmetric synthesis of either enantiomer of opium alkaloids and morphinans. ... although some more distant relatives like the morphinan series (levorphanol, dextorphan and the racemic parent chemical ...
"Enhanced morphinan alkaloid production in hairy root cultures of Papaver bracteatum by over-expression of salutaridinol 7-o- ... "Synthesis of morphinan alkaloids in Saccharomyces cerevisiae." PLoS ONE 10.4 (2015): e0124459. Galanie, Stephanie, et al. " ...
Dextrorphan Dextromethorphan Levomethorphan Morphinan Hou, Chia-Hui; Tzeng, Jann-Inn; Chen, Yu-Wen; Lin, Ching-Nan; Lin, Mao- ...
... reticulin morphine can be formed through the morphinan route, noscapine through the path of the noscapina or berberina. The ... "The opium poppy genome and morphinan production" (PDF). Science. 362 (6412): 343-347. Bibcode:2018Sci...362..343G. doi:10.1126/ ...
pp 27-41 in Martin and Isbell(1978). Fraser HF, Isbell H (1950). "Addiction liabilities of morphinan, 6-methyldihydromorphine ...
Benzylisoquinoline alkaloids include aporphines and oxoaporphines, as well as derivatives of morphinans. Essential oils include ...
... (DXA) is an opioid derivative chemical of the morphinan class that is used in scientific research. It acts as a ... Morphinan Oxilorphan Dextrorphan Dextromethorphan Levallorphan Su TP (November 1982). "Evidence for sigma opioid receptor: ... peripheral and anticholinesterase effects of some morphinan derivatives" (pdf). The Journal of Pharmacology and Experimental ...
Levallorphan Methorphan Morphinan Cyclorphan "Conversion Factors for Controlled Substances". www.deadiversion.usdoj.gov. v t e ...
"Effects of dextrorotatory morphinans on α3β4 nicotinic acetylcholine receptors expressed in Xenopus oocytes". European Journal ...
... is an opioid antagonist from the morphinan family of drugs. Cyprodime is a selective opioid antagonist which blocks ...
... is structurally related to the morphinan class of opioid analgesics. The enantioselective total synthesis of (-)- ...
... is a morphinan derivative that acts as an opioid agonist. It has potent analgesic effects and is around 10x ...
... is an opioid analgesic of the morphinan family that was never marketed. It is the levo-isomer of 3- ... hydroxymorphinan (morphinan-3-ol). Norlevorphanol is a Schedule I Narcotic controlled substance in the United States with an ...
"Crystal structure of the μ-opioid receptor bound to a morphinan antagonist". Nature. 485 (7398): 321-326. Bibcode:2012Natur.485 ...
March 2012). "Crystal structure of the µ-opioid receptor bound to a morphinan antagonist". Nature. 485 (7398): 321-6. Bibcode: ...
On the other hand, agonist activity is also shown in ligands with larger groups at the morphinan nitrogen, and therefore this ... One theory states that the morphinans biological activity could be determined by the size of the N-substituents. For example, ... antagonists usually have larger substituents, such as allyl- or cyclopropyl methyl at the morphinan nitrogen, while agonists ... "Crystal structure of the µ-opioid receptor bound to a morphinan antagonist". Nature. 485 (7398): 321-326. Bibcode:2012Natur.485 ...
It is not a morphinan derivative (in contrast to codeine and dextromethorphan). Zipeprol acts as a local anaesthetic and has ...
... (Oxymethebanol) is a morphinan derivative that acts as an opioid agonist. It was invented by Sankyo Company in Japan ...
2012). "Crystal structure of the µ-opioid receptor bound to a morphinan antagonist". Nature. 485 (7398): 321-326. Bibcode: ...
... is an opioid analgesic of the morphinan family that was never marketed. It acts as a μ-opioid receptor (MOR) weak ...
Chemically, levorphanol belongs to the morphinan class and is (−)-3-hydroxy-N-methyl-morphinan. It is the "left-handed" ( ...
... is a morphinan-type synthetic agonist-antagonist opioid analgesic developed by Bristol-Myers. Butorphanol is most ...