• Dimenhydrinate, diphenhydramine, cyclizine, or meclizine: take 1 hour before departure and continue during the trip. (tripprep.com)
  • Four over-the-counter medications that are approved in the US for this use are cyclizine (Marezine), dimenhydrinate (Dramamine), diphenhydramine (Benadryl), and meclizine (Bonine and Dramamine II). (tripprep.com)
  • Cyclizine is a piperazine derivative with histamine H1-receptor antagonist (antihistamine) activity. (wikipedia.org)
  • Cyclizine was developed in the American division of pharmacy company Burroughs Wellcome (today GlaxoSmithKline) during a research study involving many drugs of the antihistamine group. (wikipedia.org)
  • Explanation: Cyclizine is type of antihistamine that acts on the H1 receptor. (mrcoggoal.com)
  • Prescribe an antihistamine (oral cyclizine or oral promethazine), or a phenothiazine (oral prochlorperazine), and reassess after 24 hours. (patient.info)
  • 6. These data suggest that systemic injection of the 5-HT6 antagonist, Ro 04-6790, produces a stretching behaviour that appears to be mediated by an increase in cholinergic neurotransmission in the CNS and which could be a useful functional correlate for 5-HT6 receptor blockade. (lookformedical.com)
  • Cyclizine was marketed as Bonine for Kids in the US, but was discontinued in 2012, and replaced with meclizine. (wikipedia.org)
  • As cyclizine hydrochloride tablets and cyclizine lactate solution for intramuscular or intravenous injection (brand names: Valoid in UK and South Africa and Marezine, Marzine and Emoquil in US). (wikipedia.org)
  • In pregnancy NICE guidelines advise oral promethazine or oral cyclizine should be used as 1st line drug management of nausea and vomitting. (mrcoggoal.com)
  • The drug Diconal is a combination of cyclizine and the opioid dipipanone. (wikipedia.org)
  • Antihistamines like cyclizine and tripelennamine are sometimes mixed with morphine to increase both, a potentially dangerous practise via unsupervised injection but one used medically with oral opioid administration and under direct supervision of a doctor and nurse via the IV and SC routes in particular. (dieutridau.com)
  • This photosensitization of the skin may be caused by creams or ointments applied to the skin, by medications taken orally or by injection, or by the use of prescription inhalers. (wisconsin.gov)
  • Persons with nausea and vomiting may not be able to take oral drugs and may require strong sedatives that are administered by injection or suppository. (tripprep.com)
  • LD50 = mg / kg (por vía oral en ratas). (pharmacycode.com)
  • What injections can be given orally or via enteral feeding tubes? (sps.nhs.uk)
  • Cyclizine appears to be safe during pregnancy but has not been well studied. (wikipedia.org)
  • Hormonal methods of birth control include the pill, the patch, the ring, and the injection. (medsforless.co.uk)
  • CONCLUSION: The introduction of a liquid material which solidifies after injection in a short time (hydrogel) using a needle is feasible. (bvsalud.org)
  • It can be taken simply by mouth and injected directly with the help of needle injection. (anglebiopharma.com)
  • Cyclizine may be prepared by the Eschweiler-Clarke methylation of diphenylmethylpiperazine or by reaction of benzhydryl bromide with 1-methylpiperazine in acetonitrile to form the hydrobromide salt of the drug. (wikipedia.org)
  • Some people using methadone recreationally combine cyclizine with their methadone dose, a combination that is known to produce strong psychoactive effects. (wikipedia.org)
  • Cyclizine was quickly clinically found as a potent and long-acting antiemetic. (wikipedia.org)
  • Cyclizine was marketed as Bonine for Kids in the US, but was discontinued in 2012, and replaced with meclizine. (wikipedia.org)
  • Bonine For Kids (cyclizine). (drugs.com)
  • CSCIs reduce the need for bolus injections, provide comfort from stable drug plasma concentrations, and allow control of multiple symptoms with a combination of drugs. (patient.info)
  • are routinely available to astronauts primarily in oral dosage forms (tablets and capsules), but intramuscular injections, rectal suppositories, ocular preparations, and topical agents are also available in the on-board medical kit. (medscape.com)
  • Intramuscular injections are one of the most common clinical procedures. (bvsalud.org)
  • The use of intramuscular injections is not recommended. (patient.info)
  • As cyclizine hydrochloride tablets and cyclizine lactate solution for intramuscular or intravenous injection (brand names: Valoid in UK and South Africa and Marezine, Marzine and Emoquil in US). (wikipedia.org)
  • For the sixth flight (May 1963), cyclizine and meperidine injections and dextroamphetamine tablets were supplied. (medscape.com)
  • Short course antibiotic tablets, for when you can't have the injection in a clinic. (treated.com)
  • Tablets or injections. (treated.com)
  • This randomised, controlled, double-blind study examined the effectiveness of a single dose of ondansetron (0.1 mg x kg-1), cyclizine (20 mg) and placebo (normal saline) in the prevention of postoperative nausea and vomiting in 150 children (mean age 3.6 years) undergoing plastic genitourinary procedures. (nih.gov)
  • Some people using methadone recreationally combine cyclizine with their methadone dose, a combination that is known to produce strong psychoactive effects. (wikipedia.org)
  • Some can be given first off as an injection by your doctor in the hope you would then keep the next dose down orally. (pregnancysicknesssupport.org.uk)
  • Antihistamines in relatively high doses given by injection can decrease basal serum prolactin in nonlactating women and in early postpartum women. (drlact.com)
  • [6] It has also been used as an antipsychotic in doses ranging from 5 to 10 mg given as an intramuscular injection, generally in cases of severe agitation in a psychotic patient who is refusing oral medication. (cloudfront.net)
  • To describe the magnitude of the problem of abuse by self-injection of dipianone HCl/cyclizine HCl (Wellconal) and to document the associated morbidity, mortality and prevalence of HIV infection. (elsevierpure.com)
  • This document contains side effect information about cyclizine. (drugs.com)
  • epinephrine (1:1000), cyclizine for motion sickness (45 mg/0.9 mL), and meperidine for pain (90 mg/0.9 mL). (medscape.com)
  • There is a lack of anti-emetic trials performed in children, with only a few investigating the roles of the older anti-emetic agents such as cyclizine compared with newer ones such as ondansetron. (nih.gov)
  • Cyclizine, sold under a number of brand names, is a medication used to treat and prevent nausea, vomiting and dizziness due to motion sickness or vertigo. (wikipedia.org)
  • Cyclizine was introduced to many countries as a common antiemetic. (wikipedia.org)