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*  Pharmacological Stress Myocardial Perfusion Imaging With the Potent and Selective A2A Adenosine Receptor Agonists ATL193 and...
... hydroxyl group of the ribose on the ATL compounds is protected from phosphorylation by the addition of N-ethylcarboxamide. ... Maximal CF response after bolus of ATL-146e was greater and more sustained than with adenosine. Note that adenosine flow ... No pharmacodynamic half-life data were reported for the adenosine boluses owing to the fact that the adenosine response was ... because comparisons were made between the adenosine A2A receptor agonists and adenosine in the same anesthetized animal model. ...
http://circ.ahajournals.org/content/104/10/1181
*  Adenosine-5'-(N-ethylcarboxamide) - NECA Summary Report | CureHunter
N-ethylcarboxamide): A stable adenosine A1 and A2 receptor agonist. Experimentally, it inhibits cAMP and cGMP phosphodiesterase ... N-ethylcarboxamide) A stable adenosine A1 and A2 receptor agonist. Experimentally, it inhibits cAMP and cGMP phosphodiesterase ... ethylcarboxamide-adenosine (NECA), N6-phenylisopropyladenosine (PIA) and N6-cyclohexyladenosine (CHA) induced dose dependent ... N-ethylcarboxamide) (NECA). Subscribe to New Research on Adenosine-5'-( ...
http://www.curehunter.com/public/keywordSummaryD019830-Adenosine-5---N-ethylcarboxamide--NECA.do
*  Jon Mabley - Fingerprint - The University of Brighton
N-ethylcarboxamide) Oxidants Adenosine Diphosphate Ribose Interleukin-12 Cell Death ...
https://research.brighton.ac.uk/en/persons/jon-mabley/fingerprints/
*  PlumX - Adenosine A1 receptors mediate mobilization of calcium in human bronchial smooth muscle cells.
N-ethylcarboxamide); Biological Transport, Active; Bronchi; *Calcium Signaling; Cells, Cultured; Cyclic AMP; GTP-Binding ... selective agonists at adenosine A(2A) receptors and adenosine A(3) receptors, respectively. Calcium responses to NECA and CPA ... N-ethylcarboxamido-adenosine (100 nM) or N(6)-(3-iodobenzyl)-adenosine-5'-N-methyluronamide (100 nM), ... Adenosine A1 receptors mediate mobilization of calcium in human bronchial smooth muscle cells.. Citation data: American journal ...
https://plu.mx/plum/a/--9003HdxfXUceiJoLLHo6L2S2shEf66ymSBmCguGRY/
*  CLONAZEPAM | SelfDecode | Genome Analysis
Clonazepam affects the reaction [Adenosine-5'-(N-ethylcarboxamide) results in increased expression of CXCL8 protein]. R ... Gamma-aminobutyric acid receptor subunit alpha-5. Gamma-aminobutyric acid receptor subunit beta-1. Gamma-aminobutyric acid ...
https://www.selfdecode.com/chemical/clonazepam/
*  NAVER Academic > Search...
Adenosine, analogs & derivatives, chemistry, metabolism, Adenosine-5'-(N-ethylcarboxamide), Animals, Cell Membrane, Corpus ... Adenosine Triphosphatases, antagonists & inhibitors, Adenosine Triphosphate, pharmacology, Anions, Atractyloside, analogs & ... Role of cysteine residues of rat A2a adenosine receptors in agonist binding.. 1997 M R Mazzoni et al. Biochimica et biophysica ... Adenosine Monophosphate, pharmacology, Animals, Biological Transport, Caffeine, Calcium, metabolism, Calcium Channels, ...
https://academic.naver.com/search.naver?field=3&query=Biochimica+et+Biophysica+Acta+1324%EA%B6%8C+1%ED%98%B8
*  WikiGenes - Adora2a - adenosine A2a receptor
N-ethyl-carboxamide-adenos ine (CGS21680), a selective adenosine A2A receptor agonist, enhanced taurine release, while ... Purinergic P2 receptors trigger adenosine release leading to adenosine A2A receptor activation and facilitation of long-term ... Purinergic P2 receptors trigger adenosine release leading to adenosine A2A receptor activation and facilitation of long-term ... Effects of an adenosine A2A receptor blockade in the nucleus accumbens on locomotion, feeding, and prepulse inhibition in rats. ...
https://www.wikigenes.org/e/gene/e/25369.html
*  DI-fusion The role of spinal and brainstem adenosine receptors in the...
N-ethylcarboxamide). Animals. Brain Stem -- drug effects. Brain Stem -- metabolism. ... The role of spinal and brainstem adenosine receptors in the modulation of the volume-evoked micturition reflex in the ... The role of spinal and brainstem adenosine receptors in the modulation of the volume-evoked micturition reflex in the ... Assessment of the role of A1/A2 adenosine receptors mediating the purine antinociception, motor and autonomic function in the ...
https://difusion.ulb.ac.be/vufind/Record/ULB-DIPOT:oai:dipot.ulb.ac.be:2013/58752/Details
*  List of MeSH codes (D13) - Wikipedia
... adenosine monophosphate MeSH D13.695.667.138.180.080 --- adenosine phosphosulfate MeSH D13.695.667.138.236 --- adenosine ... n-ethylcarboxamide) MeSH D13.570.583.138.240 --- s-adenosylhomocysteine MeSH D13.570.583.138.264 --- s-adenosylmethionine MeSH ... adenosine monophosphate MeSH D13.695.827.068.180.080 --- adenosine phosphosulfate MeSH D13.695.827.068.236 --- adenosine ... adenosine diphosphate sugars MeSH D13.695.667.138.124.070.075 --- adenosine diphosphate glucose MeSH D13.695.667.138.124.070. ...
https://en.wikipedia.org/wiki/List_of_MeSH_codes_(D13)
*  Adenosine-generating ovarian cancer cells attract myeloid cells which differentiate into adenosine-generating tumor associated...
... we investigated the effect of adenosine on myeloid cells and explored a possible contribution of myeloid cells to adenosine ... Little, however, is known about the effect of adenosine on myeloid cells. Considering that tumor associated macrophages (TAM) ... tissues show abundant expression of the ectonucleotidases CD39 and CD73 which generate immunomodulatory adenosine, thereby ... N-ethylcarboxamide (NECA, Tocris) was employed at 100 nM. To control for effects of adenosine on chemokinesis, a control ...
https://jitc.biomedcentral.com.preview-live.oscarjournals.springer.com/articles/10.1186/s40425-016-0154-9
*  Spinal Adenosine Receptor Activation Reduces Hypersensitivity after Surgery by a Different Mechanism Than after Nerve Injury |...
... ethylcarboxamide adenosine. Brain Res 1990; 519:287-93 ... Antinociception by adenosine analogs and an adenosine kinase ... 19 Adenosine receptors are present on intrinsic interneurons in the dorsal horn. 2 It is conceivable that these adenosine ... Poon A, Sawynok J: Antinociception by adenosine analogs and inhibitors of adenosine metabolism in an inflammatory thermal ... in which adenosine is inactive. The mechanisms of norepinephrine release by activation of spinal adenosine A1 receptors after ...
http://anesthesiology.pubs.asahq.org/article.aspx?articleid=1943070
*  "Adenylyl Cyclase Type 6 Overexpression Selectively Enhances ß-Adrenerg" by Xiaoqiu Liu, Muthusamy Thangavel et al.
... adenosine (adenosine-5′-N-ethylcarboxamide, NECA), and prostacyclin (beraprost) receptors. Overexpression of AC6 increased cAMP ... cyclic adenosine monophosphate (cAMP) levels. cAMP signal generation and response is known to be compartmentalized in many cell ... Fibroblasts are activated by factors such as transforming growth factor β and inhibited by agents that elevate 3′,5′- ... N-ethylcarboxamide, NECA), and prostacyclin (beraprost) receptors. Overexpression of AC6 increased cAMP production stimulated ...
https://digitalcommons.chapman.edu/pharmacy_articles/382/
*  Adenosine A2B receptor - Wikipedia
N-ethylcarboxamide induces IL-6 expression via MAPKs and NF-kappaB activation through Akt, Ca(2+)/PKC, cAMP signaling pathways ... The adenosine A2B receptor, also known as ADORA2B, is a G-protein coupled adenosine receptor, and also denotes the human ... 2001). "Adenosine A2B receptors behave as an alternative anchoring protein for cell surface adenosine deaminase in lymphocytes ... Strohmeier GR, Reppert SM, Lencer WI, Madara JL (1995). "The A2b adenosine receptor mediates cAMP responses to adenosine ...
https://en.wikipedia.org/wiki/Adenosine_A2B_receptor
*  Adenosine A2A and A2B receptor expression in neuroendocrine tumours: potential targets for therapy -ORCA
N-ethylcarboxamide, NECA) and the A2AR agonist (CGS21680) stimulated cell proliferation by up to 20-40% which was attenuated by ... adenosine, A2A adenosine receptor, A2B adenosine receptor, human neuroendocrine tumours, cell proliferation, chromogranin A. ... Adenosine A2A and A2B receptor expression in neuroendocrine tumours: potential targets for therapy. Purinergic Signalling 8 (2 ... Adenosine, released during cellular stress, damage and hypoxia, is a major regulator of angiogenesis. Herein, we describe the ...
http://orca.cf.ac.uk/23593/
*  List of MeSH codes (D13) - Thư viện Khoa học VLOS
MeSH D13.695.667.138.124.070.075 --- adenosine diphosphate glucose * MeSH D13.695.667.138.124.070.125 --- adenosine diphosphate ... n-ethylcarboxamide) * MeSH D13.570.583.138.240 --- s-adenosylhomocysteine * MeSH D13.570.583.138.264 --- s-adenosylmethionine ... MeSH D13.695.827.068.124.070.075 --- adenosine diphosphate glucose * MeSH D13.695.827.068.124.070.125 --- adenosine diphosphate ... MeSH D13.570.583.138 --- adenosine * MeSH D13.570.583.138.025 --- adenosine-5'-( ...
https://tusach.thuvienkhoahoc.com/wiki/List_of_MeSH_codes_
*  Repeated Dosing with Oral Allosteric Modulator of Adenosine A1 Receptor Produces Tolerance in Rats with Neuropathic Pain |...
... of intrathecal injection of the adenosine receptor agonists R-phenylisopropyl-adenosine and N-ethylcarboxamide-adenosine on ... such as allosteric adenosine receptor modulation or inhibition of adenosine kinase 9,10 or adenosine deaminase, 11 have been ... Although adenosine agonists were shown to attenuate pain behaviors in a variety of animal models, adenosine agonists are also ... Keil GJ, DeLander GE: Spinally-mediated antinociception is induced in mice by an adenosine kinase-, but not by an adenosine ...
http://anesthesiology.pubs.asahq.org/article.aspx?articleid=1943048
*  NAVER Academic > Search...
Adenosine, analogs & derivatives, pharmacology, Adenosine-5'-(N-ethylcarboxamide), Animals, Caffeine, Corpus Striatum, ... Adenosine A2 receptors regulate the gene expression of striatopallidal and striatonigral neurons.. 1993 S N Schiffmann et al. ... Corticosteroids regulate brain hippocampal 5-HT1A receptor mRNA expression.. 1993 D T Chalmers et al. JOURNAL OF NEUROSCIENCE ...
https://academic.naver.com/search.naver?field=3&query=JOURNAL+OF+NEUROSCIENCE+13%EA%B6%8C+3%ED%98%B8
*  Adenosine A2B receptor-mediated leukemia inhibitory factor release from astrocytes protects cortical neurons against...
N-ethylcarboxamide (NECA) stimulation was directly correlated to de novo protein synthesis, suggesting that LIF release did not ... Adenosine from glutamate-stressed neurons induces rapid LIF release in astrocytes. This rapid release of LIF promotes the ... Mouse cortical neuronal and astrocyte cultures from wild-type and adenosine A2B receptor knock-out animals, as well as ... We show here that glutamate-stressed cortical neurons induce LIF expression through activation of adenosine A2B receptor ...
https://jneuroinflammation.biomedcentral.com/articles/10.1186/1742-2094-9-198
*  Postsynaptic dopamine/adenosine interaction: I. Adenosine analogues inhibit dopamine D2-mediated behaviour in short-term...
The adenosine agonists, L-PIA (a preferentially A-1 adenosine agonist) and NECA (an A-1 and A-2 adenosine agonist with above 10 ... Postsynaptic dopamine/adenosine interaction: I. Adenosine analogues inhibit dopamine D2-mediated behaviour in short-term ... Mice pretreated with reserpine 5 mg/kg (4 h prior to the start of motor activity recording) showed locomotor activation after ... stimulates postsynaptic D-2 receptors in dopamine-depleted mice and that this effect can be inhibited by adenosine stimulation ...
https://www.ncbi.nlm.nih.gov/pubmed/1828236?dopt=Abstract
*  8-Polycycloalkyl-1,3-dipropylxanthines as potent and selective antagonists for A1-adenosine receptors. - PubMed - NCBI
8-Polycycloalkyl-1,3-dipropylxanthines as potent and selective antagonists for A1-adenosine receptors.. Shimada J1, Suzuki F, ... Under our structure-activity relationship, the 8-substituent of xanthine antagonists and the N6-substituent of adenosine ... carbon and the conformationally restricted cyclopentyl moiety into the 8-position of xanthines enhanced the adenosine A1 ... N-ethylcarboxamide). *Animals. *Binding, Competitive. *Cell Membrane/metabolism. *Corpus Striatum/metabolism ...
https://www.ncbi.nlm.nih.gov/pubmed/1548682
*  Compound Information Page
2-[[4-(2-Carboxyethyl)phenylethyl]amino]adenosine-5'-N-ethylcarboxamide Hydrochloride; 2-p-(2-Carboxyethyl)phenethylamino-5'-N- ... a new class of highly selective adenosine A2 receptor ligands, J. Med. Chem., 33, 1914-1924 (1990).. ...
https://nimh-repository.rti.org/infosheet.cfm?rec=200411191230580360
*  Adenosine Receptor Agonist Increases Plasma Homocysteine | Leaders in Pharmaceutical Business Intelligence (LPBI) Group
N-Ethylcarboxamide-Adenosine Increases Mouse Serum Total Homocysteine Levels, Which Is a Risk Factor for Cardiovascular ... Adenosine Receptor Agonist Increases Plasma Homocysteine Larry H. Bernstein, MD, FCAP, Curator LPBI The Adenosine Receptor ... N-ethylcarboxamide-adenosine (NECA; 0.1 or 0.3 mg/kg body weight) was intraperitoneally administered to mice that had been ... N-ethylcarboxamide-adenosine (NECA) increased serum glucose levels and the expression of a glucogenic enzyme (glucose 6- ...
https://pharmaceuticalintelligence.com/2015/11/17/adenosine-receptor-agonist-increases-plasma-homocysteine/
*  Purinergic P1 Receptors - Adenosine Receptor Summary | CureHunter Mobile
N-ethylcarboxamide) (NECA) Show All ,, Therapies Related to Purinergic P1 Receptors. * Intravenous Infusions ... Also Known As: Adenosine Receptor; Purinergic P1 Receptor; Adenosine Receptors; Receptors, Adenosine; Receptors, Purinergic P1 ... Purinergic P1 Receptors (Adenosine Receptor) Summary Description: A class of cell surface receptors that prefer ADENOSINE to ... Reperfusion Injury : 5 outcomes 9 studies in 67 results * Parkinson Disease (Parkinson's Disease) : 5 outcomes 6 studies in 40 ...
http://www.curehunter.com/m/keywordSummaryD018047.do
*  Adenosine-Stimulated Atrial Natriuretic Peptide Release Through A1 Receptor Subtype | Hypertension
A relationship between adenosine and the cardiac hormone ANP is not fully studied despite the existence of adenosine receptors and their effects in the heart. Our study has revealed that adenosine increases an ANP release with negative inotropism via stimulation of A1 receptor subtype and that cellular cAMP level regulates the ANP release.. Adenosine is well known as a physiological regulator of tissue function by increasing the energy supply and decreasing the energy demand. Adenosine also exerts a protective role against ischemic injury. In addition to cardioprotective effects, adenosine inhibits a release of vasopressor hormones. These hormonal effects may be expected to exert beneficial effects on the overloaded heart. We found that adenosine increases the ANP release directly from beating atria with negative inotropism. Our results agree with other reports that ...
http://hyper.ahajournals.org/content/46/6/1381
*  NAVER Academic | Physiological and pathophysiological roles of adenosine
Adenosine is a candidate sleep substance. It can be both a distress signal of importance in pathology and a physiological regulator. Key factors in determining which of these possibilities pertain are: (i) the number of receptors expressed, and (ii) the mechanisms that establish extracellular adenosine levels. The roles of adenosine are studied by means of antagonists and/or animals (mostly mice) with targeted deletions of receptors or enzymes involved in adenosine metabolism. Whereas adaptive changes in the genetically modified mice can occur for the physiologically important effects, such adaptive changes are less likely to occur in situations where adenosine acts as a distress signal. The relevance to sleep will be covered only in general terms in this review and will be covered in other contributions to this volume.
http://academic.naver.com/article.naver?doc_id=179726312