Antazoline: An antagonist of histamine H1 receptors.Naphazoline: An adrenergic vasoconstrictor agent used as a decongestant.Names: Personal names, given or surname, as cultural characteristics, as ethnological or religious patterns, as indications of the geographic distribution of families and inbreeding, etc. Analysis of isonymy, the quality of having the same or similar names, is useful in the study of population genetics. NAMES is used also for the history of names or name changes of corporate bodies, such as medical societies, universities, hospitals, government agencies, etc.Research Report: Detailed account or statement or formal record of data resulting from empirical inquiry.Powders: Substances made up of an aggregation of small particles, as that obtained by grinding or trituration of a solid drug. In pharmacy it is a form in which substances are administered. (From Dorland, 28th ed)Commerce: The interchange of goods or commodities, especially on a large scale, between different countries or between populations within the same country. It includes trade (the buying, selling, or exchanging of commodities, whether wholesale or retail) and business (the purchase and sale of goods to make a profit). (From Random House Unabridged Dictionary, 2d ed, p411, p2005 & p283)Directories as Topic: Lists of persons or organizations, systematically arranged, usually in alphabetic or classed order, giving address, affiliations, etc., for individuals, and giving address, officers, functions, and similar data for organizations. (ALA Glossary of Library and Information Science, 1983)Manufactured Materials: Substances and materials manufactured for use in various technologies and industries and for domestic use.Nonprescription Drugs: Medicines that can be sold legally without a DRUG PRESCRIPTION.Pharmacists' Aides: Persons who perform certain functions under the supervision of the pharmacist.Pharmacy: The practice of compounding and dispensing medicinal preparations.Antitussive Agents: Agents that suppress cough. They act centrally on the medullary cough center. EXPECTORANTS, also used in the treatment of cough, act locally.United States Food and Drug Administration: An agency of the PUBLIC HEALTH SERVICE concerned with the overall planning, promoting, and administering of programs pertaining to maintaining standards of quality of foods, drugs, therapeutic devices, etc.Drug Labeling: Use of written, printed, or graphic materials upon or accompanying a drug container or wrapper. It includes contents, indications, effects, dosages, routes, methods, frequency and duration of administration, warnings, hazards, contraindications, side effects, precautions, and other relevant information.Pharmacists: Those persons legally qualified by education and training to engage in the practice of pharmacy.Prescription Drugs: Drugs that cannot be sold legally without a prescription.Self Medication: The self administration of medication not prescribed by a physician or in a manner not directed by a physician.Community Pharmacy Services: Total pharmaceutical services provided to the public through community pharmacies.3,4-Methylenedioxyamphetamine: An amphetamine derivative that inhibits uptake of catecholamine neurotransmitters. It is a hallucinogen. It is less toxic than its methylated derivative but in sufficient doses may still destroy serotonergic neurons and has been used for that purpose experimentally.N-Methyl-3,4-methylenedioxyamphetamine: An N-substituted amphetamine analog. It is a widely abused drug classified as a hallucinogen and causes marked, long-lasting changes in brain serotonergic systems. It is commonly referred to as MDMA or ecstasy.Catecholamines: A general class of ortho-dihydroxyphenylalkylamines derived from tyrosine.Hallucinogens: Drugs capable of inducing illusions, hallucinations, delusions, paranoid ideations, and other alterations of mood and thinking. Despite the name, the feature that distinguishes these agents from other classes of drugs is their capacity to induce states of altered perception, thought, and feeling that are not experienced otherwise.Amphetamines: Analogs or derivatives of AMPHETAMINE. Many are sympathomimetics and central nervous system stimulators causing excitation, vasopressin, bronchodilation, and to varying degrees, anorexia, analepsis, nasal decongestion, and some smooth muscle relaxation.Serotonin Agents: Drugs used for their effects on serotonergic systems. Among these are drugs that affect serotonin receptors, the life cycle of serotonin, and the survival of serotonergic neurons.Deoxyepinephrine: Sympathomimetic, vasoconstrictor agent.Amphetamine: A powerful central nervous system stimulant and sympathomimetic. Amphetamine has multiple mechanisms of action including blocking uptake of adrenergics and dopamine, stimulation of release of monamines, and inhibiting monoamine oxidase. Amphetamine is also a drug of abuse and a psychotomimetic. The l- and the d,l-forms are included here. The l-form has less central nervous system activity but stronger cardiovascular effects. The d-form is DEXTROAMPHETAMINE.Substance Abuse Detection: Detection of drugs that have been abused, overused, or misused, including legal and illegal drugs. Urine screening is the usual method of detection.Serotonergic Neurons: Neurons whose primary neurotransmitter is SEROTONIN.

Protection by imidazol(ine) drugs and agmatine of glutamate-induced neurotoxicity in cultured cerebellar granule cells through blockade of NMDA receptor. (1/11)

This study was designed to assess the potential neuroprotective effect of several imidazol(ine) drugs and agmatine on glutamate-induced necrosis and on apoptosis induced by low extracellular K+ in cultured cerebellar granule cells. Exposure (30 min) of energy deprived cells to L-glutamate (1-100 microM) caused a concentration-dependent neurotoxicity, as determined 24 h later by a decrease in the ability of the cells to metabolize 3-(4,5-dimethythiazol-2-yl)-2,5-diphenyltetrazoliumbromide (MTT) into a reduced formazan product. L-glutamate-induced neurotoxicity (EC50=5 microM) was blocked by the specific NMDA receptor antagonist MK-801 (dizocilpine). Imidazol(ine) drugs and agmatine fully prevented neurotoxicity induced by 20 microM (EC100) L-glutamate with the rank order (EC50 in microM): antazoline (13)>cirazoline (44)>LSL 61122 [2-styryl-2-imidazoline] (54)>LSL 60101 [2-(2-benzofuranyl) imidazole] (75)>idazoxan (90)>LSL 60129 [2-(1,4-benzodioxan-6-yl)-4,5-dihydroimidazole](101)>RX82 1002 (2-methoxy idazoxan) (106)>agmatine (196). No neuroprotective effect of these drugs was observed in a model of apoptotic neuronal cell death (reduction of extracellular K+) which does not involve stimulation of NMDA receptors. Imidazol(ine) drugs and agmatine fully inhibited [3H]-(+)-MK-801 binding to the phencyclidine site of NMDA receptors in rat brain. The profile of drug potency protecting against L-glutamate neurotoxicity correlated well (r=0.90) with the potency of the same compounds competing against [3H]-(+)-MK-801 binding. In HEK-293 cells transfected to express the NR1-1a and NR2C subunits of the NMDA receptor, antazoline and agmatine produced a voltage- and concentration-dependent block of glutamate-induced currents. Analysis of the voltage dependence of the block was consistent with the presence of a binding site for antazoline located within the NMDA channel pore with an IC50 of 10-12 microM at 0 mV. It is concluded that imidazol(ine) drugs and agmatine are neuroprotective against glutamate-induced necrotic neuronal cell death in vitro and that this effect is mediated through NMDA receptor blockade by interacting with a site located within the NMDA channel pore.  (+info)

Antazoline therapy of recurrent refractory supraventricular arrhythmias--a preliminary report. (2/11)

Seven patients with chronic or recurrent supraventricular tachyarrhythmias were selected for a trial of antazoline therapy because sinus rhythm or a controlled ventricular response could not be achieved with quinidine, procainamide, digitalis or propranolol. Sinus rhythm was established by either intravenous administration of antazoline or direct-current countershock, and has been maintained in all for 4 to 16 months by oral administration of antazoline. Side effects were minor. Antazoline is a sufficiently promising antiarrhythmic agent to warrant large-scale controlled studies.  (+info)

Imidazoline antagonists of alpha 2-adrenoceptors increase insulin release in vitro by inhibiting ATP-sensitive K+ channels in pancreatic beta-cells. (3/11)

1. Islets from normal mice were used to study the mechanisms by which imidazoline antagonists of alpha 2-adrenoceptors increase insulin release in vitro. 2. Alinidine, antazoline, phentolamine and tolazoline inhibited 86Rb efflux from islets perifused with a medium containing 3 mM glucose, i.e. under conditions where many adenosine 5'-triphosphate (ATP)-sensitive K+ channels are open in the beta-cell membrane. They also reduced the acceleration of 86Rb efflux caused by diazoxide, an opener of ATP-sensitive K+ channels. 3. ATP-sensitive and voltage-sensitive K+ currents were measured in single beta-cells by the whole-cell mode of the patch-clamp technique. Antazoline more markedly inhibited the ATP-sensitive than the voltage-sensitive current, an effect previously observed with phentolamine. Alinidine and tolazoline partially decreased the ATP-sensitive K+ current. 4. The four imidazolines reversed the inhibition of insulin release caused by diazoxide (through opening of ATP-sensitive K+ channels) or by clonidine (through activation of alpha 2-adrenoceptors) in a concentration-dependent manner. Only the former effect correlated with the ability of each drug to increase control insulin release stimulated by 15 mM glucose alone. 5. It is concluded that the ability of imidazoline antagonists of alpha 2-adrenoceptors to increase insulin release in vitro can be ascribed to their blockade of ATP-sensitive K+ channels in beta-cells rather than to their interaction with the adrenoceptor.  (+info)

Effect of histamine receptor antagonists on aminophylline-induced seizures and lethality in mice. (4/11)

The aim of this study was to evaluate the effects of H(1) (antazoline and astemizole) or H(2) (cimetidine and famotidine) histamine receptor antagonists on the clonic phase, tonic seizures and morality of mice challenged with aminophylline to induce convulsions in mice. Moreover, the total plasma and brain concentrations of theophylline were evaluated. Astemizole (1 mg/kg) did not affect the threshold for aminophylline-induced seizures, but when administered at a dose of 2 mg/kg, it significantly reduced the CD(50) value of aminophylline from 249 mg/kg to 211 mg/kg (p < 0.01). The remaining histamine receptor antagonists studied i.e., antazoline (up to 1 mg/kg), cimetidine (up to 40 mg/kg) and famotidine (up to 10 mg/kg) had no impact on seizure susceptibility in aminophylline-induced convulsions. Furthermore, astemizole (2 mg/kg) decreased latency to the clonic phase of aminophylline-induced convulsions from 51.1 +/- 4.5 to 32.1 +/- 4.3 min (p < 0.01). It is noteworthy that astemizole, a novel H(1) receptor antagonist, did not alter the brain and plasma levels of theophylline, so the existence of pharmacokinetic interactions was excluded. Our results indicate that some interactions between methylxanthines and histamine receptor antagonists may be clinically important since these drugs are usually combined during the treatment of status asthmaticus.  (+info)

A rapid derivative spectrophotometric method for simultaneous determination of naphazoline and antazoline in eye drops. (5/11)

A zero-crossing first-derivative spectrophotometric method is applied for the simultaneous determination of naphazoline hydrochloride and antazoline phosphate in eye drops. The measurements were carried out at wavelengths of 225 and 252 nm for naphazoline hydrochloride and antazoline phosphate, respectively. The method was found to be linear (r2>0.999) in the range of 0.2-1 microg/ml for naphazoline hydrochloride in the presence of 5 microg/ml antazoline phosphate at 225 nm. The same linear correlation (r2>0.999) was obtained in the range of 1-10 microg/ml of antazoline phosphate in the presence of 0.5 microg/ml of naphazoline hydrochloride at 252 nm. The limit of determination was 0.2 microg/ml and 1 microg/ml for naphazoline hydrochloride and antazoline phosphate, respectively. The method was successfully used for simultaneous analysis of naphazoline hydrochloride and antazoline phosphate in eye drops without any interference from excipients and prior separation before analysis.  (+info)

Antazoline in the treatment of cardiac arrhythmias. (6/11)

Antazoline was administered in sixty-five episodes of various types of cardiac arrhythmia. A complete suppression of the ectopic beats was achieved in five out of six episodes of premature atrial systoles and in twenty-one of the twenty-four episodes of ventricular premature systoles. Conversion to sinus rhythm was observed in seven out of ten and four out of five episodes of paroxysmal atrial and nodal tachycardia respectively. Six out of ten episodes of ventricular tachycardia were controlled by intravenous therapy. However, the drug proved to be ineffective in cases of atrial fibrillation. The side-effects were few and transitory, consisting of nausea, vomiting and drowsiness.  (+info)

Clinical efficacy of antazoline in rapid cardioversion of paroxysmal atrial fibrillation--a protocol of a single center, randomized, double-blind, placebo-controlled study (the AnPAF Study). (7/11)

 (+info)

An analysis of the purinergic component of active muscle vasodilatation obtained by electrical stimulation of the hypothalamus in rabbits. (8/11)

In anaesthetized rabbits, electrical stimulation of the hypothalamus in areas analogous to the defence area in cats produces the 'defence reaction.' This response includes signs of arousal and a large increase in blood flow to skeletal muscle in the hind limb caused by a vasodilatation in the skeletal muscle vasculature. The vasodilatation is a sympathetic response, and it is not dependent upon muscle activity in the hind limb. The muscle vasodilatation is insensitive to alpha-adrenoceptor, beta-adrenoceptor, cholinoceptor and histamine receptor antagonists. Intra-arterial injections of the purinoceptor agonists, adenosine triphosphate (ATP) and adenosine, mimic the vasodilatation produced by electrical stimulation. The P1-purinoceptor blocker, aminophylline, attenuates adenosine-induced vasodilatation, but it does not affect the vasodilatation produced by ATP or hypothalamic stimulation. The P2-purinoceptor blocker, antazoline, attenuates the vasodilatation produced by both ATP and hypothalamic stimulation. Our results suggest that the muscle vasodilatation produced by hypothalamic stimulation is mediated by purinergic nerves which release ATP and act on P2-purinoceptors.  (+info)

*ATC code R01

Oxymetazoline R01AB08 Tuaminoheptane R01AC01 Cromoglicic acid R01AC02 Levocabastine R01AC03 Azelastine R01AC04 Antazoline ...

*Antazoline

... is a 1st generation antihistamine with anticholinergic properties used to relieve nasal congestion and in eye drops ... To treat allergic conjunctivitis, antazoline can be combined in a solution with tetryzoline. The drug is a Histamine H1 ...

*P-type calcium channel

Eliprodil and antazoline are NMDA receptor antagonists and act to block P-type channels. Eliprodil can decrease P-type channel ...

*List of MeSH codes (D03)

... antazoline MeSH D03.383.129.308.080 --- biotin MeSH D03.383.129.308.090 --- bis(4-methyl-1-homopiperazinylthiocarbonyl) ...

*List of drugs: An-Ap

Antagon Antagonate antazoline (INN) antazonite (INN) antelmycin (INN) Antepar Anthra-Derm Anthraforte Anthranol Anthrascalp ...

*ATC code R06

... combinations Empty group R06AX01 Bamipine R06AX02 Cyproheptadine R06AX03 Thenalidine R06AX04 Phenindamine R06AX05 Antazoline ...
Antazoline is a first generation antihistaminic agent with chinidin-like properties. When administered intravenously, antazoline exerts a strong antiarrhythmic effect on supraventricular arrhythmia especially on atrial fibrillation (AF) facilitating rapid conversion to sinus rhythm. Despite relative lack of published data antazoline is marketed in Poland and widely used in cardiology wards and emergency rooms due to its efficacy, safety and rapid onset of action within minutes of administration.. To show superiority of antazoline over placebo a sample size of 80 patients was calculated based on following assumptions: two-tailed test, a type I error of 0.01, a power of 90%, efficacy of placebo 5%, efficacy of antazoline 50% and 20% drop-out rate to fulfill the criteria of intention-to-treat analysis. Due to presumed lack of statistical power the secondary end points and safety endpoints will be considered exploratory. ...
Looking for antazoline? Find out information about antazoline. C17H19N3 A bitter, white, crystalline powder with a melting point of 237-241°C; used as an antihistamine Explanation of antazoline
This graph shows the total number of publications written about "Antazoline" by people in this website by year, and whether "Antazoline" was a major or minor topic of these publications ...
Antazoline Phosphate is a medicine available in a number of countries worldwide. A list of US medications equivalent to Antazoline Phosphate is available on the Drugs.com website.
Lists the various brand names available for medicines containing antazoline. Find information on antazoline use, treatment, drug class and molecular formula.
[65 Pages Report] Check for Discount on antazoline hydrochloride Global Market and Forecast Research report by ChemReport. DescriptionWe provide independent and unbiased information on manufacturers, prices, production...
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Hot sale Pure powder Antazoline Phosphate CAS 154-68-7 with best price Our production and management of pharmaceutical raw materials and steroid raw materials and so on sales of products in the long-term practice, we formed a unique market...
Allergis information about active ingredients, pharmaceutical forms and doses by Nakornpatana Pharm, Allergis indications, usages and related health products lists
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Burmester liefert: pharmazeutische Rohstoffe, Wirkstoffe, Wirksubstanzen, Allantoin, PAMBA, Antazoline, Antipyrine, Arabic Gum, Baclofen, Belladonna, Bendazac, Benzbromarone, Benzocaine, Betamethasone, Calcitonin, Calcium ...
Burmester liefert: pharmazeutische Rohstoffe, Wirkstoffe, Wirksubstanzen, Allantoin, PAMBA, Antazoline, Antipyrine, Arabic Gum, Baclofen, Belladonna, Bendazac, Benzbromarone, Benzocaine, Betamethasone, Calcitonin, Calcium ...
How does cyclic AMP potentiate insulin secretion from pancreatic islet beta-cells? This question is fundamental to understanding how hormones such as glucagon, which elevates cAMP, stimulate insulin secretion and so contribute to the normal secretory response of the islet. It is well established that a rise in the cytoplasmic Ca2+ concentration ([Ca2+]i) is essential for insulin secretion and therefore cAMP has been proposed to act by elevating [Ca2+]i. But studies on permeabilized beta-cells indicate that cAMP increases insulin release even when [Ca2+]i is held constant. We have used microfluorimetry and the patch-clamp technique to measure changes simultaneously in Ca2+ currents, [Ca2+]i and exocytosis in a single beta-cell in response to cAMP. We show here that cAMP, through activation of protein kinase A, increases Ca(2+)-influx through voltage-dependent L-type Ca2+ channels, thereby elevating [Ca2+]i and accelerating exocytosis. More importantly, cAMP also promotes insulin release by a direct
Compare prices and print coupons for Naphazoline (Albalon) and other Eye Inflammation and Allergic Conjunctivitis drugs at CVS, Walgreens, and other pharmacies. Prices start at $6.64
This research report scrutinizes the major players in Naphazoline Hydrochloride, Chlorphenamine Maleate and Vitamin B12 Eye Drops market which include Novartis AG, Allergan, Inc., Meda Pharmaceuticals Inc, Bausch & Lomb Inc, Cigna, Similasan Corporation, Visine, Alcon, Viva Opti-Free, Bausch & Lomb, Systane, Rite Aid, Walgreens, Staples, Clear eyes, Refresh, Murine, Tears naturale, Genteal.
2016 Naphazoline Nitrate (CAS 5144-52-5) Industry Market Report Size and Share Published in 2016-08-30 Available for US$ 2800 at Researchmoz.us
DPP-4 inhibitors are oral medicines for people with type 2 diabetes that help control blood sugar levels, especially after eating. After eating, your gut naturally releases hormones-two important ones are GLP-1 and GIP. These hormones increase insulin release to help control blood sugar levels. GLP-1 also decreases glucagon release at meals, to further control blood sugar levels. However, these hormones are quickly broken down in the body by an enzyme called DPP-4. DPP-4 inhibitors like sitagliptin and saxagliptin block DPP-4 from breaking down GLP-1 as quickly so that GLP-1 can have a longer effect in the body.. While DPP-4 inhibitors may be used as an initial choice for a medicine to help lower blood sugar levels, they are mainly being used in combination with other diabetes medicines. This means that these medicines are usually added on when a person is already taking one or two medicines for diabetes, but their sugars are still not well controlled.. Unlike with exenatide and liraglutide, ...
DailyMed provides high quality information about marketed drugs. Drug labeling on this Web site is the most recent submitted to the Food and Drug Administration (FDA) and currently in use; it may include strengthened warnings undergoing FDA review and minor editorial changes ...
Naftazolina information about active ingredients, pharmaceutical forms and doses by Bruschettini, Naftazolina indications, usages and related health products lists
Naphazoline ophthalmic capsules also are formulated with the sodium salt spoon of Allerest eye with drops. My first theory is that a TMJ disorder is causing my blurred vision and…. ...
Naphazoline + phenylephrine + carboxymethylcellulose is used in the treatment of .get complete information about naphazoline + phenylephrine + carboxymethylcellulose including usage, side effects, drug interaction, expert advice along with medicines associated with naphazoline + phenylephrine + carboxymethylcellulose at 1mg.com
TY - JOUR. T1 - Interactions between mitochondrial bioenergetics and cytoplasmic calcium in cultured cerebellar granule cells. AU - Nicholls, David. AU - Vesce, Sabino. AU - Kirk, Liana. AU - Chalmers, Susan. PY - 2003/10. Y1 - 2003/10. N2 - The mitochondrion has moved to the center stage in the drama of the life and death of the neuron. The mitochondrial membrane potential controls the ability of the organelle to generate ATP, generate reactive oxygen species and sequester Ca(2+) entering the cell. Each of these processes interact, and their deconvolution is far from trivial. The cultured cerebellar granule cell provides a model in which knowledge gained from studies on isolated mitochondria can be applied to study the role played by the organelles in the maintenance of Ca(2+) homeostasis in the cell under resting, stimulated and pathophysiological conditions. In particular, mitochondria play a complex role in the response of the neuron to excitotoxic stimulation of NMDA and AMPA-kainate ...
A sympathomimetic with alpha-adrenergic activity. It has a vasoconstrictor effect that reduces mucosal swelling and congestion. Topical nasal use (single dose) or ophthalmological (2-4 times a day). Since the last update we have not found published data in relation to breastfeeding. The small dose and the low plasma absorption of most topical nasal or ophthalmological preparations make transfer into breastmilk in significant amounts unlikely. Do not exceed the recommended dose and time periods in order to avoid undesirable side effects and the possible decrease in milk cited by some authors (Nice 2000) for other similar drugs, although not proven in practice. It is a product which has very little literature and almost none related to pharmacokinetics. As a nasal decongestant, it is discouraged by some authors (Nice 2000), with better known drugs from the same group being preferred (Anderson 2000). Ophthalmic administration is fully compatible with breastfeeding. Absorption can be
A sympathomimetic with alpha-adrenergic activity. It has a vasoconstrictor effect that reduces mucosal swelling and congestion. Topical nasal use (single dose) or ophthalmological (2-4 times a day). Since the last update we have not found published data in relation to breastfeeding. The small dose and the low plasma absorption of most topical nasal or ophthalmological preparations make transfer into breastmilk in significant amounts unlikely. Do not exceed the recommended dose and time periods in order to avoid undesirable side effects and the possible decrease in milk cited by some authors (Nice 2000) for other similar drugs, although not proven in practice. It is a product which has very little literature and almost none related to pharmacokinetics. As a nasal decongestant, it is discouraged by some authors (Nice 2000), with better known drugs from the same group being preferred (Anderson 2000). Ophthalmic administration is fully compatible with breastfeeding. Absorption can be
ADRENOMIMETIC DRUGS: NEW DIAGNOSTIC AND THERAPEUTIC ASPECTS IN BRONCHIAL ASTHMA. V. N. Solopov, I. V. Lunichkina. Summary. It is suggested to use alfa-stimulating effect of naphthyzine and halazoline for pharmacological spirometric testing in evaluating the inflammatory-edematous componert of bronchial obstruction. Those antiedemics combined with standard bronchospasmolytics (beta-2-agonists and cholinolytics) proved effective in arresting episodes of asphyxia. Optimal doses of naphthyzine and halazoline, related side effects have been clarified in case of their addition to selective beta-2-agonists, cholinolytics and combinations thereof. In contrast to nonselective adrenomimetic drugs adrenaline and ephedrine, naphthyzine, halazoline or similar medicines do not produce cardiostimulation this justifying their use in combination with selective bronchospasmolytic berotec, salbutamole, berodual and atrovent.. «Klin. Med» (Msk) 1991, №2, с. 55-58. ...
I had to use eye allergy drops this morning, 45 minutes after I put my contacts in for the day. The drops were Opcon-A (Naphazoline). My pupils have become dilated. SHould I worry? THis has happene...
Hi all I have got some problems, and wonder if there is anybody that can help me out. I have cloned and expressed two plant proteins in E. coli with the size of 70 kDa and 97 kDa respectively. The DNA-sequences encoding the two proteins were individually cloned and their respective proteins expressed in the expression vector pET-24a. This vector provides an optional histidine-tag. The DNA-fragments were inserted in frame with the histidine-tag. Subsequently I managed to express them in inclusion bodies, (with the right size). When trying to purify the 70 kDa protein over a Ni-NTA column under denaturing conditions, the protein was eluted during a low stringency wash procedure with 50 mM imidazol. In the protocol for Qiaexpress system it is stated that proteins containing a histidine-tag will be eluted with higher concentrations of imidazol such as 250 mM. This led me to believe that something might be wrong with my his-tag. I did not fully sequence my fragment but only the ligation junctions to ...
Fosforibozilaminoimidazolna karboksilaza (EC 4.1.1.21, 5-fosforibozil-5-aminoimidazolna karboksilaza, 5-amino-1-ribozilimidazol 5-fosfatna karboksilaza, AIR karboksilaza, 1-(5-fosforibozil)-5-amino-4-imidazolkarboksilatna karboksi-lijaza, ADE2, klasa II PurE, 5-amino-1-(5-fosfo-D-ribozil)imidazol-4-karboksilatna karboksi-lijaza) je enzim sa sistematskim imenom 5-amino-1-(5-fosfo-D-ribozil)imidazol-4-karboksilat karboksi-lijaza (formira 5-amino-1-(5-fosfo-D-ribozil)imidazol).[1][2][3] Ovaj enzim katalizuje sledeću hemijsku reakciju ...
Naphcon eye drops are a kind of eye drop specially for those suffering from red scratchy eyes associated with allergies. These drops get their name from the primary ingredient, Naphazoline. The drops work by decreasing mucus in the eyes from...
Camphor + Menthol + Phenylephrine + Carboxymethylcellulose + Naphazoline is used in the treatment of .Get complete information about Camphor + Menthol + Phenylephrine + Carboxymethylcellulose + Naphazoline including usage, side effects, drug interaction, Expert Advice along with medicines associated with Camphor + Menthol + Phenylephrine + Carboxymethylcellulose + Naphazoline at 1mg.com
This page includes the following topics and synonyms: Ocular Antihistamine, Naphazoline, Vasocon, Naphcon, Epinastine, Elestat, Bepotastine, Bepreve.
Copper and tributyltin hydride catalysed cyclization, through the N-aryl bond formation, of imidazolidine-2,4-diones (11-16, 18) yielded imidazo[1,5-a]indole-1, 3-diones (5-10) in high yields (72-100%). The ease of cyclization was found to be consistent with the normal halogen reactivity and the type of substituents. The highly substituted imidazole-2,4-dione 15 gave brominated 19 and tin incorporated heterocycles 20 when treated with copper bromide and tributyltin hydride, respectively.
This topic contains 13 study abstracts on Histamine Receptor Antagonists indicating they may contribute to Pneumonia, Clostridium Infections, and Acid Reflux
Bupleurum gerardi é uma espécie de planta com flor pertencente à família Apiaceae. A autoridade científica da espécie é All., tendo sido publicada em Auctarium ad Synopsim Methodicam Stirpium Horti Reg. Taurinensis 29. 1773. Trata-se de uma espécie presente no território português, nomeadamente em Portugal Continental. Em termos de naturalidade é nativa da região atrás indicada. Não se encontra protegida por legislação portuguesa ou da Comunidade Europeia. Bupleurum gerardi - Checklist da Flora de Portugal (Continental, Açores e Madeira) - Sociedade Lusitana de Fitossociologia Checklist da Flora do Arquipélago da Madeira (Madeira, Porto Santo, Desertas e Selvagens) - Grupo de Botânica da Madeira Bupleurum gerardi - Portal da Biodiversidade dos Açores Tropicos.org. Missouri Botanical Garden. 4 de outubro de 2014 ...
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ATC code R01 Nasal preparations is a therapeutic subgroup of the Anatomical Therapeutic Chemical Classification System, a system of alphanumeric codes developed by the WHO for the classification of drugs and other medical products. Subgroup R01 is part of the anatomical group R Respiratory system. Codes for veterinary use (ATCvet codes) can be created by placing the letter Q in front of the human ATC code: for example, QR01. National issues of the ATC classification may include additional codes not present in this list, which follows the WHO version. R01AA02 Cyclopentamine R01AA03 Ephedrine R01AA04 Phenylephrine R01AA05 Oxymetazoline R01AA06 Tetryzoline R01AA07 Xylometazoline R01AA08 Naphazoline R01AA09 Tramazoline R01AA10 Metizoline R01AA11 Tuaminoheptane R01AA12 Fenoxazoline R01AA13 Tymazoline R01AA14 Epinephrine R01AA15 Indanazoline R01AB01 Phenylephrine R01AB02 Naphazoline R01AB03 Tetryzoline R01AB05 Ephedrine R01AB06 Xylometazoline R01AB07 Oxymetazoline R01AB08 Tuaminoheptane R01AC01 ...
TY - JOUR. T1 - Early diagnosis of experimental necrotizing enterocolitis using proton nuclear magnetic resonance. AU - Miller, James E.. AU - Whitman, Glenn J.R.. AU - Iozzo, Renato V.. AU - Jacobs, Danny. AU - Ziegler, Moritz M.. PY - 1985/1/1. Y1 - 1985/1/1. N2 - The purpose of this study was (1) to confirm an experimental model of aminophylline-induced necrotizing enterocolitis (NEC); and (2) to determine whether nuclear magnetic resonance (NMR) imaging, based upon proton relaxation values (T1, T2), could detect NEC during its early pathogenesis. Sixty male weanling Lewis rats (avg wt = 75 g) were randomly assigned to one of three experimental groups: (A) superior mesenteric artery (SMA) occlusion (1 min) + aminophylline treatment (40 mg/kg); (B) SMA occlusion; and (C) sham midline laparotomy (control). All surviving animals were sacrificed at 48 hr postoperation and a specimen of ileum was removed for light microscopy (LM), electron microscopy (EM), and NMR analysis. Percentage water ...
Preface xi 1 Bayesian methods and Bayesian estimation 1. 1.1 Introduction 1. 1.1.1 Summarising existing knowledge: Prior densities for parameters 2. 1.1.2 Updating information: Prior, likelihood and posterior densities 3. 1.1.3 Predictions and assessment 5. 1.1.4 Sampling parameters 6. 1.2 MCMC techniques: The Metropolis-Hastings algorithm 7. 1.2.1 Gibbs sampling 8. 1.2.2 Other MCMC algorithms 9. 1.2.3 INLA approximations 10. 1.3 Software for MCMC: BUGS, JAGS and R-INLA 11. 1.4 Monitoring MCMC chains and assessing convergence 19. 1.4.1 Convergence diagnostics 20. 1.4.2 Model identifiability 21. 1.5 Model assessment 23. 1.5.1 Sensitivity to priors 23. 1.5.2 Model checks 24. 1.5.3 Model choice 25. References 28. 2 Hierarchical models for related units 34. 2.1 Introduction: Smoothing to the hyper population 34. 2.2 Approaches to model assessment: Penalised fit criteria, marginal likelihood and predictive methods 35. 2.2.1 Penalised fit criteria 36. 2.2.2 Formal model selection using marginal ...
For eliciting contraction of rabbit aorta, the relative potency of agonists in terms of negative log molar ED50 were: oxymetazoline (8.4) greater than naphazoline (7.95) greater than phenylephrine (7.31) greater than tetrahydrozoline (6.5) greater than tolazoline (5.80). None of the imidazolines, however, produced maximal effects equal to that of phenylephrine. All agonists were directly acting agents. The interactions between oxymetazoline and phentolamine or tolazoline and phentolamine were competitive with pA2 values of 8.1 and 8.0, respectively. Phentolamine with tetrahydrozoline, naphazoline or phenylephrine produced nearly equal KB values. Thus, all the agonists and alpha adrenoceptor blockers must act at a common site in rabbit aorta. As expected, the contraction of rabbit aorta produced by an imidazole histamine was competitively antagonized by the histamine 1 antagonist, chlorpheniramine (K B 7.6 X 10(-9) M). The antagonist failed to block the contraction produced by the imidazolines ...
wherein:the H atom indicated is in the exo position;R41- represents an anion associated with the positive charge of the N atom. R1- may be but is not limited to chloride, bromide, iodide, sulfate, benzene sulfonate and toluene sulfonate;R42 and R43 are independently selected from the group consisting of straight or branched chain lower alkyl groups (having for example from 1 to 6 carbon atoms), cycloalkyl groups (having from 5 to 6 carbon atoms), cycloalkyl-alkyl (having 6 to 10 carbon atoms), heterocycloalkyl (having 5 to 6 carbon atoms) and N or O as the heteroatom, heterocycloalkyl-alkyl (having 6 to 10 carbon atoms) and N or O as the heteroatom, aryl, optionally substituted aryl, heteroaryl, and optionally substituted heteroaryl;R44 is selected from the group consisting of (C1-C6)alkyl, (C3-C12)cycloalkyl, (C3-C7)heterocycloalkyl, (C1-C6)alkyl(C3-C12)cycloalkyl, (C1-C6)alkyl(C3-C7)heterocycloalkyl, aryl, heteroaryl, (C1-C6)alkyl-aryl, (C1-C6)alkyl-heteroaryl, --OR45, --CH2OR45, --CH2OH, ...
Naive Bayes is a simple technique for constructing classifiers: models that assign class labels to problem instances, represented as vectors of feature values, where the class labels are drawn from some finite set. There is not a single algorithm for training such classifiers, but a family of algorithms based on a common principle: all naive Bayes classifiers assume that the value of a particular feature is independent of the value of any other feature, given the class variable. For example, a fruit may be considered to be an apple if it is red, round, and about 10 cm in diameter. A naive Bayes classifier considers each of these features to contribute independently to the probability that this fruit is an apple, regardless of any possible correlations between the color, roundness, and diameter features. For some types of probability models, naive Bayes classifiers can be trained very efficiently in a supervised learning setting. In many practical applications, parameter estimation for naive ...
Cetuximab will be administered intravenously prior to irinotecan at an initial dose of 400 mg/m^2 followed by weekly infusions of 250 mg/m^2. Pre-medication at the discretion of the investigator, such as with a histamine receptor antagonist or corticosteroid, will follow local, or country-specific standard of care ...
Alcaftadine is a H1 histamine receptor antagonist indicated for the prevention of itching associated with allergic conjunctivitis. This drug was approved in July 2010.
A Chlorosome is a photosynthetic antenna complex found in green sulfur bacteria (GSB) and some green filamentous anoxygenic phototrophs (FAP) (Chloroflexaceae, Oscillochloridaceae). They differ from other antenna complexes by their large size and lack of protein matrix supporting the photosynthetic pigments. Green sulfur bacteria are a group of organisms that generally live in extremely low-light environments, such as at depths of 100 metres in the Black Sea. The ability to capture light energy and rapidly deliver it to where it needs to go is essential to these bacteria, some of which see only a few photons of light per chlorophyll per day. To achieve this, the bacteria contain chlorosome structures, which contain up to 250,000 chlorophyll molecules. Chlorosomes are ellipsoidal bodies, in GSB their length varies from 100 to 200 nm, width of 50-100 nm and height of 15 - 30 nm, in FAP the chlorosomes are somewhat smaller. Chlorosome shape can vary between species, with some species containing ...
Federal government MPs have been briefed by an employee share ownership lobby group about the need for changes to the tax treatment of share schemes that impact on the start-up sector. | Strategies for Managing Your Business

Antazoline Phosphate - Drugs.comAntazoline Phosphate - Drugs.com

A list of US medications equivalent to Antazoline Phosphate is available on the Drugs.com website. ... Antazoline Phosphate is a medicine available in a number of countries worldwide. ... Ingredient matches for Antazoline Phosphate. Antazoline. Antazoline Phosphate (BANM) is known as Antazoline in the US. ... Antazoline Phosphate. Antazoline Phosphate may be available in the countries listed below. ...
more infohttps://www.drugs.com/international/antazoline-phosphate.html

Antazoline - brand name list from Drugs.comAntazoline - brand name list from Drugs.com

Find information on antazoline use, treatment, drug class and molecular formula. ... Lists the various brand names available for medicines containing antazoline. ... Medications containing antazoline:. Multi-ingredient medications containing antazoline:. antazoline/naphazoline ophthalmic. ... Antazoline. Important: The information below refers to medicines available in the United States that contain antazoline. ...
more infohttps://www.drugs.com/ingredient/antazoline.html

Antazoline | Profiles RNSAntazoline | Profiles RNS

"Antazoline" is a descriptor in the National Library of Medicines controlled vocabulary thesaurus, MeSH (Medical Subject ... This graph shows the total number of publications written about "Antazoline" by people in this website by year, and whether " ... Below are the most recent publications written about "Antazoline" by people in Profiles. ...
more infohttps://profiles.umassmed.edu/display/123927

Antazoline | Article about antazoline by The Free DictionaryAntazoline | Article about antazoline by The Free Dictionary

Find out information about antazoline. C17H19N3 A bitter, white, crystalline powder with a melting point of 237-241°C; used as ... antazoline. Also found in: Medical, Wikipedia. antazoline. [an′taz·ə‚lēn] (pharmacology) C17H19N3 A bitter, white, crystalline ... Antazoline , Article about antazoline by The Free Dictionary https://encyclopedia2.thefreedictionary.com/antazoline ... 5% phenol, portwine, quinine, urethane, 3% STDS, ethanolamine oleate, talc, antazoline, polidacanol and of late tetracycline ...
more infohttp://encyclopedia2.thefreedictionary.com/antazoline

antazoline hydrochloride Global Market and Forecast Research : ReportsnReportsantazoline hydrochloride Global Market and Forecast Research : ReportsnReports

65 Pages Report] Check for Discount on antazoline hydrochloride Global Market and Forecast Research report by ChemReport. ... The price of antazoline hydrochloride in 2016 Major end users of antazoline hydrochloride Potential users of antazoline ... antazoline hydrochloride Global Market and Forecast Research Table of Contents Part 1: General Information of antazoline ... 2.2 Construction of Industry Chain of antazoline hydrochloride Chapter 3: End User of antazoline hydrochloride List of Tables ...
more infohttp://www.reportsnreports.com/reports/618612-antazoline-hydrochloride-global-market-and-forecast-research.html

Pure Powder Antazoline Phosphate CAS 154-68-7 - Wuhan Yuancheng Gongchuang Technology Co.Ltd - ecplaza.netPure Powder Antazoline Phosphate CAS 154-68-7 - Wuhan Yuancheng Gongchuang Technology Co.Ltd - ecplaza.net

Hot sale Pure powder Antazoline Phosphate CAS 154-68-7 with best price Our production and management of pharmaceutical raw ...
more infohttps://www.ecplaza.net/products/pure-powder-antazoline-phosphate-cas-154_4198699

antazoline - oiantazoline - oi

P2697Utility of antazoline for cardioversion of recent onset atrial fibrillation in patients with a history of myocardial ... 2880Impact of antazoline on electrophysiologic properties of atrial muscle and conduction system of the heart ... Efficacy and safety of antazoline in the rapid cardioversion of paroxysmal atrial fibrillation (the AnPAF Study) ...
more infohttp://oxfordindex.oup.com/view/10.1093/oi/authority.20110803095415882

Antazoline phosphate manufacturing companiesAntazoline phosphate manufacturing companies

We are sorry, there are no companies found in " Antazoline phosphate" Listing your company for Antazoline phosphate allows ... Antazoline phosphate manufacturers and suppliers. Search. Search by Drug Name, Company, CAS, Chem formula, IUPAC Name, Country ...
more infohttp://www.poulvet.com/bulk_drugs/product_companies_india.php?sclid=1722&prefix=Y

Antazoline phosphate manufacturing companiesAntazoline phosphate manufacturing companies

We are sorry, there are no companies found in " Antazoline phosphate" Listing your company for Antazoline phosphate allows ... Antazoline phosphate manufacturers and suppliers. Search. Search by Drug Name, Company, CAS, Chem formula, IUPAC Name, Country ...
more infohttp://www.poulvet.com/bulk_drugs/product_companies_india.php?sclid=1722&prefix=A

Drug Test Kits Cross Reaction Drug ListDrug Test Kits Cross Reaction Drug List

Antazoline sulphate. Otrivine-Antistin®. Nonreactive. Antipyrine. 4-Dimethylaminoantipyrine. Nonreactive. Aripiprazole. Abilify ...
more infohttp://www.drugtestingworld.com/cross-reaction-drug-list-ezp-23.html

Antazoline - wikidocAntazoline - wikidoc

Antazoline is a 1st generation antihistamine that also anticholinergic properties used to relieve nasal congestion and in eye ... Antazoline • Azatadine • Bamipine • Cyproheptadine • Deptropine • Dimebon • Ebastine • Epinastine • Ketotifen • Mebhydrolin • ... Retrieved from "https://www.wikidoc.org/index.php?title=Antazoline&oldid=1084526" ...
more infohttps://www.wikidoc.org/index.php/Antazoline

Antazoline - WikipediaAntazoline - Wikipedia

Antazoline is a 1st generation antihistamine with anticholinergic properties used to relieve nasal congestion and in eye drops ... To treat allergic conjunctivitis, antazoline can be combined in a solution with tetryzoline. The drug is a Histamine H1 ...
more infohttps://en.wikipedia.org/wiki/Antazoline

Antazoline PhosphateAntazoline Phosphate

... contains not less than 98.0 percent and not more than 101.0 percent of C17H19N3·H3PO4, calculated on the ... Standard solutions Dissolve USP Antazoline Phosphate RS in methanol, and mix to obtain a solution having a known concentration ... Assay Dissolve about 750 mg of Antazoline Phosphate, accurately weighed, in 50 mL of glacial acetic acid, and titrate with 0.1 ... Test solution Dissolve an accurately weighed quantity of Antazoline Phosphate in methanol to obtain a solution containing 10 mg ...
more infohttps://www.drugfuture.com/Pharmacopoeia/USP32/pub/data/v32270/usp32nf27s0_m4920.html

Antazoline phosphate | VWRAntazoline phosphate | VWR

Learn more about Antazoline phosphate. We enable science by offering product choice, services, process excellence and our ...
more infohttps://us.vwr.com/store/product/20808182/antazoline-phosphate

AntazolineAntazoline

... Systematic (IUPAC) name N-(4,5-dihydro-1H-imidazol-2-ylmethyl)-N-(phenylmethyl)aniline Identifiers CAS ... Antazoline is an antihistamine used to relieve nasal congestion and in eye drops, usually in combination with naphazoline, to ... Antazoline • Azatadine • Bamipine • Cyproheptadine • Deptropine • Dimebon • Ebastine • Epinastine • Ketotifen • Mebhydrolin • ... It uses material from the Wikipedia article "Antazoline". A list of authors is available in Wikipedia. ...
more infohttps://www.chemeurope.com/en/encyclopedia/Antazoline.html

Antazoline Phosphate | BiodiscoveryAntazoline Phosphate | Biodiscovery

Antazoline Phosphate. CAS 91-75-8 (free base), 154-68-7 (phosphate), 2508-72-7 (hydrochloride). Quality: API grade , DMF ... Antazoline phosphate is a histamine H₁-receptor antagonist and is used in eye-drops (treatment of conjunctivitis etc). ...
more infohttps://biodiscovery.eu/products/antazoline-phosphate/

Antazoline | World eBook Library | Read eBooks onlineAntazoline | World eBook Library | Read eBooks online

Antazoline, is a 1st generation ,antihistamine, that also ,anticholinergic, properties ... World Heritage Encyclopedia, the ... Antazoline is a 1st generation antihistamine that also anticholinergic properties used to relieve nasal congestion and in eye ...
more infohttp://ebook.worldlibrary.net/articles/Antazoline

cholinergic antagonist (CHEBI:48873)cholinergic antagonist (CHEBI:48873)

Chemical Entities of Biological Interest (ChEBI) is a freely available dictionary of molecular entities focused on small chemical compounds.
more infohttps://www.ebi.ac.uk/chebi/chebiOntology.do?chebiId=48873

RXQ DRUGRXQ DRUG

ANTAZOLINE; NAPHAZOLINE OPHTHALMIC. d01254. ANTHRALIN TOPICAL. c00131. ANTIASTHMATIC COMBINATIONS - UNSPECIFIED. c00249. ...
more infohttps://wwwn.cdc.gov/Nchs/Nhanes/1999-2000/RXQ_DRUG.htm

Tranylcypromine (Oral Route) Before Using - Mayo ClinicTranylcypromine (Oral Route) Before Using - Mayo Clinic

Although certain medicines should not be used together at all, in other cases two different medicines may be used together even if an interaction might occur. In these cases, your doctor may want to change the dose, or other precautions may be necessary. When you are taking this medicine, it is especially important that your healthcare professional know if you are taking any of the medicines listed below. The following interactions have been selected on the basis of their potential significance and are not necessarily all-inclusive.. Using this medicine with any of the following medicines is not recommended. Your doctor may decide not to treat you with this medication or change some of the other medicines you take.. ...
more infohttps://www.mayoclinic.org/es-es/drugs-supplements/tranylcypromine-oral-route/before-using/drg-20073226

Bupropion (Oral Route) Side Effects - Mayo ClinicBupropion (Oral Route) Side Effects - Mayo Clinic

Check with your doctor before using this medicine with alcohol or other medicines that affect the central nervous system (CNS). The use of alcohol or other medicines that affect the CNS with bupropion may worsen the side effects of this medicine, such as dizziness, poor concentration, drowsiness, unusual dreams, and trouble with sleeping. Some examples of medicines that affect the CNS are antihistamines or medicine for allergies or colds, sedatives, tranquilizers, or sleeping medicines, medicine for depression, medicine for anxiety, prescription pain medicine or narcotics, medicine for attention deficit and hyperactivity disorder, medicine for seizures or barbiturates, muscle relaxants, or anesthetics, including some dental anesthetics. Bupropion may cause some people to be agitated, irritable, or display other abnormal behaviors. It may also cause some people to have suicidal thoughts and tendencies, or to become more depressed. Make sure the doctor knows if you have trouble sleeping, get upset ...
more infohttps://www.mayoclinic.org/drugs-supplements/bupropion-oral-route/side-effects/drg-20062478?p=1

Why is Twelfth Night A Comedy?Why is Twelfth Night A Comedy?

What is Antazoline? In: Science. Answer it! What is the reflection of Beowulf story? In: Beowulf ...
more infohttp://www.answers.com/Q/Why_is_Twelfth_Night_A_Comedy

Pharm.ther. Eye, Ear & Skin | Glaucoma | Human EyePharm.ther. Eye, Ear & Skin | Glaucoma | Human Eye

or formation of a steroid cataract • Antiallergics : antazoline • Local anaesthetics : lidocaine/oxybuprocaine for tonometry. ...
more infohttps://www.scribd.com/presentation/193222129/Pharm-ther-Eye-Ear-Skin
  • This graph shows the total number of publications written about "Antazoline" by people in this website by year, and whether "Antazoline" was a major or minor topic of these publications. (umassmed.edu)
  • Antazoline" is a descriptor in the National Library of Medicine's controlled vocabulary thesaurus, MeSH (Medical Subject Headings) . (umassmed.edu)