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*  Yohimbine
It behaves as an antagonist at α1-adrenergic, α2-adrenergic, 5-HT1B, 5-HT1D, 5-HT2A, 5-HT2B, and D2, and as a partial agonist ... February 2000). "Agonist and antagonist actions of yohimbine as compared to fluparoxan at alpha(2)-adrenergic receptors (AR)s, ... Yohimbine has high affinity for the α2-adrenergic receptor, moderate affinity for the α1 receptor, 5-HT1A, 5-HT1B, 5-HT1D, 5- ... "Regulation of pre-synaptic alpha adrenergic activity in the corpus cavernosum". International Journal of Impotence Research. 12 ...
*  Penbutolol
... is able to bind to both beta-1 adrenergic receptors and beta-2 adrenergic receptors (the two subtypes), thus making ... Like propanolol and pindolol, it is a serotonin 5-HT1A and 5-HT1B receptor antagonist; this discovery by several groups in the ... Penbutolol is able to bind to both beta-1 adrenergic receptors and beta-2 adrenergic receptors (the two subtypes), thus making ... Blocking β adrenergic receptors decreases the heart rate and cardiac output to lower arterial blood pressure. β blockers also ...
*  The Moscow International Medical Cluster
"Identification of adenylate cyclase-coupled beta-adrenergic receptors with radiolabeled beta-adrenergic antagonists". ...
*  Prazosin
A larger controlled Phase II "Clinical Trial of the Adrenergic Alpha-1 Antagonist Prazosin for Alcohol Dependence" is currently ... "A pilot trial of the alpha-1 adrenergic antagonist, prazosin, for alcohol dependence". Alcoholism: Clinical and Experimental ... Day, H. E.; Campeau, S.; Watson Jr, S. J.; Akil, H. (1997). "Distribution of alpha 1a-, alpha 1b- and alpha 1d-adrenergic ... Antagonist of alpha-1 adrenoceptors on vascular smooth muscle, thereby inhibiting the vasoconstrictor effect of circulating and ...
*  Hobet Coal Mine
"Identification of adenylate cyclase-coupled beta-adrenergic receptors with radiolabeled beta-adrenergic antagonists". ...
*  IronFX
"Identification of adenylate cyclase-coupled beta-adrenergic receptors with radiolabeled beta-adrenergic antagonists". ...
*  Cocaine intoxication
Schurr, James W.; Gitman, Brenda; Belchikov, Yuly (2014-12-01). "Controversial therapeutics: the β-adrenergic antagonist and ... "Death temporally related to the use of a Beta adrenergic receptor antagonist in cocaine associated myocardial infarction". ... Cocaine-induced platelet activation and thrombus formation is another deleterious effect, caused by alpha-adrenergic- and ... "Reflections on beta-adrenergic receptor blockers and cocaine use. A case in point". Revista Española De Cardiología. 62 (4): ...
*  Specific social phobia
Beta-adrenergic antagonists help to control palpitations and tremors unresponsive to the treatment of anxiolytic medication. ...
*  Olney's lesions
Conversely, coadministration of NMDA-antagonists with alpha-2 adrenergic antagonists, like yohimbine could theoretically ... D.Wozniak - NMDA Antagonist Neurotoxicity: Mechanism and Prevention] Olney J, Labruyere J, Wang G, Wozniak D, Price M, Sesma M ... The potency of the drugs in producing these neurotoxic changes corresponded with their potency as NMDA antagonists: i.e. MK-801 ... Even if the hypothesis of gross neural apoptosis proves to be false in humans, NMDA antagonists certainly have potential to ...
*  Alpha-1 blocker
Prazosin has been established as an effective and safe, brain active alpha-1 adrenergic receptor antagonist. It can be used ... Taylor, Fletcher; Raskind, Murray A. (February 2002). "The alpha1-adrenergic antagonist prazosin improves sleep and nightmares ... Alpha-1 blockers (also called alpha-adrenergic blocking agents) constitute a variety of drugs that block alpha-1-adrenergic ... By reducing α1-adrenergic activity of the blood vessels, these drugs may cause hypotension (low blood pressure) and interrupt ...
*  Alprenoxime
"Ocular delivery of the beta-adrenergic antagonist alprenolol by sequential bioactivation of its methoxime analogue". Journal of ...
*  Smith-Magenis syndrome
... "β1-adrenergic antagonists improve sleep and behavioural disturbances in a circadian disorder, Smith-Magenis syndrome" (Full ... blockade of endogenous melatonin production during the day by the adrenergic antagonist acebutolol can increase concentration, ...
*  Reflex syncope
Certain medications may also be helpful: Beta blockers (β-adrenergic antagonists) were once the most common medication given; ...
*  Rostral ventromedial medulla
Since the study using SB-269970 did not use a α2-adrenergic antagonist as a control, it is possible that some of the effects of ... One limiting factor is that SB-269970 was also found to be a potent α2-adrenergic antagonist. ... To test the effects of an NK1 antagonist during injury states, an NK1 antagonist was microinjected into the RVM after ... Based on previous experiments, a 5-HT3 antagonist, ondansetron, and a 5-HT7 antagonist, SB-269,970, were chosen to study. ...
*  Pelvic pain
Yang G, Wei Q, Li H, Yang Y, Zhang S, Dong Q (2006). "The effect of alpha-adrenergic antagonists in chronic prostatitis/chronic ...
*  Dopamine receptor D2
Piribedil - also D3 receptor agonist and α2-adrenergic antagonist Pramipexole - also D3, D4 receptor agonist Quinelorane - ... also NMDA antagonist) 2-Phenethylamine - (also a TAAR1 agonist and GABAb antagonist with effects at AMPA receptors) LSD - in ... Most of the older antipsychotic drugs such as chlorpromazine and haloperidol are antagonists for the dopamine D2 receptor, but ... Brexpiprazole Cariprazine GSK-789,472 - Also D3 antagonist, with good selectivity over other receptors Ketamine ( ...
*  Vascular dementia
... angiotensin II receptor antagonists or adrenergic antagonists. Elevated lipid levels, including HDL, were found to increase ... receptor antagonist; cholinesterase inhibitors galantamine, donepezil, rivastigmine; and ginkgo biloba extract. The general ...
*  Pharmaceutical industry
Black JW, Crowther AF, Shanks RG, Smith LH, Dornhorst AC (1964). "A new adrenergic betareceptor antagonist". The Lancet. 283 ( ...
*  Oxymetazoline
... although its pharmacological effects may be reversed by α adrenergic antagonists such as phentolamine. In the event of a ... Oxymetazoline is a selective α1 adrenergic receptor agonist and α2 adrenergic receptor partial agonist. It is a topical ... with primary effects on α adrenergic receptors and little if any effect on β adrenergic receptors. Oxymetazoline is readily ... α2 adrenergic receptors. Since vascular beds widely express α1 receptors, the action of oxymetazoline results in ...
*  Pacrinolol
... is a beta adrenergic receptor antagonist. Stache, U; Fritsch, W; Fehlhaber, HW (1987). "Synthesis of the highly ...
*  Tienoxolol
... is a beta adrenergic receptor antagonist. Mahé, N; Do, B; Nicolaï, B; Rietveld, IB; Barrio, M; Tamarit, JL; Céolin, ...
*  Tiprenolol
... is a beta adrenergic receptor antagonist. Allen, JD; Shanks, RG (1974). "Effects of tiprenolol, practolol and ...
*  Spirendolol
... is a beta adrenergic receptor antagonist. Mostaghim, R; Maddox, YT; Ramwell, PW (1986). "Endothelial potentiation ...
*  Tamsulosin
It is an α1a adrenergic receptor antagonist. Tamsulosin was developed by Yamanouchi Pharmaceuticals (now part of Astellas ... Tamsulosin is a selective α1 receptor antagonist that has preferential selectivity for the α1A receptor in the prostate versus ...
*  Pyogenic granuloma
Several reports have demonstrated the efficacy of topical application of the beta-adrenergic antagonist timolol in the ... Treatment of pediatric pyogenic granulomas using B-adrenergic receptor antagonists. Pediatr Dermatol. 2014 Mar;31(2)203-7. ...
*  Corynanthine
... acts as an α1-adrenergic and α2-adrenergic receptor antagonist with approximately 10-fold selectivity for the ... This is in contrast to yohimbine and rauwolscine which have around 30-fold higher affinity for α2-adrenergic over α1-adrenergic ... Doxey JC, Lane AC, Roach AG, Virdee NK (February 1984). "Comparison of the alpha-adrenoceptor antagonist profiles of idazoxan ( ... Dual effects of yohimbine, rauwolscine and corynanthine as alpha-adrenoceptor antagonists and 5-HT-receptor agonists". Naunyn- ...
*  C17H19N3O
... a reversible nonselective alpha-adrenergic antagonist Piberaline, a psychoactive drug. ...