Allosteric RegulationAllosteric SiteReceptor, Metabotropic Glutamate 5CyclohexylaminesReceptors, Metabotropic GlutamateErythrocebus patasReceptors, Calcium-SensingReceptors, NicotinicStructure-Activity RelationshipPyridinesBenzamidesDose-Response Relationship, DrugCalciumRadioligand AssayReceptors, GABA-AAlcuroniumGABA ModulatorsHEK293 CellsBinding SitesCricetinaePhthalimidesModels, MolecularProtein Bindingalpha7 Nicotinic Acetylcholine ReceptorGallamine TriethiodideBinding, CompetitiveN-MethylscopolamineRats, Sprague-DawleyIsoxazolesCell LineKineticsReceptor, Muscarinic M4MSH Release-Inhibiting HormoneLigandsCholinergic AgentsGABA-A Receptor AgonistsReceptor, Muscarinic M1BenzothiadiazinesBenzodiazepinesPregnanoloneCricetulusNootropic AgentsCHO CellsReceptor, Muscarinic M2Bicyclo CompoundsPhenylurea CompoundsNicotinic AgonistsGABA-B Receptor AgonistsObidoxime ChlorideExcitatory Amino Acid AgentsDiazepamXenopus laevisMolecular StructureNicotinic AntagonistsDrug DiscoveryReceptor, Muscarinic M5ThiophenesGalantaminePiperidinesGABA AgentsProtein Structure, TertiaryDrug DesignHydrocarbons, BrominatedReceptors, GABA-BProtein ConformationDrug Partial AgonismExcitatory Amino Acid AgonistsReceptors, G-Protein-CoupledReceptors, AMPAMuscarinic AgonistsPentobarbitalGABA AgonistsGlutamic AcidOocytesReceptor, Adenosine A1Central Nervous System AgentsProtein SubunitsXanthenesPeptidomimeticsThiadiazolesHigh-Throughput Screening AssaysPatch-Clamp TechniquesPregnanedionesAniline CompoundsQuinolizidinesReceptors, MuscarinicAmino Acid SequenceAlprazolamReceptor, Adenosine A3Molecular Sequence DataMutagenesis, Site-DirectedDrug Evaluation, PreclinicalReceptors, GlycineSelective Estrogen Receptor ModulatorsBaclofenExcitatory Amino Acid AntagonistsAnti-Anxiety AgentsCarbolinesgamma-Aminobutyric AcidBicyclo Compounds, Heterocyclic