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*  Alpha-1A adrenergic receptor
2001). "Agonist-regulated Interaction between alpha2-adrenergic receptors and spinophilin". J. Biol. Chem. 276 (18): 15003-8. ... The alpha-1A adrenergic receptor (α1A adrenoreceptor), also known as ADRA1A, formerly known also as the alpha-1C adrenergic ... a potent alpha 1-adrenergic receptor agonist, selective for the alpha 1A receptor subtype". J. Pharmacol. Exp. Ther. 274 (1): ... "Entrez Gene: ADRA1A adrenergic, alpha-1A-, receptor". Roberts LR, Fish PV, Ian Storer R, Whitlock GA (April 2009). "6,7-Dihydro ...
*  Norepinephrine
ISBN 1-4684-3171-4. Griffith RK (2013). "Chapter 10: Adrenergic Receptors and Drugs Affecting Adrenergic Neurotransmission". In ... Alpha-2 agonists often have a sedating effect, and are commonly used as anesthesia-enhancers in surgery, as well as in ... These are sympatholytic drugs that block the effects of beta adrenergic receptors while having little or no effect on alpha ... These are sympatholytic drugs that block the effects of adrenergic alpha receptors while having little or no effect on beta ...
*  Alpha blocker
... inverse agonist) Tamsulosin Terazosin Silodosin Selective α2-adrenergic receptor antagonists include: Atipamezole Idazoxan ... Beta blocker Adrenergic antagonists Katzung, Bertram; Masters, Susan (2013). Basic and Clinical Pharmacology. Lange. ISBN 978-0 ... Non-selective α-adrenergic receptor antagonists include: Phenoxybenzamine Phentolamine Tolazoline Trazodon Selective α1- ... The proposed mechanism for yohimbine is stimulation of the adrenergic receptors that are associated with penile erection and ...
*  Adrenergic agonist
... the adrenergic receptors). Directly acting adrenergic agonists act on adrenergic receptors. All adrenergic receptors are G- ... An adrenergic agonist is a drug that stimulates a response from the adrenergic receptors. The five main categories of ... Agonists of each class of receptor elicit these downstream responses. Indirectly acting adrenergic agonists affect the uptake ... Virtual Chembook article on adrenergic drugs adrenergic agonists at the US National Library of Medicine Medical Subject ...
*  Beta-adrenergic agonist
Beta adrenergic agonists or beta agonists are medications that relax muscles of the airways, which widen the airways and result ... In general, pure beta-adrenergic agonists have the opposite function of beta blockers. Beta adrenoreceptor agonist ligands ... "WHAT ARE BETA-AGONISTS?". Thoracic.org. American Thoracic Society. Retrieved 17 October 2014. Adrenergic beta-Agonists at the ... "The beta-adrenergic receptors". Yoo, B.; et al. "Beta1-adrenergic receptors stimulate cardiac contractility and CaMKII ...
*  Beta1-adrenergic agonist
Beta1-adrenergic agonists, also known as Beta1-adrenergic receptor agonists, are a class of drugs that bind selectively to the ... February 2001). "Beta1-adrenergic agonist is a potent stimulator of alveolar fluid clearance in hyperoxic rat lungs". Jpn. J. ... September 1998). "Denopamine, a beta1-adrenergic agonist, prolongs survival in a murine model of congestive heart failure ... Beta-adrenoceptors typically bind to norepinephrine release by sympathetic adrenergic nerves and to circulating epinephrine. ...
*  Alpha-adrenergic agonist
Alpha blocker Adrenergic agonist Beta-adrenergic agonist Declerck I, Himpens B, Droogmans G, Casteels R (September 1990). "The ... An adrenergic alpha-agonist (or alpha-adrenergic agonists) are a class of sympathomimetic agents that selectively stimulates ... α Adrenergic agonists have the opposite function of alpha blockers. Alpha adrenoreceptor ligands mimic the action of ... MeSH list of agents 82000316 Adrenergic alpha-Agonists at the US National Library of Medicine Medical Subject Headings (MeSH). ...
*  Beta2-adrenergic agonist
... adrenergic receptor agonists, also known as adrenergic β2 receptor agonists, are a class of drugs that act on the β2 adrenergic ... Like other β adrenergic agonists, they cause smooth muscle relaxation. β2 adrenergic agonists' effects on smooth muscle cause ... 9 Beta Adrenergic Drugs beta-Adrenergic Receptor Agonists at the US National Library of Medicine Medical Subject Headings (MeSH ... Discovery and development of β2 agonists Ramanujan K. Common beta-agonist inhalers more than double death rate in COPD patients ...
*  Use of beta-adrenergic agonists livestock
Beta-adrenergic agonists, or β-agonists, are non-hormonal growth promotants that help animals put on muscle instead of fat. ... "Beta-agonists: What are they and should I be concerned?". Retrieved 9 January 2017. "Beta agonists in cattle debate beefs up". ... "Use of Beta-Agonists in Cattle Feed". Retrieved 9 January 2017. "Broad screening and identification of β-agonists in feed and ... But problems may exist with all β-agonists supplementation, and not just for animals. The family of β-agonists includes β1-, β2 ...
*  Benzodiazepine
Gross ME (2001). "Tranquilizers, α2-adrenergic agonists, and related agents". In Adams RH. Veterinary Pharmacology and ... These long-acting metabolites are partial agonists. Short-acting compounds have a median half-life of 1-12 hours. They have few ... Ballenger JC (2000). "Benzodiazepine receptors agonists and antagonists". In Sadock VA, Sadock BJ, Kaplan HI. Kaplan & Sadock's ...
*  Orexigenic
α2 adrenergic antagonists[citation needed] - mirtazapine, mianserin Mixed α1/β blockers - carvedilol α2 Adrenergic agonists - ... quetiapine Adrenergic antagonists: β blockers - propranolol, etc. Paradoxically, β-adrenergic agonists are also listed. ... Agents with orexigenic effects include the following: 5-HT2C receptor antagonists/inverse agonists - mirtazapine, olanzapine, ... pregabalin Ghrelin receptor agonists such as anamorelin, GHRP-6, ibutamoren, ipamorelin, and pralmorelin MC4 receptor ...
*  Bronchospasm
Beta2-adrenergic agonists are recommended for bronchospasm. Short acting (SABA) Terbutaline Salbutamol Levosalbutamol Long ... Both of these medications activate alpha-1 adrenergic receptors that result in smooth muscle constriction. Non-selective beta ...
*  Brimonidine
... is an α2 adrenergic agonist. α2 agonists, through the activation of a G protein-coupled receptor, inhibit the ... Peripheral α2 agonist activity results in vasoconstriction of blood vessels (as opposed to central α2 agonist activity that ... The increased uveoscleral outflow from prolonged use may be explained by increased prostaglandin release due to α adrenergic ...
*  Tretoquinol
... is a beta-adrenergic agonist. "Synthesis of 6,7-dihydrox-1,2,3,4-tetrahydroisoquinoline derivatives". Tetrahedron. ...
*  Mivazerol
... is an alpha-adrenergic agonist. Fox K, Dargie HJ, de Bono DP, Oliver MF, Wülfert E, Kharkevitch T (September 1999). " ... "Effect of an alpha(2) agonist (mivazerol) on limiting myocardial ischaemia in stable angina". Heart. 82 (3): 383-5. doi:10.1136 ...
*  Zinterol
... is a beta-adrenergic agonist. Its structure is based on soterenol (antiarrhythmic) and phentermine. Heubach JF, Graf ...
*  Dexmedetomidine
Similar to clonidine, it is an agonist of α2-adrenergic receptors in certain parts of the brain. Dexmedetomidine hydrochloride ... Dexmedetomidine is a highly selective α2-adrenergic agonist. Unlike opioids and other sedatives such as propofol, ...
*  Xylazine
... is a potent α2 adrenergic agonist. When xylazine and other α2 adrenergic receptor agonists are administered, they ... Xylazine is an analogue of clonidine and an agonist at the α2 class of adrenergic receptor. It is used for sedation, anesthesia ... Park, JW; Chung, HW; Lee, EJ; Jung, KH; Paik, JY; Lee, KH (29 April 2013). "α2-Adrenergic agonists including xylazine and ... As an agonist, xylazine leads to a decrease in neurotransmission of norepinephrine and dopamine in the central nervous system. ...
*  Talipexole
... is a D2 dopamine receptor agonist and interacts both pre- and post-synaptic receptors. It also is an α2-adrenergic ... Dopamine agonists in schizophrenia: a review. Eur Neuropsychopharmacol. 1995;5 Suppl:43-53. PMID 8775758 Japanese Ministry of ... Talipexole (B-HT920, Domnin) is a dopamine agonist that is marketed as a treatment for Parkinson's Disease in Japan by ... agonist. The main side effects are drowsiness, dizziness, hallucinations and minor gastrointestinal complaints. In 2008 the ...
*  Alifedrine
... is a partial beta-adrenergic agonist. Effects of the novel beta-adrenergic partial agonist alifedrine on cardiac ...
*  Cimaterol
... is a beta-adrenergic agonist. Dichloroisoprenaline Byrem TM, Beermann DH, Robinson TF (April 1998). "The beta-agonist cimaterol ...
*  Nasal congestion
Alpha-adrenergic agonists are the first treatment of choice. They relieve congestion by constricting the blood vessels in the ...
*  Opioid use disorder
"Alpha₂-adrenergic agonists for the management of opioid withdrawal". The Cochrane Database of Systematic Reviews (5): CD002024 ...
*  Zilpaterol
... (zilpaterol hydrochloride; codenamed RU 42173) is a β2 adrenergic agonist. Under its trade name, Zilmax, it is used ... Verhoeckx KC, Doornbos RP, Witkamp RF, van der Greef J, Rodenburg RJ (January 2006). "Beta-adrenergic receptor agonists induce ... A. Plascencia; N. Torrentera & R.A. Zinn (1999). "Influence of the β-Agonist, Zilpaterol, on Growth Performance and Carcass ...
*  Gabriella Campadelli-Fiume
"Assessment of compliance in children using inhaled beta adrenergic agonists". Ann Allergy. 62 (5): 406-9. PMID 2566291. Herpes ...
*  Saba (disambiguation)
Jedi Master in the fictional Star Wars Expanded Universe Short-acting beta2-adrenergic agonist, a class of drug primarily used ...
*  Phenylpropanolamine
Although originally thought to act as a direct agonist of adrenergic receptors, PPA was subsequently found to show only weak or ... However, such substitution greatly enhances agonist activity at both α- and β- adrenergic receptors. Although ephedrine is less ... Westfall DP, Westfall TC (2010). "Chapter 12: Adrenergic Agonists and Antagonists: CLASSIFICATION OF SYMPATHOMIMETIC DRUGS". In ... The stereoisomers of the drug have only weak or negligible affinity for α- and β-adrenergic receptors. Many sympathetic ...