Another key identifying feature is its ability to split benzamide. M. hassiacum can also split urea, nicotinamide, and ...
Chemically, it is a substituted benzamide, closely related to metoclopramide. A small Spanish study found that more adverse ...
Kuş C, Özer E, Korkmaz Y, Yurtcu E, Dağalp R (2018). "Benzamide and Benzamidine Compounds as New Inhibitors of Urokinasetype ...
"AH-7921: 3,4-dichloro-N-[[1-(dimethylamino)cyclohexyl]methyl]benzamide". PubChem. U.S. National Library of Medicine. Retrieved ...
Benzamide Gastroprokinetic agent Robert M, Salvà M, Segarra R, et al. (July 2007). "The prokinetic cinitapride has no ... Cinitapride (trade names Cintapro, Pemix) is a gastroprokinetic agent and antiemetic agent of the benzamide class which is ...
Dose M, Lange HW (January 2000). "The benzamide tiapride: treatment of extrapyramidal motor and other clinical syndromes". ...
February 2005). "Discovery and structure-activity relationship of quinuclidine benzamides as agonists of alpha7 nicotinic ... Benzamides, Chloroarenes, All stub articles, Nervous system drug stubs). ...
May 2010). "Exploration of the HDAC2 foot pocket: Synthesis and SAR of substituted N-(2-aminophenyl)benzamides". Bioorganic & ...
A range of related benzamides exhibited activity, of which compound number 40 is shown here. ML252: channel inhibitor, IC50 = ... Pyridyl and Pyrimidine Benzamides as KCNQ2/Q3 Potassium Channel Openers for the Treatment of Epilepsy". ACS Medicinal Chemistry ...
... ethyl benzamides as transient receptor potential ankyrin 1 (TRPA1) antagonists". Molecular Pain. 3: 1744-8069-3-39. doi:10.1186 ...
"Ab-initiocrystal structure analysis and refinement approaches of oligop-benzamides based on electron diffraction data" (PDF). ...
... benzamide (AP24534), a Potent, Orally Active Pan-Inhibitor of Breakpoint Cluster Region-Abelson (BCR-ABL) Kinase Including the ... "Design and synthesis of 3-substituted benzamide derivatives as Bcr-Abl kinase inhibitors". Bioorganic & Medicinal Chemistry ... "Structural factors contributing to the Abl/Lyn dual inhibitory activity of 3-substituted benzamide derivatives". Bioorganic & ...
May 2007). "Structural factors contributing to the Abl/Lyn dual inhibitory activity of 3-substituted benzamide derivatives". ... "Design and synthesis of 3-substituted benzamide derivatives as Bcr-Abl kinase inhibitors". Bioorganic & Medicinal Chemistry ...
Antiemetic Benzamide Grant SC, Kris MG, Gralla RJ, Clark RA, Tyson LB (1993). "Dose-ranging evaluation of the substituted ... Dazopride (AHR-5531) is an antiemetic and gastroprokinetic agent of the benzamide class which was never marketed. It acts as a ... by use of tryptamine and benzamide derivatives, of the putative 5-HT4 receptor mediating tachycardia in the pig". British ... benzamide dazopride when used as an antiemetic in patients receiving anticancer chemotherapy". Cancer Chemotherapy and ...
... benzamide with Morpholine". Pharmaceutical Chemistry Journal. 0091-150X. 38 (7): 381-384. doi:10.1023/B:PHAC.0000048439.38383. ...
... benzamide with Morpholine". Pharmaceutical Chemistry Journal. 0091-150X. 38 (7): 381-384. doi:10.1023/B:PHAC.0000048439.38383. ... Benzamides, Chloroarenes, Russian drugs, All stub articles, Nervous system drug stubs). ...
... benzamides] and Benzisothiazolones". Journal of Medicinal Chemistry. 39 (21): 4313-4320. doi:10.1021/jm960253w. PMID 8863808. ...
... undergoes Beckmann rearrangement to form benzamide, catalyzed by nickel salts or photocatalyzed by BODIPY. ... "Kinetic and mechanistic studies of the rearrangement of benzaldoxime to benzamide catalysed by nickel acetate". Inorganica ...
design and in vitro/in vivo evaluation of a benzamide-type cyclooxygenase-1 selective inhibitor". Journal of Medicinal ...
... a novel azabicyclononane benzamide selective for D2-like dopamine receptors". Synapse. 38 (4): 438-449. doi:10.1002/1098-2396( ...
Trimebutine Amoproxan Bernzamide 3,4,5-trimethoxy-N-(pyridin-4-yl)benzamide [31638-97-8]. Butobendine Capobenic acid Dilazep ...
Some of these prokinetic agents, such as mosapride and cisapride, classic benzamides, have only moderate affinity for 5HT4 ... Benzamide Cisapride Domperidone Itopride Mosapride Metoclopramide Prucalopride Renzapride Tegaserod Mitemcinal Levosulpiride ...
It was originally synthesized to prove that the removal of a single methylene spacer of the benzamide would alter a κ-opioid ... benzamide analgesics". The Upjohn Company. "Properties Viewer". chemicalize.org. v t e (CS1 maint: multiple names: authors list ... Benzamides, Bromoarenes, Synthetic opioids, Mu-opioid receptor agonists, All stub articles, Analgesic stubs). ... hydrogen-bond acceptors and substituted aromatic system to find the compound with the lowest Ki value in a series of benzamide ...
Typical antipsychotic Benzamide Grind M, Nilsson MI, Nilsson L, Oxenstierna G, Sedvall G, Wahlén A (1989). "Remoxipride--a new ... Benzamides, Organobromides, Phenol ethers, Pyrrolidines, Withdrawn drugs, All stub articles, Nervous system drug stubs). ...
"Orally Active Benzamide Antipsychotic Agents with Affinity for Dopamine D2, Serotonin 5-HT1A, and Adrenergic α1Receptors". ... "Orally Active Benzamide Antipsychotic Agents with Affinity for Dopamine D2, Serotonin 5-HT1A, and Adrenergic α1Receptors". ...
The benzamide antipsychotics-amisulpride, nemonapride, etc.-have been shown to bind to these GHB-activated receptors in vivo. ... gamma-hydroxybutyrate binding by benzamide neuroleptics and prochlorperazine but not by other antipsychotics". European Journal ...
They replaced the imidazopyridine with benzimidazole and the benzhydril group was swapped out for a benzamide. The outcome was ...
... γ-hydroxybutyrate binding by benzamide neuroleptics and prochlorperazine but not by other antipsychotics". European Journal of ...
Domperidone Drug of last resort Serotonin-agonising laxatives Benzamide Itopride Metoclopramide Mosapride Anvisa (2023-03-31 ...
... (trade names Barnetil, Barnotil, Topral) is an atypical antipsychotic of the benzamide chemical class used in Europe ... gamma-hydroxybutyrate binding by benzamide neuroleptics and prochlorperazine but not by other antipsychotics". European Journal ...