Structure-Activity RelationshipMolecular StructureLobelineMolecular Sequence DataDrug DesignModels, MolecularStereoisomerismProtein ConformationAmino Acid SequenceDrug Screening Assays, AntitumorMass SpectrometryKineticsInhibitory Concentration 50Protein BindingBinding SitesMagnetic Resonance SpectroscopyChromatography, High Pressure LiquidLigandsCircular DichroismSpectrometry, FluorescenceProdrugsEscherichia coliMolecular ConformationBinding, CompetitiveMicroscopy, ElectronMutationCell Line, TumorProtein Structure, SecondaryAntineoplastic AgentsDNADrug Evaluation, PreclinicalCell LineOxidation-ReductionProtein Processing, Post-TranslationalModels, ChemicalBase SequenceDose-Response Relationship, DrugHydrogen-Ion ConcentrationCrystallography, X-RayProtein Structure, TertiaryNucleic Acid ConformationModels, BiologicalPeptide FragmentsCells, CulturedCell SurvivalSubstrate SpecificityTemperatureSequence Homology, Amino AcidElectrophoresis, Polyacrylamide GelAnti-Bacterial AgentsTime FactorsThermodynamicsCricetinaeBacterial ProteinsRecombinant ProteinsPhosphorylationRats, Sprague-DawleyCattleEnzyme InhibitorsCell MembraneLiverHistonesMethylationLysineAcetylationEpigenesis, GeneticSUMO-1 ProteinCysteineChromatinDiethyl PyrocarbonateGlycosylationDNA MethylationProtein Modification, TranslationalSmall Ubiquitin-Related Modifier ProteinsSulfhydryl CompoundsAcetylglucosamineSumoylationPhenylglyoxalBromosuccinimideTranscription, GeneticProteinsChromatin Assembly and DisassemblySpectrometry, Mass, Matrix-Assisted Laser Desorption-IonizationHistone CodeChromatin ImmunoprecipitationPeptidesMutagenesis, Site-DirectedRNA, TransferTetranitromethaneEpigenomicsHeLa CellsSaccharomyces cerevisiaeMethyltransferasesProteomicsUbiquitinationPromoter Regions, GeneticGene Expression RegulationCarbodiimidesHistone-Lysine N-MethyltransferaseEthylmaleimide