... (INN) is an anticholinergic and antispasmodic atropine derivative. In the US its patent number is 3,356,682. ...
... hyoscyamine or laevo-atropine (1831), opium salts mixtures (c. 1840s), chloral derivatives (1831 et seq.), ephedrine (1836?), ... The atropine may very well not present a problem, and there is the possibility of atropine content reduction of soluble tablets ... Unlike naloxone, atropine does indeed help morphine and other narcotics combat neuralgia. ... Some manufacturers add the narcotic antagonist naloxone or the anticholinergics atropine and homatropine (in lower than ...
... (NVP) is a naphthalene derivative that possesses anticholinergic activity similar to that of atropine. ... Several NVP derivatives have been synthesized and evaluated for their ability to inhibit choline acetyltransferase and protect ... Cozzari, Costantino; Hartman, BK (1983). "Synthesis of a naphthylvinylpyridine derivative and its use for affinity ...
For example, atropine, stylopine, europine, and lycopine belong to different classes of molecules. Opines and opine-like ... Similar derivatives have been isolated from muscle tissue of certain marine invertebrates: alanopine, strombine, and tauropine ... Leucinopine Leucinopine (N2-(D-1,3-dicarboxypropyl) derivative of leucine) is a member of the nopaline family isolated from ... Chemically, opines fall into two major structural classes: 1. The vast majority are secondary amine derivatives resulting from ...
An O-acylpseudotropine is any derivative of pseudotropine in which the alcohol group is substituted with an acyl group. ... Tropine Pseudotropine benzoate (tropacocaine) Atropine Tropinone Rabot S, Peerless AC, Robins RJ (1995). "Tigloyl-CoA: ...
Isoetarine is yet another medicinally useful derivative of ethanolamine. Heptaminol, a cardiac stimulant Propanolamines Most ... Veratridine and veratrine Tropane alkaloids such as atropine hormones and neurotransmitters epinephrine (adrenaline) and ...
... (3β-tropanol, ψ-tropine, 3-pseudotropanol, or PTO) is a derivative of tropane and an isomer of tropine. ... Atropine Tropine Tropinone Biondich AS, Joslin JD (2016). "Coca: The History and Medical Significance of an Ancient Andean ...
... was first synthesized in 1952 as a chemical analogue of atropine. It was one of several derivatives of an ... Cyclopentolate derivatives can be used as an antidote for organophosphate poisoning. Lethality of cyclopentolate has been ... Treves GR, Testa FC (1952). "Basic Esters and Quaternary Derivatives of β-Hydroxy Acids as Antispasmodics1". Journal of the ... Cyclopentolate or atropine can also be administered to reverse muscarinic and central nervous system effects of indirect ...
For example, atropine is isolated from the plant Atropa belladonna; strychnine is obtained from the seed of the Strychnine tree ... It is another derivative dimer of vindoline and catharanthine and is synthesised from anhydrovinblastine, starting either from ... Alkaloids can be toxic too (e.g. atropine, tubocurarine). Although alkaloids act on a diversity of metabolic systems in humans ... Hesse, p. 5 The suffix "ine" is a Greek feminine patronymic suffix and means "daughter of"; hence, for example, "atropine" ...
Because of its highly polar nature it penetrated less readily into the central nervous system than did atropine; hence it was ... Methylatropine (trade name Eumydrin) is a belladonna derivative. In 1902, the Bayer Company introduced methylatropine, a ... The blocking potency of methylatropine is approximately 10-20 times higher than that of atropine at neuromuscular and ... Gyermek L (1998). "Semisynthetic Derivatives of Tropane Alkaloids and of other Tropane Esters". Pharmacology of Antimuscarinic ...
... atropine MeSH D03.132.889.180.297.297 - atropine derivatives MeSH D03.132.889.180.297.297.400 - ipratropium MeSH D03.132. ... atropine MeSH D03.605.869.189.297 - atropine derivatives MeSH D03.605.869.189.297.400 - ipratropium MeSH D03.605.869.270 - ... atropine MeSH D03.132.760.180.848 - scopolamine MeSH D03.132.760.200 - capsaicin MeSH D03.132.760.570 - nicotine MeSH D03.132. ... morphine derivatives MeSH D03.132.610.422.547.547.149 - codeine MeSH D03.132.610.422.547.547.149.287 - hydrocodone MeSH D03.132 ...
C08CA Dihydropyridine derivatives) Includes atenolol, carvedilol, and metoprolol as alternatives. Atenolol should not be used ... Ephedrineα Atropine Midazolam Morphine Oxygen Acetylsalicylic acid (aspirin) Ibuprofen Paracetamol (acetaminophen) Codeine ... C08CA Dihydropyridine derivatives) (for amlodipine) Alternatives are 4th level ATC chemical subgroup (C09AA ACE inhibitors, ... C08CA Dihydropyridine derivatives) (for amlodipine) Alternatives are 4th level ATC chemical subgroup (C09CA Angiotensin II ...
Atropine Epinephrine (adrenaline)α No listings in this section. No listings in this section. No listings in this section. No ... D08AE Phenol and derivatives) Alternatives limited to chlorothiazide and chlorthalidone Alternatives limited to 4th level ATC ... activated Acetylcysteine Atropine Calcium gluconate Naloxone Deferoxamineα Dimercaprolα Fomepizoleα Sodium calcium edetateα ... purified protein derivative (PPD) Anti-rabies virus monoclonal antibodies Antivenom immunoglobulin Diphtheria antitoxin Equine ...
Ipratropium is a derivative of atropine but is a quaternary amine and therefore does not cross the blood-brain barrier, which ... obtained by treating atropine with isopropyl bromide, thus the name: isopropyl + atropine.[citation needed] It is chemically ... The main contraindication for inhaled ipratropium is hypersensitivity to atropine and related substances. Previously Atrovent ...
Varghese, S.; Vettath, N.; Iyer, K.; Puliyel, J. M.; Puliyel, M. M. (1990). "Ocular atropine induced psychosis--is there a ... The related quinoline derivative mefloquine (Lariam) has also been associated with psychosis. some over-the-counter drugs, ... Bergman, K. R.; Pearson, C.; Waltz, G. W.; Evans R. III (1980). "Atropine-induced psychosis. An unusual complication of therapy ... Prednisone and other corticosteroids Isotretinoin Anticholinergic drugs atropine scopolamine antidepressants L-dopa ...
Research supported in part by the US Army has led to a US patent application for the use of galantamine and/or its derivatives ... Increasing the dose of galantamine from 5 to 8 mg/kg decreased the dose of atropine needed to protect experimental animals from ... According to the investigators, an unexpected synergistic interaction occurred between galantamine and atropine in an amount of ... studied in the research cited in the patent application for use along with the well-recognized nerve agent antidote atropine. ...
It can be prepared by hydrolysis of atropine or other solanaceous alkaloids. Pseudotropine Atropine Tropinone Tropane alkaloid ... Tropine is a derivative of tropane containing a hydroxyl group at the third carbon. It is also called 3-tropanol. It is a ...
Atropine is a parasympathetic blocker. The common premedication dose for atropine is 0.01-0.02 mg/kg. With standard intravenous ... Etomidate - It is an imidazole-derivative that stimulates GABA receptors. The dosage is between 0.2 and 0.6 mg/kg (commonly 20 ... Atropine is a muscarinic receptor antagonist, thus blocking the vagal response. The dose is 10 mcg/kg. It has quick onset of ... Atropine may also be used as a premedication agent in pediatrics to prevent bradycardia caused by hypoxia, laryngoscopy, and ...
Mechanisms of alpha-methylated substrate derivatives". Neurotoxicology. 25 (1-2): 223-32. doi:10.1016/S0161-813X(03)00101-3. ... atropine and cannabinoid receptor antagonists. As well, compounds such as 5-HTP, fenfluramine, 1-Methylpsilocin, Ergometrine, ...
Its derivatives include the triarylmethane dyes. An arenium ion is a cyclohexadienyl cation that appears as a reactive ... itself named for the molecule atropine). Salts of the tropylium cation can be stable, e.g. tropylium tetrafluoroborate. It can ...
Chinotto Tree, N-Methylated tryptamine derivative in leaf Citrus medica, N-Methylated tryptamine derivative in leaf Species, ... "Atropine". The American Society of Health-System Pharmacists. Archived from the original on 2015-07-12. Retrieved Aug 13, 2015 ... N-Methylated tryptamine derivative in leaves Citrus sinesis,DMT, N-Methylated tryptamine derivative Citrus bergamia,DMT, N- ... Methylated tryptamine derivative Mandarin orange Traces of N-methylated tryptamine derivative in leaf. ...
He wanted to convince chemists that organic bases could be described in terms of derivatives of ammonia. Hofmann successfully ... atropine, and tubocurarine, among others. Coniine eventually became the first of the alkaloids to be artificially synthesised. ... In 1863, Hofmann showed that aniline blue is a triphenyl derivative of rosaniline and discovered that different alkyl groups ... He also examined its derivative, allyl isothiocyanate (mustard oil), in 1868, and studied various other isocyanates and ...
Additionally, morphine-atropine pre-medication usually prevents this problem. The recovery from vinyl ether is rapid with only ... Many divinyl ether derivatives of fatty acids exist in nature. Wollweber, Hartmund (2000). "Anesthetics, General". Ullmann's ...
Caffeoyl derivatives from the roots of Aconitum coreanum have been shown to have at least some anti-inflammatory effect in ... The major physiological antidote is atropine, which is used to treat bradycardia. Other drugs used for ventricular arrhythmia ... 2009). "The anti-oxidative and anti-inflammatory effects of caffeoyl derivatives from the roots of Aconitum coreanum R. RAYMOND ...
Given specific circumstances this mechanism (which is intended to protect the heart) may cause atropine-resistant refractory ... Like other methylated xanthine derivatives, aminophylline is both a competitive nonselective phosphodiesterase inhibitor which ... "A randomized controlled trial of intravenous aminophylline for atropine-resistant out-of-hospital asystolic cardiac arrest". ...
... (Pro-Diazepam) is a water-soluble prodrug of the benzodiazepine derivative diazepam. It can be administered ... influence of atropine dose". Toxicology. 188 (2-3): 197-209. doi:10.1016/s0300-483x(03)00086-6. PMID 12767691. v t e (Articles ...
The side effects noted were atropine-like, and most patients experienced dizziness. Imipramine was first tried for treating ... an ethyl cyclohexanol derivative". Biochemical Pharmacology. 35 (24): 4493-4497. doi:10.1016/0006-2952(86)90769-0. PMID 3790168 ... but no pharmacological assessment of this compound or any substituted derivatives was undertaken until the late 1940s. ...
A popular derivative, crack cocaine is typically smoked. When transformed into its freebase form, crack, the cocaine vapour may ... Deliriants atropine (alkaloid found in plants of the family Solanaceae, including datura, deadly nightshade, henbane and ... LSD: A popular ergoline derivative, that was first synthesized in 1938 by Albert Hofmann. However, he failed to notice its ... For instance, in the music industry, the musical genres hip hop, hardcore rap, and trap, alongside their derivative subgenres ...
It is the N,N,N-trimethyl derivative of the well-known biogenic amine tyramine, and, being a natural product with a positively ... but inhibited by atropine pre-treatment. Concentrations of 3-6 μg/mL produced contractions of the isolated guinea pig ileum ... J. S. Buck, R. Baltzly and W. S. Ide (1938). "β-Phenethylamine derivatives. Tertiary and quaternary salts." 60 1789-1792. G. ... or atropine, but completely counteracted by sparteine or tetrapropylammonium iodide. No muscarinic action was seen. Doses of 6 ...
Further, it produces hypotension of 1-2 hours in duration that is not prevented by treatment with atropine or propranolol. Most ... acetic acid derivatives as protein kinase inhibitors. Surugatoxin has not been demonstrated to be effective in either of these ...