GABA AgonistsGABA AntagonistsGABA Agentsgamma-Aminobutyric AcidChromatography, AffinityGABA ModulatorsReceptors, GABA-AGABA Plasma Membrane Transport ProteinsProtein BindingBinding SitesKineticsMolecular Sequence DataBinding, CompetitiveAmino Acid SequenceReceptors, GABA-BAntibody AffinityGABA Uptake InhibitorsAffinity LabelsLigandsGABA-A Receptor AgonistsRecombinant ProteinsGABA-A Receptor AntagonistsRadioligand AssayMuscimolModels, MolecularBaclofenBase SequenceBicucullineNipecotic AcidsStructure-Activity RelationshipCell LineProtein Structure, TertiaryCarrier ProteinsProtein ConformationSurface Plasmon ResonanceDose-Response Relationship, DrugCell MembraneGABA-B Receptor AgonistsMutagenesis, Site-DirectedReceptors, Cell SurfacePicrotoxinPhosphinic AcidsNeuronsSubstrate Specificity4-Aminobutyrate TransaminaseRecombinant Fusion ProteinsSequence Homology, Amino AcidGABA-B Receptor AntagonistsNeural InhibitionMutationPatch-Clamp TechniquesElectrophoresis, Polyacrylamide GelRats, Sprague-DawleyCalciumPeptidesCloning, MolecularCHO CellsCells, CulturedCricetinaeMolecular WeightGlutamate DecarboxylaseEscherichia coliPyridazinesPeptide FragmentsCattleDiazepamTransfectionProtein SubunitsRabbitsInhibitory Postsynaptic PotentialsBrainDNABiological TransportSynaptic TransmissionHydrogen-Ion ConcentrationGlutamic AcidMembrane ProteinsMacromolecular SubstancesIodine RadioisotopesMembrane Transport ProteinsPeptide LibraryProtein Structure, SecondaryBenzodiazepinesGlycineAllosteric RegulationSpectrometry, FluorescenceAntibodies, MonoclonalXenopus laevisHippocampusDimerizationMembrane PotentialsRats, WistarMolecular StructureFlunitrazepamAdenosine TriphosphateVigabatrinHeparinCrystallography, X-RayBacterial ProteinsOrganic Anion Transporters