Derivative butyrophenones. Medical search. Frequent questions

It is structurally similar to terfenadine and haloperidol (a butyrophenone antipsychotic ). (wikidoc.org)

Phenothiazines or butyrophenones are known to act at both pre and post-synaptic dopamine receptors, whereas butaclamol or thioxanthenes are supposed to act preferentially at post-synaptic receptors. (erowid.org)
The anticholinergic effect of drugs such as tri- and tetracyclic antidepressants, antihistamines, quinidine, amantadine, antipsychotics (e.g. butyrophenones, phenothiazines), disopyramide and other anticholinergics (e.g. tiotropium, ipratropium, atropine-like compounds) may be intensified by Buscopan. (janusinfo.se)

Other neuroleptics, phenothiazine thioxantene, and butyrophenone derivatives do not affect brain 5-HT levels. (erowid.org)

Trifluperidol is a typical antipsychotic of the butyrophenone chemical class. (wikipedia.org)
Haldol antipsychotic remedy, butyrophenone derivative. (happyfamilymedstore.com)
The atypical antipsychotic risperidone , although not a butyrophenone, was developed with the structures of benperidol and lenperone as a basis. (wikidoc.org)

Combinations of concentrations of butyrophenones or control EPI (chlorpromazine) along with ciprofloxacin (CIP) were utilized in checkerboard assays to determine their minimum inhibitory concentration (MIC) and fractional inhibitory concentration (FIC). (confex.com)

Domperidone , an dopamine-antagonist antiemetic , derived further from butyrophenone (not being a butyrophenone itself). (wikidoc.org)
1) Rabbit retinae in vitro were used to test potential dopamine agonist- and or antagonist-activity of a synthetic derivative, meter-goline, by measuring the formation of cAMP in intact- or homogenized-tissue. (erowid.org)
Parlodel® (bromocriptine mesylate) is an ergot derivative with potent dopamine receptor agonist activity. (rxlist.com)
Two calcium channel blockers available in Europe and South America , which are piperazine derivatives, are thought to cause drug-induced parkinsonism by blocking dopamine receptors. (parkinsonsinfoclub.com)

Consequently, the reports of toxicologic and pharmacologic effects of crude extracts or synthetic derivatives of cannabis published before 1968 lack precision and uniformity and preclude any quantitative correlation between physiological effects and chemical composition. (unodc.org)
These effects are less likely to occur with synthetic derivatives when used in large doses. (recallguide.org)
Opioids are either made from naturally occurring opiates (extracted from the poppy plant) or synthetic derivatives of them (synthetic opioids). (anrclinic.com)

For all of our butyrophenone compounds we observed a reduction in the MIC of ciprofloxacin in S. aureus 1199B reversing its susceptibility from resistant to susceptible. (confex.com)

some of its derivatives (called commonly butyrophenones ) are used to treat various psychiatric disorders such as schizophrenia , as well as acting as antiemetics . (wikidoc.org)

With neuroleptic drugs, the most significant changes in 5-HT metabolism in the brain are produced by Rauwolfia serpentine alkaloids and benzoquinoline derivatives. (erowid.org)
The MICs for all three butyrophenones, was greater than 200 ug/mL in both strains, demonstrating that on their own, these drugs would be considered non-antibiotics. (confex.com)
Butyrophenones are a class of pharmaceutical drugs derived from butyrophenone. (wikidoc.org)

All together these results show that butyrophenones are inhibitors of the NorA efflux pump , and its derivatives have potential for treating ciprofloxacin resistant S. aureus infections in combination therapy. (confex.com)

The efflux assays demonstrated that butyrophenones were able to reduce the loss of ethidium bromide fluorescence over time, confirming a blockage of the NorA efflux pump. (confex.com)

Haloperidol (hal" oh per' i dol) is a butyrophenone derivative which appears to act as a dopamine type 2 (D2) receptor antagonist, but has other central and peripheral effects. (nih.gov)

Since Cabaser exerts its therapeutic effect by direct stimulation of dopamine receptors, it should not be concurrently administered with drugs which have dopamine antagonist activity (such as phenothiazines, butyrophenones, thioxanthines, metoclopramide) as these might reduce the therapeutic effect of Cabaser. (restarajasthan.com)
It has potential in the treatment of hepatitis C . Silymarin reduces liver damage caused by lipid peroxidation in patients taking butyrophenones or phenothiazines. (joyfoodshop.com)

11. TLC differentiation of butyrophenone and diphenylbutylpiperidine compounds from phenothiazine derivatives. (nih.gov)

By analogy with other ergot derivatives, Cabaser should not be used in association with macrolide antibiotics (e. (restarajasthan.com)

Derivatives of the simplest aromatic ketone acetophenone (of general formula C6H5C(O)CH3). (nih.gov)

18. Which of the following xanthine derivative has bronchodilator action? (rankfiles.com)

Increased sensitivity to the drug, other sulfonamide derivatives or other ingredients, anuria, refractory hypokalemia, severe liver failure (including encephalopathy) and / or severe renal impairment (creatinine clearance less than 30 mL / min), pregnancy, breast feeding, age and 18 years (effectiveness and safety have been established). (pharmru.com)

AHR -1900 hydrochloride is a butyrophenone derivative used in the treatment of schizophrenia. (targetmol.com)
A butyrophenone used in the treatment of PSYCHOSES. (bvsalud.org)
The invention discloses novel aminopyrimidine derivatives, synthesis and uses thereof for the treatment of diseases mediated directly or indirectly by the tachykinin receptors. (justia.com)

A triazene derivative with antineoplastic activity. (blogspot.com)
Azaperone is a butyrophenone tranquilizer that exhibits sedative activity through the inhibition of α-adrenergic receptors. (lktlabs.com)