Small Molecule LibrariesNeurotransmitter AgentsCell Adhesion MoleculesModels, MolecularMolecular Sequence DataProtein BindingHigh-Throughput Screening AssaysMolecular StructureSignal TransductionDrug Evaluation, PreclinicalSerotoninAmino Acid Sequencegamma-Aminobutyric AcidDrug DesignBinding SitesLigandsNeuronsDopamineDrug DiscoveryCells, CulturedCell LineGlutamic AcidStructure-Activity RelationshipBiogenic MonoaminesKineticsCell Line, TumorBrainNeuropeptidesCombinatorial Chemistry TechniquesProtein ConformationEnzyme InhibitorsNorepinephrineProtein Structure, TertiaryDose-Response Relationship, DrugCrystallography, X-RayModels, BiologicalBase SequencePeptidesSynaptic TransmissionRats, Sprague-DawleyNeurochemistryMutationMice, Inbred C57BLInhibitory Concentration 50CalciumRecombinant ProteinsCatecholaminesProteinsAcetylcholineFluorescent DyesAntineoplastic AgentsProtein Kinase InhibitorsCell MembraneTime FactorsSynaptic VesiclesGlycineRNA, MessengerReceptors, NeurotransmitterPhosphorylationPeptide FragmentsBrain ChemistryMolecular ConformationImmunohistochemistryTransfectionGlutamatesMembrane ProteinsMolecular Docking SimulationIndolesAntibodies, MonoclonalCell ProliferationGene Expression RegulationApoptosisNeurotransmitter Transport ProteinsOctopamineCarrier ProteinsSynaptosomesAmino AcidsCell SurvivalDNANerve Tissue ProteinsBlotting, WesternMonoamine OxidaseMagnetic Resonance SpectroscopyChromatography, High Pressure LiquidNeurosecretory SystemsNeural Cell Adhesion MoleculesPiperazinesMice, KnockoutRats, WistarBiological TransportExocytosisDrug Screening Assays, AntitumorAdenosine TriphosphateMicrodialysisCell AdhesionMolecular WeightVasoactive Intestinal PeptideHydroxyindoleacetic AcidNeuropeptide YReceptors, G-Protein-Coupled