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*  Alpha-1A adrenergic receptor
... a potent alpha 1-adrenergic receptor agonist, selective for the alpha 1A receptor subtype". J. Pharmacol. Exp. Ther. 274 (1): ... 1994). "Cloning, expression and characterization of human alpha adrenergic receptors alpha 1a, alpha 1b and alpha 1c". Biochem ... The alpha-1A adrenergic receptor (α1A adrenoreceptor), also known as ADRA1A, formerly known also as the alpha-1C adrenergic ... There are 3 alpha-1 adrenergic receptor subtypes: alpha-1A, -1B and -1D, all of which signal through the Gq/11 family of G- ...
*  Alpha-adrenergic agonist
An adrenergic alpha-agonist (or alpha-adrenergic agonists) are a class of sympathomimetic agents that selectively stimulates ... Alpha blocker Adrenergic agonist Beta-adrenergic agonist Declerck I, Himpens B, Droogmans G, Casteels R (September 1990). "The ... α Adrenergic agonists have the opposite function of alpha blockers. Alpha adrenoreceptor ligands mimic the action of ... alpha adrenergic receptors. The alpha-adrenergic receptor has two subclasses α1 and α2. Alpha 2 receptors are associated with ...
*  Mivazerol
... is an alpha-adrenergic agonist. Fox K, Dargie HJ, de Bono DP, Oliver MF, Wülfert E, Kharkevitch T (September 1999). " ... "Effect of an alpha(2) agonist (mivazerol) on limiting myocardial ischaemia in stable angina". Heart. 82 (3): 383-5. doi:10.1136 ...
*  Allergic rhinitis
For nocturnal symptoms, intranasal corticosteroids can be combined with nightly oxymetazoline, an adrenergic alpha-agonist, or ...
*  Nasal congestion
Alpha-adrenergic agonists are the first treatment of choice. They relieve congestion by constricting the blood vessels in the ...
*  Vasoactivity
Important vasoactive substances are angiotensin-11, endothelin-1, and alpha-adrenergic agonists. Various vasoactive agents, ...
*  Ciliary body
Alpha-adrenergic agonists work by decreasing production of fluid and increasing drainage. Brimonidine and Apraclonidine are two ... less selective alpha agonists such as [epinephrine] may decrease the production of aqueous humor through vasoconstriction of ... commonly prescribes alpha agonists for glaucoma treatment. Alphagan P uses a purite preservative, which is better tolerated ...
*  Tetrodotoxin
Alpha adrenergic agonists are recommended in addition to intravenous fluids to combat hypotension; anticholinesterase agents " ...
*  Amitraz
Adverse effects in mammals are caused by amitraz' alpha-adrenergic agonist activity. Symptoms can include low blood pressure ... Its effectiveness is traced back on alpha-adrenergic agonist activity, interaction with octopamine receptors of the central ...
*  Xylometazoline
... is in the decongestant and alpha-adrenergic agonist families of medication. Xylometazoline was patented in 1956 ... It binds to α1 and α2 adrenergic receptors in the nasal mucosa. Due to its sympathomimetic effects, it should not be used by ... The drug works by stimulating adrenergic receptors on the lamina propria of blood vessels in the nose. The decongestant effect ... Haenisch, B.; Walstab, J.; Herberhold, S.; Bootz, F.; Tschaikin, M.; Ramseger, R.; Bönisch, H. (2009). "Alpha-adrenoceptor ...
*  List of MeSH codes (D16)
... adrenergic agents MeSH D27.505.519.625.050.100 --- adrenergic agonists MeSH D27.505.519.625.050.100.100 --- adrenergic alpha- ... adrenergic agents MeSH D27.505.696.577.050.100 --- adrenergic agonists MeSH D27.505.696.577.050.100.100 --- adrenergic alpha- ... agonists MeSH D27.505.519.625.050.100.200 --- adrenergic beta-agonists MeSH D27.505.519.625.050.200 --- adrenergic antagonists ... agonists MeSH D27.505.696.577.050.100.200 --- adrenergic beta-agonists MeSH D27.505.696.577.050.200 --- adrenergic antagonists ...
*  Overflow incontinence
Alpha-adrenergic agonists may cause urinary retention by stimulating the contraction of the urethral sphincter. Calcium channel ...
*  Benign prostatic hyperplasia
Alpha-adrenergic agonist medications, such as decongestants with pseudoephedrine can increase bladder outlet resistance. In ... Effects may take longer to appear than alpha blockers, but they persist for many years. When used together with alpha blockers ... As men age, the enzymes aromatase and 5-alpha reductase increase in activity. Aromatase and 5-alpha reductase are responsible ... Alpha blockers relax smooth muscle in the prostate and the bladder neck, thus decreasing the blockage of urine flow. Common ...
*  Beta blocker
... s must not be used in the treatment of selective alpha-adrenergic agonist overdose. The blockade of only beta ... β1-adrenergic receptors are located mainly in the heart and in the kidneys. β2-adrenergic receptors are located mainly in the ... Newer, third-generation beta blockers can cause vasodilation through blockade of alpha-adrenergic receptors. Accordingly, ... These agents are capable of exerting low-level agonist activity at the β-adrenergic receptor while simultaneously acting as a ...
*  General anaesthesia
One commonly used premedication is clonidine, an alpha-2 adrenergic agonist. Clonidine premedication reduces the need for ... Halothane has been found to be a GABA agonist, and ketamine is an NMDA receptor antagonist. Prior to a planned procedure, the ... Another example of anaesthetic premedication is the preoperative administration of beta adrenergic antagonists to reduce the ... evidence for slowed agonist unbinding". J. Neurosci. 20 (3): 899-907. PMID 10648694. Harrison, N.; Simmonds, M. (1985). " ...
*  Alpha-2 adrenergic receptor
"Inhibition of the lipolytic action of beta-adrenergic agonists in human adipocytes by alpha-adrenergic agonists". J. Lipid Res ... Agonists 4-NEMD 7-Me-marsanidine (also I1 agonist) Agmatine (also I agonist, NMDA, 5-HT3, nicotinic antagonist and NOS ... The alpha-2 (α2) adrenergic receptor (or adrenoceptor) is a G protein-coupled receptor (GPCR) associated with the Gi ... Agonists (activators) of the α2-adrenergic receptor are frequently used in veterinary anaesthesia where they affect sedation, ...
*  Hydromorphone
"Simultaneous treatment of hypertension and opiate withdrawal using an alpha 2 adrenergic agonist" (PDF). J Natl Med Assoc. 75: ... Hydromorphone is a semi-synthetic μ-opioid agonist. As a hydrogenated ketone of morphine, it shares the pharmacologic ...
*  Micro-g environment
Another countermeasure includes administration of Midodrine, which is a selective alpha-1 adrenergic agonist. Midodrine ... The use of beta-2 adrenergic agonists to increase muscle mass, and the use of essential amino acids in conjunction with ...
*  Methyldopa
... is in the alpha-2 adrenergic receptor agonist family of medication. It works by stimulating the brain to decrease ... α-methylnorepinephrine is an agonist of presynaptic central nervous system α2 adrenergic receptors. Activation of these ... with increased use of other safer and more tolerable agents such as alpha blockers, beta blockers, and calcium channel blockers ... This inhibition results in reduced dopaminergic and adrenergic neurotransmission in the peripheral nervous system. This effect ...
*  4-NEMD
... is a potent sedative drug which acts as a selective alpha-2 adrenergic agonist. It is closely related to dexmedetomidine ... ethyl-1H-imidazoles on alpha 1- and alpha 2-adrenergic receptors". Journal of Medicinal Chemistry. 37 (15): 2328-33. doi: ... Like other alpha-2 agonists, it produces sedative and muscle relaxant effects but without producing respiratory depression. It ... "Medetomidine analogs as alpha 2-adrenergic ligands. 3. Synthesis and biological evaluation of a new series of medetomidine ...
*  Attention deficit hyperactivity disorder
Medications used include stimulants, atomoxetine, alpha-2 adrenergic receptor agonists, and sometimes antidepressants. In those ...
*  C10H16N2O3S
The molecular formula C10H16N2O3S (molar mass : 244.31 g/mol) may refer to : Amidephrine, an alpha-adrenergic agonist Biotin, a ...
*  Urinary retention
... alpha-adrenergic agonists, opiates, nonsteroidal anti-inflammatories (NSAIDs), calcium-channel blockers and beta-adrenergic ... BPH may respond to alpha blocker and 5-alpha-reductase inhibitor therapy, or surgically with prostatectomy or transurethral ... 2010-02-10 Fisher, Euan; Subramonian, Kesavapillai; Omar, Muhammad Imran (2014-06-10). "The role of alpha blockers prior to ... agonists, may increase the risk. Anesthesia: General anesthetics during surgery may cause bladder atony by acting as a smooth ...
*  TEAD3
... is a transcriptional activator in alpha 1-adrenergic agonist-stimulated cardiac myocytes". The Journal of Biological Chemistry ...
*  Alpha agonist
... may refer to: Alpha-adrenergic agonist, drugs that selectively stimulate alpha adrenergic receptors PPAR ... modulator, drugs which act upon the Peroxisome proliferator-activated receptor alpha. ...
*  Cannabigerol
CBG has been found to act as a high affinity α2-adrenergic receptor agonist, moderate affinity 5-HT1A receptor antagonist, and ... "Evidence that the plant cannabinoid cannabigerol is a highly potent alpha(2)-adrenoceptor agonist and moderately potent 5HT ... Evidence that the plant cannabinoid cannabigerol is a highly potent α2-adrenoceptor agonist and moderately potent 5HT1A ...
*  Beta-adrenergic agonist
Alpha-adrenergic agonist "WHAT ARE BETA-AGONISTS?". Thoracic.org. American Thoracic Society. Retrieved 17 October 2014. ... Beta adrenergic agonists or beta agonists are medications that relax muscles of the airways, which widen the airways and result ... In general, pure beta-adrenergic agonists have the opposite function of beta blockers. Beta adrenoreceptor agonist ligands ... Adrenergic beta-Agonists at the US National Library of Medicine Medical Subject Headings (MeSH) Delbruck, Max. "The beta- ...