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*  Efficacy and Safety of Vortioxetine (Lu AA21004) in the Treatment of Patients With Major Depressive Disorder - Full Text View -...
Serotonin Uptake Inhibitors. Serotonin Agents. Serotonin 5-HT1 Receptor Agonists. Serotonin Receptor Agonists. Serotonin 5-HT1 ... Serotonin and Noradrenaline Reuptake Inhibitors. Neurotransmitter Uptake Inhibitors. Membrane Transport Modulators. Molecular ... Experimental: Vortioxetine 5 mg Vortioxetine 5 mg, encapsulated tablets, orally, once daily for up to 8 weeks, then placebo- ... Has a significant risk of suicide according to the investigator's opinion or has a score ≥5 on item 10 (suicidal thoughts) of ...
https://clinicaltrials.gov/ct2/show/NCT00672620
*  Long-Term Extension Study of Lu AA21004 in Participants With Major Depressive Disorder - Full Text View - ClinicalTrials.gov
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https://clinicaltrials.gov/ct2/show/NCT01395147
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Serotonin Receptor Agonists. Serotonin 5-HT1 Receptor Antagonists. Serotonin Antagonists. Serotonin 5-HT3 Receptor Antagonists ... Serotonin Uptake Inhibitors. Neurotransmitter Uptake Inhibitors. Membrane Transport Modulators. Molecular Mechanisms of ... Vortioxetine, 5, 10, and 20 mg, Relapse Prevention Study in Adults With Major Depressive Disorder. The safety and scientific ... The purpose of this study is to evaluate the efficacy of vortioxetine (5, 10, and 20 mg) versus placebo during the first 28 ...
https://www.clinicaltrials.gov/ct2/show/study/NCT02371980?show_locs=Y
*  Study of Efficacy and Safety of Vortioxetine (Lu AA21004) in Treating Generalized Anxiety Disorder - Full Text View -...
Serotonin Receptor Agonists. Serotonin 5-HT1 Receptor Antagonists. Serotonin Antagonists. Serotonin 5-HT3 Receptor Antagonists ... Has previously failed to respond to adequate treatment with selective serotonin reuptake inhibitors and/or serotonin- ... Serotonin Uptake Inhibitors. Neurotransmitter Uptake Inhibitors. Membrane Transport Modulators. Molecular Mechanisms of ... 5. General mental health (psychological distress and well-being). 6. Limitations in usual role activities because of emotional ...
https://www.clinicaltrials.gov/ct2/show/NCT00731120?term=LuAA21004_309&rank=1
*  The Effects of Serotonin Receptor Antagonists on Contraction and Relaxation Responses Induced by Electrical Stimulation in the...
The Effects of Serotonin Receptor Antagonists on Contraction and Relaxation Responses Induced by Electrical Stimulation in the ... Mashhadi, Farzaneh Farajian, Naylor, Robert J. and Javid, Farideh A. (2014) The Effects of Serotonin Receptor Antagonists on ... In the presence of SB258585 1.0 µM (a 5-HT6 receptor antagonist) there was a trend to enhance contraction in the proximal part ... Pre-treatment with SB269970A 1.0 µM (5-HT7 receptor antagonist) induced a greater contractile response to EFS at 0.4 Hz only in ...
http://eprints.hud.ac.uk/id/eprint/21653/
*  Gene, Cell and Tissue | The Effects of Serotonin Receptor Antagonists on Contraction and Relaxation Responses Induced by...
Receptor-binding properties in vitro and in vivo of ritanserin: A very potent and long acting serotonin-S2 antagonist. Mol ... The Effects of Serotonin Receptor Antagonists on Contraction and Relaxation Responses Induced by Electrical Stimulation in the ... Peripheral neural serotonin receptors: identification and characterization with specific antagonists and agonists. Proc Natl ... Development of neural receptors for serotonin in the murine bowel. J Comp Neurol. 1987; 258(4): 597-610[DOI][ PubMed ] ...
http://genecelltissue.com/en/articles/14787.html
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*  Molindone - DrugBank
It has only low to moderate affinity for cholinergic and alpha-adrenergic receptors. Some electrophysiologic data from animals ... Molindone has much lower affinity for D2 receptors than most antipsychotic agents and has a relatively low affinity for D1 ... Antagonist. General Function. Serotonin receptor activity. Specific Function. G-protein coupled receptor for 5- ... Virus receptor activity. Specific Function. G-protein coupled receptor for 5-hydroxytryptamine (serotonin). Also functions as a ...
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*  Alverine - DrugBank
Antagonist. General Function. Serotonin receptor activity. Specific Function. G-protein coupled receptor for 5- ... hydroxytryptamine (serotonin). Also functions as a receptor for various drugs and psychoactive substances. Ligand binding ... 5-methoxy-N,N-dimethyltryptamine. The risk or severity of adverse effects can be increased when Alverine is combined with 5- ... 2,5-Dimethoxy-4-ethylthioamphetamine. The risk or severity of adverse effects can be increased when Alverine is combined with 2 ...
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*  Evidence that the plant cannabinoid cannabigerol is a highly potent alpha2-adrenoceptor agonist and moderately potent 5HT1A...
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https://www.ncbi.nlm.nih.gov/pubmed/20002104
*  Pediatric Headache Medication: Analgesics, Other, Sedative/Hypnotics, Serotonin 5-HT-Receptor Agonists, Antiemetic Agents, Beta...
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https://emedicine.medscape.com/article/2110861-medication
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*  McN-5652: a highly potent inhibitor of serotonin uptake. | Journal of Pharmacology and Experimental Therapeutics
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*  Indian Patents. 214875:'ARALKYL AND ARALKYLIDENE HETEROCYCLIC LACTAMS AND IMIDES'
treatment or prevention a serotonin receptor antagonizing or agonizing effective amount of a compound of the formula I or a ... J. Pharmacol.. 94, 1128 (1988)]. This effect can be blocked by methiothepin, a known serotonin antagonist. Sumatriptan is known ... The "affinities of the compounds of this invention for the various serotonin-1 receptors can be determined using standard ... Glennon's article "Serotonin Receptors: Clinical Implications", Neuroscienceand Behavioral Reviews, 14, 35-47 (1990), refers to ...
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*  A selective 5-HT1a receptor agonist improves respiration in a mouse model of Rett syndrome. - PubMed - NCBI
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*  Metergoline - Liquid Serotonin Antagonist For Lab/R&D | Ray Peat Forum
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https://raypeatforum.com/community/threads/metergoline-liquid-serotonin-antagonist-for-lab-r-d.12908/
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*  A role of 5-HT2 receptors in the gill vasculature of the antarctic fish Pagothenia borchgrevinki. | Journal of Experimental...
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http://jeb.biologists.org/content/201/14/2129