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*  Ketanserin
ISBN 978-1-56019-100-1. ATC/DDD Index Ketanserin van der Starre PJ, Solinas C (1996). "Ketanserin in the treatment of protamine ... Ketanserin is a high-affinity non-selective antagonist of 5-HT2 receptors in rodents, with Ki values of 2-3 nM for the 5-HT2A ... Ketanserin (INN, USAN, BAN) (brand name Sufrexal; former developmental code name R41468) is a drug used clinically as an ... Ketanserin is classified as an antihypertensive by the World Health Organization and the National Institute of Health. It has ...
*  Serotonin receptor antagonist
Ketanserin Antihypertensive. Blocks 5-HT2A, 5-HT2C and Alpha 1 (A1) adrenoreceptors. Risperidone antipsychotic Trazodone ...
*  Ritanserin
Ketanserin Dr. Ian Morton; I.K. Morton; Judith M. Hall (31 October 1999). Concise Dictionary of Pharmacological Agents: ...
*  Naftidrofuryl
Ketanserin Sarpogrelate Peter Lanzer; Eric J. Topol (20 December 2013). Pan Vascular Medicine: Integrated Clinical Management. ...
*  Altanserin
Other ligands for other parts of the serotonin system used in PET studies are, e.g., DASB, ketanserin, and WAY-100635. As of ...
*  Lidanserin
Ketanserin Richard C. Allen (1989). Annual Reports in Medicinal Chemistry. Academic Press. p. 56. ISBN 978-0-12-040524-4. ...
*  Atiprosin
Prazosin Ketanserin David J. Triggle (1996). Dictionary of Pharmacological Agents. Boca Raton: Chapman & Hall/CRC. ISBN 0-412- ...
*  RH-34
5-MeO-NBpBrT Ketanserin Efavirenz Ralf Heim. Synthese und Pharmakologie potenter 5-HT2A-Rezeptoragonisten mit N-2-Methoxybenzyl ... It was derived by structural modification of the selective 5-HT2A antagonist ketanserin, with the 4-(p-fluorobenzoyl)piperidine ...
*  Cinanserin
The preparation is effective against an atypical pneumonia (SARS). Ketanserin Ritanserin Neuman RS, Zebrowska G (December 1992 ...
*  Streptomyces calvus
"The acute antihypertensive effect of ketanserin increases with age". Journal of cardiovascular pharmacology. 7 Suppl 7: S126-7 ...
*  Phenoxybenzamine
Ketanserin Pindobind Phentolamine Caine M, Perlberg S, Meretyk S (1978). "A placebo-controlled double-blind study of the effect ...
*  KML-010
"Ketanserin and spiperone as templates for novel serotonin 5-HT(2A) antagonists". Current Topics in Medicinal Chemistry. 2 (6): ...
*  Quipazine
"Neurochemical and behavioral evidence that quipazine-ketanserin discrimination is mediated by serotonin2A receptor". The ...
*  Vesicular monoamine transporter
Ketanserin (KET) and the drug Lobeline also bind to the TBZ binding site conformation. Three to four glycosolation sites exist ... Tetrabenazine (branded Nitoman and Xenazine), dihydrotetrabenazine, ketanserin, and the drug lobeline bind to the TBZ binding ... VMAT inhibitors include: Reserpine(RES), bietaserpine, and ketanserin(KET) (potent inhibitors of VMAT2 mediated serotonin ... Tetrabenazine (TBZ, also called Nitoman and Xenazine), Dihydrotetrabenazine (DTBZOH), Ketanserin (KET), and the drug Lobeline ...
*  5-HT2A receptor
The discovery of ketanserin was a landmark in the pharmacology of 5-HT2 receptors. Ketanserin, though capable of blocking 5-HT ... Compounds chemically related to ketanserin such as ritanserin are more selective 5-HT2A receptor antagonists with low affinity ...
*  Lenperone
Chemically related drugs containing the same 4-(p-fluorobenzoyl)piperidine group: Altanserin Ketanserin Lidanserin Setoperone. ...
*  Volinanserin
Eplivanserin Glemanserin Ketanserin Pimavanserin Ritanserin Schmidt CJ, Fadayel GM, Sullivan CK, Taylor VL (November 1992). "5- ...
*  5-I-R91150
... ketanserin displacement". Journal of Nuclear Medicine. 47 (6): 929-937. PMID 16741301. ...
*  Risperidone
Although not a butyrophenone, it was developed with the structures of benperidol and ketanserin as a basis. It has actions at ...
*  Positron emission tomography
2010). "Imaging cortical dopamine D1 receptors using 11C NNC112 and ketanserin blockade of the 5-HT 2A receptors". J Cereb ...
*  Latrepirdine
... ketanserin and quinuclidinyl benzilate in the rat brain]". Eksperimental'naia I Klinicheskaia Farmakologiia (in Russian). 56 (1 ...
*  Vesicular monoamine transporter 1
... and ketanserin (KET). It is thought that RES exhibits competitive inhibition, binding to the same site as the monoamine ...
*  Bath salts (drug)
This effect is mediated by an increase in synaptic dopamine, as haloperidol, but not ketanserin, was capable of blocking the ...
*  5-HT2C receptor
Cinanserin Deramciclane Ketanserin LY-53,857 Metergoline Methiothepin Pizotifen Ritanserin S-32212 SB-206,553 SB-228,357 SB- ...
*  2C-TFM
... displaced radiolabelled ketanserin from 5-HT2A/C receptors with a Ki of 74.5nM, as compared to a Ki of 80.9nM for the ...