Drug DesignMolecular StructureStructure-Activity RelationshipDrug DiscoveryInhibitory Concentration 50Drug Evaluation, PreclinicalSmall Molecule LibrariesCombinatorial Chemistry TechniquesHigh-Throughput Screening AssaysDrug Screening Assays, AntitumorModels, MolecularEnzyme InhibitorsAntineoplastic AgentsMolecular Docking SimulationStereoisomerismSpiro CompoundsBiological ProductsCell Line, TumorQuantitative Structure-Activity RelationshipPlant ExtractsDatabases, ChemicalLigandsDose-Response Relationship, DrugMagnetic Resonance SpectroscopyAzo CompoundsParasitic Sensitivity TestsTrypanocidal AgentsHeterocyclic CompoundsCrystallography, X-RayAntiprotozoal AgentsProtein BindingAntiparasitic AgentsSulfur CompoundsAxinellaBinding SitesChalconeAgelasFuransAdamantaneVolatile Organic CompoundsCell SurvivalChalconesCell LineNitrofuransThiazolesMolecular ConformationAntiviral AgentsTriterpenesPoriferaCoccidiostatsIndolespara-AminobenzoatesMicrobial Sensitivity TestsMolecular Sequence DataKineticsChemistry Techniques, SyntheticThiosemicarbazonesPharmaceutical PreparationsPyransProdrugsAnti-Bacterial AgentsBenzophenonesLeadCell ProliferationAntimalarialsThiostreptonAziridinesBenzofuransPeptidesChromatography, High Pressure LiquidCatalytic DomainAmino Acid SequenceDiterpenesModels, ChemicalPlants, MedicinalPyridinesIndicators and ReagentsTerpenesPlasmodium falciparumEnoyl-(Acyl-Carrier-Protein) Reductase (NADH)CoumarinsTubulin ModulatorsBiological AssayApoptosisAntitubercular AgentsBiological AvailabilityChemistry, PharmaceuticalTriazolesAmidesBenzothiazolesSubstrate SpecificityThiophenesAminopyridinesAlkaloidsPhenolsQuinolinesPyrazolesMass SpectrometryBiphenyl CompoundsNeoplasms