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*  Benzazepine
Benzazepines are heterocyclic chemical compounds consisting of a benzene ring fused to an azepine ring. Examples include: ... Benazepril Fenoldopam GSK-189,254 Ivabradine Lorcaserin Semagacestat Varenicline Benzodiazepine Dibenzazepine Benzazepines at ...
*  2,3,4,5-Tetrahydro-1,5-methano-1H-3-benzazepine
... is a drug originally researched as a potential opioid analgesic, but was found ... 5-methano-1H-3-benzazepine, it seems unlikely that this is actually the compound being sold. Corey lactone 4-phenylbenzoate ... 5-methano-1H-3-benzazepines". Journal of Medicinal Chemistry. 22 (4): 455-7. doi:10.1021/jm00190a020. PMID 430484. Singer, R. A ... 5-methano-1H-3-benzazepine via Oxidative Cleavage and Reductive Amination Strategies". Synthesis. 2004 (11): 1755. doi:10.1055/ ...
*  Azepine
Azepane Benzazepines Diazepine Oxepin Borepin. ...
*  List of dopaminergic drugs
Adamantanes: Amantadine • Memantine • Rimantadine Aminotetralins: 7-OH-DPAT • 8-OH-PBZI • Rotigotine • UH-232 Benzazepines: 6- ...
*  Oxazepine
Azepine Benzazepines Diazepine Oxepin Borepin CR gas(dibenzoxazepine). ...
*  Dibenzazepine
Benzazepine Dibenzothiazepine Dibenzothiepin Dibenzoxepin Yagiela, John; Dowd, Frank; Johnson, Bart; Mariotti, Angelo; Neidle, ...
*  Heterocyclic compound
For azepine, benzazepine is the preferred name. Likewise, the compounds with two benzene rings fused to the central heterocycle ...
*  Dopamine receptor D1
Benzazepine derivatives SCH-23,390 - 100-fold selectivity for D1 over D5 SKF-83,959 - 7-fold selectivity for D1 over D5 with ... Some of the benzazepines have high intrinsic activity whereas others do not. In 2015 the first positive allosteric modulator ... the D5 receptor, but the benzazepines generally are more selective for the D1 and D5 receptors versus the D2-like family. ... To date, most of the known ligands are based on dihydrexidine or the prototypical benzazepine partial agonist SKF-38393 (one ...
*  Povarov reaction
Treatment of these compounds with TBAF invokes a ring-expansion that provides the corresponding benzazepines. One variation of ... "Tetrahydroquinolines and Benzazepines through Catalytic Diastereoselective Formal [4 + 2]-Cycloaddition Reactions between Donor ...
*  2-Bromomescaline
5-tetrahydro-1H-3-benzazepines". J Het Chem. 9 (3): 609-616. Alexander Shulgin; Tania Manning; Paul F Daley (2011). The Shulgin ...
*  Benzhydryl compounds
Benzazepine: mianserin Tetracyclic: dizocilpine Aromatic alkoxy: bifemelane, phenyltoloxamine Keto: phenadoxone, methadone, ...
*  SKF-82,958
... is a synthetic compound of the benzazepine class that acts as a D1/D5 receptor full agonist. SKF-82,958 and similar ... 1982). "Dopaminergic activity of substituted 6-chloro-1-phenyl-2,3,4,5-tetrahydro-1H-3-benzazepines". Journal of Medicinal ...
*  Trepipam
... (INN) is a dopamine receptor agonist of the benzazepine group that was never marketed. Daniel Lednicer (4 March 2009 ...
*  5-HT2C receptor agonist
A series of 3-benzazepine derivatives, such as Lorcaserin (Figure 6) have been evaluated for their potency and selectivity for ... "Discovery and SAR of new benzazepines as potent and selective 5-HT2C receptor agonists for the treatment of obesity". ...
*  Lorcaserin
"Benzazepine derivatives and methods of prophylaxis or treatment of 5ht2c receptor associated diseases", published 2004-16-06, ... "Discovery and SAR of new benzazepines as potent and selective 5-HT2C receptor agonists for the treatment of obesity". ... 5-tetrahydro-1-methyl-1H-3-benzazepine (Lorcaserin), a Selective Serotonin 5-HT2CReceptor Agonist for the Treatment of Obesity ...
*  Corey lactone 4-phenylbenzoate
5-methano-1H-3-benzazepine Vionnet, J. P.; Renaud, P. (1994). "Facile Preparation of (-)-12-Epiprostaglandins from 7-Oxabicyclo ...
*  Aldose reductase inhibitor
3 (6). Sebastian, Jomon (2016). "Structure-Activity Relationship Study Reveals Benzazepine Derivatives of Luteolin as New ...
*  Fenoldopam
... mesylate (Corlopam) is a drug and synthetic benzazepine derivative which acts as a selective D1 receptor partial ...
*  SKF-38,393
... is a synthetic compound of the benzazepine chemical class which acts as a selective D1/D5 receptor partial agonist. ...
*  SKF-83,959
... is a synthetic benzazepine derivative used in scientific research which acts as an agonist at the D1-D2 dopamine ...
*  Anilopam
... (INN; PR 786-723) is an opioid analgesic of the benzazepine class which was developed by Pentwell in the 1960s but was ...
*  6-Br-APB
5-tetrahydro-1H-3-benzazepine and its 6-bromo analogue". Journal of Medicinal Chemistry. 35 (8): 1466-71. doi:10.1021/ ...
*  List of MeSH codes (D03)
8-dihydroxy-1-phenyl-1h-3-benzazepine MeSH D03.438.103.070 --- albendazole MeSH D03.438.103.105 --- astemizole MeSH D03.438. ...
*  Ecopipam
... (SCH-39166) is a synthetic benzazepine derivative drug that acts as a selective dopamine D1/D5 receptor antagonist, ...
*  SKF-81,297
... is a synthetic drug of the benzazepine chemical class that acts as a selective dopamine D1/D5 receptor full agonist ...