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*  Norepinephrine
ISBN 1-4684-3171-4. Griffith RK (2013). "Chapter 10: Adrenergic Receptors and Drugs Affecting Adrenergic Neurotransmission". In ... In most cases when the term "alpha blocker" is used without qualification, it refers to a selective alpha-1 antagonist. ... These are sympatholytic drugs that block the effects of beta adrenergic receptors while having little or no effect on alpha ... These are sympatholytic drugs that block the effects of adrenergic alpha receptors while having little or no effect on beta ...
*  Alpha blocker
Beta blocker Adrenergic antagonists Katzung, Bertram; Masters, Susan (2013). Basic and Clinical Pharmacology. Lange. ISBN 978-0 ... Non-selective α-adrenergic receptor antagonists include: Phenoxybenzamine Phentolamine Tolazoline Trazodon Selective α1- ... are a class of pharmacological agents that act as antagonists on α-adrenergic receptors (α-adrenoceptors). Historically, alpha- ... adrenergic receptor antagonists include: Alfuzosin Doxazosin Prazosin (inverse agonist) Tamsulosin Terazosin Silodosin ...
*  Phentolamine
... (Regitine) is a reversible nonselective α-adrenergic antagonist. Its primary action is vasodilation due to α1 ... In response, the β1 adrenergic receptors on the heart increase its rate, contractility, and dromotropy, which help to offset ... as they can cause unopposed α-adrenergic mediated coronary vasoconstriction, worsening myocardial ischemia and hypertension. It ...
*  Adrenergic antagonist
The α-adrenergic antagonists have different effects from the β-adrenergic antagonists. Adrenergic ligands are endogenous ... While a only a few α-adrenergic antagonists are competitive, all β-adrenergic antagonists are competitive antagonists. ... an α1-adrenergic antagonist will result in vasodilation. Some adrenergic antagonists, mostly β antagonists, passively diffuse ... An adrenergic antagonist is a drug that inhibits the function of adrenergic receptors. There are five adrenergic receptors, ...
*  Beta-2 adrenergic antagonist
A Beta-2 adrenergic antagonist (β2-adrenoceptor antagonist) is an adrenergic antagonist which blocks the beta-2 adrenergic ... ICI-118,551 Butaxamine Propranolol Betablocker Beta-2 adrenergic receptor Beta2-adrenergic agonist Bilski, AJ; Halliday, SE; ... an antagonist for β2 and for β1 or β3 adrenoceptors) like the non-selective betablocker Propranolol. ... Fitzgerald, JD; Wale, JL (1983). "The pharmacology of a beta 2-selective adrenoceptor antagonist (ICI 118,551)". J Cardiovasc ...
*  Beta-3 adrenergic antagonist
A Beta-3 adrenergic antagonist (β3-adrenoceptor antagonist) is an adrenergic antagonist which blocks the Beta-3 adrenergic ... adrenergic receptor antagonists". The Journal of Pharmacology and Experimental Therapeutics. 290 (2): 649-55. PMID 10411574. ... SR 59230A Carvedilol Betablocker Beta-3 adrenergic receptor Candelore MR, Deng L, Tota L, Guan XM, Amend A, Liu Y, Newbold R, ... an antagonist for β3 and for β1 or β2 adrenoceptors) like the non-selective betablocker Carvedilol. ...
*  Brefonalol
... is a beta-adrenergic antagonist. Halabi, A; Endell, W; Halabi, I; Kirch, W (1990). "Hemodynamic effects of ...
*  Bucumolol
... is a beta-adrenergic antagonist. Nakayama, K; Oshima, T; Koike, H (1981). "Assessment of beta-blockade and the non- ... specific effect of bucumolol, a beta-adrenergic blocking agent, on atrioventricular conduction in anesthetized dogs". Archives ...
*  Moxisylyte
It is an α1-adrenergic antagonist. In the United Kingdom, Moxisylte is marketed as Opilon (Archimedes Pharma UK Ltd) and is ...
*  Metazosin
... is an antihypertensive alpha-adrenergic antagonist. Trcka, V; König, J; Mácová, S; Smíd, M; Helfert, I; Votavová, M; ... a novel alpha-adrenergic antagonist". Biopharmaceutics & drug disposition. 10 (6): 581-9. PMID 2575403. ...
*  Cetamolol
... is a beta adrenergic antagonist. Cardioselective b1-adrenergic blocker. Klausner, MA; Irwin, C; Mullane, JF; Shand, ...
*  Bornaprolol
... is a beta-adrenergic antagonist. Cheymol, G; Jaillon, P; Lecoq, B; Lecoq, V; Cheymol, A; Krumenacker, M (1987). " ... "Cardiovascular beta-adrenergic blocking effects of bornaprolol in humans: Relation to dose and plasma concentration". Journal ...
*  Bunitrolol
... is a beta-adrenergic antagonist. Haddad, S; Poulin, P; Funk, C (2010). "Extrapolating in vitro metabolic ...
*  Levomoprolol
... is a beta adrenergic antagonist. It is the (S)-enantiomer of moprolol. Gianesello, V; Brenn, E; Figini, G; ...
*  Pseudoephedrine
Beta-adrenergic antagonists may also interact with sympathomimetics. Increase of ectopic pacemaker activity can occur when ... α-adrenergic receptors are located on the muscles lining the walls of blood vessels. When these receptors are activated, the ... Activation of β2-adrenergic receptors produces relaxation of smooth muscle of the bronchi, causing bronchial dilation and in ... Its principal mechanism of action relies on its direct action on the adrenergic receptor system. The vasoconstriction that ...
*  Dorzolamide/timolol
Timolol is a non-selective beta-adrenergic antagonist. Common adverse effects include temporarily blurred vision, cloudy vision ...
*  Diprafenone
... is an antiarrhythmic beta adrenergic antagonist. Koytchev, R; Alken, RG; Mayer, O; Smith, I; Greenwood, M (1996). " ...
*  Piribedil
Dopamine receptor antagonist, selective for subtypes D4. Adrenergic receptor antagonist, subtypes α2A and α2C: could be the ... It also has α2-adrenergic antagonist properties. Treatment of Parkinson's disease (PD), either as monotherapy (without levodopa ... Dopamine antagonists reduce the effect of piribedil. At very high doses, piribedil has an emetic action on the chemoreceptor ... Agonist and Antagonist Properties at Subtypes of Dopamine D2-Like Receptor and α1/α2-Adrenoceptor" (PDF). J. Pharmacol. Exp. ...
*  Synephrine
... β2 antagonist): 3.58 μM; SR-5923A (β3 antagonist): 17 μM. The binding of racemic synephrine to cloned human adrenergic ... An adrenergic antagonist selective for α1 receptors. Reversal of reserpine-induced hypothermia by a drug is a classical test ... Referred to here as "oxedrine". A drug often used as a selective 5-HT2A antagonist. Used as a non-selective β-antagonist ... a standard α1 antagonist) and ketanserin, with prazosin being the more potent antagonist (pA2 = 9.38, vs pA2 = 8.23 for ...
*  Tiodazosin
... is an alpha-1 adrenergic antagonist. Terazosin Chiang, J; Hermodsson, G; Oie, S (1991). "The effect of alpha 1-acid ... glycoprotein on the pharmacological activity of alpha 1-adrenergic antagonists in rabbit aortic strips". The Journal of ...
*  Allium neapolitanum
... seems to have beta-adrenergic antagonist properties. The Plant List "BSBI List 2007". Botanical Society of ...
*  Radiocontrast agent
Adverse experience with cimetidine and safety of beta-adrenergic antagonists". Arch Intern Med. 145 (12): 2197-200. doi:10.1001 ...
*  Isoxaprolol
... is an adrenergic antagonist with antiarrhythmic and antihypertensive properties. C.R. Ganellin, David J. Triggle ( ...
*  Moprolol
... is a beta-adrenergic antagonist, or beta blocker. Typically moprolol is prescribed to treat hypertension, high blood ...
*  Pathophysiology of asthma
Medications, including aspirin, β-adrenergic antagonists (beta blockers), ibuprofen, and penicillin. Food allergies such as ... Szentivanyi's Beta Adrenergic Theory is a citation classic using the Science Citation Index and has been cited more times than ... In 1968 Andor Szentivanyi first described The Beta Adrenergic Theory of Asthma; in which blockage of the Beta-2 receptors of ... Szentivanyi, Andor (1968). "The Beta Adrenergic Theory of the Atopic Abnormality in Asthma". J. Allergy. 42: 203-232. doi: ...
*  List of investigational anxiolytics
... α1-adrenergic, α2-adrenergic, and H1 receptor antagonist [10] Cyclobenzaprine (TNX-102) - undefined mechanism of action [11] ... and α1-adrenergic receptor antagonist [12] Midomafetamine (MDMA; "ecstasy") - serotonin-norepinephrine-dopamine releasing agent ... 5-HT2A receptor antagonist [18] Verucerfont (GSK-561679, NBI-77860) - CRF1 receptor antagonist [19] Vilazodone (EMD-68843, SB- ... Agomelatine (AGO-178; Valdoxan) - melatonin MT1 and MT2 receptor agonist, 5-HT2C receptor antagonist[1] Riluzole sublingual ( ...
*  Cirazoline
... is an α1 adrenergic agonist and an α2 adrenergic antagonist". Journal of Pharmacology and Experimental Therapeutics ... a partial agonist at both the α1B and α1D adrenergic receptors, and a nonselective antagonist to the α2 adrenergic receptor. It ... Cirazoline is a full agonist at the α1A adrenergic receptor, ...