TY - JOUR. T1 - Protein phosphorylation in primary astrocyte cultures treated with and without dibutyryl cyclic AMP. AU - Neary, Joseph T.. AU - Gutierrez, Maria del Pilar. AU - Norenberg, Luz Oliva B.. AU - Norenberg, Michael D.. PY - 1987/4/28. Y1 - 1987/4/28. N2 - Protein phosphorylation was investigated in primary rat astrocyte cultures treated with and without dibutyryl cyclic AMP. Astrocytes maintained in dibutyryl cyclic AMP for several weeks displayed increased phosphate incorporation in 5 protein bands (55, 52, 45, 43 and 28 kDa) while incorporation in one band (42 kDa) was decreased. Phosphate incorporation in several other protein bands was unchanged. Calcium-dependent phosphate incorporation was also altered by prior exposure of the cells to dibutyryl cyclic AMP: addition of calcium to broken cell preparations resulted in increased incorporation in 75, 53 and 52 kDa while decreased incorporation occurred in 100 kDa. These differences in protein phosphorylation may be related to the ...
DYMPNA M. P. MORROW, MICHAEL P. RYAN, HUGH Mc GLYNN; Downregulation of intracellular cyclic AMP levels by tumour promoting agents. Biochem Soc Trans 1 February 1997; 25 (1): 148S. doi: https://doi.org/10.1042/bst025148s. Download citation file:. ...
Glial fibrillary acidic protein (GFA) expression was induced in rat C6 glioma in chemically defined medium by the addition of N6,O2-dibutyryl cyclic AMP (dbcAMP). Induction was dependent on the increase in intracellular cyclic AMP (cAMP), which was linearly correlated with added dbcAMP. Contrary to GFA mRNA synthesis, which can be obtained by cAMP-dependent and -independent pathways, translation of mRNA into GFA was observed only above a cellular cAMP concentration of approximately 0.2 fmol/cell. dbcAMP stimulation did not affect the vimentin concentration, which remained at a low level, but changed the cellular morphology from a bipolar to a stellate shape. A similar morphological change was observed after stimulation of C6 with lipopolysaccharide (LPS). However, LPS did not significantly increase the intracellular concentration of cAMP and the LPS-induced mRNA was not translated into GFA. Our results indicate that GFA synthesis is regulated at the mRNA level and at the translational level and ...
1. Cyclic AMP-stimulated protein kinase activity phosphorylating intrinsic substrates in preparations of synaptic-membrane fragments from ox cerebral cortex was examined in relation to (a) the content of membrane-bound Ca2+in the preparations and (b) added Ca2+in the assay medium. 2. Centrifugal washing of synaptic-membrane fragments with buffered ethane dioxybis(ethylamine)tetra-acetate solutions decreased bound Ca2+from 2.8±0.4 (s.d.) to 0.9±0.3nmol/mg of protein. In washed preparations basal protein kinase activity was increased by about 40% and the cyclic AMP-stimulated activity by about 15%. Addition of Ca2+in the concentration range 5-50μm to the assay medium progressively inhibited the kinase activity of the washed preparations; in this range of Ca2+concentration the basal activity was inhibited more than the stimulated activity. 3. In unwashed preparations concentrations of Ca2+above 100μm inhibited the cyclic AMP-stimulated activity more than the basal activity. 4. The inhibitory ...
Innovative genomic test for bucladesine personalised pharmacogenomic analysis to explore how your genes can affect and modulate your response to bucladesine ...
The detector detects the ion as it creates an electric current as it attracts electrons. This creates a mass spectra showing the mass to charge ratio (m/z). This shows the abundance of each isotope. There are also ghost results - this is when a +2 ion is detected and due to its higher charge this means it is much lower than the other detections ...
TY - JOUR. T1 - Immunocytochemical expression of human muscle cell p75 neurotrophin receptor is down-regulated by cyclic adenosine 3,5-monophosphate. AU - Baron, Pierluigi. AU - Scarpini, Elio. AU - Pizzul, Silvia. AU - Zotti, Fabrizio. AU - Conti, Giancarlo. AU - Pleasure, David E. AU - Scarlato, Guglielmo. PY - 1997/10/3. Y1 - 1997/10/3. N2 - To investigate whether the immunocytochemical expression of low affinity neurotrophin receptor (p75) in human muscle is modulated by increased levels of intracellular cyclic adenosine 3,5-monophoshate (cAMP), human cultured myogenic cells were treated with cAMP analogues dibutyryl cAMP (dbcAMP 0.5-1 mM) and 8-bromo cAMP (1 mM) or the adenylate cyclase activator forskolin (10- 100 μM). Cultures were processed for indirect immunofluorescence microscopy using an anti-human p75 mAb. The treatment of cultured muscle cells with cAMP analogues or forskolin for two days induced a decrease of immunoreactivity for p75 and a reduction of both myotube formation ...
TY - JOUR. T1 - Contribution of stored rat growth hormone to restoration of depleted rat pituitary immediate release pools. AU - Stachura, M. E.. AU - Tyler, J. M.. PY - 1990/1/1. Y1 - 1990/1/1. N2 - Stored rat pituitary growth hormone (GH) is functionally divided into immediately releasable and more stable compartments. These observations are consistent with either intracellular hormone compartmentalization within cells of a functionally homogeneous somatotroph population or summed responses from a heterogeneous population of functionally specialized cell subgroups. We investigated the pituitarys ability to recruit stored rGH to replenish depleted immediate release pools. We used perifused pituitary fragments whose stored rGH was labeled during pre-incubation in the presence of [3H] leucine. Initial immediate release pool depletion was accomplished by continuous exposure to combined 21 mM potassium ion (K+) and 1 mM dibutyryl cyclic AMP (dbcAMP). During a subsequent perifusion period in the ...
Juurlink, B H.; Hertz, L; and Fedoroff, S, Effects of high serum levels, dibutyryl cyclic amp and hydrocortisone on glutamine synthetase activity in primary mouse astroglial cultures. Abstr. (1979). Subject Strain Bibliography 1979. 1485 ...
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Supplementary MaterialsVideo S1. with ER. mmc4.mp4 (2.6M) GUID:?C82852C9-015D-4E49-90EA-F519F399A2BB Video S4. Dynamic Lysosomes Preferentially Linger at IP3R1 Puncta: Example 1, Linked to Shape?4 TIRFM video (acquisition 0.3 fps, displayed at 5 …. ...
an enzyme that phosphorylates target proteins in response to a rise in intracellular cyclic AMP. See cyclic AMP‐dependent protein
Looking for online definition of cyclic adenosine monophosphate (cyclic AMP, cAMP, 3',5'-cAMP) in the Medical Dictionary? cyclic adenosine monophosphate (cyclic AMP, cAMP, 3',5'-cAMP) explanation free. What is cyclic adenosine monophosphate (cyclic AMP, cAMP, 3',5'-cAMP)? Meaning of cyclic adenosine monophosphate (cyclic AMP, cAMP, 3',5'-cAMP) medical term. What does cyclic adenosine monophosphate (cyclic AMP, cAMP, 3',5'-cAMP) mean?
To test whether angiotensinogen might be targeted to dense core secretory granules in cells containing a regulated secretory pathway, we expressed rat angiotensinogen in AtT-20 cells, a mouse pituitary cell line that has the demonstrated ability to correctly sort proteins to the constitutive or regulated pathway. We compared the pattern of secretion of angiotensinogen with that of endogenous adrenocorticotropin hormone, which is secreted by AtT-20 cells through the regulated pathway. When cells were incubated for 5 hours with dibutyryladenosine cyclic monophosphate or KCl, adrenocorticotropin hormone secretion was significantly higher than control, whereas monensin had no effect. In contrast, angiotensinogen secretion was markedly reduced by monensin, but no stimulation was observed with dibutyryladenosine cyclic monophosphate or KCl. These results make it unlikely that angiotensinogen could be cotargeted with active renin in the dense core granules of the regulated pathway. Alternative ...
Induction of neural differentiation in cultures of undetermined presumptive epidermis from three amphibian species was achieved by the addition of 1 millimolar dibutyryl adenosine 3,5-monophosphate, 8-bromadenosine 3,5-monophosphate, or adenosine C,E-monophosphate together with theophylline. Adenosine 5-monophosphate, adenosine 2,3-monophosphate, dibutyryl guanosine 3,5-monophosphate, and butyrate at 1 millimolar are ineffective. These results suggest that the action of the primary inductor or inductors may be mediated via adenosine 3,5-monophosphate. ...
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Both treatments resulted in improvements in lung function that were sustained throughout the study. As compared with treatment with high-dose budesonide, treatment with low-dose budesonide plus theophylline resulted in greater improvements in forced
ค่ายนี้เป็นค่ายระดับมัธยมศึกษา สำหรับเยาวชนที่สนใจการศึกษาต่อในสาขาชีวเคมี. จัดขึ้นเป็นครั้งแรกเมื่อเดือนมกราคม 2558 โดยนิสิตภาควิชาชีวเคมี คณะวิทยาศาสตร์ จุฬาลงกรณ์มหาวิทยาลัย. ชมมิวสิควิดิโอ What is the pathway? ซึ่งจัดทำขึ้นโดยนิสิตภาควิชาชีวเคมี คณะวิทยาศาสตร์ จุฬาลงกรณ์มหาวิทยาลัย. ...
TY - JOUR. T1 - AMP deaminase and thymidine kinase deficiencies in a mutant mouse S49 cell clone.. AU - Hanson, S.. AU - Ullman, B.. N1 - Copyright: This record is sourced from MEDLINE/PubMed, a database of the U.S. National Library of Medicine. PY - 1989. Y1 - 1989. N2 - From a mutagenized population of wild type S49 cells, a clone was isolated in a single step that possessed functional and biochemical deficiencies in both AMP deaminase and thymidine kinase activities. This mutant cell line, DTB6, was selected in semi-solid medium containing 1mM thymidine and 1mM dibutyryl cyclic AMP. In comparative growth rate experiments, DTB6 cells were considerably less sensitive than parental cells to the growth inhibitory effects of thymidine. In contrast, DTB6 cells were much more sensitive to the cytotoxic effects of adenine and adenosine. The supersensitivity of DTB6 cells toward adenine could be ameliorated by the addition of hypoxanthine to the culture medium. The growth phenotype of the mutant cells ...
Available data indicate that the liver is a target organ for parathyroid hormone (PTH) and that this effect is most likely mediated by PTH-induced calcium entry into hepatocytes. The present study examined the effects of both PTH-(1-84) and its amino-terminal fragment [PTH-(1-34)] on cytosolic calcium concentration ([Ca2+]i) of hepatocytes and explored the cellular pathways that mediate this potential action of PTH. Both moieties of PTH produced a dose-dependent rise in [Ca2+]i, but the effect of PTH-(1-84) was greater (P | 0.01) than an equimolar amount of PTH-(1-34). This effect required calcium in the medium and was totally [PTH-(1-34)] or partially [PTH-(1-84)] blocked by PTH antagonist ([Nle8,18,Tyr34]bPTH-(7-34)-NH2] and by verapamil or nifedipine. Sodium or chloride channel blockers did not modify this effect. 12-O-tetradecanoylphorbol 13-acetate (TPA), an activator of protein kinase C, dibutyryl adenosine 3,5-cyclic monophosphate (DBcAMP), and G protein activator also produced a dose-dependent
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The kinetics for activation of the cyclic adenosine 3′:5′-monophosphate (cyclic AMP)-dependent protein kinase (PKA) and thymidine incorporation into DNA was investigated in epinephrine- and prostaglandin E1 (PGE1)-treated murine P1798 lymphosarcoma cells. A positive correlation between the duration and extent of PKA activation and Accumulation of cyclic AMP and inhibition of thymidine incorporation into DNA was observed with both hormones. Epinephrine and PGE1 elevated intracellular cyclic AMP 34- and 14-fold, respectively. All hormone concentrations which increased cyclic AMP accumulation also promoted inhibition of thymidine incorporation into DNA. In addition, dibutyryl cyclic AMP (50 µm) inhibited thymidine incorporation.. No difference in the kinetics for activation of PKA was observed when cells were treated with µm epinephrine or PGE1. With both agents, 50% PKA activation was observed when intracellular cyclic AMP concentrations were elevated 6.5-fold, or to 9 pmol/106 cells. In the ...
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Cyclic 3,5-adenosine monophosphate modulates vascular endothelial cell migration in vitro.: Using a modified Boyden chamber assay, we have examined the effect
15731-72-3 - UEUPTUCWIHOIMK-RRKCRQDMSA-N - 2-Deoxy-3-adenosine monophosphate - Similar structures search, synonyms, formulas, resource links, and other chemical information.
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Synaptic-membrane fragments from ox cerebral cortex contain basal and cyclic AMP-stimulated protein kinase activity catalysing the phosphorylation of endogenous substrates. Extraction of membrane fragments with Triton X-100 solubilized less than 20% of the kinase activity and left the major part of the endogenous substrates in the insoluble fraction.. ...
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Gandelman, K.Y., S.E. Pfeiffer, and J.H. Carson. Cyclic AMP regulation of P0 glycoprotein and myelin basic protein gene expression in semi-differentiated peripheral neurinoma cell line D6P2T. Development 106.2 (1989): 389-398. Web. 05 April. 2020. ...