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*  Anthelmintic
Benzimidazoles: Albendazole - effective against threadworms, roundworms, whipworms, tapeworms, hookworms Mebendazole - ...
*  Benzimidazole
This method afford 2-substituted benzimidazoles. Benzimidazole is a base: C6H4N(NH)CH + H+ → [C6H4(NH)2CH]+ It can also be ... Several dyes are derived from benzimidazoles. Benzimidazole is involved in the synthesis of the antiandrogen Galeterone. ... The benzimidazole opioid family includes a number of strong agents e.g. etonitazene, whose article discusses the family in some ... Benzimidazole fungicides are commercialized. They act by binding to the fungal microtubules and stopping hyphal growth. It also ...
*  Benzimidazole fungicide
The solubility of benzimidazole fungicides is low at physiological pH and becomes high at low pH. In plants, carbendazim, ... Benzimidazole fungicides are a class of fungicides including benomyl, carbendazim (MBC), thiophanate-methyl, thiabendazole and ... Mutant pathogens resistant to one benzimidazole fungicide are usually resistant to all of them. The F200Y and E198A,G,K ... Because there is only one target site, benzimidazole resistance quickly became a serious problem. When they were the only ...
*  Triclabendazole
It is a member of the benzimidazole family of anthelmintics. The benzimidazole drugs share a common molecular structure, ... Benzimidazoles such as triclabendazole are generally accepted to bind to beta-tubulin and prevent the polymerization of the ... It is a member of the benzimidazole family of medications for worms. It is on the World Health Organization's List of Essential ... Wolfe, M. Michael; Lowe, Robert C. (2014). "Benzimidazoles". Pocket Guide to GastrointestinaI Drugs. John Wiley & Sons. p. ...
*  Ancylostoma braziliense
Most benzimidazoles are effective. Mebendazole, triclabendazole and fenbendazole are commonly used. Ivermectin and pyrantel ...
*  Diethyl azodicarboxylate
P. N. Preston (1980). Benzimidazoles and congeneric tricyclic compounds. John Wiley and Sons. pp. 475-. ISBN 978-0-471-08189-0 ...
*  Cooperia oncophora
There are several benzimidazoles were successful in clearing infection, including albendazole, febantel, fenbendazole, ... Broad spectrum anthelmintics include benzimidazoles (BZs). BZs have been used since the 1960s, and resistance was detected in ... Infections are usually treated with broad-spectrum anthelmintics such as benzimidazole, but resistance to these drugs has ... Resistance has been reported to all broad spectrum anthelmintics, which are benzimidazoles (BZs), levamisole/morantel (LEV) and ...
*  AZ-11713908
Verbist BM, De Cleyn MA, Surkyn M, Fraiponts E, Aerssens J, Nijsen MJ, Gijsen HJ (April 2008). "5-Sulfonyl-benzimidazoles as ... WO patent 2004/108688, LIU Z, PAGÈ D, WALPOLE C, YANG H, "BENZIMIDAZOLE DERIVATIVES, COMPOSITIONS CONTAINING THEM, PREPARATION ... A large number of related benzimidazole derived cannabinoid ligands are known. AM-6545 CB-13 Yu XH, Cao CQ, Martino G, Puma C, ... "Novel benzimidazole derivatives as selective CB2 agonists". Bioorganic & Medicinal Chemistry Letters. 18 (13): 3695-700. doi: ...
*  Etonitazene
Synthese neuer 2-Amino-benzimidazole" [Benzimidazole Derivatives and related Heterocycles VII. Synthesis of new 2-amino- ... The benzimidazole is then alkylated with the desired 1-chloro-2-dialkylaminoethane, forming the final product. This particular ... It is one of several benzimidazole opioids, and is structurally related to clonitazene (where the p-ethoxybenzyl group is ... Etonitazene and its related opioid agonist benzimidazoles were discovered in the late 1950s, by a team of Swiss researchers ...
*  Tiabendazole
2-(4'-Thiazolyl)-Benzimidazole, A New Anthelmintic". Journal of the American Chemical Society. 83 (7): 1764-1765. doi:10.1021/ ... Grenda, V. J.; Jones, R. E.; Gal, G.; Sletzinger, M. (1965). "Novel Preparation of Benzimidazoles from N-Arylamidines. New ... 5-isopropoxycarbonylamino-benzimidazole". Experientia. 26 (5): 550-551. doi:10.1007/BF01898506. Chronicles of Drug Discovery, ...
*  Clonorchis sinensis
However, benzimidazoles are very weak as vermicide. As with other trematodes, praziquantel is the drug of choice. Lately, ...
*  Benzimidazoline
Grimmett, M. R. (1997). Imidazole and Benzimidazole Synthesis. Academic Press. pp. 71ff. ISBN 9780080534459. ...
*  Apple scab
Benzimidazole fungicides, e.g., Benlate (now banned in many countries due to its containing the harmful chemical benzene) work ...
*  Clemizole
Benzimidazoles substituted with an alkylamine at position 2 have a venerable history as H1 antihistaminic agents. The standard ... Imide formation with the remaining free amino group closes the ring to afford 2-chloromethyl benzimidazole (3). Displacement of ... "Zur Darstellung der Benzimidazole". Justus Liebigs Annalen der Chemie. 575 (2): 162. doi:10.1002/jlac.19525750204. GB 703272 ; ... starting material for many benzimidazoles consists of phenylenediamine, or its derivatives. Reaction of that compound with ...
*  Imidazole
Grimmett, M. Ross (1997). Imidazole and Benzimidazole Synthesis. Academic Press. Brown, E. G. (1998). Ring Nitrogen and Key ... Benzimidazole, an analog with a fused benzene ring Dihydroimidazole or imidazoline, an analog where 4,5-double bond is ...
*  Discovery and development of proton pump inhibitors
Though all have a substituted pyridine part, one group has it linked to various benzimidazoles but the other has it linked to a ... Optimization of substituted benzimidazoles and their antisecretory effects were studied on the newly discovered proton pump to ... It is similar to lansoprazole in having no substituents on its benzimidazole part and a methyl group at site 3 on the pyridine ... Addition of a trifluoromethyl group to the benzimidazole moiety led to a series of very active compounds with varying solution- ...
*  Echinococcus multilocularis
Currently, benzimidazoles (such as albendazole) are used to treat AE: only halt their proliferation and do not actually kill ... Jura H, Bader A, Frosch M (May 1998). "In vitro activities of benzimidazoles against Echinococcus multilocularis metacestodes ... best results in reducing parasite burden Despite the improvements in the chemotherapy of echinococcosis with benzimidazole ...
*  Ascaridia
Piperazine salts, levamisole and benzimidazoles are all reported treatments. Ascarid eggs are resistant to desiccation, persist ...
*  Oxfendazole
It comes under the chemical class of the benzimidazoles. This drug is barely used in horses, goats, sheep, and cattle. It is ... Oxfendazole is a broad spectrum benzimidazole anthelmintic. Its main use is for protecting livestock against roundworm, ...
*  O-Phenylenediamine
Reactions with carboxylic acids and their derivatives afford benzimidazoles. The herbicide benomyl is prepared in this manner. ...
*  Chlorflurazole
"Benzimidazole, 4,5-dichloro-2-(trifluoromethyl)-". WebBook. NIST. Chlorflurazole, alanwood.net "40 C.F.R.: Appendix A to Part ...
*  Taenia asiatica
The commonly used drugs for tapeworms, benzimidazoles are relatively ineffective. Praziquantel at a single dose of 150 mg is ...
*  Ancylostoma duodenale
... can be treated with albendazole, mebendazole and benzimidazoles. Pyrantel pamoate is an alternative. In ...
*  Janus kinase inhibitor
Kyoung Kim M, Shin H, Kwang-su P, Kim H, Park J, Kim K, Nam J, Choo H, Chong Y (2015). "Benzimidazole Derivatives as Potent ... Some JAK1 inhibitors are based on a benzimidazole core. Ruxolitinib (trade names Jakafi/Jakavi) against JAK1/JAK2 for psoriasis ...
*  BIM-018
... is a synthetic cannabinoid that is the benzimidazole analog of JWH-018. It is presumed to be a potent agonist of the ... Related benzimidazole derivatives have been reported to be highly selective agonists for the CB2 receptor. AM-2201 FUBIMINA ... "Novel benzimidazole derivatives as selective CB2 agonists". Bioorganic & Medicinal Chemistry Letters. 18 (13): 3695-3700. doi: ...