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*  Phentolamine
... (Regitine) is a reversible nonselective α-adrenergic antagonist. Its primary action is vasodilation due to α1 ... In response, the β1 adrenergic receptors on the heart increase its rate, contractility, and dromotropy, which help to offset ... as they can cause unopposed α-adrenergic mediated coronary vasoconstriction, worsening myocardial ischemia and hypertension. It ...
*  Alpha-1D adrenergic receptor
Antagonists A-315456 BMY 7378 (also α2C antagonist) Adrenergic receptor GRCh38: Ensembl release 89: ENSG00000171873 - Ensembl, ... The alpha-1D adrenergic receptor (α1D adrenoreceptor), also known as ADRA1D, is an alpha-1 adrenergic receptor, and also ... This gene encodes alpha-1D-adrenergic receptor. Similar to alpha-1B-adrenergic receptor gene, this gene comprises 2 exons and a ... 2004). "Cell surface expression of alpha1D-adrenergic receptors is controlled by heterodimerization with alpha1B-adrenergic ...
*  Osemozotan
This molecules bind with almost 1000 times greater affinity to 5-HT1A receptors than most other 5-HT, dopamine, or adrenergic ... Modification of cocaine-induced behavioral and neurochemical effects by serotonin1A receptor agonist/antagonist in mice. ...
*  Beta blocker
Adverse effects associated with β2-adrenergic receptor antagonist activity (bronchospasm, peripheral vasoconstriction, ... β1-adrenergic receptors are located mainly in the heart and in the kidneys. β2-adrenergic receptors are located mainly in the ... β3-adrenergic receptors are located in fat cells. Beta receptors are found on cells of the heart muscles, smooth muscles, ... Some block activation of all types of β-adrenergic receptors and others are selective for one of the three known types of beta ...
*  Tolamolol
... is a beta adrenergic receptor antagonist. Curtis-Prior, PB; Gadd, AL (1990). "Beta-adrenoceptor antagonists and human ...
*  Pafenolol
... is a beta adrenergic receptor antagonist. Lennernäs, H; Regårdh, CG (1993). "Dose-dependent intestinal absorption and ...
*  Sulfinalol
... is a beta adrenergic receptor antagonist. The methyl group on a sulfoxide is sufficiently acidic to substitute for ... "Studies on the mechanism of the acute antihypertensive and vasodilator actions of several beta-adrenoceptor antagonists". J. ...
*  Procinolol
... is a beta adrenergic receptor antagonist. Singh, KP (1983). "Influence of beta-adrenoceptor antagonists on ...
*  Ronactolol
... is a beta adrenergic receptor antagonist. Mannucci, C; Caviglioli, G; Perico, A; Triolo, A (1992). "High-performance ...
*  Toliprolol
... is a beta adrenergic receptor antagonist. Stephenson, KA; Wilson, AA; Meyer, JH; Houle, S; Vasdev, N (2008). "Facile ...
*  Soquinolol
... is a beta adrenergic receptor antagonist. Gries, J; Unger, L; Einig, H; Friedrich, L; Hofmann, HP; Kreiskott, H; ... "Pharmacological characterization of the new highly potent beta-adrenergic receptor blocker soquinolol". Arzneimittel-Forschung ...
*  Primidolol
... is a beta adrenergic receptor antagonist. J. Augstein, D. A. Cox and A. L. Ham., DE 2238504 (1973). Chem. Abstr. jte ...
*  Pamatolol
... is a beta adrenergic receptor antagonist. Ban, T; Sada, S; Takahashi, Y; Sada, H; Fujita, T (1985). "Effects of para- ...
*  Ridazolol
... is a beta adrenergic receptor antagonist. Fach, WA; Starke, E; Becker, HJ (1992). "Duration of the effect and dose- ...
*  Pargolol
... is a beta adrenergic receptor antagonist. Hugues, FC; Julien, D; Bors, V; Mougeot, G; Marche, J (1980). "Determination ...
*  Antidepressant
Additionally, most also act as α1-adrenergic receptor antagonists. The majority of the currently marketed SARIs belong to the ... Serotonin antagonist and reuptake inhibitors (SARIs) while mainly used as antidepressants, are also anxiolytics and hypnotics. ... Bupropion, a weak NDRI and nicotinic antagonist, may be useful in treating reduced libido as a result of SSRI treatment. ... and antagonist of the 5-HT3 and 5-HT7 receptors. However, it can also technically be applied to vilazodone, which is an ...
*  Abanoquil
... (INN) is an α1-adrenergic receptor antagonist. Alpha blocker Tham, TC; Guy, S; Shanks, RG; Harron, DW (1992). "Dose- ... dependent alpha 1-adrenoceptor antagonist activity of the anti-arrhythmic drug, abanoquil (UK-52,046), without reduction in ...
*  Rauwolscine
... acts predominantly as a α2-adrenergic receptor antagonist. It has also been shown to function as a 5-HT1A receptor ... a specific antagonist radioligand for brain alpha 2-adrenergic receptors". European Journal of Pharmacology. 76 (4): 461-4. doi ... Wainscott DB, Sasso DA, Kursar JD, Baez M, Lucaites VL, Nelson DL (January 1998). "[3H]Rauwolscine: an antagonist radioligand ... partial agonist and 5-HT2A and 5-HT2B receptor antagonist. Ajmalicine Corynanthine Spegatrine Yohimbine KOHLI JD, DE NN (June ...
*  Flestolol
... is a short-acting beta adrenergic receptor antagonist. Acylation of glycidol (2) with the acid chloride 1 produces ...
*  Boldine
In addition, it has alpha-adrenergic antagonist activities in vascular tissue, and it has also been reported to have ...
*  Transurethral needle ablation of the prostate
... needle ablation of the prostate as an alternative to transurethral resection of the prostate when alpha-adrenergic antagonist ...
*  Spegatrine
... is an adrenergic receptor antagonist isolated from Rauvolfia verticillata. Ajmalicine Corynanthine Rauwolscine ...
*  Tolazoline
... is a non-selective competitive α-adrenergic receptor antagonist. It is a vasodilator that is used to treat spasms of ...
*  Niguldipine
... is a calcium channel blocker and a1-adrenergic receptor antagonist. Boer R, Grassegger A, Schudt C, Glossmann H ( ...
*  Iodopindolol
... is a beta-adrenergic selective antagonist tagged by radioisotopic iodine. Pindolol Ezrailson, E. G.; Garber, A. J ... Munson, P. J.; Swartz, T. L.; Birnbaumer, L; Entman, M. L. (1981). "125Iiodopindolol: A new beta adrenergic receptor probe". ...
*  Ritanserin
It has relatively low affinity for the H1, D2, α1-adrenergic, and α2-adrenergic receptors (39-, 77-, 107-, and 166-fold lower ... Ritanserin (INN, USAN, BAN) is a serotonin receptor antagonist which was never marketed for clinical use but has been used in ... Ritanserin acts as a selective 5-HT2A (Ki = 0.45 nM) and 5-HT2C receptor (Ki = 0.71 nM) antagonist. ... a 5HT2A/2C antagonist, on negative symptoms of schizophrenia: A double-blind randomized placebo-controlled study". Progress in ...
*  Intraoperative floppy iris syndrome
Schwinn, D.; Afshari, N. (2006). "α1-Adrenergic Receptor Antagonists and the Iris: New Mechanistic Insights into Floppy Iris ...