Names
Personal names, given or surname, as cultural characteristics, as ethnological or religious patterns, as indications of the geographic distribution of families and inbreeding, etc. Analysis of isonymy, the quality of having the same or similar names, is useful in the study of population genetics. NAMES is used also for the history of names or name changes of corporate bodies, such as medical societies, universities, hospitals, government agencies, etc.
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The interchange of goods or commodities, especially on a large scale, between different countries or between populations within the same country. It includes trade (the buying, selling, or exchanging of commodities, whether wholesale or retail) and business (the purchase and sale of goods to make a profit). (From Random House Unabridged Dictionary, 2d ed, p411, p2005 & p283)
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Scopolamine Hydrobromide
An alkaloid from SOLANACEAE, especially DATURA and SCOPOLIA. Scopolamine and its quaternary derivatives act as antimuscarinics like ATROPINE, but may have more central nervous system effects. Among the many uses are as an anesthetic premedication, in URINARY INCONTINENCE, in MOTION SICKNESS, as an antispasmodic, and as a mydriatic and cycloplegic.
Antitussive Agents
United States Food and Drug Administration
Drug Labeling
Use of written, printed, or graphic materials upon or accompanying a drug container or wrapper. It includes contents, indications, effects, dosages, routes, methods, frequency and duration of administration, warnings, hazards, contraindications, side effects, precautions, and other relevant information.
Protection by imidazol(ine) drugs and agmatine of glutamate-induced neurotoxicity in cultured cerebellar granule cells through blockade of NMDA receptor. (1/11)
This study was designed to assess the potential neuroprotective effect of several imidazol(ine) drugs and agmatine on glutamate-induced necrosis and on apoptosis induced by low extracellular K+ in cultured cerebellar granule cells. Exposure (30 min) of energy deprived cells to L-glutamate (1-100 microM) caused a concentration-dependent neurotoxicity, as determined 24 h later by a decrease in the ability of the cells to metabolize 3-(4,5-dimethythiazol-2-yl)-2,5-diphenyltetrazoliumbromide (MTT) into a reduced formazan product. L-glutamate-induced neurotoxicity (EC50=5 microM) was blocked by the specific NMDA receptor antagonist MK-801 (dizocilpine). Imidazol(ine) drugs and agmatine fully prevented neurotoxicity induced by 20 microM (EC100) L-glutamate with the rank order (EC50 in microM): antazoline (13)>cirazoline (44)>LSL 61122 [2-styryl-2-imidazoline] (54)>LSL 60101 [2-(2-benzofuranyl) imidazole] (75)>idazoxan (90)>LSL 60129 [2-(1,4-benzodioxan-6-yl)-4,5-dihydroimidazole](101)>RX82 1002 (2-methoxy idazoxan) (106)>agmatine (196). No neuroprotective effect of these drugs was observed in a model of apoptotic neuronal cell death (reduction of extracellular K+) which does not involve stimulation of NMDA receptors. Imidazol(ine) drugs and agmatine fully inhibited [3H]-(+)-MK-801 binding to the phencyclidine site of NMDA receptors in rat brain. The profile of drug potency protecting against L-glutamate neurotoxicity correlated well (r=0.90) with the potency of the same compounds competing against [3H]-(+)-MK-801 binding. In HEK-293 cells transfected to express the NR1-1a and NR2C subunits of the NMDA receptor, antazoline and agmatine produced a voltage- and concentration-dependent block of glutamate-induced currents. Analysis of the voltage dependence of the block was consistent with the presence of a binding site for antazoline located within the NMDA channel pore with an IC50 of 10-12 microM at 0 mV. It is concluded that imidazol(ine) drugs and agmatine are neuroprotective against glutamate-induced necrotic neuronal cell death in vitro and that this effect is mediated through NMDA receptor blockade by interacting with a site located within the NMDA channel pore. (+info)Antazoline therapy of recurrent refractory supraventricular arrhythmias--a preliminary report. (2/11)
Seven patients with chronic or recurrent supraventricular tachyarrhythmias were selected for a trial of antazoline therapy because sinus rhythm or a controlled ventricular response could not be achieved with quinidine, procainamide, digitalis or propranolol. Sinus rhythm was established by either intravenous administration of antazoline or direct-current countershock, and has been maintained in all for 4 to 16 months by oral administration of antazoline. Side effects were minor. Antazoline is a sufficiently promising antiarrhythmic agent to warrant large-scale controlled studies. (+info)Imidazoline antagonists of alpha 2-adrenoceptors increase insulin release in vitro by inhibiting ATP-sensitive K+ channels in pancreatic beta-cells. (3/11)
1. Islets from normal mice were used to study the mechanisms by which imidazoline antagonists of alpha 2-adrenoceptors increase insulin release in vitro. 2. Alinidine, antazoline, phentolamine and tolazoline inhibited 86Rb efflux from islets perifused with a medium containing 3 mM glucose, i.e. under conditions where many adenosine 5'-triphosphate (ATP)-sensitive K+ channels are open in the beta-cell membrane. They also reduced the acceleration of 86Rb efflux caused by diazoxide, an opener of ATP-sensitive K+ channels. 3. ATP-sensitive and voltage-sensitive K+ currents were measured in single beta-cells by the whole-cell mode of the patch-clamp technique. Antazoline more markedly inhibited the ATP-sensitive than the voltage-sensitive current, an effect previously observed with phentolamine. Alinidine and tolazoline partially decreased the ATP-sensitive K+ current. 4. The four imidazolines reversed the inhibition of insulin release caused by diazoxide (through opening of ATP-sensitive K+ channels) or by clonidine (through activation of alpha 2-adrenoceptors) in a concentration-dependent manner. Only the former effect correlated with the ability of each drug to increase control insulin release stimulated by 15 mM glucose alone. 5. It is concluded that the ability of imidazoline antagonists of alpha 2-adrenoceptors to increase insulin release in vitro can be ascribed to their blockade of ATP-sensitive K+ channels in beta-cells rather than to their interaction with the adrenoceptor. (+info)Effect of histamine receptor antagonists on aminophylline-induced seizures and lethality in mice. (4/11)
The aim of this study was to evaluate the effects of H(1) (antazoline and astemizole) or H(2) (cimetidine and famotidine) histamine receptor antagonists on the clonic phase, tonic seizures and morality of mice challenged with aminophylline to induce convulsions in mice. Moreover, the total plasma and brain concentrations of theophylline were evaluated. Astemizole (1 mg/kg) did not affect the threshold for aminophylline-induced seizures, but when administered at a dose of 2 mg/kg, it significantly reduced the CD(50) value of aminophylline from 249 mg/kg to 211 mg/kg (p < 0.01). The remaining histamine receptor antagonists studied i.e., antazoline (up to 1 mg/kg), cimetidine (up to 40 mg/kg) and famotidine (up to 10 mg/kg) had no impact on seizure susceptibility in aminophylline-induced convulsions. Furthermore, astemizole (2 mg/kg) decreased latency to the clonic phase of aminophylline-induced convulsions from 51.1 +/- 4.5 to 32.1 +/- 4.3 min (p < 0.01). It is noteworthy that astemizole, a novel H(1) receptor antagonist, did not alter the brain and plasma levels of theophylline, so the existence of pharmacokinetic interactions was excluded. Our results indicate that some interactions between methylxanthines and histamine receptor antagonists may be clinically important since these drugs are usually combined during the treatment of status asthmaticus. (+info)A rapid derivative spectrophotometric method for simultaneous determination of naphazoline and antazoline in eye drops. (5/11)
A zero-crossing first-derivative spectrophotometric method is applied for the simultaneous determination of naphazoline hydrochloride and antazoline phosphate in eye drops. The measurements were carried out at wavelengths of 225 and 252 nm for naphazoline hydrochloride and antazoline phosphate, respectively. The method was found to be linear (r2>0.999) in the range of 0.2-1 microg/ml for naphazoline hydrochloride in the presence of 5 microg/ml antazoline phosphate at 225 nm. The same linear correlation (r2>0.999) was obtained in the range of 1-10 microg/ml of antazoline phosphate in the presence of 0.5 microg/ml of naphazoline hydrochloride at 252 nm. The limit of determination was 0.2 microg/ml and 1 microg/ml for naphazoline hydrochloride and antazoline phosphate, respectively. The method was successfully used for simultaneous analysis of naphazoline hydrochloride and antazoline phosphate in eye drops without any interference from excipients and prior separation before analysis. (+info)Antazoline in the treatment of cardiac arrhythmias. (6/11)
Antazoline was administered in sixty-five episodes of various types of cardiac arrhythmia. A complete suppression of the ectopic beats was achieved in five out of six episodes of premature atrial systoles and in twenty-one of the twenty-four episodes of ventricular premature systoles. Conversion to sinus rhythm was observed in seven out of ten and four out of five episodes of paroxysmal atrial and nodal tachycardia respectively. Six out of ten episodes of ventricular tachycardia were controlled by intravenous therapy. However, the drug proved to be ineffective in cases of atrial fibrillation. The side-effects were few and transitory, consisting of nausea, vomiting and drowsiness. (+info)Clinical efficacy of antazoline in rapid cardioversion of paroxysmal atrial fibrillation--a protocol of a single center, randomized, double-blind, placebo-controlled study (the AnPAF Study). (7/11)
(+info)An analysis of the purinergic component of active muscle vasodilatation obtained by electrical stimulation of the hypothalamus in rabbits. (8/11)
In anaesthetized rabbits, electrical stimulation of the hypothalamus in areas analogous to the defence area in cats produces the 'defence reaction.' This response includes signs of arousal and a large increase in blood flow to skeletal muscle in the hind limb caused by a vasodilatation in the skeletal muscle vasculature. The vasodilatation is a sympathetic response, and it is not dependent upon muscle activity in the hind limb. The muscle vasodilatation is insensitive to alpha-adrenoceptor, beta-adrenoceptor, cholinoceptor and histamine receptor antagonists. Intra-arterial injections of the purinoceptor agonists, adenosine triphosphate (ATP) and adenosine, mimic the vasodilatation produced by electrical stimulation. The P1-purinoceptor blocker, aminophylline, attenuates adenosine-induced vasodilatation, but it does not affect the vasodilatation produced by ATP or hypothalamic stimulation. The P2-purinoceptor blocker, antazoline, attenuates the vasodilatation produced by both ATP and hypothalamic stimulation. Our results suggest that the muscle vasodilatation produced by hypothalamic stimulation is mediated by purinergic nerves which release ATP and act on P2-purinoceptors. (+info)
Antazoline | Article about antazoline by The Free Dictionary
Antazoline | Profiles RNS
Antazoline Phosphate - Drugs.com
Antazoline - brand name list from Drugs.com
antazoline hydrochloride Global Market and Forecast Research : ReportsnReports
Pure Powder Antazoline Phosphate CAS 154-68-7 - Wuhan Yuancheng Gongchuang Technology Co.Ltd - ecplaza.net
Antazoline phosphate manufacturing companies
Antazoline phosphate manufacturing companies
antazoline - oi
eye pain | Symptoms | Sickness Finder
Burmester Pharmatrade GmbH
Burmester Pharmatrade GmbH
Calcium-independent potentiation of insulin release by cyclic AMP in single beta-cells. - Oxford Neuroscience
Bamberger咪唑合成 - 化学慧
Naphazoline | REACH
Discover the naphazoline hydrochloride,chlorphenamine maleate and vitamin B12 eye drops market - WhaTech
adrenergic blocker Vasoconstrictor Naphazoline hydrochloride from wuhan yuancheng pharmaceutical company Manufacturers &...
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Naftazolina (Naphazoline Hydrochloride) Bruschettini
Albalon Liquifilm (Naphazoline) Allergan
October 2019 * Page 2 of 3 * We have answers to all your questions.
Divorcing Exercise this Summer - Green Mountain at Fox Run
Mechanisms of the Stimulation of Insulin Release by Saturated Fatty Acids: A Study of Palmitate Effects in Mouse β-cells |...
Interactions between mitochondrial bioenergetics and cytoplasmic calcium in cultured cerebellar granule cells<...
Naphazoline Hydrochloride and breastfeeding. Are they compatible?
Naphazoline and breastfeeding. Are they compatible?
Fosforibozilaminoimidazolna karboksilaza - Википедија
Allergy eye drops p height - akvo.flypole.ru
clear eyes maximum redness relief active ingredients
Sabinet | Synthesis of Imidazol[1,5-a]indole-1,3-diones from Imidazolidene-2,4-diones
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SelectiveN-methylation of ethyl esters of 3-(1H-imidazol-4-yl)-2-propenoic acid - oatao
Outsourcing-a dental laboratory business model - Dentsply Sirona Implants
Histamine Receptor Antagonists | GreenMedInfo | Toxic Ingredient
Histamine Receptor Antagonists | GreenMedInfo | Toxic Ingredient
Histamine Receptor Antagonists | GreenMedInfo | Toxic Ingredient
ATC code R01 - Wikipedia
Early diagnosis of experimental necrotizing enterocolitis using proton nuclear magnetic resonance<...
Zincfrin a scene is affected with its constituent ergotamine
Wiley: Applied Bayesian Modelling, 2nd Edition - Peter Congdon
Plus it
Histamine Receptor Antagonists Comprising an Azepin Core - Patent application
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A Trial of Dalotuzumab in Combination With Irinotecan Versus Cetuximab and Irinotecan for Participants With Metastatic Rectal...
Alcaftadine - DrugBank
Study of the Clinical and Biological Efficacity of NAAXIA SINE® in Vernal Keratoconjunctivitis - Full Text View -...
Chlorosome - Wikipedia
Changes to employee share schemes briefing to c...
Tetryzoline
To treat allergic conjunctivitis, tetryzoline can be combined in a solution with antazoline. In an overdose, slow heart rate ...
P-type calcium channel
Eliprodil and antazoline are NMDA receptor antagonists and act to block P-type channels. Eliprodil can decrease P-type channel ...
List of MeSH codes (D03)
... antazoline MeSH D03.383.129.308.080 - biotin MeSH D03.383.129.308.090 - bis(4-methyl-1-homopiperazinylthiocarbonyl)disulfide ...
List of drugs: An-Ap
Antagon Antagonate antazoline (INN) antazonite (INN) antelmycin (INN) Antepar Anthra-Derm Anthraforte Anthranol Anthrascalp ...
ATC code R01
Oxymetazoline R01AB08 Tuaminoheptane R01AC01 Cromoglicic acid R01AC02 Levocabastine R01AC03 Azelastine R01AC04 Antazoline ...
C17H19N3
The molecular formula C17H19N3 (molar mass : 265.35 g/mol) may refer to: Acridine orange Antazoline Esmirtazapine Mirtazapine A ...
ATC code R06
... combinations Empty group R06AX01 Bamipine R06AX02 Cyproheptadine R06AX03 Thenalidine R06AX04 Phenindamine R06AX05 Antazoline ...
Ethylenediamine
... and antazoline. The other classes are derivatives of ethanolamine, alkylamine, piperazine, and others (primarily tricyclic and ...
Antazoline
... is a 1st generation antihistamine with anticholinergic properties used to relieve nasal congestion and in eye drops ... To treat allergic conjunctivitis, antazoline can be combined in a solution with tetryzoline. The drug is a Histamine H1 ...
Captodiame
... (INN), also known as captodiamine, is an antihistamine sold under the trade names Covatine, Covatix, and Suvren which is used as a sedative and anxiolytic. The structure is related to diphenhydramine.[1] A 2004 study suggested captodiame may be helpful in preventing benzodiazepine withdrawal syndrome in people discontinuing benzodiazepine treatment.[1] In addition to its actions as an antihistamine, captodiamine has been found to act as a 5-HT2C receptor antagonist and σ1 receptor and D3 receptor agonist.[2] It produces antidepressant-like effects in rats.[2] However, captodiamine is unique among antidepressant-like drugs in that it increases brain-derived neurotrophic factor (BDNF) levels in the hypothalamus but not in the frontal cortex or hippocampus.[2] This unique action may be related to its ability to attenuate stress-induced anhedonia and corticotropin-releasing factor (CRF) signaling in the hypothalamus.[2] ...
Decongestant
Antazoline. *Thonzylamine). *mast cell stabilizer (some are also antihistamines) (Cromoglicic acid. *Nedocromil ...
Ranitidine
... was first prepared as AH19065 by John Bradshaw in the summer of 1977 in the Ware research laboratories of Allen & Hanburys, part of the Glaxo organization.[36][37] Its development was a response to the first in class histamine H2 receptor antagonist, cimetidine, developed by Sir James Black at Smith, Kline and French, and launched in the United Kingdom as Tagamet in November 1976. Both companies would eventually become merged as GlaxoSmithKline following a sequence of mergers and acquisitions starting with the integration of Allen & Hanbury's Ltd and Glaxo to form Glaxo Group Research in 1979, and ultimately with the merger of Glaxo Wellcome and SmithKline Beecham in 2000. Ranitidine was the result of a rational drug-design process using what was by then a fairly refined model of the histamine H2 receptor and quantitative structure-activity relationships. Glaxo refined the model further by replacing the imidazole ring of cimetidine with a furan ring with a nitrogen-containing ...
Oxmetidine
Text is available under the Creative Commons Attribution-ShareAlike License; additional terms may apply. By using this site, you agree to the Terms of Use and Privacy Policy. Wikipedia® is a registered trademark of the Wikimedia Foundation, Inc., a non-profit organization ...
Loratadine
As of 2017 brands included: Actalor, Actidin, Aerotina, Alaspan, Alavert, Albatrina, Alerdina, Alerfast, Alergan, Alergiano, Alergiatadina, Alergin Ariston, Alergipan, Alergit, Alergitrat L, Aleric Lora, Alermuc, Alernitis, Alerpriv, Alertadin, Alertine, Aleze, Algac, Algecare, Algistop, Alledryl, Aller-Tab, Allerfre, Allerget, Allergex Non Drowsy, Allergyx, Allerhis, Allernon, Allerta, Allertyn, Allohex, Allor, Allorat, Alloris, Alor, Analor, Anhissen, Anti-Sneeze, Antial, Antil, Antimin, Ao Hui Feng, Ao Mi Xin, Ao Shu, Ardin, Atinac, Avotyne, Axcel Loratadine, Bai Wei Le, Bang Nuo, Bedix, Belodin, Benadryl, Besumin, Bi Sai Ning, Bi Yan Tong, Biliranin, Biloina, Biolorat, Bollinol, Boots Hayfever Relief, Boots Hooikoortstabletten, Boots Once-a-Day Allergy Relief, Carin, Carinose, Chang Ke, Civeran, Clara, Claratyne, Clarid, Clarihis, Clarihist, Clarilerg, Clarinese, Claritin, Claritine, Clarityne, Clarityne SP, Clarotadine, Clatatin, Clatine, Clear-Atadine, Clear-Atadine Children's, Clistin, ...
Mesoridazine
... (Serentil) is a piperidine neuroleptic drug belonging to the class of drugs called phenothiazines, used in the treatment of schizophrenia. It is a metabolite of thioridazine. The drug's name is derived from the methylsulfoxy and piperidine functional groups in its chemical structure. It has central antiadrenergic, antidopaminergic, antiserotonergic and weak muscarinic anticholinergic effects. Serious side effects include akathisia, tardive dyskinesia and the potentially fatal neuroleptic malignant syndrome. Mesoridazine was withdrawn from the United States market in 2004 due to dangerous side effects, namely irregular heart beat and QT-prolongation of the electrocardiogram.[1] It currently appears to be unavailable worldwide. ...
Phenyltoloxamine
... is widely used in preparations as an enhancing agent for some analgesics and antitussives (acetaminophen, dihydrocodeine, codeine, hydrocodone). It is widely used in certain parts of the world as cough suppressant usually with codeine, and sometimes by itself or in addition to dextromethorphan as it, like diphenhydramine, possesses antitussive action of its own and is particularly useful in semi-productive coughs because of its moderate drying action. Phenyltoloxamine has analgesic and anti-spasmodic properties of its own[citation needed] and is used in combination with paracetamol, aspirin and other salicylates and other drugs in proprietary preparations available over the counter for backache, muscle strains and similar conditions. In this respect, it is similar to a closely related antihistamine, orphenadrine, and both drugs are very closely related to diphenhydramine and to doxylamine, the latter of which is the active ingredient in NyQuil and many other cough ...
Histidine
When both imidazole ring nitrogens are protonated, their 15N chemical shifts are similar (about 200 ppm, relative to nitric acid on the sigma scale, on which increased shielding corresponds to increased chemical shift). NMR shows that the chemical shift of N1-H drops slightly, whereas the chemical shift of N3-H drops considerably (about 190 vs. 145 ppm). This indicates that the N1-H tautomer is preferred, it is presumed due to hydrogen bonding to the neighboring ammonium. The shielding at N3 is substantially reduced due to the second-order paramagnetic effect, which involves a symmetry-allowed interaction between the nitrogen lone pair and the excited π* states of the aromatic ring. As the pH rises above 9, the chemical shifts of N1 and N3 become approximately 185 and 170 ppm. An entirely deprotonated form of the imidazole ring, the imidazolate ion, would be formed only above a pH of 14, and is therefore not physiologically relevant. This change in chemical shifts can be explained by the ...
Trifluoperazine
Brand names include Eskazinyl, Eskazine, Jatroneural, Modalina, Stelazine, Terfluzine, Trifluoperaz, Triftazin. In the United Kingdom and some other countries, trifluoperazine is sold and marketed under the brand 'Stelazine'. The drug is sold as tablet, liquid and 'Trifluoperazine-injectable USP' for deep intramuscular short-term use. GP studying pharmacological data has indicated cases of neck vertebrae irreversible fusing leading to NHS preparations being predominantly of the liquid form trifluoperazine as opposed to the tablet form as in Stela zine etc. In the past, trifluoperazine was used in fixed combinations with the MAO inhibitor (antidepressant) tranylcypromine (tranylcypromine/trifluoperazine) to attenuate the strong stimulating effects of this antidepressant. This combination was sold under the brand name Jatrosom N. Likewise a combination with amobarbital (potent sedative/hypnotic agent) for the amelioration of psychoneurosis and insomnia existed under the brand name Jalonac. In ...
Terfenadine
In the United States, Seldane was brought to market in 1985 as the first nonsedating antihistamine for the treatment of allergic rhinitis.[1][4] In June 1990, evidence of serious ventricular arrhythmias among those taking Seldane prompted the FDA to issue a report on the risk factors associated with concomitant use of the drug with macrolide antibiotics and ketoconazole.[1] Two months later, the FDA required the manufacturer to send a letter to all physicians, alerting them to the problem; in July 1992, the existing precautions were elevated to a black box warning[1] and the issue attracted mass media attention in reports that people with liver disease or who took ketoconazole, an antifungal agent, or the antibiotic erythromycin, could suffer cardiac arrhythmia if they also took Seldane.[4] In January 1997, the same month when the U.S. Food and Drug Administration (FDA) had earlier approved a generic version of Seldane made by IVAX Corporation of Miami, the FDA recommended terfenadine-containing ...
Sufotidine
... (INN,[1] USAN, codenamed AH25352) is a long-acting competitive H2 receptor antagonist which was under development as an antiulcerant by Glaxo (now GlaxoSmithKline).[2] It was planned to be a follow-up compound to ranitidine (Zantac).[3] When taken in doses of 600 mg twice daily it induced virtually 24-hour gastric anacidity[4] thus closely resembling the antisecretory effect of the proton pump inhibitor omeprazole.[5] Its development was terminated in 1989[6] from phase III clinical trials based on the appearance of carcinoid tumors in long-term toxicity testing in rodents.[7] ...
Bisulepin
Polívka, Zdeněk; Rajšner, Miroslav; Metyš, Jan; Holubek, Jiří; Svátek, Emil; Ryska, Miroslav; Protiva, Miroslav (1983). "Antiaminic agents derived from thieno[2,3-c]-2-benzothiepin: 4-(1-Methyl-4-piperidylidene)-4,9-dihydrothieno[2,3-c]-2-benzothiepin and some related compounds". Collection of Czechoslovak Chemical Communications. 48 (2): 623-641. doi:10.1135/cccc19830623 ...
Ipratropium bromide
Antazoline. *Thonzylamine). *mast cell stabilizer (some are also antihistamines) (Cromoglicic acid. *Nedocromil ...
GSK-189,254
Medhurst AD, Atkins AR, Beresford IJ, Brackenborough K, Briggs MA, Calver AR, Cilia J, Cluderay JE, Crook B, Davis JB, Davis RK, Davis RP, Dawson LA, Foley AG, Gartlon J, Gonzalez MI, Heslop T, Hirst WD, Jennings C, Jones DN, Lacroix LP, Martyn A, Ociepka S, Ray A, Regan CM, Roberts JC, Schogger J, Southam E, Stean TO, Trail BK, Upton N, Wadsworth G, Wald JA, White T, Witherington J, Woolley ML, Worby A, Wilson DM. GSK189254, a novel H3 receptor antagonist that binds to histamine H3 receptors in Alzheimer's disease brain and improves cognitive performance in preclinical models. Journal of Pharmacology and Experimental Therapeutics. 2007 Jun;321(3):1032-45. PMID 17327487 ...
Methapyrilene
... is an antihistamine and anticholinergic of the pyridine chemical class which was developed in the early 1950s. It was sold under the trade names Co-Pyronil and Histadyl EC.[1] It has relatively strong sedative effects, to the extent that its primary use was as a medication for insomnia rather than for its antihistamine action. Together with scopolamine, it was the main ingredient in Sominex, Nytol, and Sleep-Eze. It also provided the sedative component of Excedrin PM. All of these products were reformulated in the late 1970s when methapyrilene was demonstrated to cause liver cancer in rats when given chronically.[2] ...
Pipofezine
... , sold under the brand name Azafen or Azaphen, is an antidepressant approved in Russia for the treatment of depression.[1][2][3][4] It was introduced in the late 1960s and is still used today.[5][6] Pipofezine has been shown to act as a potent inhibitor of the reuptake of serotonin.[7][8] In addition to its antidepressant action, pipofezine has sedative effects as well, suggesting antihistamine activity.[4] Other properties such as anticholinergic or antiadrenergic actions are less clear but are likely.[citation needed] ...
Cinnarizine
It acts by interfering with the signal transmission between vestibular apparatus of the inner ear and the vomiting centre of the hypothalamus by limiting the activity of the vestibular hair cells which send signals about movement.[10] The disparity of signal processing between inner ear motion receptors and the visual senses is abolished, so that the confusion of brain whether the individual is moving or standing is reduced. Vomiting in motion sickness could be a physiological compensatory mechanism of the brain to keep the individual from moving so that it can adjust to the signal perception, but the true evolutionary reason for this malady is currently unknown.[11] When prescribed for balance problems and vertigo, cinnarizine is typically taken two or three times daily depending on the amount of each dose and when used to treat motion sickness, the pill is taken at least two hours before travelling and then again every four hours during travel.[12] However, a recent 2012 study comparing the ...
Loratadine
As of 2017, loratadine was available under many brand names and dosage forms worldwide, including several combination drug formulations with pseudoephedrine, paracetamol, betamethasone, ambroxol, salbutamol, phenylephrine, and dexamethasone.[25] As of 2017[update] brands included: Actalor, Actidin, Aerotina, Alaspan, Alavert, Albatrina, Alerdina, Alerfast, Alergan, Alergiano, Alergiatadina, Alergin Ariston, Alergipan, Alergit, Alergitrat L, Aleric Lora, Alermuc, Alernitis, Alerpriv, Alertadin, Alertine, Aleze, Algac, Algecare, Algistop, Alledryl, Aller-Tab, Allerfre, Allerget, Allergex Non Drowsy, Allergyx, Allerhis, Allernon, Allerta, Allertyn, Allohex, Allor, Allorat, Alloris, Alor, Analor, Anhissen, Anti-Sneeze, Antial, Antil, Antimin, Ao Hui Feng, Ao Mi Xin, Ao Shu, Ardin, Atinac, Avotyne, Axcel Loratadine, Bai Wei Le, Bang Nuo, Bedix, Belodin, Benadryl, Besumin, Bi Sai Ning, Bi Yan Tong, Biliranin, Biloina, Biolorat, Bollinol, Boots Hayfever Relief, Boots Hooikoortstabletten, Boots ...
Novartis
Spersallerg (antazoline/tetrahydrozoline). Allergic conjunctivitis. Stalevo (carbidopa/levodopa/entacapone). Parkinson's ...
بازدارنده آنزیم - ویکیپدیا، دانشنامهٔ آزاد
Antagonists: ۱st generation: ۴-Methyldiphenhydramine • Alimemazine • Antazoline • Azatadine • Bamipine • Benzatropine ( ...
组氨酸脱羧酶 - 维基百科,自由的百科
Antazoline(英语:Antazoline). *Azatadine(英语:Azatadine). *Bamipine(英语:Bamipine) ...
Antazoline Phosphate - Drugs.com
A list of US medications equivalent to Antazoline Phosphate is available on the Drugs.com website. ... Antazoline Phosphate is a medicine available in a number of countries worldwide. ... Ingredient matches for Antazoline Phosphate. Antazoline. Antazoline Phosphate (BANM) is known as Antazoline in the US. ... Antazoline Phosphate. Antazoline Phosphate may be available in the countries listed below. ...
Antazoline - Wikipedia
Antazoline - brand name list from Drugs.com
Find information on antazoline use, treatment, drug class and molecular formula. ... Lists the various brand names available for medicines containing antazoline. ... Medications containing antazoline:. Multi-ingredient medications containing antazoline:. antazoline/naphazoline ophthalmic. ... Antazoline. Important: The information below refers to medicines available in the United States that contain antazoline. ...
Antazoline - wikidoc
Antazoline is a 1st generation antihistamine that also anticholinergic properties used to relieve nasal congestion and in eye ... Antazoline • Azatadine • Bamipine • Cyproheptadine • Deptropine • Dimebon • Ebastine • Epinastine • Ketotifen • Mebhydrolin • ... Retrieved from "https://www.wikidoc.org/index.php?title=Antazoline&oldid=1084526" ...
Cas 91-75-8,Antazoline | lookchem
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Antazoline Phosphate and Xylometazoline Hydrochloride Ophthalmic Drops
A formulation for preparing Antazoline Phosphate and Xylometazoline Hydrochloride Ophthalmic Drops. Includes ingredients, ... Antazoline Phosphate and Xylometazoline Hydrochloride Ophthalmic Drops. Allen Loyd V Jr Jul/Aug 2010. 336. Buy. ... Related Keywords: Loyd V. Allen Jr., PhD, RPh, formulation, antazoline phosphate, xylometazoline hydrochloride, ophthalmic ... Abstract: A formulation for preparing Antazoline Phosphate and Xylometazoline Hydrochloride Ophthalmic Drops. Includes ...
antazoline hydrochloride Global Market and Forecast Research : ReportsnReports
65 Pages Report] Check for Discount on antazoline hydrochloride Global Market and Forecast Research report by ChemReport. ... The price of antazoline hydrochloride in 2016 Major end users of antazoline hydrochloride Potential users of antazoline ... antazoline hydrochloride Global Market and Forecast Research Table of Contents Part 1: General Information of antazoline ... 2.2 Construction of Industry Chain of antazoline hydrochloride Chapter 3: End User of antazoline hydrochloride List of Tables ...
Antazoline | Article about antazoline by The Free Dictionary
Find out information about antazoline. C17H19N3 A bitter, white, crystalline powder with a melting point of 237-241°C; used as ... antazoline. Also found in: Medical, Wikipedia. antazoline. [an′taz·ə‚lēn] (pharmacology) C17H19N3 A bitter, white, crystalline ... Antazoline , Article about antazoline by The Free Dictionary https://encyclopedia2.thefreedictionary.com/antazoline ... 5% phenol, portwine, quinine, urethane, 3% STDS, ethanolamine oleate, talc, antazoline, polidacanol and of late tetracycline ...
Antazoline HCl
Antazoline | Profiles RNS
"Antazoline" is a descriptor in the National Library of Medicines controlled vocabulary thesaurus, MeSH (Medical Subject ... This graph shows the total number of publications written about "Antazoline" by people in this website by year, and whether " ... Below are the most recent publications written about "Antazoline" by people in Profiles. ...
Pure Powder Antazoline Phosphate CAS 154-68-7 - Wuhan Yuancheng Gongchuang Technology Co.Ltd - ecplaza.net
Antazoline Phosphate
... contains not less than 98.0 percent and not more than 101.0 percent of C17H19N3·H3PO4, calculated on the ... Standard solutions Dissolve USP Antazoline Phosphate RS in methanol, and mix to obtain a solution having a known concentration ... Assay Dissolve about 750 mg of Antazoline Phosphate, accurately weighed, in 50 mL of glacial acetic acid, and titrate with 0.1 ... Test solution Dissolve an accurately weighed quantity of Antazoline Phosphate in methanol to obtain a solution containing 10 mg ...
Antazoline phosphate | VWR
Antazoline
... Systematic (IUPAC) name N-(4,5-dihydro-1H-imidazol-2-ylmethyl)-N-(phenylmethyl)aniline Identifiers CAS ... Antazoline is an antihistamine used to relieve nasal congestion and in eye drops, usually in combination with naphazoline, to ... Antazoline • Azatadine • Bamipine • Cyproheptadine • Deptropine • Dimebon • Ebastine • Epinastine • Ketotifen • Mebhydrolin • ... It uses material from the Wikipedia article "Antazoline". A list of authors is available in Wikipedia. ...
antazoline - oi
P2697Utility of antazoline for cardioversion of recent onset atrial fibrillation in patients with a history of myocardial ... 2880Impact of antazoline on electrophysiologic properties of atrial muscle and conduction system of the heart ... Efficacy and safety of antazoline in the rapid cardioversion of paroxysmal atrial fibrillation (the AnPAF Study) ...
Antazoline Phosphate | Biodiscovery
Antazoline phosphate manufacturing companies
Antazoline | World eBook Library | Read eBooks online
Antazoline | histamine H1 receptors antagonist | CAS#91-75-8 | 154-68-7 | MedKoo
Antazoline is an ethylenediamine derivative with histamine H1 antagonistic and sedative properties. Antazoline antagonizes ... Antazoline is a 1st generation antihistamine with also anticholinergic properties used to relieve nasal congestion and in eye ... Antazoline is an ethylenediamine derivative with histamine H1 antagonistic and sedative properties. Antazoline antagonizes ... Name: Antazoline CAS#: 91-75-8 (free base) Chemical Formula: C17H19N3 Exact Mass: 265.1579 Molecular Weight: 265.35 Elemental ...
cholinergic antagonist (CHEBI:48873)
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Tranylcypromine (Oral Route) Before Using - Mayo Clinic
Although certain medicines should not be used together at all, in other cases two different medicines may be used together even if an interaction might occur. In these cases, your doctor may want to change the dose, or other precautions may be necessary. When you are taking this medicine, it is especially important that your healthcare professional know if you are taking any of the medicines listed below. The following interactions have been selected on the basis of their potential significance and are not necessarily all-inclusive.. Using this medicine with any of the following medicines is not recommended. Your doctor may decide not to treat you with this medication or change some of the other medicines you take.. ...
Bupropion (Oral Route) Side Effects - Mayo Clinic
Check with your doctor before using this medicine with alcohol or other medicines that affect the central nervous system (CNS). The use of alcohol or other medicines that affect the CNS with bupropion may worsen the side effects of this medicine, such as dizziness, poor concentration, drowsiness, unusual dreams, and trouble with sleeping. Some examples of medicines that affect the CNS are antihistamines or medicine for allergies or colds, sedatives, tranquilizers, or sleeping medicines, medicine for depression, medicine for anxiety, prescription pain medicine or narcotics, medicine for attention deficit and hyperactivity disorder, medicine for seizures or barbiturates, muscle relaxants, or anesthetics, including some dental anesthetics. Bupropion may cause some people to be agitated, irritable, or display other abnormal behaviors. It may also cause some people to have suicidal thoughts and tendencies, or to become more depressed. Make sure the doctor knows if you have trouble sleeping, get upset ...
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Phosphate10
- Antazoline Phosphate may be available in the countries listed below. (drugs.com)
- Antazoline Phosphate (BANM) is known as Antazoline in the US. (drugs.com)
- In the same systematic review, 9 RCTs with 313 patients compared topical antihistamines (levocabastine, azelastine hydrochloride, emedastine, and antazoline phosphate) with placebo. (thefreedictionary.com)
- Antazoline Phosphate contains not less than 98.0 percent and not more than 101.0 percent of C 17 H 19 N 3 ·H 3 PO 4 , calculated on the dried basis. (drugfuture.com)
- Standard solutions Dissolve USP Antazoline Phosphate RS in methanol, and mix to obtain a solution having a known concentration of 0.10 mg per mL. (drugfuture.com)
- Test solution Dissolve an accurately weighed quantity of Antazoline Phosphate in methanol to obtain a solution containing 10 mg per mL. (drugfuture.com)
- Antazoline phosphate is a histamine H₁-receptor antagonist and is used in eye-drops (treatment of conjunctivitis etc). (biodiscovery.eu)
- Listing your company for Antazoline phosphate allows buyers to find your information through our directory pages which appear in the top positions when a search is conducted in Google, Yahoo! (poulvet.com)
- Combination of antazoline phosphate & naphazoline HCl in soln with polyvinyl alcohol, edetate sodium & benzalkonium chloride. (nih.gov)
- Antihistamine eye drops, such as over-the-counter antazoline phosphate (Vasocon-A) or prescription olopatadine ophthalmic (Patanol) may reduce swelling or itching. (aspirus.org)
Hydrochloride5
- We provide independent and unbiased information on manufacturers, prices, production news and consumers for the global and regional (North America, Asia and Europe) market of antazoline hydrochloride. (reportsnreports.com)
- Antazoline hydrochloride can be also produced. (biodiscovery.eu)
- 3: Wang R, Chu Y, Li X, Wan B, Yu T, Wang L, Hao L, Guo M. Determination of antazoline hydrochloride in rat plasma and excreta by reversed-phase ion-pair chromatography and its application to pharmacokinetics. (medkoo.com)
- 4: Li X, Chu Y, Ke Y, Wang L, Yu T, Hao L. Determination of antazoline hydrochloride in Beagle dog plasma by HPLC-UV and its application to pharmacokinetics. (medkoo.com)
- Maybe I should refer to some more references, such as antazoline hydrochloride. (biology-online.org)
Antihistamine3
- Antazoline is a 1st generation antihistamine with anticholinergic properties used to relieve nasal congestion and in eye drops, usually in combination with naphazoline, to relieve the symptoms of allergic conjunctivitis. (wikipedia.org)
- Topical antihistamine/sympathomimetic combination drops, such as antazoline 0. (thefreedictionary.com)
- Independent assortment refers to a cephalosporin ceftazidime plus an antihistamine naphazoline antazoline, a nonsteroidal antiinflammatory drug is administered. (pacoimabeautiful.org)
Drops3
- Sometimes antazoline is called Vasocon a eye drops. (ljseek.com)
- Souri E, Amanlou M, Farsam H, Afshari A (2006) A rapid derivative spectrophotometric method for simultaneous determination of naphazoline and antazoline in eye drops. (springer.com)
- Eye drops containing antazoline and naphazoline are considered safe to use. (wa.gov.au)
Ophthalmic1
- 25% vasocon vasocon-a antazoline-naphazoline ophthalmic ointment shelf life. (fentek-ind.com)
Treat allergic conjunctivitis1
- To treat allergic conjunctivitis, antazoline can be combined in a solution with tetryzoline. (wikipedia.org)
Amphetamine1
- antazoline, as it blocks alongside the amphetamine receptors, stimulates a later reflex activation of the sympathetic system in conscious patients. (ljseek.com)
Tripelennamine2
- Diphenhydramine and doxylamine ii ethylenediamines where x = n, e.G., tripelennamine, mepyramine and antazoline. (cadasb.org)
- Usually, the pill may be the smallest unit of benzylpenicillin necessitates its parenteral administration of diphenhydramine, antazoline, and tripelennamine may cause drowsiness, dizziness, blurring of vision. (dsaj.org)
Histamine2
- Antazoline is an ethylenediamine derivative with histamine H1 antagonistic and sedative properties. (medkoo.com)
- Antazoline antagonizes histamine H1 receptor and prevents the typical allergic symptoms caused by histamine activities on capillaries, skin, mucous membranes, and gastrointestinal and bronchial smooth muscles. (medkoo.com)
Imidazoline1
- Adrenaline-collagen-induced elevation of [TXB 2 ] i in canine platelets was not inhibited by the non-imidazoline α 2 -adrenoceptor agonist xylazine, but was inhibited by α 2 -adrenoceptor antagonists, an imidazoline α 2 -adrenoceptor agonist (naphazoline) and an imidazoline compound (antazoline). (scialert.net)
Refers1
- The information below refers to medicines available in the United States that contain antazoline. (drugs.com)
Article1
- It uses material from the Wikipedia article "Antazoline" . (chemeurope.com)
Found1
- Antazoline is only found in individuals that have taken the drug. (lookchem.com)
Library1
- Antazoline" is a descriptor in the National Library of Medicine's controlled vocabulary thesaurus, MeSH (Medical Subject Headings) . (umassmed.edu)
Major1
- This graph shows the total number of publications written about "Antazoline" by people in this website by year, and whether "Antazoline" was a major or minor topic of these publications. (umassmed.edu)
Naphazoline3
- Determination of Antazoline, Naphazoline. (gazi.edu.tr)
- Safely Buy Vasocon (Antazoline phosphate/naphazoline hydrochloride - non Rx) from Canada Prescriptions Plus. (canadaprescriptionsplus.com)
- Antazoline phosphate/naphazoline HCL (Vasocon-A). Do not use eye drops for allergies if you have an eye infection. (conexao.fm)