Labetalol
... is typically given as a racemic mixture to achieve both α- and β-adrenergic receptor blocking activity. Labetalol ... "Labetalol". Drug Information Portal. U.S. National Library of Medicine. "Labetalol hydrochloride". Drug Information Portal. U.S ... Geriatric: the elderly are more likely to experience dizziness when taking labetalol. Labetalol should be dosed with caution in ... The peripheral vascular resistance decreases when labetalol is first administered. Continuous labetalol use further decreases ...
Beta blocker
"Labetalol Hydrochloride Monograph for Professionals". Drugs.com. American Society of Health-System Pharmacists. Retrieved March ... Some beta blockers (e.g., labetalol and carvedilol) exhibit mixed antagonism of both β- and α1-adrenergic receptors, which ... The mixed alpha- and beta blocker labetalol is especially useful for treatment of concomitant tachycardia and hypertension ... Butaxamine ICI-118,551 SR 59230A Nebivolol Agents with intrinsic sympathomimetic action (ISA) Acebutolol, pindolol, labetalol, ...
Alpha blocker
... such as Labetalol or carvedilol. In low doses, labetalol and carvedilol can decrease the peripheral resistance and block the ... Blockers that have both the ability to block both α and β receptors, such as carvedilol, bucindolol, and labetalol, have the ... Brogden, R. N.; Heel, R. C.; Speight, T. M.; Avery, G. S. (1978-04-01). "Labetalol: A Review of its Pharmacology and ... Finally, in drugs with both alpha and beta blocking properties, such as carvedilol and labetalol, interactions with other alpha ...
Cocaine intoxication
Furthermore, the use of labetalol is approved by a AHA/ACC guideline for people who have used cocaine and methamphetamine with ... Richards, John R.; Lange, Richard A. (2016-02-01). "Labetalol and cardiovascular consequences of cocaine use". Trends in ... "Influence of labetalol on cocaine-induced coronary vasoconstriction in humans". The American Journal of Medicine. 94 (6): 608- ... the intravenous racemic mixture of labetalol, a non-selective β blocker and selective α1 blocker is recommended for treating ...
Medroxalol
Labetalol Dage RC, Cheng HC, Woodward JK (1981). "Cardiovascular properties of medroxalol, a new antihypertensive drug". ...
Subarachnoid hemorrhage
Medications such as labetalol may be required to lower the blood pressure until repair can occur. Efforts to treat fevers are ... Medications to achieve this may include labetalol or nicardipine. People whose CT scan shows a large hematoma, depressed level ...
Pheochromocytoma
... labetalol, carvedilol) combined alpha-beta-adrenoceptor antagonists. These agents should be avoided whenever possible as there ...
Me-too drug
It was followed by propranolol, sotalol, practolol, metoprolol, labetalol, acebutolol and bisoprolol. Successive differences ...
Anterior cerebral artery syndrome
Hypotensive agents that can be options include labetalol, nicardipine, clevidipine, hydralazine, enalaprilat.[21] For the ...
Pre-eclampsia
Labetalol, hydralazine and nifedipine are commonly used antihypertensive agents for hypertension in pregnancy. ACE inhibitors ... Blood pressure medication, such as labetalol and methyldopa, may be used to improve the mother's condition before delivery. ...
Intravenous therapy
Peacock WF, Hilleman DE, Levy PD, Rhoney DH, Varon J (July 2012). "A systematic review of nicardipine vs labetalol for the ...
Hypertensive urgency
Recommended medications for hypertensive urgencies include: captopril, labetalol, amlodipine, felodipine, isradipine, and ...
Gestational hypertension
Methyldopa, hydralazine, nifedipine, and labetalol are most commonly used for severe pregnancy hypertension. The fetus is at ...
Hypertensive emergency
Labetalol is a beta-blocker with mild alpha antagonism, decreasing the ability of catecholamine activity to increase systemic ... Medications include labetalol, nicardipine, hydralazine, sodium nitroprusside, esmolol, nifedipine, minoxidil, isradipine, ...
Hypertensive encephalopathy
Labetalol - an alpha- and beta-adrenergic blocker, given as an intravenous bolus or infusion. Bolus followed by infusion. ... This may be done with labetalol or sodium nitroprusside given by injection into a vein. In those who are pregnant, magnesium ...
Salicylamide
Derivatives of salicylamide include ethenzamide, labetalol, medroxalol, lopirin, otilonium, oxyclozanide, salicylanilide, ...
Alpha-1 adrenergic receptor
Fahed S, Grum DF, Papadimos TJ (May 2008). "Labetalol infusion for refractory hypertension causing severe hypotension and ...
Adrenergic antagonist
A review of the animal pharmacology of labetalol, a combined alpha-and beta-adrenoceptor-blocking drug. British journal of ... Atenolol Oxprenolol Metoprolol Timolol Pindolol Nadolol Pindolol Esmolol Acebutolol Sotalol Talinolol Betaxolol Labetalol ...
Hydralazine
... is often used to treat hypertension in pregnancy, though, with either labetalol and/or methyldopa. Hydralazine is ...
Antihypertensive drug
Although α-methyldopa is generally regarded as a first-line agent, labetalol and metoprolol are also acceptable. Atenolol has ... Beta blockers acebutolol atenolol bisoprolol betaxolol carteolol carvedilol labetalol metoprolol nadolol nebivolol oxprenolol ... bucindolol carvedilol labetalol clonidine (indirectly) Although beta blockers lower blood pressure, they do not have a positive ...
Hyperkalemia
Examples of drugs that can raise the serum potassium are non-selective beta-blockers such as propranolol and labetalol. Beta-1 ...
Methamphetamine
Beta blockers with lipophilic properties and CNS penetration such as metoprolol and labetalol may be useful for treating CNS ... and cardiovascular toxicity.[failed verification] The mixed alpha- and beta-blocker labetalol is especially useful for ...
Tetanus
... and may require IV labetalol, magnesium, clonidine, or nifedipine. Drugs such as diazepam or other muscle relaxants can be ...
Nebivolol
Along with labetalol, celiprolol and carvedilol, it is one of four beta blockers to cause dilation of blood vessels in addition ...
Aortic dissection
... or labetalol) is preferred. Vasodilators such as sodium nitroprusside can be considered for people with ongoing high blood ...
Eclampsia
Common drugs used for blood pressure control during eclampsia are hydralazine or labetalol, due to their effectiveness, lack of ...
List of adrenergic drugs
N-Isopropyloctopamine Isoxsuprine Labetalol Levonordefrin Levosalbutamol Mabuterol Methoxyphenamine Methyldopa Norepinephrine ( ... DL-017 Domesticine Doxazosin Eugenodilol Fenspiride GYKI-12,743 GYKI-16,084 Indoramin Ketanserin L-765,314 Labetalol ... Hydroxytertatolol ICI-118,551 Idropranolol Indenolol Indopanolol Iodocyanopindolol Iprocrolol Isoxaprolol Isamoltane Labetalol ...
Sympatholytic
Labetalol (has additional α-blocking activity) Nadolol Penbutolol (has intrinsic sympathomimetic activity) Pindolol (has ...
List of drugs: La
Ls-Ly labetalol (INN) labetuzumab (INN) Labid (Warner Chilcott) labradimil (USAN) Lac-Hydrin lacidipine (INN) lacosamide (INN) ...
Discovery and development of beta-blockers
... for example labetalol and carvedilol) and additional direct vasodilator activity (nebivolol). In addition, long-acting and ...