Acetamides
Etanidazole
Acetanilides
Cryoprotective Agents
Phenoxypropanolamines
Hares
Amides
Thiourea
A photographic fixative used also in the manufacture of resins. According to the Fourth Annual Report on Carcinogens (NTP 85-002, 1985), this substance may reasonably be anticipated to be a carcinogen (Merck Index, 9th ed). Many of its derivatives are ANTITHYROID AGENTS and/or FREE RADICAL SCAVENGERS.
Indoleacetic Acids
Urea
Dimethyl Sulfoxide
A highly polar organic liquid, that is used widely as a chemical solvent. Because of its ability to penetrate biological membranes, it is used as a vehicle for topical application of pharmaceuticals. It is also used to protect tissue during CRYOPRESERVATION. Dimethyl sulfoxide shows a range of pharmacological activity including analgesia and anti-inflammation.
Semen Preservation
Molecular Structure
Iodoacetates
Alkylation
Structure-Activity Relationship
Glycerol
Cryopreservation
Fluorine Radioisotopes
Pyrazoles
Receptors, Opioid, kappa
Pseudomonas
Pyrimidines
Cell Membrane Permeability
Magnetic Resonance Spectroscopy
Gas Chromatography-Mass Spectrometry
Receptors, GABA-A
Stereoisomerism
Carbon Radioisotopes
Binding Sites
Water
Positron-Emission Tomography
An imaging technique using compounds labelled with short-lived positron-emitting radionuclides (such as carbon-11, nitrogen-13, oxygen-15 and fluorine-18) to measure cell metabolism. It has been useful in study of soft tissues such as CANCER; CARDIOVASCULAR SYSTEM; and brain. SINGLE-PHOTON EMISSION-COMPUTED TOMOGRAPHY is closely related to positron emission tomography, but uses isotopes with longer half-lives and resolution is lower.
Culture Media
Any liquid or solid preparation made specifically for the growth, storage, or transport of microorganisms or other types of cells. The variety of media that exist allow for the culturing of specific microorganisms and cell types, such as differential media, selective media, test media, and defined media. Solid media consist of liquid media that have been solidified with an agent such as AGAR or GELATIN.
delta-Aminolevulinate synthetases in the liver cytosol fraction and mitochondria of mice treated with allylisopropylacetamide and 3,5-dicarbethoxyl-1,4-dihydrocollidine. (1/1656)
Hepatic delta-aminolevulinate (ALA) synthetase was induced in mice by the administration of allylisopropylacetamide (AIA) and 3,5-dicarbethoxy-1,4-dihydrocollidine (DDC). In both cases, a significant amount of ALA synthetase accumulated in the liver cytosol fraction as well as in the mitochondria. The apparent molecular weight of the cytosol ALA synthetase was estimated to be 320,000 by gel filtration, but when the cytosol ALA synthetase was subjected to sucrose density gradient centrifugation, it showed a molecular weight of 110,000. In the mitochondria, there were two different sizes of ALA synthetase with molecular weights of 150,000 and 110,000, respectively; the larger enzyme was predominant in DDC-treated mice, whereas in AIA-treated mice and normal mice the enzyme existed mostly in the smaller form. When hemin was injected into mice pretreated with DDC, the molecular size of the mitochondrial ALA synthetase changed from 150,000 to 110,000. The half-life of ALA synthetase in the liver cytosol fraction was about 30 min in both the AIA-treated and DDC-treated mice. The half-life of the mitochondrial ALA synthetase in AIA-treated mice and normal mice was about 60 min, but in DDC-treated mice the half-life was as long as 150 min. The data suggest that the cytosol ALA synthetase of mouse liver is a protein complex with properties very similar to those of the cytosol ALA synthetase of rat liver, which has been shown to be composed of the enzyme active protein and two catalytically inactive binding proteins, and that ALA synthetase may be transferred from the liver cytosol fraction to the mitochondria with a size of about 150,000 daltons, followed by its conversion to enzyme with a molecular weight of 110,000 within the mitochondria. The process of intramitochondrial enzyme degradation seems to be affected in DDC-treated animals. (+info)Properties of 5-aminolaevulinate synthetase and its relationship to microsomal mixed-function oxidation in the southern armyworm (Spodoptera eridania). (2/1656)
1. Activity of 5-aminolaevulinate synthetase was measured in the midgut and other tissues of the last larval instar of the southern armyworm (Spodoptera eridania Cramer, formerly Prodenia eridania Cramer). 2. Optimum conditions for measuring the activity were established with respect to all variables involved and considerable differences from those reported for mammalian enzyme preparations were found. 3. Maximum activity (20 nmol/h per mg of protein) occurs 18-24 h after the fifth moult and thereafter decreases to trace amounts as the larvae age and approach pupation. 4. Synthetase activity was rapidly induced by oral administration (in the diet) of pentamethylbenzene, phenobarbital, diethyl 1,4-dihydro-2,4,6-trimethylpyridine-3, 5-dicarboxylate, and 2-allyl-2-isopropylacetamide. 5. Puromycin inhibited the induction of synthetase by pentamethylbenzene. 6. Induction of 5-aminolaevulinate synthetase correlated well with the induction of microsomal N-demethylation of p-chloro-N-methylaniline, except for phenobarbital, which induced the microsomal oxidase relatively more than the synthetase. (+info)The in-vitro activity of linezolid (U-100766) and tentative breakpoints. (3/1656)
The in-vitro activity of linezolid, a novel oxazolidinone, was investigated in comparison with those of amoxycillin, cefuroxime, quinupristin/dalfopristin, trovafloxacin and vancomycin against 420 recent Gram-positive and anaerobic clinical isolates. Linezolid was equally active (MIC90 1 mg/L) against methicillin-susceptible and -resistant Staphylococcus aureus. It demonstrated uniform activity against streptococci and enterococci and no cross-resistance with other agents. The time-kill kinetic data demonstrated that the in-vitro activity of linezolid was predominantly bacteriostatic; slow bactericidal activity was only observed at the higher concentration with streptococci. An increase in inoculum from 10(4) to 10(6) cfu on selected strains had little effect on the MICs (MIC90 within one dilution step) of linezolid and an increase in inoculum from 10(5) to 10(7) cfu/mL had no notable effect on the in-vitro bactericidal activity. A tentative linezolid breakpoint of 2 mg/L was chosen after analysis of distribution of susceptibilities. (+info)Aldehyde oxidase-dependent marked species difference in hepatic metabolism of the sedative-hypnotic, zaleplon, between monkeys and rats. (4/1656)
A marked difference in hepatic activity of aldehyde oxidase between rats and monkeys was found to be responsible for the previously reported marked species difference in the metabolism of Zaleplon in vivo. In the postmitochondrial fractions, S-9s, from liver homogenates of these animals, Zaleplon was transformed in the presence of NADPH into the side chain oxidation product, N-desethyl-Zaleplon, and the aromatic ring oxidation product, 5-oxo-Zaleplon. In the rat S-9, N-desethyl-Zaleplon and 5-oxo-Zaleplon were a major and a very minor metabolites, respectively. However, in the monkey S-9, Zaleplon was transformed into 5-oxo-Zaleplon at a much higher rate than that for N-desethyl-Zaleplon formation. N-Desethyl-Zaleplon was formed in the monkey S-9 at a rate almost equal to that in the rat S-9. N-Desethyl-5-oxo-Zaleplon was formed at a minor rate only in the monkey S-9 through N-desethyl-Zaleplon as an obligatory intermediate. The hepatic activity for the formation of 5-oxo-Zaleplon in the monkey and rat was localized in cytosol and did not require NADPH. Sensitivity to various inhibitors and requirement of water as oxygen source, using H218O, strongly suggested that the hepatic cytosolic formation of 5-oxo-Zaleplon was mediated by aldehyde oxidase. N-Desethyl-Zaleplon was formed in the presence of NADPH by microsomes from the liver of rats and monkeys, and its formation was strongly suggested using various cytochrome P-450 inhibitors to be mediated by a number of cytochrome P-450 isoforms, such as 3A, 2C, and 2D subfamilies. (+info)Increased transcriptional activity of prostate-specific antigen in the presence of TNP-470, an angiogenesis inhibitor. (5/1656)
Prostate-specific antigen, PSA, is regarded as a reliable surrogate marker for androgen-independent prostate cancer (AIPC). Concern has been raised that investigational agents may affect PSA secretion without altering tumour growth or volume. In a phase I trial, several patients with AIPC had elevated serum PSA levels while receiving TNP-470 that reversed upon discontinuation. TNP-470 inhibits capillary growth in several angiogenesis models. These observations prompted us to determine if TNP-470, or its metabolite, AGM-1883, altered PSA secretion. Intracellular protein and transcriptional levels of PSA and androgen receptor were also determined. The highest TNP-470 concentration produced a 40.6% decrease in cell number; AGM-1883 had minimal effects on cell viability. PSA secretion per cell was induced 1.1- to 1.5-fold following TNP-470 exposure. The same trend was observed for AGM-1883. PSA and AR were transcriptionally up-regulated within 30 min after exposure to TNP-470. PSA transcription was increased 1.4-fold, while androgen receptor (AR) transcription was induced 1.2-fold. The increased PSA transcriptional activity accounts for the increased PSA secretion. Increased AR transcription was also reflected at the protein level. In conclusion, TNP-470 and AGM-1883 both up-regulated PSA making clinical utilization of this surrogate marker problematic. (+info)Bcl-XL induction during terminal differentiation of friend erythroleukaemia cells correlates with delay of apoptosis and loss of proliferative capacity but not with haemoglobinization. (6/1656)
Friend murine erythroleukaemia (F-MEL) cells are a useful model for studying the processes that regulate erythroid differentiation since exposure of these cells to chemical inducers (DMSO or HMBA) results in commitment to terminal cell division and synthesis of haemoglobin. This study examined the relationship between differentiation and apoptosis in DMSO sensitive and resistant F-MEL cells. Clear apoptosis was not observed in DMSO-treated sensitive F-MEL (strain 745A) cells during the induction of differentiation. In contrast, DMSO-induced 745A cells exhibited delayed apoptosis compared to uninduced cells. Since the Bcl-2 family members play a major role in the control of apoptosis and/or differentiation, we determined their expression before and after DMSO or HMBA treatment. Neither untreated nor chemically-induced 745A cells expressed the Bcl-2 protein. The levels of Bax and Bad proteins remained relatively constant during DMSO-induced differentiation. DMSO or HMBA treatment of 745A cells induced a marked increase of Bcl-XL expression during the late phase of differentiation which persisted even when the cells began to die. This upregulation of Bcl-XL was independent of cell density but was correlated with cell arrest in G0/G1. DMSO treatment induced a similar delay of apoptosis and enhancement of Bcl-XL expression in F-MEL (strain TFP10) cells which fail to synthesize haemoglobin in the presence of DMSO. Dexamethasone, which blocks DMSO-induced differentiation of F-MEL cells, prevented the induction of Bcl-XL. Inhibitors such as imidazole or succinylacetone, which inhibit haemoglobin synthesis but not commitment to terminal cell division, did not suppress Bcl-XL induction in DMSO-induced cells. Taken together, these results indicate that DMSO treatment of F-MEL cells induces a marked increase in Bcl-XL expression suggesting a role for this anti-apoptotic protein in the process of erythroid differentiation in F-MEL cells. Moreover, induction of Bcl-XL during this process seems to be associated with loss of proliferative capacity rather than with haemoglobin synthesis. (+info)Activation of three types of voltage-independent Ca2+ channel in A7r5 cells by endothelin-1 as revealed by a novel Ca2+ channel blocker LOE 908. (7/1656)
1. We have shown that in addition to voltage-operated Ca2+ channel (VOC), endothelin-1 (ET-1) activates two types of Ca2+-permeable nonselective cation channel (NSCC) in A7r5 cells: its lower concentrations (< or = 1 nM; lower [ET-1]) activate only an SK&F 96365-resistant channel (NSCC-1), whereas its higher concentrations (> or = 10 nM; higher [ET-1]) activate an SK&F 96365-sensitive channel (NSCC-2) as well. 2. We now characterized the effects of a blocker of Ca2+ entry channel LOE 908 on NSCCs and store-operated Ca2+ channel (SOCC) in A7r5 cells, and using two drugs, clarified the involvement of these channels in the ET-1-induced increase in the intracellular free Ca2+ concentrations ([Ca2+]i). Whole-cell recordings and [Ca2+]i monitoring with fluo-3 were used. 3. LOE 908 up to 10 microM had no effect on increases in [Ca2+]i induced by thapsigargin or ionomycin, but SK&F 96365 abolished them. 4. In the cells clamped at -60 mV, both lower and higher [ET-1] induced inward currents with linear iv relationships and the reversal potentials of -15.0 mV. Thapsigargin induced no currents. 5. In the presence of nifedipine, lower [ET-1] induced a sustained increase in [Ca2+]i, whereas higher [ET-1] induced a transient peak and a sustained increase. The sustained increases by lower and higher [ET-1] were abolished by removal of extracellular Ca2+, and they were suppressed by LOE 908 to 0 and 35%, respectively, with the LOE 908-resistant part being abolished by SK&F 96365. 6. These results show that LOE 908 is a blocker of NSCCs without effect on SOCC, and that the increase in [Ca2+]i at lower [ET-1] results from Ca2+ entry through NSCC-1 in addition to VOC, whereas the increase at higher [ET-1] involves NSCC-1, NSCC-2 and SOCC in addition to VOC. (+info)Mechanisms of melatonin-induced vasoconstriction in the rat tail artery: a paradigm of weak vasoconstriction. (8/1656)
1. Vasoconstrictor effects of melatonin were examined in isolated rat tail arteries mounted either in an isometric myograph or as cannulated pressurized segments. Melatonin failed by itself to mediate observable responses but preactivation of the arteries with vasopressin (AVP) reliably uncovered vasoconstriction responses to melatonin with maxima about 50% of maximum contraction. Further experiments were conducted with AVP preactivation to 5-10% of the maximum contraction. 2. Responses to melatonin consisted of steady contractions with superimposed oscillations which were large and irregular in isometric but small in isobaric preparations. Nifedipine (0.3 microM) reduced the responses and abolished the oscillations. Charybdotoxin (30 nM) increased the magnitude of the oscillations with no change in the maximum response. 3. Forskolin (0.6 microM) pretreatment increased the responses to melatonin compared to control and sodium nitroprusside (1 microM) treated tissues. The AVP concentration required for preactivation was 10 fold higher than control in both the forskolin and nitroprusside treated groups. 4. In isometrically-mounted arteries treated with nifedipine, melatonin receptor agonists had the potency order 2-iodomelatonin > melatonin > S20098 > GR196429, and the MT2-selective antagonist luzindole antagonized the effects of melatonin with a low pK(B) of 6.1+/-0.1. 5. It is concluded that melatonin elicits contraction of the rat tail artery via an mt1 or mt1-like receptor that couples via inhibition of adenylate cyclase and opening of L-type calcium channels. Calcium channels and charybdotoxin-sensitive K channels may be recruited into the responses via myogenic activation rather than being coupled directly to the melatonin receptors. 6. It is proposed that the requirement of preactivation for overt vasoconstrictor responses to melatonin results from the low effector reserve of the melatonin receptors together with the tail artery having threshold inertia. Potentiative interactions between melatonin and other vasoconstrictor stimuli probably also result from the threshold inertia. A simple model is presented and a general framework for consideration of interactions between weak vasoconstrictor agonists and other vasoconstrictor stimuli is discussed. (+info)
N,N-dimethylacetamide - Registration Dossier - ECHA
CCCC 1983, Volume 48, Issue 11, Abstracts pp. 3214-3222 | Collection of Czechoslovak Chemical Communications
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Acetylation
Acetate esters and acetamides are generally prepared by acetylations. Acetylations are often used in making C-acetyl bonds in ...
DPA-713
... pyrimidine acetamides: 4-Phenyl alkyl ether derivatives as potent ligands for the 18 kDa translocator protein (TSPO)". ... pyrimidin-3-yl acetamides. New potent and selective peripheral benzodiazepine receptor ligands". Bioorg. Med. Chem. 9 (10): ...
Hypocretin (orexin) receptor 2
October 2008). "Synthesis of (3,4-dimethoxyphenoxy)alkylamino acetamides as orexin-2 receptor antagonists". Bioorganic & ... alkylamino acetamides Compound 1m - Selective OX2 antagonist Orexin receptor GRCh38: Ensembl release 89: ENSG00000137252 - ...
Chitin-glucan complex
v t e (Acetamides, Biomolecules, Biopesticides, Polysaccharides, All stub articles, Biochemistry stubs). ...
Acetyl bromide
It also reacts with alcohols and amines to produce acetate esters and acetamides, respectively. Acetyl bromide[permanent dead ...
Phosphoramidite ligand
These ligands afford a very active and productive catalyst, which efficiently reduces a various acetamides. It is worth noting ...
PD-168,077
... acetamides: selective dopamine D4 receptor agonists". Bioorganic & Medicinal Chemistry. 12 (13): 3471-83. doi:10.1016/j.bmc. ...
1-Tetralone
... acetamides", J. Org. Chem. (in German), vol. 38, no. 23, pp. 4073-4074, doi:10.1021/jo00987a029 "1-Phenylnaphthalene". Organic ...
Ro07-5220
Structure-activity relationship between substituted 2-amino-N-(2-benzoyl-4-chlorophenyl)acetamides and 1,4-benzodiazepinones". ...
Alpidem
... acetamides as Probes of Mitochondrial Steroidogenesis-A New Mechanism for GABAA Receptor Modulation". Angewandte Chemie ...
Ethenone
It does for example react with water to acetic acid or with primary or secondary amines to the corresponding acetamides. In ...
DPA-714
... pyrimidine acetamides: 4-Phenyl alkyl ether derivatives as potent ligands for the 18 kDa translocator protein (TSPO)". Bioorg. ...
Passerini reaction
... acetamides by a ThreeComponent Reaction between an Isocyanide, Quinoline-4-carbaldehyde, and Arenecarboxylic Acids". Helvetica ... acetamides by a ThreeComponent Reaction between an Isocyanide, Quinoline-4-carbaldehyde, and Arenecarboxylic Acids". Helvetica ... acetamides by a ThreeComponent Reaction between an Isocyanide, Quinoline-4-carbaldehyde, and Arenecarboxylic Acids". Helvetica ... acetamides by a ThreeComponent Reaction between an Isocyanide, Quinoline-4-carbaldehyde, and Arenecarboxylic Acids". Helvetica ...
Valrubicin
Acetamides, Withdrawn drugs). ...
Cefadroxil
Acetamides). ...
List of benzimidazole opioids
US 2944062, Hoffman K, Hunger A, "Certain Alpha (1-diethylaminoethyl (2), Alpha Aryl Acetamides", issued 5 July 1960, assigned ...
Dirlotapide
Acetamides, Biphenyls). ...
Thioacetic acid
Salts of thioacetic acid such as potassium thioacetate can be used to do one-step conversion of nitroarenes to aryl acetamides ...
Phenylpiracetam
Acetamides, Drugs in sport, Drugs in the Soviet Union, Nicotinic agonists, Nootropics, Norepinephrine-dopamine reuptake ...
Modafinil sulfone
Acetamides, Anticonvulsants, Benzhydryl compounds, Human drug metabolites, Sulfones, All stub articles, Nervous system drug ...
Pirenzepine
Acetamides, Peripherally selective drugs, All stub articles, Gastrointestinal system drug stubs). ...
Oxetacaine
Acetamides, Primary alcohols, All stub articles, Cardiovascular system drug stubs, Nervous system drug stubs). ...
TIK-301
Acetamides, Phenol ethers, Melatonin receptor agonists). ...
Acetoxolutamide
Acetamides, Selective androgen receptor modulators, Trifluoromethyl compounds, Nitro compounds, Tertiary alcohols, All stub ...
Melatonin
Acetamides, Antioxidants, Aromatase inhibitors, Circadian rhythm, Hormones of the pineal gland, Melatonin receptor agonists, ...
Melatonin as a medication and supplement
Acetamides, Antidepressants, Antioxidants, Aromatase inhibitors, Circadian rhythm, Drugs acting on the nervous system, ...
Ketoconazole
Acetamides, Aldosterone synthase inhibitors, Antifungals for dermatologic use, Antiglucocorticoids, Aromatase inhibitors, ...
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Acetamides, Drugs acting on the cardiovascular system, Japanese brands, Pyrazines, Sulfonamides, Isopropyl compounds, ...
ALD-52
Acetamides). ...
Indantadol
Acetamides). ...
Browsing Technical Documents by Subject "Acetamides"
Browsing by Subject "Acetamides"
Silicon‐Mediated Synthesis of Acetamides - ChemistryViews
Silicon‐Mediated Synthesis of Acetamides. Author: Angewandte Chemie International Edition. The activation and coupling of small ... Silicon-Mediated Coupling of Carbon Monoxide, Ammonia, and Primary Amines to Form Acetamides,. Marcel-Philip Luecke, Arseni ... and primary amines to form acetamides. The transformation starts with the deoxygenative homocoupling of two CO molecules at two ...
IMSEAR at SEARO: Synthesis and anticonvulsant activity of 6-methyl-2-thioxo-2, 3-dihydropyrimidin-4(1H)-one acetamides
Synthesis and anticonvulsant activity of 6-methyl-2-thioxo-2, 3-dihydropyrimidin-4(1H)-one acetamides. Journal of Applied ... Synthesis and anticonvulsant activity of 6-methyl-2-thioxo-2, 3-dihydropyrimidin-4(1H)-one acetamides. ... thio-acetamides. An initial intermediate 6-methyl-2-thioxo-2,3-dihydro-pyrimidin-4(1Н)-one was obtained by thereaction of ...
N-alkylation of azoles disubstituted acetamides under microwave and Mannich reaction conditions | Abstract
... acetamides, was carried out under different conditions basic, micro.. ... The N-alkylation of some secondary amides, 2-(1H-azol-1-yl)-N-(substituted phenyl) acetamides, was carried out under different ... N-alkylation of azoles disubstituted acetamides under microwave and Mannich reaction conditions. Author(s): Ambarsing P. Rajput ...
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Synthesis3
- Synthesis of acetamides 2 . (beilstein-journals.org)
- Synthesis and evaluation of 3-ylideneoxindole acetamides as potent anticancer agents. (cocites.com)
- Note also that the widely used synthesis of acetyl - acetamides by the addition of primary or secondary amines to diketene is not relevant to this section. (thieme.com)
Amides1
- The N-alkylation of some secondary amides, 2-(1H-azol-1-yl)-N-(substituted phenyl) acetamides, was carried out under different conditions basic, microwave and Mannich reaction. (derpharmachemica.com)
Herbicides1
- Growth regulators and acetamides are the herbicides most commonly associated with twisted whorls or 'buggy-whipping. (pioneer.com)
Phenyl2
- A series of Schiff's bases N'-(substituted benzylidene)-2-(naphthalen-1-yloxy) acetohydrazides (3a-f) and azetidinones N-[3-chloro-2-oxo-4-(substituted phenyl)-azetidin-1-yl]-2-(naphthalen-1-yloxy) acetamides (4a-b) were synthesized and tested for antimicrobial activity. (technologynetworks.com)
- Identification of new compounds with anticonvulsant and antinociceptive properties in a group of 3-substituted (2,5-dioxo-pyrrolidin-1-yl)(phenyl)-acetamides. (krakow.pl)
Amino1
- In the current work, new 2-[(4-amino-5-aryl-4H-1,2,4-triazol-3-yl)thio]-N-(thiazol/benzothiazol-2-yl)acetamides (1-18) were synthesized and evaluated for their inhibitory capacities on AR. (bilecik.edu.tr)
Amines1
- Matthias Driess and colleagues, Technische Universität Berlin, Germany, have developed a silicon-mediated direct coupling of carbon monoxide, ammonia, and primary amines to form acetamides. (chemistryviews.org)
Reaction2
- Glorius, F. Palladium-catalyzed Heck-type reaction of 2-chloro acetamides with olefins. (mpg.de)
- The method offers mild reaction conditions, as well as wide substrate scope that is particularly compatible with some internal aromatic alkynes and acetamides. (organic-chemistry.org)
Library1
- A small library of quinazolin-4-one clubbed thiazole acetates/acetamides lacking toxicity-producing functionalities was designed, synthesized, and evaluated for antidiabetic potential as glucokinase activators (GKA). (springeropen.com)
Aromatic1
- Chemical modification of 10E8 with aromatic acetamides facilitates the productive and specific recognition of the native antigen, partially buried in the crowded environment of the viral membrane, resulting in a dramatic increase of its capacity to block viral infection. (pasteur.fr)
Compounds1
- So some new compounds, substituted acetamides bearing indole moiety which are related to rivastigmine were designed and synthesized. (manipal.edu)
Inhibitors4
- 2-((1H-indol-3-yl)thio)-N-phenyl-acetamides: SARS-CoV-2 RNA-dependent RNA polymerase inhibitors. (amedeo.com)
- 1. Potent dual EGFR/Her4 tyrosine kinase inhibitors containing novel (1,2-dithiolan-4-yl)acetamides. (nih.gov)
- Discovery of inhibitors of the mitotic kinase TTK based on N-(3-(3-sulfamoylphenyl)-1H-indazol-5-yl)-acetamides and carboxamides. (sigmaaldrich.com)
- Discovery of pyrazolo-thieno[3,2-d]pyrimidinylamino-phenyl acetamides as type-II pan-tropomyosin receptor kinase (TRK) inhibitors: Design, synthesis, and biological evaluation. (uams.edu)
Order1
- The DNA-cleaving ability of conjugates does not directly follow the order of the photocycloaddition of their acetamides. (cytologycongress.org)