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*  Folliculogenesis
... primarily estradiol. Consequently, estrogen levels begin to rise. At this point, the majority of the group of follicles that ...
*  Challenge hypothesis
Berg, S. J.; Wynne-Edwards, K. E. (2001). "Changes in testosterone, cortisol, and estradiol levels in men becoming fathers". ... Estradiol (E2), a type of non gonadal estrogen, seems to play a key role in regulating aggressive behavior during the non- ...
*  Ovarian follicle activation
... and estradiol production in human granulosa-lutein cells". Fertility and Sterility. 100 (2): 585-592.e1. doi:10.1016/j. ...
*  Epiestriol
... also known as 16β-epiestriol or simply 16-epiestriol as well as 16β-hydroxy-17β-estradiol, is a minor and weak endogenous ... estrogen, and the 16β-epimer of estriol (which is 16α-hydroxy-17β-estradiol). Epiestriol is (or has previously been) used ...
*  Gonadotropin-releasing hormone antagonist
Gustofson RL, Segars JH, Larsen FW (November 2006). Ganirelix acetate causes a rapid reduction in estradiol levels without ...
*  Estradiol
... is additionally conjugated with an ester into lipoidal estradiol forms like estradiol palmitate and estradiol ... Estradiol is conjugated in the liver to form estrogen conjugates like estradiol sulfate, estradiol glucuronide and, as such, ... While estradiol levels in men are much lower compared to those in women, estradiol has important roles in men as well. Aside ... Estradiol (E2), also spelled oestradiol, is an estrogen steroid hormone and the major female sex hormone. It is involved in the ...
*  Estradiol sulfamate
Unlike estradiol and other estradiol esters, due to its unique sulfamate ester, E2MATE is not hydrolyzed during first-pass ... Estradiol sulfamate (E2MATE; developmental code names J995, PGL-2, PGL-2001, ZK-190628), or estradiol-3-O-sulfamate, is a ... It is the 3-sulfamate ester of estradiol, and in terms of its estrogenic activity, acts as a prodrug of estradiol. The drug ... In accordance, the systemic potency of oral E2MATE is increased approximately 100-fold relative to that of oral estradiol, ...
*  Estradiol furoate
It is an estrogen ester, specifically, an ester of estradiol. Estradiol benzoate, another estradiol ester, has also been ... Estradiol furoate (brand name Di-Folliculine), also known as 17-furoylestradiol or 17-(2-furancarbonyl)estradiol, is a ...
*  Estradiol stearate
Estradiol palmitate Estradiol undecanoate Hochberg RB, Pahuja SL, Larner JM, Zielinski JE (1990). "Estradiol-fatty acid esters ... It occurs in the body as a very long-lasting metabolite and prohormone of estradiol. In addition, estradiol stearate is or has ... Estradiol stearate (brand name Depofollan), or estradiol octadecanoate, is a naturally occurring steroidal estrogen and an ... estrogen ester - specifically, the C17β stearate ester of estradiol. ...
*  Estradiol dienanthate
... , or estradiol 3,17-dihepanoate, is a semisynthetic, steroidal estrogen. It is an estrogen ester, ... and estradiol benzoate that is used in the treatment of menopausal symptoms in women. Estradiol enanthate J. Elks (14 November ... The drug is a component of Climacteron, an injectable combination formulation of testosterone enanthate, estradiol dienanthate ...
*  Estradiol decanoate
... (E2D), or estradiol decylate, also known as estradiol 17β-decanoate or as estra-1,3,5(10)-triene-3,17β-diol ... Estradiol enanthate Estradiol undecanoate Luisi M, Kicovic PM, Alicicco E, Franchi F (1978). "Effects of estradiol decanoate in ... ester of estradiol - which has been studied for use in hormone replacement therapy for ovariectomized women but was never ...
*  Estradiol phenylpropionate
... (EPP), also known as estradiol 17β-phenylpropionate, is a semisynthetic, steroidal estrogen. It is ... EPP is marketed in combination with estradiol benzoate under the brand name Dimenformon Prolongatum in the Netherlands and in ... a balanced mixture of estradiol and testosterone esters).[1] Both of these drug combinations are long-acting injectables ... combination with estradiol benzoate, testosterone propionate, testosterone phenylpropionate, and testosterone isocaproate under ...
*  Estradiol valerate
Other common esters of estradiol in use include estradiol cypionate, estradiol enanthate, and estradiol acetate, the former two ... Estradiol valerate is an estradiol ester, or a prodrug of estradiol. As such, it is an estrogen, or an agonist of the estrogen ... Along with estradiol cypionate, it is one of the most widely used esters of estradiol. Estradiol valerate is used in the United ... and estradiol cypionate (1952), has since become one of the most widely used esters of estradiol. Estradiol valerate is the ...
*  Estradiol diundecylate
... (brand names Estrolent), or estradiol diundecanoate, also known as 17β-estradiol 3,17β-diundecylate, is ... Estradiol diundecylenate Estradiol undecylate J. Elks (14 November 2014). The Dictionary of Drugs: Chemical Data: Chemical Data ... a semisynthetic, steroidal estrogen and an estrogen ester - specifically, the 3,17β-diundecylate ester of estradiol - which is ...
*  Estradiol diundecylenate
... (brand name Etrosteron), or estradiol diundecenoate, also known as 17β-estradiol 3,17β-diundec-10- ... 17β-diundecylenate ester of estradiol - which is marketed in Argentina. Estradiol diundecylate Estradiol undecylate J. Elks (14 ...
*  Estradiol monopropionate
Estradiol dipropionate Estradiol 3-propionate J. Elks (14 November 2014). The Dictionary of Drugs: Chemical Data: Chemical Data ... also known as estradiol 17β-propionate or estradiol 17β-propanoate, as well as estra-1,3,5(10)-trien-3,17β-diol 17β-propionate ... Estradiol monopropionate (brand names Acrofollin, Agofollin, Akrofollin, Di-Ovahormon Depot, Follhormon, Ovocylin), ... is a synthetic, steroidal estrogen and an estrogen ester - specifically, the C17β propionate ester of estradiol - which was ...
*  Estradiol butyrylacetate
It is an estrogen ester, specifically, an ester of estradiol. J. Elks (14 November 2014). The Dictionary of Drugs: Chemical ... Estradiol butyrylacetate (brand name Follikoside), also known as 17-butanoylacetylestradiol, is a semisynthetic, steroidal ...
*  Estradiol dipropionate
... estradiol dipropionate and estradiol benzoate were the most widely used estradiol esters. Estradiol monopropionate Estradiol 3- ... Along with estradiol benzoate, estradiol dipropionate was one of the first estradiol esters to be developed, having been ... Relative to estradiol benzoate, estradiol dipropionate has enhanced and very prolonged effects. Prior to the development and ... Erwin Schwenk of the Schering Corporation for the estradiol benzoate (Progynon B), estradiol dipropionate (Progynon DP), ...
*  Estradiol pivalate
... (brand name Estrotate), also known as estradiol trimethyl acetate, trimethyl estradiol acetate, or estradiol ... It is an estrogen ester, specifically, an ester of estradiol. J. Elks (14 November 2014). The Dictionary of Drugs: Chemical ...
*  Estradiol hexahydrobenzoate
... (INN) (brand names Benzo-Ginoestril A.P., BenzoGynoestryl Retard, Ginestryl-15-Depot, Menodin, ... It is an estrogen ester, specifically, an ester of estradiol. J. Elks (14 November 2014). The Dictionary of Drugs: Chemical ... Tardoginestryl), also known as 17-hexahydrobenzoylestradiol or estradiol 17-cyclohexanecarboxylate, is a semisynthetic, ...
*  Estradiol propoxyphenylpropionate
... (brand name Durovex), also known as estradiol 17-(4-propoxyphenyl)propanoate or estradiol p- ... It is an estrogen ester, specifically, an ester of estradiol. J. Elks (14 November 2014). The Dictionary of Drugs: Chemical ...
*  Estradiol glucuronide
... , or estradiol 17β-D-glucuronide, is a conjugated metabolite of estradiol. It is formed from estradiol in ... of estradiol is excreted in the urine as estradiol glucuronide. The positional isomer of estradiol glucuronide, estradiol 3- ... Estradiol glucuronide can be converted back into estradiol, and a large circulating pool of estrogen glucuronide and sulfate ... A single administered dose of estradiol is absorbed 15% as estrone, 25% as estrone sulfate, 25% as estradiol glucuronide, and ...
*  Estradiol benzoate
17β dipropionate ester of estradiol, and estradiol acetate, the C3 acetate ester of estradiol. Estradiol benzoate was one of ... Esters of estradiol like estradiol benzoate are readily hydrolyzed prodrugs of estradiol, but have an extended duration when ... As prodrugs of estradiol, estradiol benzoate and other estradiol esters are estrogens, or agonists of the estrogen receptors ( ... Two estradiol esters that are related to estradiol benzoate are estradiol dipropionate, the C3, ...
*  Estradiol/progesterone
... (developmental code name TX-001HR, formerly TX-12-001HR) is an oral combination of estradiol, an ... Oral Estradiol + Progesterone) - TherapeuticsMD Estradiol/progesterone - TherapeuticsMD - AdisInsight. ... The drug is the first combination of estradiol and progesterone in oral capsule form that has been developed for clinical use. ... A combination formulation of estradiol and progesterone for use by intramuscular injection has been developed and approved for ...
*  Estradiol undecylate
A few related estradiol esters include estradiol decanoate, estradiol diundecylate, and estradiol diundecylenate. Estradiol ... Along with estradiol valerate, estradiol cypionate, and estradiol benzoate, estradiol undecylate is or has been used as an ... Esters of estradiol like estradiol undecylate are readily hydrolyzed prodrugs of estradiol, but have an extended duration when ... As prodrugs of estradiol, estradiol undecylate and other estradiol esters are estrogens. A phase III clinical trial comparing ...