*  Brimonidine/timolol
... a selective alpha-2 adrenergic receptor agonist, and timolol, a non-selective beta-adrenergic receptor inhibitor. Elevated IOP ... It is a combination of brimonidine (an α2 adrenergic agonist) and timolol (a β adrenergic blocker), in concentrations of 0.2% ...
*  Physical dependence
... including beta blockers such as propanolol and alpha-adrenergic agonists such as clonidine androgenic-anabolic steroids ... a k-opioid agonist), nor opioid antagonists or inverse agonists, such as naltrexone (a universal opioid inverse agonist) All[ ... All µ-opioids with any (even slight) agonist effect, such as (partial list) morphine, heroin, codeine, oxycodone, buprenorphine ... citation needed] GABA agonists and positive allosteric modulators of both the GABA-A ionotropic receptor and GABA-B ...
*  Postural orthostatic tachycardia syndrome
In these patients the selective Alpha-1 Adrenergic receptor agonist Midodrine may increase venous return, enhance stroke volume ... The selective alpha 1 agonist phenylephrine has been used successfully to enhance venous return and stroke volume in some ...
*  Drug class
5-Alpha-reductase inhibitor Angiotensin II receptor antagonist ACE inhibitor Alpha-adrenergic agonist Beta blocker Dopamine ... For receptors, these activities include agonist, antagonist, inverse agonist, or modulator. Enzyme target mechanisms include ... Conversely not all PPAR agonists are fibrates, not all triglyceride lowering agents are PPAR agonists, and not all drugs that ... PPAR agonist), mode of action (reducing blood triglycerides), and are used to prevent and to treat the same disease ( ...
*  Hypnotic
First-generation Chlorpromazine Second-generation Clozapine Olanzapine Quetiapine Risperidone Zotepine Alpha-adrenergic agonist ...
*  Guanfacine
doi:10.1111/j.1365-2125.1983.tb00311.x. PMC 1427667 . Arnsten AF (October 2010), "The use of α2A adrenergic agonists for the ... Belkin, MR; Schwartz, TL (2015). "Alpha-2 receptor agonists for the treatment of posttraumatic stress disorder". Drugs in ... Guanfacine is a highly selective agonist of the α2A adrenergic receptor, with negligible affinity for any other receptor. ... Adrenergic Receptor Agonist For Attention-Deficit/Hyperactivity Disorder". P & T : a peer-reviewed journal for formulary ...
*  Alpha-1A adrenergic receptor
... a potent alpha 1-adrenergic receptor agonist, selective for the alpha 1A receptor subtype". J. Pharmacol. Exp. Ther. 274 (1): ... 1994). "Cloning, expression and characterization of human alpha adrenergic receptors alpha 1a, alpha 1b and alpha 1c". Biochem ... The alpha-1A adrenergic receptor (α1A adrenoreceptor), also known as ADRA1A, formerly known also as the alpha-1C adrenergic ... There are 3 alpha-1 adrenergic receptor subtypes: alpha-1A, -1B and -1D, all of which signal through the Gq/11 family of G- ...
*  Adrenergic agonist
Tyramine Nicotine Caffeine Methylphenidate Ephedrine Pseudoephedrine Adrenergic receptor Alpha adrenergic agonist Siegel, ... the adrenergic receptors). Directly acting adrenergic agonists act on adrenergic receptors. All adrenergic receptors are G- ... An adrenergic agonist is a drug that stimulates a response from the adrenergic receptors. The five main categories of ... Agonists of each class of receptor elicit these downstream responses. Indirectly acting adrenergic agonists affect the uptake ...
*  Tiamenidine
"Quantitative relationships between alpha-adrenergic activity and binding affinity of alpha-adrenoceptor agonists and ... "Electrophysiologic and Hemodynamic Effects of Chronic Oral Therapy With the Alpha 2-agonists Clonidine and Tiamenidine in ... It acts as a centrally-acting α1 and α2 adrenergic receptor antagonist (with IC50 4.85 μM and 0.0091 μM, respectively). In ...
*  Alpha-1 adrenergic receptor
"Quantitative relationships between alpha-adrenergic activity and binding affinity of alpha-adrenoceptor agonists and ... The alpha-1 (α1) adrenergic receptor is a G protein-coupled receptor (GPCR) associated with the Gq heterotrimeric G-protein. It ... Note that only active muscle α1-adrenergic receptors will be blocked. Resting muscle will not have its α1-adrenergic receptors ... Adrenergic receptor Graham, Robert (May 1, 1996). "α1-Adrenergic Receptor Subtypes Molecular Structure, Function, and Signaling ...
*  Primary polydipsia
... an alpha-2 adrenergic agonist Irbesartan, an angiotensin II receptor antagonist Propranolol, a sympatholytic beta blocker ... Such medications include antipsychotics, antidepressants, anticonvulsants, alpha agonists and anticholinergics. It should also ... a carbonic anhydrase inhibitor Lithium was previously used for treatment of PPD as a direct competitive ADH agonist, but is now ...
*  Aortic insufficiency
Alpha/Beta Adrenergic Agonists, Calcium Channel Blockers, Anticoagulants, Cardiovascular, Opioid Analgesics". emedicine. ... "Heart Failure Medication: Beta-Blockers, Alpha Activity, Beta-Blockers, Beta-1 Selective, ACE Inhibitors, ARBs, Inotropic ... "Dopamine agonists and the risk of cardiac-valve regurgitation". N. Engl. J. Med. 356 (1): 29-38. doi:10.1056/NEJMoa062222. PMID ... "Valvular heart disease and the use of dopamine agonists for Parkinson's disease". N. Engl. J. Med. 356 (1): 39-46. doi:10.1056/ ...
*  Methylergometrine
... is a partial agonist/antagonist on serotonergic, dopaminergic and alpha-adrenergic receptors. Its specific ... dopaminergic and adrenergic receptors". In Vladimír Křen,Ladislav Cvak. Ergot: the genus Claviceps. CRC Press. pp. 411-440. ... which is also an agonist at the 5HT2A-mGlu2 receptor protomer and increases the chances of a patient experiencing ...
*  Arotinolol
"Beta-3 Adrenergic Agonist, BRL-26830A, and Alpha/Beta Blocker, Arotinolol, Markedly Increase Regional Blood Flow in the Brown ... "Arotinolol is a weak partial agonist on beta 3-adrenergic receptors in brown adipocytes". Can J Physiol Pharmacol. 79 (7): 585- ... Arotinolol (INN, marketed under the tradename Almarl) is a medication in the class of mixed alpha/beta blockers. It also acts ... "β-adrenergic blocking, antiarrhythmic compound S-596". It is used in the treatment of high blood pressure and essential tremor ...
*  List of veterinary drugs
... α2-adrenergic antagonist used to reverse the sedative and analgesic effects of alpha-2 adrenergic receptor agonists benazepril ... α2-adrenergic agonist (used to temporarily sedate animals) yohimbine - used to reverse effects of xylazine, also called an " ... mu agonist/kappa antagonist, used as a cough suppressant and for a muscle relaxation effect in horses carprofen - COX-2 ... Pure mu agonist/opioid analgesic used as a premedication moxifloxacin - Antibiotic used for the treatment of acute bacterial ...
*  Generalized anxiety disorder
... α2-adrenergic receptor agonist. Guanfacine - Sympatholytic, α2-adrenergic receptor agonist. Prazosin - Sympatholytic, alpha ... 5-HT1A receptor partial agonists, such as buspirone and tandospirone. Serotonin-norepinephrine reuptake inhibitors (SNRIs), ...
*  Olney's lesions
Drugs that work to suppress NAN include anticholinergics, benzodiazepines, barbiturates and agonists at the alpha-2 adrenergic ... Conversely, coadministration of NMDA-antagonists with alpha-2 adrenergic antagonists, like yohimbine could theoretically ...
*  Adrenergic antagonist
Alpha-2 Adrenergic Receptor Agonists: A Review of Current Clinical Applications, Giovannitti Jr, J. A., Thoms, S. M., & ... Alpha-2 Adrenergic Receptor Agonists: A Review of Current Clinical Applications, Giovannitti Jr, J. A., Thoms, S. M., & ... This is because adrenergic stimulation by agonists, results in normal calcium channel regulation. If these adrenergic receptors ... There are few non-cardiovascular uses for adrenergic antagonists. Alpha-adrenergic antagonists are also used for treatment of ...
*  Anosmia
Idiopathic intracranial hypertension Suprasellar meningioma Refsum's disease Adrenergic agonists or withdrawal from alpha ...
*  Discovery and development of beta2 agonists
Beta2-adrenergic agonist Alpha-adrenergic agonist Asthma Beta blocker Beta-1 adrenergic receptor Beta-2 adrenergic receptor ... Adrenergic agonists that are selective for the β2 subtype cause bronchial dilation and might be expected to relieve the ... β2-agonists are used to treat asthma and COPD, diseases that cause obstruction in the airways. The first β2-agonist ... Long-lasting β2-agonists are often given in a combination with corticosteroids to treat asthma. Short-acting β2-agonists are ...
*  Guanabenz
... (pronounced GWAHN-a-benz, sold under the trade name Wytensin) is an alpha agonist of the alpha-2 adrenergic receptor ...
*  Oxytocin/ergometrine
... an alpha-adrenergic, dopaminergic and serotonin (5-HT2) receptor agonist. Both substances cause the uterus to contract. An ...
*  Alpha-2C adrenergic receptor
3.1 (R)-(+)-m-nitrobiphenyline, a new efficient and alpha2C-subtype selective agonist". Journal of Medicinal Chemistry. 50 (16 ... The alpha-2C adrenergic receptor (α2C adrenoceptor), also known as ADRA2C, is an alpha-2 adrenergic receptor, and also denotes ... "Human alpha 2-adrenergic receptor subtype distribution: widespread and subtype-selective expression of alpha 2C10, alpha 2C4, ... Alpha-2-adrenergic receptors include 3 highly homologous subtypes: alpha2A, alpha2B, and alpha2C. These receptors have a ...
*  TDIQ
It is thought these effects are mediated via a partial agonist action at Alpha-2 adrenergic receptors, and TDIQ has been ...
*  Methamphetamine
... is also an agonist of the alpha-2 adrenergic receptors and sigma receptors with a greater affinity for σ1 than ... alpha-methoxy-alpha-(trifluoromethy)phenylacetyl chloride (MTPA)". J Anal Toxicol. 28 (6): 449-455. doi:10.1093/jat/28.6.449. ... The mixed alpha- and beta-blocker labetalol is especially useful for treatment of concomitant tachycardia and hypertension ... Because neither of these agonists alone can open this ion channel, glutamate and glycine are referred to as coagonists of the ...
*  Prostaglandin DP1 receptor
2007). "Synergistic effect of PGD2 via prostanoid DP receptor on TNF-alpha-induced production of MCP-1 and IL-8 in human ... also known as β-Adrenergic receptor kinase 2 [BARK1]) and arrestin 2 (also known as Arrestin beta 1 [ARRB1]). These agents act ... a novel selective DP agonist". British Journal of Pharmacology. 123 (7): 1317-24. doi:10.1038/sj.bjp.0701708. PMC 1565289 . ...